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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T130428 Destruxin CHL

Destruxin CHL 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T130428。
T20525 Chloramphenicol palmitate

Antibacterial; Antibiotic Microbiology/Virology
Chloramphenicol palmitate 是一种广谱抗生素,对革兰氏阳性和革兰氏阴性细菌具有活性。 Chloramphenicol palmitate 可用于在含有氯霉素抗性基因的转化细胞中作为细菌选择剂的研究。
T28229 Olanexidine hydrochloride

OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045

Antibacterial Microbiology/Virology
Olanexidine hydrochloride (OPB-2045 HCl) 对革兰氏阳性菌和革兰氏阴性菌具有杀菌活性。 Olanexidine hydrochloride 破坏金黄色葡萄球菌的膜完整性。
T7470 6-Chloropurine

6-氯嘌呤,6-Chloro-9H-purine

Others Others
6-Chloropurine (6-Chloro-9H-purine) 是一种制备9-烷基嘌呤和6-巯基嘌呤的中间体,是化学合成的砌块,具有抗肿瘤作用。
T61338 MS023 dihydrochloride

MS023 2HCl

Histone Methyltransferase Chromatin/Epigenetic
MS023 dihydrochloride (MS023 2HCl) 是一种具有选择性、细胞活性和高效性的人I 型蛋白精氨酸甲基转移酶 (PRMTs)抑制剂,具有抗肿瘤活性,抑制 PRMT1,PRMT3,PRMT4,PRMT6和PRMT8,增加离体培养的 MuSC 的增殖能力,可用于研究乳腺癌。
T72322 R 59-022 hydrochloride

DKGI-I hydrochloride,Diacylglycerol kinase inhibitor I hydrochloride,DKGI-I hydrochloride ; Diacylglycerol kinase inhibitor I hydrochloride

5-HT Receptor; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; GPCR/G Protein; Neuroscience
R 59-022 hydrochloride (DKGI-I hydrochloride) 是一种 5-HT Receptor 拮抗剂,可激活蛋白激酶 C (PKC)。R 59-022 hydrochloride 是一种 DGK 抑制剂 (IC50:2.8 µM),可抑制 OAG 磷酸化为 OAPA。R 59-022 增强血小板中凝血酶诱导的甘油二酯的产生,并抑制嗜中性粒细胞中磷脂酸的产生。
T22831 Protein kinase inhibitor H-7 dihydrochloride

H-7 dihydrochloride

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride0) 是一种有效的蛋白激酶 C(PKC)抑制剂。Protein kinase inhibitor H-7 dihydrochloride(100 μM)显著抑制 TPA (皮肤肿瘤启动子,12-O-tetradecanoylphorbol-13-acetate) 和磷脂酶 C 促使的 ODC (鸟氨酸脱羧酶),抑制 PMA 诱导的混杂细胞溶解活性。
T14333 Asoxime dichloride

Tert-Butyl2-(2-hydroxyethyl)-1-pyrrolidinecarboxylate,Asoxime (dichloride),HI-6

AChR Neuroscience
Asoxime dichloride (Tert-Butyl2-(2-hydroxyethyl)-1-pyrrolidinecarboxylate) 是乙酰胆碱受体 (AChRs) 拮抗剂,包括烟碱受体,α7 乙酰胆碱受体。Asoxime dichloride 参与调节免疫应答。Asoxime dichloride 可作为抗原使用,改善神经系统的免疫效果。
T38846 Vevorisertib trihydrochloride

ARQ 751 trihydrochloride

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Vevorisertib trihydrochloride(ARQ 751 trihydrochloride) 是一种具有选择性和有效性的 pan-AKT 和 AKT1-E17K 突变抑制剂,抑制 AKT1 、AKT2 和 AKT3 。 Vevorisertib trihydrochloride 可用于研究肝癌和晚期实体瘤。
T60248 4-Aminobenzamidine dihydrochloride

p-Aminobenzamidine dihydrochloride

Serine Protease Proteases/Proteasome
4-Aminobenzamidine dihydrochloride (p-Aminobenzamidine dihydrochloride) 是一种强胰蛋白酶 (trypsin)抑制剂,也是一种相对较弱的尿激酶型纤溶酶原激活剂 (uPA) 抑制剂 (Ki=82 μM)。4-Aminobenzamidine 可抑制 SCID 小鼠体内前列腺肿瘤的生长。
T14954 Chlorthal-dimethyl

Dimethyl tetrachloroterephthalate

Others Others
Chlorthal-dimethyl (Dimethyl tetrachloroterephthalate) 用作农药中间体。
T37034 H-Gly-Arg-pNA dihydrochloride

H-Gly-Arg-Pna 2HCl

H-Gly-Arg-pNA dihydrochloride (H-Gly-Arg-Pna 2HCl) 属于多肽类,可与1,2凝血酶结合,可通过 405 纳米波长的比色检测进行定量,作为凝血酶活性的测量指标。
T12414 PF-00356231 hydrochloride

MMP Proteases/Proteasome
PF-00356231 hydrochloride 是基质金属蛋白酶 MMP-12 的抑制剂,IC50 为 1.4 μM。
T12352 Oxidopamine hydrochloride

6-Hydroxydopamine hydrochloride,6-OHDA hydrochloride,6-羟基多巴胺盐酸盐

Mitophagy; Dopamine Receptor; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) 是一种神经递质多巴胺拮抗剂,可选择性地破坏多巴胺能神经元,是一种广泛使用的神经毒素。
T12032 Mibefradil dihydrochloride

盐酸米贝地尔,Ro 40-5967 (dihydrochloride),米贝拉地尔

Calcium Channel Membrane transporter/Ion channel; Metabolism
Mibefradil dihydrochloride (Ro 40-5967 (dihydrochloride)) 是一种钙离子通道抑制剂,选择性作用于 T 型 Ca2+通道,对 T 型和 L 型通道的IC50分别为 2.7 和 18.6 μM。
T12156 N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea

Others Others
N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea 是一种抗惊厥剂,对广泛强直和部分性发作挛性具有潜在的研究价值。
T6507 Gabapentin hydrochloride

加巴喷丁盐酸盐,Neurontin HCl,Gabapentin HCl

Calcium Channel; GABA Receptor Membrane transporter/Ion channel; Metabolism; Neuroscience
Gabapentin hydrochloride (Neurontin HCl) 是GABA 类似物,可用于缓解神经性疼痛。
T22501 2-Pyridylethylamine dihydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
2-Pyridylethylamine dihydrochloride 是一种组胺 H1 受体激动剂。
T21652 RN-1 dihydrochloride

Histone Demethylase; MAO Chromatin/Epigenetic; Metabolism; Neuroscience
RN-1 dihydrochloride 是血脑屏障通透性的、不可逆的赖氨酸特异性脱甲基酶 1 (LSD1) 选择性抑制剂,IC50为 70 nM,对 LSD1 的选择性高于 MAO-A 和 MAO-B,IC50分别为 0.51 μM 和 2.785 μM。
T37348 6-Chloro-7-deazapurine-β-D-riboside

Antifungal Microbiology/Virology
6-Chloro-7-deazapurine-β-D-riboside 是核苷的衍生物,显示出抗真菌活性。
T8747 Levofloxacin hydrochloride

DNA gyrase; Topoisomerase DNA Damage/DNA Repair
Levofloxacin hydrochloride 是一种广谱的第三代氟喹诺酮类抗生素,是氧氟沙星的光学活性 L-异构体,具有抗菌活性。左氧氟沙星通过细菌细胞壁扩散并通过抑制 DNA 促旋酶(细菌拓扑异构酶 II)起作用,这是一种 DNA 复制、RNA 转录和细菌 DNA 修复所需的酶。 DNA 促旋酶活性的抑制导致细菌细胞生长受阻。
T72112 Clozapine N-oxide dihydrochloride

AChE Neuroscience
Clozapine N-oxide dihydrochloride 是一种 Clozapine 的衍生物,也是一种可穿过血脑屏障的人毒蕈碱设计受体 (DREADDs) 激动剂。Clozapine N-oxide dihydrochloride 诱导 DREADD 受体 hM3Dq 和 hM4Di激活。
T1702 Nortropinone hydrochloride

Others Others
Nortropinone hydrochloride 用作药物中间体。
T17924 (S,R,S)-AHPC-PEG2-NH2 hydrochloride

VH032-PEG2-NH2 hydrochloride,VHL Ligand-Linker Conjugates 3 hydrochloride,E3 ligase Ligand-Linker Conjugates 6

Others; E3 Ligase Ligand-Linker Conjugate Others; PROTAC
(S,R,S)-AHPC-PEG2-NH2 hydrochloride (E3 ligase Ligand-Linker Conjugates 6) 包含基于 (S,R,S)-AHPC 的 VHL 配体和 2 个单元 PEG linker,是一种合成的 E3 连接酶配体-linker 偶联物,可用于 PROTAC 的合成分子。
T35326 Labetalone hydrochloride

Labetalone hydrochloride,Benzoic amide

Others Others
Labetalone hydrochloride (Benzoic amide) 是 Labetalol 的一种杂质。Labetalol 是一种口服有效的肾上腺素能受体阻断药物,对 α 和 β 受体部位都有竞争性拮抗作用。
T10718L CCT241533 hydrochloride

Chk Cell Cycle/Checkpoint
CCT241533 hydrochloride is an effective and selective ATP competitive inhibitor of CHK2 (Ki: 1.16 nM; IC50: 3 nM).
T22538 A-7 hydrochloride

CaMK Neuroscience
A-7 hydrochloride 是一种钙调蛋白拮抗剂,会引起 MDA-MB-231细胞中 CD44+CD24-亚群的改变。
T1254 Chlorophyllin sodium copper salt

Chlorophyllin copper sodium complex,Chlorophyllin,叶绿素铜钠盐,Chlorophyllin coppered trisodium salt,Sodium-copper chlorin e6

Others Others
Chlorophyllin sodium copper salt (Chlorophyllin coppered trisodium salt) 是一种由 Chlorophyll 衍生的铜钠盐的半合成混合物,常用作食品添加剂。
T23072 NNC 05-2090 hydrochloride

Transaminase Metabolism
NNC 05-2090 hydrochloride 是一种 betaine/GABA transporter (BGT-1) 抑制剂,IC50 值为 10.6 μM。NNC 05-2090 hydrochloride 可用于研究癫痫和神经疾病。
T22456 Voreloxin hydrochloride

SNS-595 hydrochloride,Vosaroxin,(3S-反式)-1,4-二氢-7-[3-甲氧基-4-(甲基氨基)-1-吡咯烷基]-4-氧代-1-(2-噻唑基)-1,8-萘啶-3-羧酸单盐酸盐

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
Voreloxin hydrochloride (SNS-595 hydrochloride) 是一种新型拓扑异构酶 II 抑制剂,能够诱导 DNA 双链断裂,阻滞 G2 期,引起细胞凋亡。
T20684 2',7'-Dichlorofluorescein diacetate

Diacetyldichlorofluorescein,Leuco-dcf diacetate,Dcfh-DA,双氯荧光黄乙酸乙酯,DCFDA

Others Others
2',7'-Dichlorofluorescein diacetate (Diacetyldichlorofluorescein) 是一种可渗透细胞的荧光探针,可用于检测一氧化氮和活性氧以及确定总体氧化应激的程度。
T8867 RO2959 Hydrochloride

RO2959 HCl

IL Receptor; Calcium Channel; Interleukin Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
RO2959 Hydrochloride (RO2959 HCl) 是选择性CRAC 通道抑制剂,IC50为 402 nM。它是人IL-2产生的有效抑制剂,有效阻断 T 细胞受体触发的基因表达和 T 细胞功能途径。它是由Orai1/Stim1通道介导的钙存储进入的有效阻滞剂,IC50为 25 nM。
T3491 1400W dihydrochloride

1400W 2HCl,N-(3-(Aminomethyl)benzyl)acetamidine

NOS; NO Synthase Immunology/Inflammation
1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) 是高效选择性的诱导型一氧化氮合成酶抑制剂(Ki:7 nM)。
T4068 E6446 dihydrochloride

TLR Immunology/Inflammation
E6446 dihydrochloride 是一种新型合成拮抗剂,用于核酸感应 TLR;有效抑制对 HEK:TLR9 细胞的 DNA 刺激,IC50 为 10 nM。
T3462 BMS-582949 hydrochloride

BMS-582949 HCl

p38 MAPK; Autophagy Autophagy; MAPK
BMS-582949 hydrochloride (BMS-582949 HCl) 是一种高度特异性的 p38α MAPK 抑制剂,其 IC50值为13 nM,可研究炎症性疾病。
T6592 ML133 hydrochloride

ML133 HCl,(4-甲氧基苄基)(1-萘基甲基)胺盐酸盐

Potassium Channel Membrane transporter/Ion channel
ML133 hydrochloride (ML133 HCl) 是选择性的Kir2家族通道抑制剂,在pH 7.4 和pH 8.5 时的IC50值分别为1.8 μM 和290 nM。
T62385 Befiradol hydrochloride

NLX-112 hydrochloride,F 13640 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Befiradol hydrochloride (NLX-112 hydrochloride) 是一种具有选择性的5-羟色胺 1A (5-HT)1A 受体激动剂,具有抗焦虑活性。Befiradol hydrochloride 抑制突变ATXN3聚集。
T4093 Fabomotizole hydrochloride

Afobazole hydrochloride,CM346 hydrochloride

MAO Metabolism; Neuroscience
Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。
T5856 Barnidipine hydrochloride

盐酸巴尼地平,YM-09730-5 hydrochloride,Mepirodipine (hydrochloride)

Calcium Channel Membrane transporter/Ion channel; Metabolism
Barnidipine hydrochloride (YM-09730-5 hydrochloride) 是一种二氢吡啶类钙通道阻滞剂,对 CaA 受体具有选择性作用。它是一种抗高血压药物,通过减少其血管扩张作用继发的外周血管阻力起作用。
T3281 Delapril hydrochloride

indalapril,地拉普利盐酸盐,Alindapril Hydrochloride,Delapril Hydrochloride,盐酸地拉普利,CV 3317

RAAS Endocrinology/Hormones
Delapril hydrochloride (indalapril) 是一种血管紧张素转化酶抑制剂,能够用于心血管疾病的研究。
T22324 Ensartinib hydrochloride

Ensartinib dihydrochloride,X-396 dihydrochloride

Others; Trk receptor; c-Met/HGFR; ALK Angiogenesis; Others; Tyrosine Kinase/Adaptors
Ensartinib hydrochloride (X-396 dihydrochloride) 是双重的 ALK/MET 抑制剂,IC50分别 <0.4 nM 和 0.74 nM。
T2191 Tacrine hydrochloride (hydrate)

Tacrine,他克林盐酸盐水合物,Tacrine hydrochloride hydrate,Tetrahydroaminacrine,Tetrahydroaminoacridine

AChR; AChE Neuroscience
Tacrine hydrochloride hydrate (Tetrahydroaminacrine) 是一种乙酰胆碱酯酶 (AChE) 和丁酰胆碱酯酶 (BChE) 的抑制剂,它们的IC50值分别为 31 nM 和 25.6 nM。
T5820 Amsacrine hydrochloride

acridinyl anisidide hydrochloride,盐酸胺苯吖啶,m-AMSA hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Amsacrine hydrochloride (acridinyl anisidide hydrochloride) 是一种拓扑异构酶 II 抑制剂,用于治疗急性髓细胞性白血病。
T12482 Pipendoxifene hydrochloride

Estrogen Receptor/ERR Endocrinology/Hormones
Pipendoxifene hydrochloride 是雌激素受体的选择性调节剂。
T13423 (1R,2R)-2-PCCA hydrochloride

(1R,2R)-2-PCCA(hydrochloride)

Others Others
(1R,2R)-2-PCCA hydrochloride 是一种具有有效性、选择性和可穿过血脑屏障的 GPR88 受体激动剂,在 WT 小鼠纹状体膜中 EC50 值为1140 n。(1R,2R)-2-PCCA hydrochloride 可用于研究中枢神经系统。
T7739 L-Leucyl-L-Leucine methyl ester hydrochloride

Leu-Leu-ome hydrochloride

Others; Endogenous Metabolite Metabolism; Others
L-Leucyl-L-Leucine methyl ester hydrochloride (Leu-Leu-ome hydrochloride) 是一种人单核细胞或多形核白细胞产生的 L-亮氨酸甲酯的二肽缩合产物,能够选择性消除具有细胞毒性潜能的淋巴细胞,也能够诱导溶酶体途径应激。
T8677 3,4 Dichloroisocoumarin

Others; Serine Protease; Cysteine Protease Others; Proteases/Proteasome
3,4 Dichloroisocoumarin 是一种颗粒酶、组织蛋白酶 G 和中性粒细胞弹性蛋白酶抑制剂
T3217 PF-CBP1 hydrochloride

PF-CBP1 HCl

Epigenetic Reader Domain; Histone Acetyltransferase Chromatin/Epigenetic
PF-CBP1 hydrochloride (PF-CBP1 HCl) 是 CREB 结合蛋白溴结构域的一种高选择性抑制剂,抑制 CREBBP 和 EP300溴结构域的 IC50分别为 125 和 363 nM。它降低 LPS 诱导的巨噬细胞中炎症因子的表达,也可下调皮质神经元 RGS4 的表达,可用于癫痫和帕金森病等神经疾病的研究。
T4391 Syk Inhibitor II dihydrochloride

Syk Inhibitor II (hydrochloride)

Others; Tyrosine Kinases; Syk; PKC; BTK Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; Others; Tyrosine Kinase/Adaptors
Syk Inhibitor II (hydrochloride) 是一种非受体酪氨酸激酶,磷酸化后,它与 FcRγ 链的基于免疫受体酪氨酸的激活基序结合,并介导与血小板功能和炎症相关的下游信号传导。 Syk inhibitor II 是一种可渗透细胞的嘧啶-甲酰胺化合物,以 ATP 竞争性方式选择性和可逆地阻断 Syk (IC50 = 41 nM)。它对 PKCε、PKCβII、ZAP-70、Btk 和 Itk 的效力要低得多(IC50s 分别为5.1、11、11.2、15.5 和 22.6 μM)。
T4383 GSK-J4 Hydrochloride

GSK J4 HCl,GSK J4 HCl (1373423-53-0 free base)

Histone Demethylase Chromatin/Epigenetic
GSK-J4 Hydrochloride (GSK J4 HCl) 是 H3K27me3/me2 去甲基化酶 JMJD3/KDM6B 和 UTX/KDM6A 双抑制剂,IC50分别为 8.6 和 6.6 μM。它是 GSK-J1 的乙酯衍生物,体外 IC50 值大于 50 μM。它抑制 LPS 诱导的人原代巨噬细胞产生 TNF-α,IC50值为 9 μM。

化合物

Destruxin CHL
Cat.No: T130428
Synonym:
Target:
Chloramphenicol palmitate
Cat.No: T20525
Synonym:
Target: Antibacterial, Antibiotic
Olanexidine hydrochloride
Cat.No: T28229
Synonym: OPB2045,OPB-2045,OPB-2045 HCl,OPB 2045
Target: Antibacterial
6-Chloropurine
Cat.No: T7470
Synonym: 6-氯嘌呤,6-Chloro-9H-purine
Target: Others
MS023 dihydrochloride
Cat.No: T61338
Synonym: MS023 2HCl
Target: Histone Methyltransferase
R 59-022 hydrochloride
Cat.No: T72322
Synonym: DKGI-I hydrochloride,Diacylglycerol kinase inhibitor I hydrochloride,DKGI-I hydrochloride ; Diacylglycerol kinase inhibitor I hydrochloride
Target: 5-HT Receptor, PKC
Protein kinase inhibitor H-7 dihydrochloride
Cat.No: T22831
Synonym: H-7 dihydrochloride
Target: PKC
Asoxime dichloride
Cat.No: T14333
Synonym: Tert-Butyl2-(2-hydroxyethyl)-1-pyrrolidinecarboxylate,Asoxime (dichloride),HI-6
Target: AChR
Vevorisertib trihydrochloride
Cat.No: T38846
Synonym: ARQ 751 trihydrochloride
Target: Akt
4-Aminobenzamidine dihydrochloride
Cat.No: T60248
Synonym: p-Aminobenzamidine dihydrochloride
Target: Serine Protease
Chlorthal-dimethyl
Cat.No: T14954
Synonym: Dimethyl tetrachloroterephthalate
Target: Others
H-Gly-Arg-pNA dihydrochloride
Cat.No: T37034
Synonym: H-Gly-Arg-Pna 2HCl
Target:
PF-00356231 hydrochloride
Cat.No: T12414
Synonym:
Target: MMP
Oxidopamine hydrochloride
Cat.No: T12352
Synonym: 6-Hydroxydopamine hydrochloride,6-OHDA hydrochloride,6-羟基多巴胺盐酸盐
Target: Mitophagy, Dopamine Receptor, Autophagy
Mibefradil dihydrochloride
Cat.No: T12032
Synonym: 盐酸米贝地尔,Ro 40-5967 (dihydrochloride),米贝拉地尔
Target: Calcium Channel
N-(2-Chloro-6-methylphenyl)-N'-4-pyridinylurea
Cat.No: T12156
Synonym:
Target: Others
Gabapentin hydrochloride
Cat.No: T6507
Synonym: 加巴喷丁盐酸盐,Neurontin HCl,Gabapentin HCl
Target: Calcium Channel, GABA Receptor
2-Pyridylethylamine dihydrochloride
Cat.No: T22501
Synonym:
Target: Histamine Receptor
RN-1 dihydrochloride
Cat.No: T21652
Synonym:
Target: Histone Demethylase, MAO
6-Chloro-7-deazapurine-β-D-riboside
Cat.No: T37348
Synonym:
Target: Antifungal
Levofloxacin hydrochloride
Cat.No: T8747
Synonym:
Target: DNA gyrase, Topoisomerase
Clozapine N-oxide dihydrochloride
Cat.No: T72112
Synonym:
Target: AChE
Nortropinone hydrochloride
Cat.No: T1702
Synonym:
Target: Others
(S,R,S)-AHPC-PEG2-NH2 hydrochloride
Cat.No: T17924
Synonym: VH032-PEG2-NH2 hydrochloride,VHL Ligand-Linker Conjugates 3 hydrochloride,E3 ligase Ligand-Linker Conjugates 6
Target: Others, E3 Ligase Ligand-Linker Conjugate
Labetalone hydrochloride
Cat.No: T35326
Synonym: Labetalone hydrochloride,Benzoic amide
Target: Others
CCT241533 hydrochloride
Cat.No: T10718L
Synonym:
Target: Chk
A-7 hydrochloride
Cat.No: T22538
Synonym:
Target: CaMK
Chlorophyllin sodium copper salt
Cat.No: T1254
Synonym: Chlorophyllin copper sodium complex,Chlorophyllin,叶绿素铜钠盐,Chlorophyllin coppered trisodium salt,Sodium-copper chlorin e6
Target: Others
NNC 05-2090 hydrochloride
Cat.No: T23072
Synonym:
Target: Transaminase
Voreloxin hydrochloride
Cat.No: T22456
Synonym: SNS-595 hydrochloride,Vosaroxin,(3S-反式)-1,4-二氢-7-[3-甲氧基-4-(甲基氨基)-1-吡咯烷基]-4-氧代-1-(2-噻唑基)-1,8-萘啶-3-羧酸单盐酸盐
Target: Apoptosis, Topoisomerase
2',7'-Dichlorofluorescein diacetate
Cat.No: T20684
Synonym: Diacetyldichlorofluorescein,Leuco-dcf diacetate,Dcfh-DA,双氯荧光黄乙酸乙酯,DCFDA
Target: Others
RO2959 Hydrochloride
Cat.No: T8867
Synonym: RO2959 HCl
Target: IL Receptor, Calcium Channel, Interleukin
1400W dihydrochloride
Cat.No: T3491
Synonym: 1400W 2HCl,N-(3-(Aminomethyl)benzyl)acetamidine
Target: NOS, NO Synthase
E6446 dihydrochloride
Cat.No: T4068
Synonym:
Target: TLR
BMS-582949 hydrochloride
Cat.No: T3462
Synonym: BMS-582949 HCl
Target: p38 MAPK, Autophagy
ML133 hydrochloride
Cat.No: T6592
Synonym: ML133 HCl,(4-甲氧基苄基)(1-萘基甲基)胺盐酸盐
Target: Potassium Channel
Befiradol hydrochloride
Cat.No: T62385
Synonym: NLX-112 hydrochloride,F 13640 hydrochloride
Target: 5-HT Receptor
Fabomotizole hydrochloride
Cat.No: T4093
Synonym: Afobazole hydrochloride,CM346 hydrochloride
Target: MAO
Barnidipine hydrochloride
Cat.No: T5856
Synonym: 盐酸巴尼地平,YM-09730-5 hydrochloride,Mepirodipine (hydrochloride)
Target: Calcium Channel
Delapril hydrochloride
Cat.No: T3281
Synonym: indalapril,地拉普利盐酸盐,Alindapril Hydrochloride,Delapril Hydrochloride,盐酸地拉普利,CV 3317
Target: RAAS
Ensartinib hydrochloride
Cat.No: T22324
Synonym: Ensartinib dihydrochloride,X-396 dihydrochloride
Target: Others, Trk receptor, c-Met/HGFR, ALK
Tacrine hydrochloride (hydrate)
Cat.No: T2191
Synonym: Tacrine,他克林盐酸盐水合物,Tacrine hydrochloride hydrate,Tetrahydroaminacrine,Tetrahydroaminoacridine
Target: AChR, AChE
Amsacrine hydrochloride
Cat.No: T5820
Synonym: acridinyl anisidide hydrochloride,盐酸胺苯吖啶,m-AMSA hydrochloride
Target: Topoisomerase, Autophagy
Pipendoxifene hydrochloride
Cat.No: T12482
Synonym:
Target: Estrogen Receptor/ERR
(1R,2R)-2-PCCA hydrochloride
Cat.No: T13423
Synonym: (1R,2R)-2-PCCA(hydrochloride)
Target: Others
L-Leucyl-L-Leucine methyl ester hydrochloride
Cat.No: T7739
Synonym: Leu-Leu-ome hydrochloride
Target: Others, Endogenous Metabolite
3,4 Dichloroisocoumarin
Cat.No: T8677
Synonym:
Target: Others, Serine Protease, Cysteine Protease
PF-CBP1 hydrochloride
Cat.No: T3217
Synonym: PF-CBP1 HCl
Target: Epigenetic Reader Domain, Histone Acetyltransferase
Syk Inhibitor II dihydrochloride
Cat.No: T4391
Synonym: Syk Inhibitor II (hydrochloride)
Target: Others, Tyrosine Kinases, Syk, PKC, BTK
GSK-J4 Hydrochloride
Cat.No: T4383
Synonym: GSK J4 HCl,GSK J4 HCl (1373423-53-0 free base)
Target: Histone Demethylase
Cat. No. Product Name Target Signaling Pathways
T9862 Pseudocoptisine chloride

盐酸异黄连碱,Isocoptisine chloride

AChE Neuroscience
Pseudocoptisine chloride (Isocoptisine chloride) 是从 Corydalis Tuber 中分离出来的,具有抗炎和抗健忘的作用。 Pseudocoptisine chloride 抑制乙酰胆碱酯酶 (AChE) 活性 (IC50 = 12.8 μM)。
T6631 Quinine hydrochloride dihydrate

奎宁单盐酸盐二水合物,Quinine HCl Dihydrate,奎宁盐酸盐二水合物

Potassium Channel; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Quinine hydrochloride dihydrate (Quinine HCl Dihydrate) 是一种白色结晶 K+ 通道阻滞剂,用于治疗疟疾,具有退热,抗疟,止痛,抗炎等特性。
T4895 Pentane-1,5-diamine dihydrochloride

5-diamine dihydrochloride,Cadaverine dihydrochloride,1,5-戊二胺盐酸盐,Pentane-1

Endogenous Metabolite Metabolism
Pentane-1,5-diamine dihydrochloride (Cadaverine dihydrochloride) 是内源性代谢产物的一种。
TN1106 Cyanidin-3-O-galactoside chloride

Ideain chloride

Antioxidant oxidation-reduction
Cyanidin-3-O-galactoside chloride (Ideain chloride)是从山楂果皮 (EPHF)中提取的小分子化合物,具有抗氧化和抗肿瘤作用,可用于研究肥胖。
T7557 Guvacine hydrochloride

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Guvacine hydrochloride 是从槟榔中得到的一种生物碱,是 GABA 摄取抑制剂,IC50为 10 μM。它对几种克隆的 GABA 转运体具有适度的选择性。
T5S1530 Isochlorogenic acid C

金银花,异绿原酸C

Antioxidant oxidation-reduction
Isochlorogenic acid C 具有抗氧化活性。
TN7202 3-Chloro-6-Bromo Indole

6-溴-3-氯-1H-吲哚,6-bromo-3-chloro-1H-indole,3-CHLORO-6-BROMOINDOLE

Others Others
3-Chloro-6-Bromo Indole (3-CHLORO-6-BROMOINDOLE) 是一种海洋来源的天然产物,存在于 Ptychodera flava。
T3406 Kuromanin chloride

Glucocyanidin chloride,Chrysontemin,矢车菊素-3-O-葡萄糖苷,Chrysontemin chloride,Cyanidin 3-O-glucoside chloride

NF-κB NF-κB
Kuromanin chloride (Chrysontemin chloride) 是从桑叶中获得,能够提高血糖浓度、维持脂质代谢平衡,表现出降低肥胖的作用。
T2921 Sinomenine hydrochloride

盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride

Apoptosis; NF-κB; Opioid Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; GPCR/G Protein; Neuroscience; NF-κB
Sinomenine hydrochloride (Kukoline hydrochloride) 是来自汉防己的一种生物碱,是NF-κB 活化的阻断剂。Sinomenine 也是一种 μ 阿片受体激活剂。
T1680 Tolazoline hydrochloride

Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Tolazoline hydrochloride (NSC35110(hydrochloride)) 是一种 α 肾上腺素受体抑制剂。
T4826 L-Histidine monohydrochloride monohydrat

Others; Endogenous Metabolite Metabolism; Others
L-Histidine monohydrochloride monohydrat 是一种 α-氨基酸。 L-异构体是 22 种蛋白质氨基酸之一,即蛋白质的组成部分。
T0019 Betaine chloride

Betaine hydrochloride,盐酸甜菜碱

Others; Chloride channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
Betaine chloride (Betaine hydrochloride) 是一种天然化合物,在许多食物中能够发现,也是能够维持正常 DNA 甲基化模式的特性甲基供体。
T7851 Tyramine hydrochloride

盐酸酪胺,酪胺盐酸盐

Others; Endogenous Metabolite Metabolism; Others
Tyramine hydrochloride 是一种氨基酸,有助于调节血压。其中 Tyramine 天然存在于体内,并存在于某些食物中。
T6S1537 Cryptochlorogenic acid

隐绿原酸,4-O-Caffeoylquinic acid,4-Caffeoylquinic acid,金银花

Antioxidant; Endogenous Metabolite Metabolism; oxidation-reduction
Cryptochlorogenic acid (4-O-Caffeoylquinic acid) 是一种天然产物,具有抗氧化活性。
T1205 Chloramphenicol

Chlornitromycin,Levomycetin,Chloromycetin,氯霉素

ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
T0810 Ethambutol dihydrochloride

Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Ethambutol dihydrochloride (CL40881) 能抗分枝杆菌,可抑制阿拉伯糖基转移酶活性来阻止细胞壁形成。
T8048 Diphenylamine Hydrochloride

Others Others
Diphenylamine hydrochloride 分离自 coriander ,具有抗氧化作用。在农业中,它可用作杀菌剂及抗菌剂;在工业中,它可用作抗氧化剂及染料媒染剂。
T2718 Palmatine chloride

Others; Indoleamine 2,3-Dioxygenase (IDO); Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Others
Palmatine chloride 是口服具有活力的不可逆 IDO-1抑制剂。它能够减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,并改善 DSS 诱发的结肠炎。
T0268 Lobeline hydrochloride

盐酸洛贝林,α-Lobeline hydrochloride,L-Lobeline hydrochloride

AChR Neuroscience
Lobeline hydrochloride (α-Lobeline hydrochloride) 是一种烟碱样受体激动剂,是神经元烟碱受体α3β2和α4β2拮抗剂。
T0788 Spectinomycin dihydrochloride

淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Spectinomycin dihydrochloride (Actinospectacin) 是一种能与细菌核糖体的30S 亚基结合,干扰蛋白质合成的抗生素。
T0486 Irinotecan hydrochloride trihydrate

Irinotecan HCl Trihydrate,CPT-11 HCl Trihydrate,盐酸伊立替康三水合物

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan hydrochloride trihydrate (CPT-11 HCl Trihydrate) 通过抑制拓扑异构酶 1 来防止 DNA 展开,可研究结肠癌和直肠癌。
T0129 Sanguinarine chloride

Pseudochelerythrine chloride,血根碱,氯化血根碱,Sanguinarium chloride

Apoptosis; EGFR; VEGFR; Antibacterial; Parasite; Autophagy Angiogenesis; Apoptosis; Autophagy; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Sanguinarine chloride (Pseudochelerythrine chloride) 是一种来源于 Sanguinaria Canadensis 的生物碱,通过激活活性氧的产生,诱导细胞凋亡。
T1591 Ancitabine hydrochloride

NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C

Others; DNA/RNA Synthesis; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。
T3604 Sodium dichloroacetate

Sodium Dichloroacetate,DCA,bichloroacetic acid,二氯乙酸钠,Sodium dichloroacetate (DCA),二氯醋酸酯

Apoptosis; Dehydrogenase; Reactive Oxygen Species; PDK Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Sodium dichloroacetate (BCA) 是癌细胞线粒体中的一种代谢调节剂,具有抗癌活性。它抑制丙酮酸脱氢酶激酶,从而导致肿瘤微环境中的乳酸减少。它增加活性氧的产生并促进癌细胞凋亡,还可作为NKCC 抑制剂。
T0415 Guanidine hydrochloride

Guanidine HCl,Aminoformamidine HCl,盐酸胍,Aminoformamidine Hydrochloride,Guanidinium chloride

Others; Arginase; DNA/RNA Synthesis; Endogenous Metabolite; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Others
Guanidine hydrochloride (Aminoformamidine Hydrochloride) 是一种强离液剂和一种蛋白质的强变性剂。
T2219 Puromycin dihydrochloride

CL13900 dihydrochloride,Puromycin 2HCl,嘌呤霉素二盐酸盐水合物,嘌呤霉素二盐酸盐

ribosome; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Puromycin dihydrochloride (CL13900 dihydrochloride) 属于肉桂酰胺腺苷抗生素,是一种蛋白质合成的抑制剂。Puromycin dihydrochloride 通过与 RNA 结合来抑制蛋白质合成,具有抗肿瘤和抗锥虫活性。
TN3497 Benzylamine hydrochloride

Others Others
Benzylamine hydrochloride 由卞胺和盐酸制的, 可用于治疗晕动病和蛔虫病,具有止吐特性。
T4614 Ellipticine hydrochloride

Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐

Topoisomerase DNA Damage/DNA Repair
Ellipticine hydrochloride (NSC-71795 (hydrochloride)) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 的活性。
T1020 Doxorubicin hydrochloride

Adriamycin,Doxorubicin (Adriamycin) HCl,Hydroxydaunorubicin hydrochloride,盐酸多柔比星,盐酸阿霉素,NSC 123127

Apoptosis; Mitophagy; HBV; HIV Protease; Topoisomerase; Antibacterial; Antibiotic; AMPK; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Doxorubicin hydrochloride (Adriamycin) 属于蒽环类抗生素,是人类 DNA 拓扑异构酶 I/II 抑制剂 (IC50=0.8/2.67 μM)。Doxorubicin hydrochloride 具有细胞毒性和抗肿瘤活性。Doxorubicin hydrochloride 可降低 AMPK 及其下游靶蛋白乙酰辅酶 A 羧化酶的磷酸化,还可诱导凋亡和自噬。
T13302 Viquidil hydrochloride

Quinotoxine hydrochloride

Others Others
Viquidil hydrochloride (Quinotoxine hydrochloride) 是奎尼丁的同分异构体,是一种脑血管扩张剂,具有抗血栓作用。
T2762 Kasugamycin hydrochloride

Kasumin,盐酸春雷霉素

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Kasugamycin hydrochloride (Kasumin) 是一种能结合 30s 和 70s 核糖体,但不能结合 50s 亚基的抗生素。它模拟 mRNA 核苷酸以破坏 tRNA 结合并抑制经典翻译起始。
T2O2701 L-Ornithine hydrochloride

L(+)-Ornithine hydrochloride,(S)-2,5-Diaminopentanoic acid,L-鸟氨酸盐酸盐;L-2,5-二氨基戊酸盐酸盐;L-鸟氨酸单盐酸盐;鸟氨酸盐酸盐;L-盐酸鸟氨酸;L-鸟粪氨基酸盐酸盐

Others; Endogenous Metabolite Metabolism; Others
L-Ornithine hydrochloride ((S)-2,5-Diaminopentanoic acid) 通过提高能量消耗效率和促进氨的排泄而具有抗疲劳作用。它是尿素循环中的关键反应物之一。
T4925 Thiamine monophosphate chloride (dihydrate)

Thiamine monophosphate chloride dihydrat,胺氯化亚磷酸酯,Aneurine monophosphate chloride

Others; Endogenous Metabolite Metabolism; Others
Thiamine monophosphate chloride dihydrate (Aneurine monophosphate chloride) 是内源性代谢产物的一种。
T4592 TOMATIDINE HYDROCHLORIDE

Tomatidine,Tomatidine HCl,盐酸番茄碱

Others; NF-κB; JNK; Autophagy Autophagy; MAPK; NF-κB; Others
Tomatidine hydrochloride (Tomatidine HCl) 是一种甾体生物碱,可防止肌肉萎缩并促进肌肉生长。它通过阻断 NF-κB 和JNK 信号发挥抗炎作用,可激活哺乳动物细胞或秀丽隐杆线虫中的自噬。
T8298 Vasicine hydrochloride

鸭嘴花碱盐酸盐,Peganine hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Vasicine hydrochloride (Peganine hydrochloride) 是从Justicia adhatoda 中分离得到的一种喹唑啉类生物碱,有抗结核活性。
T2811 Harmine hydrochloride

telepathine hydrochloride,盐酸哈尔明碱

5-HT Receptor; DYRK; GluR Cell Cycle/Checkpoint; GPCR/G Protein; Neuroscience; Tyrosine Kinase/Adaptors
Harmine hydrochloride (telepathine hydrochloride) 是一种 DYRK 抑制剂,具有抗癌和抗炎活性。它对5-HT2A 血清素受体具有高亲和力,Ki 值为 397 nM。
T2S2043 Dracorhodin perchlorate

Dracorhodin perochlorate,血竭素高氯酸盐,Dracohodin perochlorate

Apoptosis; Others Apoptosis; Others
Dracorhodin perchlorate 是来源于中药血竭的一种天然产物。它抑制细胞生长,并以剂量和时间依赖性方式诱导成纤维细胞凋亡,将细胞周期阻滞在 G1 期,可作为抗乳腺癌的候选药物。
T5807 Stylopine hydrochloride

NOS; COX Immunology/Inflammation; Neuroscience
Stylopine hydrochloride 是一种生物碱类化合物,从紫堇属之植物块茎中分离得到,具有抗炎症和抗寄生虫作用。
T0896 Furaltadone hydrochloride

Furaltadone HCl,盐酸呋喃它酮

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Furaltadone hydrochloride (Furaltadone HCl) 是硝基呋喃药,可研究肠沙门氏菌感染,治疗球虫病。Furaltadone 具有体外抑制葡萄球菌作用。
T8787 Drotaverine hydrochloride

PDE Metabolism
Drotaverine hydrochloride 是磷酸二酯酶 4 (PDE4)的抑制剂,也是 L 型电压依赖钙通道(L-VDCC)的阻滞剂,可阻断3',5'-环腺苷单磷酸的降解。它在体内有抗痉挛效果,但无抗胆碱能的效果。
T10990 Dehydrocorydaline chloride

盐酸脱氢紫堇碱,13-Methylpalmatine chloride

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline chloride (13-Methylpalmatine chloride) 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达;激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
TN7197 6-Chloro-2,4-dibromophenol

2,4-dibromo-6-chloro-phenol,2,4-二溴-6-氯苯酚,2,4-dibromo-6-chlorophenol,ZINC397569

Others Others
6-Chloro-2,4-dibromophenol (2,4-dibromo-6-chlorophenol) 是一种海洋来源的天然产物,存在于Pseudoalteromonas luteoviolacea。
T0266 Quinidine hydrochloride monohydrate

奎宁树,奎尼丁盐酸盐一水合物,奎尼丁盐酸盐,Quinidine hydrochloride

Potassium Channel; Sodium Channel; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Quinidine hydrochloride monohydrate 是一种抗心律失常剂,也是 K+通道 (K+channel) 的有效阻断剂,其IC50值为 19.9 μM。它是一种有效且选择性的细胞色素 P450db (cytochrome P450db) 抑制剂,也可用作疟疾的研究。
T5S0761 Nitidine chloride

Apoptosis; ERK; FAK; p38 MAPK; NF-κB; Topoisomerase; STAT; Parasite Angiogenesis; Apoptosis; Cytoskeletal Signaling; DNA Damage/DNA Repair; JAK/STAT signaling; MAPK; Microbiology/Virology; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Nitidine chloride 是从Zanthoxylum nitidum (Roxb) DC 中分离得到的,具有抗疟疾活性。它通过多个靶点通路,起抗癌作用,抑制STAT3、DNA 拓扑异构酶1和2A、ERK 和c-Src/FAK 相关信号通路。它通过MAPK 和NF-kB 途径抑制Lps 诱导的炎性细胞因子的产生。
T0330 Diphenhydramine hydrochloride

盐酸苯海拉明,Diphenhydramine HCl,DPH

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenhydramine hydrochloride (DPH) 是一种组胺 H1 拮抗剂,用作镇咳药和止吐药。它还用于治疗瘙痒和皮肤病、过敏反应、抗帕金森病、催眠药和普通感冒制剂的成分。
T1221 Acetylcholine chloride

ACh chloride,Pilofrin,氯化乙酰胆碱

Calcium Channel; Endogenous Metabolite; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience
Acetylcholine chloride (Pilofrin) 是一种神经递质,是胆碱能激动剂,通过刺激烟碱乙酰胆碱受体调节多巴胺能神经元活性,在体外抑制 p53 突变肽的聚集。
T4333 Quinine dihydrochloride

盐酸奎宁,Quinine bimuriate

Others Others
Quinine dihydrochloride (Quinine bimuriate) 是Cinchona(Rubiaceae) 各种物种的主要生物碱。它也是一种抗疟药和肌肉松弛剂(骨骼)。
T6475 (±)-Carnitine chloride

Monocamin,DL-Carnitine HCl,Bicarnesine,混旋肉碱盐酸盐,DL-Carnitine chloride

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
(±)-Carnitine chloride (Monocamin) 有D 和L 两种异构体。其中 L-carnitine 在脂肪酸的 β-氧化中起重要作用,也具有抗氧化作用和抗炎活性。
TN1564 Delphinidin 3-glucoside chloride

Delphinidin-3-O-glucoside chloride

Apoptosis; EGFR Angiogenesis; Apoptosis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Delphinidin 3-glucoside chloride (Delphinidin-3-O-glucoside chloride) 是从 Hibiscus sabdariffa 提取物中发现的膳食酚类物质。Delphinidin 3-glucoside chloride 具有抗氧化活性,可诱导 B 细胞慢性淋巴细胞性白血病 (B CLL) 的促凋亡作用,抑制 EGFR,抑制血小板聚集。Delphinidin 3-glucoside chloride 具有抗肿瘤活性,通过调节 pAKT/IRF1/HOTAIR 通路发挥作用。
T60789 L-Cystine dihydrochloride

L-Cystine dihydrochloride 是合成谷胱甘肽 (GSH) 的含硫前体。L-Cystine dihydrochloride 的稳态对谷胱甘肽的功能很重要。L-Cystine dihydrochloride 可用作细胞培养组分。
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天然产物

Pseudocoptisine chloride
Cat.No: T9862
Synonym: 盐酸异黄连碱,Isocoptisine chloride
Target: AChE
Quinine hydrochloride dihydrate
Cat.No: T6631
Synonym: 奎宁单盐酸盐二水合物,Quinine HCl Dihydrate,奎宁盐酸盐二水合物
Target: Potassium Channel, Parasite
Pentane-1,5-diamine dihydrochloride
Cat.No: T4895
Synonym: 5-diamine dihydrochloride,Cadaverine dihydrochloride,1,5-戊二胺盐酸盐,Pentane-1
Target: Endogenous Metabolite
Cyanidin-3-O-galactoside chloride
Cat.No: TN1106
Synonym: Ideain chloride
Target: Antioxidant
Guvacine hydrochloride
Cat.No: T7557
Synonym:
Target: GABA Receptor
Isochlorogenic acid C
Cat.No: T5S1530
Synonym: 金银花,异绿原酸C
Target: Antioxidant
3-Chloro-6-Bromo Indole
Cat.No: TN7202
Synonym: 6-溴-3-氯-1H-吲哚,6-bromo-3-chloro-1H-indole,3-CHLORO-6-BROMOINDOLE
Target: Others
Kuromanin chloride
Cat.No: T3406
Synonym: Glucocyanidin chloride,Chrysontemin,矢车菊素-3-O-葡萄糖苷,Chrysontemin chloride,Cyanidin 3-O-glucoside chloride
Target: NF-κB
Sinomenine hydrochloride
Cat.No: T2921
Synonym: 盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride
Target: Apoptosis, NF-κB, Opioid Receptor, Autophagy
Tolazoline hydrochloride
Cat.No: T1680
Synonym: Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)
Target: Adrenergic Receptor
L-Histidine monohydrochloride monohydrat
Cat.No: T4826
Synonym:
Target: Others, Endogenous Metabolite
Betaine chloride
Cat.No: T0019
Synonym: Betaine hydrochloride,盐酸甜菜碱
Target: Others, Chloride channel, Endogenous Metabolite
Tyramine hydrochloride
Cat.No: T7851
Synonym: 盐酸酪胺,酪胺盐酸盐
Target: Others, Endogenous Metabolite
Cryptochlorogenic acid
Cat.No: T6S1537
Synonym: 隐绿原酸,4-O-Caffeoylquinic acid,4-Caffeoylquinic acid,金银花
Target: Antioxidant, Endogenous Metabolite
Chloramphenicol
Cat.No: T1205
Synonym: Chlornitromycin,Levomycetin,Chloromycetin,氯霉素
Target: ribosome, HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
Ethambutol dihydrochloride
Cat.No: T0810
Synonym: Ethambutol 2HCl,盐酸乙胺丁醇,Emb dihydrochloride,CL40881
Target: Antibacterial, Antibiotic, Antifungal
Diphenylamine Hydrochloride
Cat.No: T8048
Synonym:
Target: Others
Palmatine chloride
Cat.No: T2718
Synonym:
Target: Others, Indoleamine 2,3-Dioxygenase (IDO), Aurora Kinase
Lobeline hydrochloride
Cat.No: T0268
Synonym: 盐酸洛贝林,α-Lobeline hydrochloride,L-Lobeline hydrochloride
Target: AChR
Spectinomycin dihydrochloride
Cat.No: T0788
Synonym: 淋必治,Spectinomycin 2HCl,盐酸奇霉素,Actinospectacin
Target: ribosome, Antibacterial, Antibiotic
Irinotecan hydrochloride trihydrate
Cat.No: T0486
Synonym: Irinotecan HCl Trihydrate,CPT-11 HCl Trihydrate,盐酸伊立替康三水合物
Target: Topoisomerase, Autophagy
Sanguinarine chloride
Cat.No: T0129
Synonym: Pseudochelerythrine chloride,血根碱,氯化血根碱,Sanguinarium chloride
Target: Apoptosis, EGFR, VEGFR, Antibacterial, Parasite, Autophagy
Ancitabine hydrochloride
Cat.No: T1591
Synonym: NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C
Target: Others, DNA/RNA Synthesis, Autophagy
Sodium dichloroacetate
Cat.No: T3604
Synonym: Sodium Dichloroacetate,DCA,bichloroacetic acid,二氯乙酸钠,Sodium dichloroacetate (DCA),二氯醋酸酯
Target: Apoptosis, Dehydrogenase, Reactive Oxygen Species, PDK
Guanidine hydrochloride
Cat.No: T0415
Synonym: Guanidine HCl,Aminoformamidine HCl,盐酸胍,Aminoformamidine Hydrochloride,Guanidinium chloride
Target: Others, Arginase, DNA/RNA Synthesis, Endogenous Metabolite, Autophagy
Puromycin dihydrochloride
Cat.No: T2219
Synonym: CL13900 dihydrochloride,Puromycin 2HCl,嘌呤霉素二盐酸盐水合物,嘌呤霉素二盐酸盐
Target: ribosome, DNA/RNA Synthesis, Antibacterial, Antibiotic
Benzylamine hydrochloride
Cat.No: TN3497
Synonym:
Target: Others
Ellipticine hydrochloride
Cat.No: T4614
Synonym: Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐
Target: Topoisomerase
Doxorubicin hydrochloride
Cat.No: T1020
Synonym: Adriamycin,Doxorubicin (Adriamycin) HCl,Hydroxydaunorubicin hydrochloride,盐酸多柔比星,盐酸阿霉素,NSC 123127
Target: Apoptosis, Mitophagy, HBV, HIV Protease, Topoisomerase, Antibacterial, Antibiotic, AMPK, Autophagy
Viquidil hydrochloride
Cat.No: T13302
Synonym: Quinotoxine hydrochloride
Target: Others
Kasugamycin hydrochloride
Cat.No: T2762
Synonym: Kasumin,盐酸春雷霉素
Target: Antibacterial, Antibiotic, Antifungal
L-Ornithine hydrochloride
Cat.No: T2O2701
Synonym: L(+)-Ornithine hydrochloride,(S)-2,5-Diaminopentanoic acid,L-鸟氨酸盐酸盐;L-2,5-二氨基戊酸盐酸盐;L-鸟氨酸单盐酸盐;鸟氨酸盐酸盐;L-盐酸鸟氨酸;L-鸟粪氨基酸盐酸盐
Target: Others, Endogenous Metabolite
Thiamine monophosphate chloride (dihydrate)
Cat.No: T4925
Synonym: Thiamine monophosphate chloride dihydrat,胺氯化亚磷酸酯,Aneurine monophosphate chloride
Target: Others, Endogenous Metabolite
TOMATIDINE HYDROCHLORIDE
Cat.No: T4592
Synonym: Tomatidine,Tomatidine HCl,盐酸番茄碱
Target: Others, NF-κB, JNK, Autophagy
Vasicine hydrochloride
Cat.No: T8298
Synonym: 鸭嘴花碱盐酸盐,Peganine hydrochloride
Target: Antibacterial, Antibiotic
Harmine hydrochloride
Cat.No: T2811
Synonym: telepathine hydrochloride,盐酸哈尔明碱
Target: 5-HT Receptor, DYRK, GluR
Dracorhodin perchlorate
Cat.No: T2S2043
Synonym: Dracorhodin perochlorate,血竭素高氯酸盐,Dracohodin perochlorate
Target: Apoptosis, Others
Stylopine hydrochloride
Cat.No: T5807
Synonym:
Target: NOS, COX
Furaltadone hydrochloride
Cat.No: T0896
Synonym: Furaltadone HCl,盐酸呋喃它酮
Target: Antibacterial, Antibiotic, Parasite
Drotaverine hydrochloride
Cat.No: T8787
Synonym:
Target: PDE
Dehydrocorydaline chloride
Cat.No: T10990
Synonym: 盐酸脱氢紫堇碱,13-Methylpalmatine chloride
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
6-Chloro-2,4-dibromophenol
Cat.No: TN7197
Synonym: 2,4-dibromo-6-chloro-phenol,2,4-二溴-6-氯苯酚,2,4-dibromo-6-chlorophenol,ZINC397569
Target: Others
Quinidine hydrochloride monohydrate
Cat.No: T0266
Synonym: 奎宁树,奎尼丁盐酸盐一水合物,奎尼丁盐酸盐,Quinidine hydrochloride
Target: Potassium Channel, Sodium Channel, Parasite
Nitidine chloride
Cat.No: T5S0761
Synonym:
Target: Apoptosis, ERK, FAK, p38 MAPK, NF-κB, Topoisomerase, STAT, Parasite
Diphenhydramine hydrochloride
Cat.No: T0330
Synonym: 盐酸苯海拉明,Diphenhydramine HCl,DPH
Target: Histamine Receptor
Acetylcholine chloride
Cat.No: T1221
Synonym: ACh chloride,Pilofrin,氯化乙酰胆碱
Target: Calcium Channel, Endogenous Metabolite, AChR
Quinine dihydrochloride
Cat.No: T4333
Synonym: 盐酸奎宁,Quinine bimuriate
Target: Others
(±)-Carnitine chloride
Cat.No: T6475
Synonym: Monocamin,DL-Carnitine HCl,Bicarnesine,混旋肉碱盐酸盐,DL-Carnitine chloride
Target: Reactive Oxygen Species
Delphinidin 3-glucoside chloride
Cat.No: TN1564
Synonym: Delphinidin-3-O-glucoside chloride
Target: Apoptosis, EGFR
L-Cystine dihydrochloride
Cat.No: T60789
Synonym:
Target:
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