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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T4093 Fabomotizole hydrochloride

Afobazole hydrochloride,CM346 hydrochloride

MAO Metabolism; Neuroscience
Fabomotizole hydrochloride (CM346 hydrochloride) 是一种具有抗焦虑和神经保护作用的化合物。
T62385 Befiradol hydrochloride

NLX-112 hydrochloride,F 13640 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Befiradol hydrochloride (NLX-112 hydrochloride) 是一种具有选择性的5-羟色胺 1A (5-HT)1A 受体激动剂,具有抗焦虑活性。Befiradol hydrochloride 抑制突变ATXN3聚集。
T4045 Epetraborole hydrochloride

GSK2251052 hydrochloride

Antibacterial Microbiology/Virology
Epetraborole hydrochloride (GSK2251052 hydrochloride) 是一个新型 LeuRS 抑制剂,通过绑定 leucyl-tRNA 合成酶终端的腺苷核糖抑制蛋白合成,可研究 Gram-negative 细菌引起的感染。
T2092 Amitifadine hydrochloride

DOV-21947 hydrochloride,EB-1010 hydrochloride

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine GPCR/G Protein; Neuroscience
Amitifadine hydrochloride (EB-1010 hydrochloride) 是一种 5-羟色胺-去甲肾上腺素-多巴胺的再摄取抑制剂(SNDRI),其在 HEK 293 细胞中测得的 IC50值分别为 12, 23, 96 nM。
T8617 GMQ hydrochloride

NSC 403387 hydrochloride

Others Others
GMQ hydrochloride (NSC-403387 hydrochloride) 是一种有效的选择性酸感应离子通道 (ASIC) 调节剂。它在中性 pH 值下激活 ASIC3 通道并阻止酸引起的最大峰值电流。
T11872L LMP744 hydrochloride

NSC706744 hydrochloride,MJ-III65 hydrochloride

Topoisomerase DNA Damage/DNA Repair
LMP744 hydrochloride (NSC-706744 hydrochloride) 是一种是拓扑异构酶 1 抑制剂,显示出抗肿瘤的活性。
T12225L Nevanimibe hydrochloride

PD-132301 hydrochloride,ATR101 hydrochloride

Apoptosis; Acyltransferase Apoptosis; Metabolism
Nevanimibe hydrochloride (PD-132301 hydrochloride) 是一种口服有效的,选择性酰基辅酶 A:胆固醇 O-酰基转移酶 1 抑制剂,EC50为 9 nM。它抑制 ACAT2,EC50为 368 nM。它诱导细胞凋亡,具有抗肾上腺皮质癌的潜力。
T10898 Samuraciclib hydrochloride

ICEC0942 hydrochloride,CT7001 hydrochloride

Apoptosis; CDK Apoptosis; Cell Cycle/Checkpoint
Samuraciclib hydrochloride (ICEC0942 hydrochloride) 是一种具有选择性,ATP 竞争性和口服活性的CDK7抑制剂,IC50为 41 nM。它以 GI50值为 0.2-0.3 µM 来抑制乳腺癌细胞系的生长,具有抗肿瘤作用。
T11508L Camicinal hydrochloride

GSK962040 hydrochloride

Others; Motilin Receptor GPCR/G Protein; Others
Camicinal hydrochloride (GSK962040 hydrochloride) 是胃动素受体的特异性激动剂 (pEC50 = 7.9)。
T10797 Chlormidazole hydrochloride

Clomidazole hydrochloride

Antifungal Microbiology/Virology
Chlormidazole hydrochloride (Clomidazole hydrochloride) 是一种抗真菌剂,抑制多种真菌和部分革兰氏阳性球菌,可治疗指甲和皮肤的真菌和细菌感染。
T4370 Resminostat hydrochloride

4SC-201 hydrochloride,RAS2410 hydrochloride

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
Resminostat hydrochloride (RAS2410 hydrochloride) 是HDAC1,HHDAC3和HDAC6抑制剂,IC50值分别为 42.5、50.1和71.8 nM,对 HDAC8 的活性较低,IC50值为 877 nM。
T11213 Epertinib hydrochloride

S-22611 hydrochloride

EGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Epertinib hydrochloride (S-22611 hydrochloride) 是口服可逆的选择性EGFR、HER2和HER4抑制剂,IC50值分别为 1.48、7.15 和 2.49 nM,具有抗肿瘤活性。
T13202 Trilaciclib hydrochloride

G1T28 hydrochloride

CDK Cell Cycle/Checkpoint
Trilaciclib hydrochloride (G1T28 hydrochloride) 是一种CDK4/6的抑制剂,对 CDK4 和 CDK6 的IC50值分别为 1 nM 和 4 nM。
T11188L Emixustat hydrochloride

ACU-4429 hydrochloride

Others Others
Emixustat hydrochloride (ACU-4429 hydrochloride) 能够高效抑制11-顺式-视黄醇的生产(IC50:232±3 nM)。
T15378L Gemcitabine elaidate hydrochloride

CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride

Others Others
Gemcitabine elaidate (CP-4126) hydrochloride 是 Gemcitabine 的亲脂性前药。Gemcitabine elaidate hydrochloride 通过酯酶转化为 Gemcitabine 以被磷酸化。Gemcitabine elaidate hydrochloride 可以口服给药,具有抗肿瘤活性。
T11004 Desformylflustrabromine hydrochloride

dFBr hydrochloride,Deformylflustrabromine hydrochloride

AChR Neuroscience
Desformylflustrabromine hydrochloride (dFBr hydrochloride) 是α4β2神经元中烟碱乙酰胆碱受体(nAChR)的选择性激动剂,pEC50为6.48。
T6104 Cerdulatinib hydrochloride

Cerdulatinib,PRT2070,PRT062070 hydrochloride,PRT062070,PRT2070 hydrochloride

MLK; c-Fms; Tyrosine Kinases; Hippo pathway; JAK; Syk Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; MAPK; Stem Cells; Tyrosine Kinase/Adaptors
Cerdulatinib hydrochloride (PRT2070 hydrochloride) 是一种选择性可逆,具有口服活性、 ATP 竞争性的 SYK 和 JAK 的双重抑制剂,抑制 JAK1、2、3、SYK 和 Tyk2的 IC50值分别为12、6、8、32 和 0.5 nM。它可用于研究自身免疫性疾病和B 细胞恶性肿瘤。
T12311 Tirabrutinib hydrochloride

ONO-4059 (hydrochloride),GS-4059 (hydrochloride)

BTK Angiogenesis; Tyrosine Kinase/Adaptors
Tirabrutinib hydrochloride (GS-4059 (hydrochloride)) 是一种有选择性的、新颖的抑制剂 (IC50:2.2 nM)。 在 B 细胞中 ONO-4059 结合 BTK,因此阻止 B 细胞受体信号和阻碍 B 细胞的发展。
T10221 Abeprazan hydrochloride

DWP14012 hydrochloride,Fexuprazan hydrochloride

Proton pump Membrane transporter/Ion channel
Abeprazan hydrochloride (Fexuprazan hydrochloride) 是一种有效的、可逆的、具有口服活性的potassium-competitive acid 阻滞剂,通过竞争性的与钾离子结合抑制 H+,K+- ATPase,而无需酸激活。Abeprazan hydrochloride 是一种质子泵抑制剂(PPI),通过减少胃酸的产生而起作用,可用于治疗胃酸相关疾病,如胃食管反流病(GERD)和消化性溃疡。
T4081 MPTP hydrochloride

MPTP-hydrochloride

Apoptosis; Dopamine Receptor Apoptosis; GPCR/G Protein; Neuroscience
MPTP hydrochloride 是 MPP+ 的前体,是一种多巴胺神经毒素,具有血脑屏障渗透性。MPTP hydrochloride 对多巴胺能神经元有毒,可以导致帕金森症,被广泛应用于帕金森动物模型的构建。
T10305 Amiselimod hydrochloride

MT-1303 hydrochloride

S1P Receptor; LPL Receptor GPCR/G Protein
Amiselimod hydrochloride (MT-1303 hydrochloride) 是一种鞘氨醇 1-磷酸受体 1 (S1P1) 调节剂。
T11353L Gallopamil hydrochloride

Methoxyverapamil hydrochloride

Calcium Channel Membrane transporter/Ion channel; Metabolism
Gallopamil hydrochloride (Methoxyverapamil hydrochloride) 是苯烷基胺钙的拮抗剂。Gallopamil hydrochloride 可用于抗心律失常和血管扩张剂研究。
T21969 ML-095 hydrochloride

CID-25067483 hydrochloride,MLS-0315848 hydrochloride

Phospholipase Metabolism
ML-095 hydrochloride (CID-25067483 hydrochloride) 是一种特异性胎盘碱性磷酸酶抑制剂。它抑制 PLAP、TNAP 和 IAP,IC50 分别为 2.1、>100 和 53 μM。
T13278 Valecobulin hydrochloride

CKD-516 hydrochloride

Microtubule Associated Cytoskeletal Signaling
Valecobulin hydrochloride (CKD-516 hydrochloride) 是 S516 的缬氨酸前体药和血管阻断剂。Valecobulin hydrochloride 对β-微管蛋白聚合有强效的抑制作用,对小鼠和人类的实体肿瘤具有显著的抗肿瘤活性。
T12266L2 Ilginatinib hydrochloride

NS-018 hydrochloride

Tyrosine Kinases; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Ilginatinib hydrochloride (NS-018 hydrochloride) 是一种可口服的 JAK2强效抑制剂,IC50值为 0.72 nM,对其选择性是对 JAK1、JAK3和 Tyk2 的 46、54 和 22 倍,IC50分别为 33、39 和 22 nM。
T12565 PRX933 hydrochloride

BVT-933 hydrochloride,GW876167 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
PRX933 hydrochloride (GW876167 hydrochloride) 是一种 5-HT2C 受体激动剂,可用于高血压急性期治疗的研究。
T39740 Acoramidis hydrochloride

AG10 hydrochloride,Alxn2060 hydrochloride

Others Others
Acoramidis hydrochloride (Alxn2060 hydrochloride) 是具有口服活性的、选择性的甲状腺素转运蛋白 (TTR (transthyretin)) 的稳定剂,对野生型和 V1221 突变型均有效。Acoramidis hydrochloride 可用于转体甲状腺素淀粉样变性的研究。
T10758L Centanafadine hydrochloride

EB-1020 hydrochloride

Dopamine Receptor; Serotonin Transporter; Adrenergic Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Centanafadine hydrochloride (EB-1020 hydrochloride) 是一种去甲肾上腺素(NE)/多巴胺(DA)转运的双抑制剂,还能抑制5-羟色胺(serotonin)转运体。它对人 NE,DA 和5-羟色胺转运体的 IC50值分别为6 nM,38 nM 和 83 nM。
T35326 Labetalone hydrochloride

Labetalone hydrochloride,Benzoic amide

Others Others
Labetalone hydrochloride (Benzoic amide) 是 Labetalol 的一种杂质。Labetalol 是一种口服有效的肾上腺素能受体阻断药物,对 α 和 β 受体部位都有竞争性拮抗作用。
T3184 Kevetrin hydrochloride

Thioureidobutyronitrile HCl,thioureido butyronitrile hydrochloride,4-Isothioureidobutyronitrile hydrochloride

Mdm2; p53 Apoptosis
Kevetrin hydrochloride (4-Isothioureidobutyronitrile hydrochloride) 是一种小分子,是肿瘤抑制蛋白 p53 的激活剂,具有潜在的抗肿瘤活性。
T9251 Fedratinib hydrochloride hydrate

TG-101348 hydrochloride hydrate,SAR 302503 hydrochloride hydrate

Apoptosis; JAK Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Fedratinib hydrochloride hydrate (SAR 302503 hydrochloride hydrate) 是一种选择性的,ATP 竞争性和具有口服活性的JAK2抑制剂,对于JAK2和JAK2V617F 激酶的IC50均为 3 nM。它可诱导癌细胞凋亡,可研究骨髓增生性疾病。
T61233 Penehyclidine hydrochloride

Penequinine hydrochloride

NF-κB; AChR Neuroscience; NF-κB
Penehyclidine hydrochloride (Penequinine hydrochloride) 是M1和M3拮抗剂,并激活肺组织中的NF-κB。 Penehyclidine hydrochloride 抑制炎症因子的释放,并显示出抗胆碱能特性。
T15207 Eleclazine hydrochloride

GS 6615 hydrochloride

Sodium Channel Membrane transporter/Ion channel
Eleclazine hydrochloride (GS 6615 hydrochloride) 是新型 Na+电流抑制剂,IC50是0.7 uM。
T29645 Adatanserin hydrochloride

WY50324 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Adatanserin hydrochloride (WY50324 hydrochloride) 是一种新型 5-HT(1A)/5-HT(2) 受体配体,具有潜在的神经保护作用,抑制内源性氨基酸缺血性外排,可用于研究抑郁症和焦虑症。
T4134 OTS514 hydrochloride

OTS-514 hydrochloride,OTS514 hydrochloride(1338540-63-8(free base))

Apoptosis; TOPK Apoptosis; MAPK
OTS514 hydrochloride 是一种高效的TOPK 抑制剂,IC50为 2.6 nM。它可强效抑制 TOPK 阳性的肿瘤细胞生长,诱导细胞周期停滞和凋亡。
T7000 Tiagabine hydrochloride

NO328 hydrochloride,盐酸噻加宾,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Tiagabine hydrochloride (NO050328 hydrochloride) 是具有抗惊厥特性的选择性GABA 再摄取抑制剂,在突触体、神经元和神经胶质中,能够抑制 [3H]GABA 的重摄取,IC50值分别为 67、446 和 182 nM。
T4369 SCH-23390 hydrochloride

R-(+)-SCH23390 hydrochloride

Potassium Channel; Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) 是一种选择性多巴胺 D1样受体拮抗剂,对 D1和 D5受体的Ki 分别为 0.2 和 0.3 nM。它还抑制 G 蛋白偶联的内向整流钾通道,IC50为 268 nM。它与5-HT2和5-HT1C 受体具有高亲和力,是人5-HT2C 受体激动剂,Ki 为 9.3 nM。
T22689 CP94253 hydrochloride

CP 94253 hydrochloride

Others; 5-HT Receptor GPCR/G Protein; Neuroscience; Others
CP94253 hydrochloride (CP 94253 hydrochloride) 是一种有效的、特异性的和中枢活性的 5-HT1B 受体激动剂,Ki 为 2 nM。5-HT1A、5-HT1D、5-HT1C 和 5-HT2 的 Ki 分别为 89、49、860 和 1600 nM 。
T4423 LY 303511 hydrochloride

LY303511 hydrochloride

Potassium Channel; TNF; mTOR Apoptosis; Membrane transporter/Ion channel; PI3K/Akt/mTOR signaling
LY 303511 hydrochloride 是LY294002 的一种结构类似物。LY 303511 hydrochloride 可增强 SHEP-1 神经母细胞瘤细胞的TRAIL 敏感性,还可逆地阻断 MIN6 胰岛瘤细胞中的K+电流。
T12201 Nebracetam hydrochloride

WEB 1881 FU hydrochloride

AChR Neuroscience
Nebracetam hydrochloride (WEB 1881 FU hydrochloride) 是促智 M1-毒蕈碱的激动剂。 它诱导细胞内 Ca2+ 浓度升高, EC50 为 1.59 mM。
T60523 Agomelatine hydrochloride

S-20098 hydrochloride

MT Receptor Neuroscience
Agomelatine hydrochloride (S-20098 hydrochloride) (S-20098 hydrochloride) 是特异性的MT1和MT2受体激动剂,对 CHO-hMT1的Ki 值为0.1 nM,对HEK-hMT1的Ki 值为0.06 nM,对CHO-hMT2的Ki 值为0.12 nM,对HEK-hMT2 的Ki 值为0.27 nM。Agomelatine hydrochloride 是选择性的5-羟色胺2C(5-HT2C)受体拮抗剂,对天然 (猪) 和克隆的人 5-HT2C 受体的pKi 值分别为 6.4 和 6.2。
T68113 Naluzotan hydrochloride

PRX 00023 hydrochloride

EGFR; 5-HT Receptor Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Neuroscience; Tyrosine Kinase/Adaptors
Naluzotan hydrochloride (PRX 00023 hydrochloride) 是一种小分子、非氮杂吡酮、5-羟色胺(5-HT)1A 受体激动剂和sigma-1受体拮抗剂。在之前的临床试验中,该化合物在400多名患者中被证明安全且耐受性良好。
T15456 GYKI 53655 hydrochloride

GYKI53655 hydrochloride,LY300168 hydrochloride

GluR Neuroscience
GYKI 53655 hydrochloride (LY300168 hydrochloride) 是一种 AMPA 的拮抗剂,可用于研究神经系统疾病。
T1272L Cytarabine hydrochloride

Ara-C hydrochloride,Cytosine Arabinoside hydrochloride

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Cytarabine hydrochloride (Ara-C hydrochloride) 是一种核苷类似物,可导致 S 期细胞周期停滞并抑制DNA 聚合酶。Cytarabine 抑制DNA 合成,IC50为 16 nM。Cytarabine hydrochloride 对HSV 具有抗病毒作用。
T9189 Iptacopan hydrochloride

Iptacopan HCl,LNP023 hydrochloride

Complement System Immunology/Inflammation
Iptacopan hydrochloride (LNP023 hydrochloride) 是一种可口服、高效和高选择性的因子 B 抑制剂,IC50 为 10 nM。 LNP023 显示与人因子 B 的直接、可逆和高亲和力结合,KD 为 7.9 nM。
T1778 AT7519 Hydrochloride

AT7519 HCl,AT 7519 hydrochloride salt

Apoptosis; GSK-3; CDK Apoptosis; Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells
AT7519 Hydrochloride (AT7519 HCl) 是一种多CDK 抑制剂,对 CDK1、CDK2、CDK4-CDK6 以及 CDK9 的IC50值分别为 210、47、100、13、170 和 <10 nM。
T4230 PF-3758309 hydrochloride

PF-03758309 hydrochloride

Apoptosis; PAK Apoptosis; Cytoskeletal Signaling
PF-3758309 hydrochloride (PF-03758309 hydrochloride) 是一种口服的、可逆的 ATP 竞争性PAK4抑制剂,Kd 为 2.7 nM,Ki 为 18.7 nM。它抑制锚定独立生长、诱导凋亡、细胞骨架重塑和抑制增殖,具有 PAK4 抑制剂的预期细胞功能。
T4361 CBL0137 hydrochloride

CBL0137,CBLC137,Curaxin 137,CBL-C137 hydrochloride,Curaxin-137 hydrochloride

Others; NF-κB; p53 Apoptosis; NF-κB; Others
CBL0137 hydrochloride (Curaxin-137 hydrochloride) 是一种组蛋白分子伴侣FACT 的抑制剂,也可激活p53并抑制NF-κB,对于它们的EC50值分别为 0.37 和 0.47 μM。
T0766 Promazine hydrochloride

Romtiazin hydrochloride,Sinophenin hydrochloride,盐酸丙嗪

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR GPCR/G Protein; Neuroscience
Promazine hydrochloride (Romtiazin hydrochloride) 是一种抗精神病药,也是一种多巴胺受体 (D2) 拮抗剂,能够抑制多巴胺能神经传递。
T22486 Vesamicol hydrochloride

(±)-AH5183 hydrochloride

AChR Neuroscience
Vesamicol hydrochloride ((±)-AH5183 hydrochloride) ((±)-AH5183 hydrochloride) 是一种有效的囊泡乙酰胆碱转运 (vesicular acetylcholine transport) 抑制剂,Ki 为 2 nM。(±)-Vesamicol hydrochloride 也对 σ1 和 σ2 受体具有高亲和力,Ki 值分别为 26 nM 和 34 nM。

化合物

Fabomotizole hydrochloride
Cat.No: T4093
Synonym: Afobazole hydrochloride,CM346 hydrochloride
Target: MAO
Befiradol hydrochloride
Cat.No: T62385
Synonym: NLX-112 hydrochloride,F 13640 hydrochloride
Target: 5-HT Receptor
Epetraborole hydrochloride
Cat.No: T4045
Synonym: GSK2251052 hydrochloride
Target: Antibacterial
Amitifadine hydrochloride
Cat.No: T2092
Synonym: DOV-21947 hydrochloride,EB-1010 hydrochloride
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine
GMQ hydrochloride
Cat.No: T8617
Synonym: NSC 403387 hydrochloride
Target: Others
LMP744 hydrochloride
Cat.No: T11872L
Synonym: NSC706744 hydrochloride,MJ-III65 hydrochloride
Target: Topoisomerase
Nevanimibe hydrochloride
Cat.No: T12225L
Synonym: PD-132301 hydrochloride,ATR101 hydrochloride
Target: Apoptosis, Acyltransferase
Samuraciclib hydrochloride
Cat.No: T10898
Synonym: ICEC0942 hydrochloride,CT7001 hydrochloride
Target: Apoptosis, CDK
Camicinal hydrochloride
Cat.No: T11508L
Synonym: GSK962040 hydrochloride
Target: Others, Motilin Receptor
Chlormidazole hydrochloride
Cat.No: T10797
Synonym: Clomidazole hydrochloride
Target: Antifungal
Resminostat hydrochloride
Cat.No: T4370
Synonym: 4SC-201 hydrochloride,RAS2410 hydrochloride
Target: HDAC
Epertinib hydrochloride
Cat.No: T11213
Synonym: S-22611 hydrochloride
Target: EGFR, HER
Trilaciclib hydrochloride
Cat.No: T13202
Synonym: G1T28 hydrochloride
Target: CDK
Emixustat hydrochloride
Cat.No: T11188L
Synonym: ACU-4429 hydrochloride
Target: Others
Gemcitabine elaidate hydrochloride
Cat.No: T15378L
Synonym: CO-101 hydrochloride,Gemcitabine elaidate hydrochloride(210829-30-4(free base)),Gemcitabine 5'-elaidate hydrochloride,CP-4126 hydrochloride
Target: Others
Desformylflustrabromine hydrochloride
Cat.No: T11004
Synonym: dFBr hydrochloride,Deformylflustrabromine hydrochloride
Target: AChR
Cerdulatinib hydrochloride
Cat.No: T6104
Synonym: Cerdulatinib,PRT2070,PRT062070 hydrochloride,PRT062070,PRT2070 hydrochloride
Target: MLK, c-Fms, Tyrosine Kinases, Hippo pathway, JAK, Syk
Tirabrutinib hydrochloride
Cat.No: T12311
Synonym: ONO-4059 (hydrochloride),GS-4059 (hydrochloride)
Target: BTK
Abeprazan hydrochloride
Cat.No: T10221
Synonym: DWP14012 hydrochloride,Fexuprazan hydrochloride
Target: Proton pump
MPTP hydrochloride
Cat.No: T4081
Synonym: MPTP-hydrochloride
Target: Apoptosis, Dopamine Receptor
Amiselimod hydrochloride
Cat.No: T10305
Synonym: MT-1303 hydrochloride
Target: S1P Receptor, LPL Receptor
Gallopamil hydrochloride
Cat.No: T11353L
Synonym: Methoxyverapamil hydrochloride
Target: Calcium Channel
ML-095 hydrochloride
Cat.No: T21969
Synonym: CID-25067483 hydrochloride,MLS-0315848 hydrochloride
Target: Phospholipase
Valecobulin hydrochloride
Cat.No: T13278
Synonym: CKD-516 hydrochloride
Target: Microtubule Associated
Ilginatinib hydrochloride
Cat.No: T12266L2
Synonym: NS-018 hydrochloride
Target: Tyrosine Kinases, JAK
PRX933 hydrochloride
Cat.No: T12565
Synonym: BVT-933 hydrochloride,GW876167 hydrochloride
Target: 5-HT Receptor
Acoramidis hydrochloride
Cat.No: T39740
Synonym: AG10 hydrochloride,Alxn2060 hydrochloride
Target: Others
Centanafadine hydrochloride
Cat.No: T10758L
Synonym: EB-1020 hydrochloride
Target: Dopamine Receptor, Serotonin Transporter, Adrenergic Receptor, Norepinephrine
Labetalone hydrochloride
Cat.No: T35326
Synonym: Labetalone hydrochloride,Benzoic amide
Target: Others
Kevetrin hydrochloride
Cat.No: T3184
Synonym: Thioureidobutyronitrile HCl,thioureido butyronitrile hydrochloride,4-Isothioureidobutyronitrile hydrochloride
Target: Mdm2, p53
Fedratinib hydrochloride hydrate
Cat.No: T9251
Synonym: TG-101348 hydrochloride hydrate,SAR 302503 hydrochloride hydrate
Target: Apoptosis, JAK
Penehyclidine hydrochloride
Cat.No: T61233
Synonym: Penequinine hydrochloride
Target: NF-κB, AChR
Eleclazine hydrochloride
Cat.No: T15207
Synonym: GS 6615 hydrochloride
Target: Sodium Channel
Adatanserin hydrochloride
Cat.No: T29645
Synonym: WY50324 hydrochloride
Target: 5-HT Receptor
OTS514 hydrochloride
Cat.No: T4134
Synonym: OTS-514 hydrochloride,OTS514 hydrochloride(1338540-63-8(free base))
Target: Apoptosis, TOPK
Tiagabine hydrochloride
Cat.No: T7000
Synonym: NO328 hydrochloride,盐酸噻加宾,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride
Target: GABA Receptor
SCH-23390 hydrochloride
Cat.No: T4369
Synonym: R-(+)-SCH23390 hydrochloride
Target: Potassium Channel, Dopamine Receptor, 5-HT Receptor
CP94253 hydrochloride
Cat.No: T22689
Synonym: CP 94253 hydrochloride
Target: Others, 5-HT Receptor
LY 303511 hydrochloride
Cat.No: T4423
Synonym: LY303511 hydrochloride
Target: Potassium Channel, TNF, mTOR
Nebracetam hydrochloride
Cat.No: T12201
Synonym: WEB 1881 FU hydrochloride
Target: AChR
Agomelatine hydrochloride
Cat.No: T60523
Synonym: S-20098 hydrochloride
Target: MT Receptor
Naluzotan hydrochloride
Cat.No: T68113
Synonym: PRX 00023 hydrochloride
Target: EGFR, 5-HT Receptor
GYKI 53655 hydrochloride
Cat.No: T15456
Synonym: GYKI53655 hydrochloride,LY300168 hydrochloride
Target: GluR
Cytarabine hydrochloride
Cat.No: T1272L
Synonym: Ara-C hydrochloride,Cytosine Arabinoside hydrochloride
Target: DNA/RNA Synthesis
Iptacopan hydrochloride
Cat.No: T9189
Synonym: Iptacopan HCl,LNP023 hydrochloride
Target: Complement System
AT7519 Hydrochloride
Cat.No: T1778
Synonym: AT7519 HCl,AT 7519 hydrochloride salt
Target: Apoptosis, GSK-3, CDK
PF-3758309 hydrochloride
Cat.No: T4230
Synonym: PF-03758309 hydrochloride
Target: Apoptosis, PAK
CBL0137 hydrochloride
Cat.No: T4361
Synonym: CBL0137,CBLC137,Curaxin 137,CBL-C137 hydrochloride,Curaxin-137 hydrochloride
Target: Others, NF-κB, p53
Promazine hydrochloride
Cat.No: T0766
Synonym: Romtiazin hydrochloride,Sinophenin hydrochloride,盐酸丙嗪
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR
Vesamicol hydrochloride
Cat.No: T22486
Synonym: (±)-AH5183 hydrochloride
Target: AChR
Cat. No. Product Name Target Signaling Pathways
T8769 Harmaline hydrochloride

Harmidine hydrochloride

Others Others
Harmaline hydrochloride (Harmidine hydrochloride) 是一种荧光吲哚生物碱,来自 harmala 生物碱和 β-咔啉。它是 harmine 的部分氢化形式。 Harmaline 通过诱导下橄榄神经元的节律性放电在正常大鼠中产生全身性震颤。
T13302 Viquidil hydrochloride

Quinotoxine hydrochloride

Others Others
Viquidil hydrochloride (Quinotoxine hydrochloride) 是奎尼丁的同分异构体,是一种脑血管扩张剂,具有抗血栓作用。
T2774 Lycorine hydrochloride

石蒜碱,Licorine hydrochloride,Galanthidine hydrochloride,Narcissine hydrochloride,Lycorine chloride,Amarylline hydrochloride,盐酸石蒜碱

Virus Protease; HCV Protease; Antibacterial; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Lycorine hydrochloride (Narcissine hydrochloride) 是黑色素瘤血管生成抑制剂,是一种来自石蒜的主要活性成分,抑制 Hey1B 细胞的有丝分裂增殖,IC50值为 1.2 μM,具有抗肿瘤活性。
T6460 Cysteamine hydrochloride

2-Mercaptoethylamine Hydrochloride,β-Mercaptoethylamine Hydrochloride,半胱胺盐酸盐,Thioethanolamine Hydrochloride,2-Aminoethanethiol Hydrochloride,Cysteamine HCl,Bekaptan

Apoptosis; Others; Reactive Oxygen Species; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB; Others
Cysteamine hydrochloride (Thioethanolamine Hydrochloride) 是一种可口服的,用于肾病型胱胺酸症的小分子药物,也可作为抗氧化剂。
TN1519L (-)-Coclaurine hydrochloride

(-)-Coclaurine hydrochloride (486-39-5 Free base)

AChR Neuroscience
(-)-Coclaurine hydrochloride 是从 Sarcopetalum harveyanum 中分离出来的,是一种 nAChR 拮抗剂。
TN1724 Harmalol hydrochloride

Harmidol hydrochloride

P450; Antioxidant Metabolism; oxidation-reduction
Harmalol hydrochloride (Harmidol hydrochloride) 是一种可从Peganum harmala L.的种子中提取出来的β-咔啉生物碱。Harmalol hydrochloride 是Harmaline 的主要代谢产物,在转录和翻译后水平上显著抑制二恶英介导的 CYP1A1 诱导。Harmalol hydrochloride 在去氧肾上腺素或KCl 预先收缩的分离大鼠胸主动脉制剂中显示出血管松弛活性。 Harmalol hydrochloride 具有抗氧化活性.
T3232 Higenamine hydrochloride

Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Higenamine hydrochloride (norcoclaurine HCl) 是一种 β2-AR 激动剂,是用于心力衰竭相关研究的中药乌头的关键成分,具有抗凋亡活性。
T2921 Sinomenine hydrochloride

盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride

Apoptosis; NF-κB; Opioid Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; GPCR/G Protein; Neuroscience; NF-κB
Sinomenine hydrochloride (Kukoline hydrochloride) 是来自汉防己的一种生物碱,是NF-κB 活化的阻断剂。Sinomenine 也是一种 μ 阿片受体激活剂。
T1680 Tolazoline hydrochloride

Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Tolazoline hydrochloride (NSC35110(hydrochloride)) 是一种 α 肾上腺素受体抑制剂。
T1549 Raloxifene hydrochloride

LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl

Estrogen Receptor/ERR; Others; MAO; Estrogen/progestogen Receptor; Autophagy Autophagy; Endocrinology/Hormones; Metabolism; Neuroscience; Others
Raloxifene hydrochloride (LY156758 hydrochloride) 是一种选择性且可口服的雌激素受体调节剂,用于预防绝经后妇女的骨质疏松症。它对骨骼和胆固醇代谢具有雌激素激动作用,但对乳腺和子宫组织具有完全的雌激素拮抗作用。
T4429 Rauwolscine hydrochloride

Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) 是一种高选择性的 α2 adrenergic 受体拮抗剂,Ki=12 nM。
T2953 Ligustrazine hydrochloride

Tetramethylpyrazine hydrochloride,Tetramethylpyrazine HCl,Chuanxiongzine hydrochloride,Tetrapyrazine HCl,盐酸川芎嗪

Others Others
Ligustrazine hydrochloride (Chuanxiongzine hydrochloride) 是一种天然产物。
T0268 Lobeline hydrochloride

盐酸洛贝林,α-Lobeline hydrochloride,L-Lobeline hydrochloride

AChR Neuroscience
Lobeline hydrochloride (α-Lobeline hydrochloride) 是一种烟碱样受体激动剂,是神经元烟碱受体α3β2和α4β2拮抗剂。
T22911 β-N-methylamino-L-alanine hydrochloride

L-BMAA hydrochloride

Others Others
β-N-methylamino-L-alanine hydrochloride (L-BMAA hydrochloride) 是由蓝细菌产生的一种神经毒素,既有导致肌萎缩性侧索硬化症 (ALS) 以及其他可能的神经退行性疾病可能性。
T2203 D-Carnitine hydrochloride

(S)-Carnitine Hydrochloride,L-Carnitine hydrochloride

Others; Endogenous Metabolite Metabolism; Others
D-Carnitine hydrochloride ((S)-Carnitine Hydrochloride) 已被用于研究麦角硫因素转运蛋白 SLC22A4 和肉毒碱转运蛋白 SLC22A5,也被用于使棕榈酸进入线粒体。
T0486L Irinotecan Hydrochloride

盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan Hydrochloride (CPT-11 hydrochloride) 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。
T8384 Gatifloxacin hydrochloride

AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Gatifloxacin hydrochloride (AM-1155 hydrochloride) 是一种氟喹诺酮类抗生素,有广谱抗菌活性。它可抑制大肠杆菌 DNA 解旋酶 (IC50=0.109 μg/ml)和细菌 II 型拓扑异构酶(IC50=13.8 μg/ml) 。它在动物模型中,可研究细菌性结膜炎。
TN6787L N-Noratherosperminine hydrochloride

N-Noratherosperminine hydrochloride (74606-53-4 free base)

Others Others
N-Noratherosperminine hydrochloride 是生物碱盐酸盐。 Noratherosperminine 可从 Cryptocarya nigra 中提取。
TQ0296L N-Nornuciferine hydrochloride(4846-19-9 free base)

N-Nornuciferine hydrochloride

P450 Metabolism
N-Nornuciferine hydrochloride(4846-19-9 free base) (N-Nornuciferine hydrochloride) 是荷叶中的一种 aporphine 生物碱,显着抑制 CYP2D6(IC50:3.76 μM,Ki:2.34 μM)。
T1591 Ancitabine hydrochloride

NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C

Others; DNA/RNA Synthesis; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。
T8298 Vasicine hydrochloride

鸭嘴花碱盐酸盐,Peganine hydrochloride

Antibacterial; Antibiotic Microbiology/Virology
Vasicine hydrochloride (Peganine hydrochloride) 是从Justicia adhatoda 中分离得到的一种喹唑啉类生物碱,有抗结核活性。
T21344 1-Deoxynojirimycin hydrochloride

Moranoline,去氧野艽霉素盐酸盐,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin

PI3K; Antibacterial; Antibiotic; Glucosidase Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
1-Deoxynojirimycin hydrochloride (Moranoline) 是一种口服有效的 α-葡萄糖苷酶抑制剂,具有降血糖、减肥和抗病毒的作用,可抑制餐后血糖,预防糖尿病。
T8149 Dobutamine hydrochloride

盐酸多巴酚丁胺,Dobutamine (hydrochloride)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Dobutamine hydrochloride (Dobutamine(hydrochloride)) 是一种合成的儿茶酚胺,可作用于肾上腺素能受体α1-AR、β1-AR 和β2-AR,是一种选择性的 β1-AR 受体激动剂,对 α1-AR 和 β2-AR 作用相对较弱。它能够增加心输出量,矫正低灌注。
T2941 Glucosamine hydrochloride

Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride

Reactive Oxygen Species; HIF/HIF Prolyl-Hydroxylase; Endogenous Metabolite; Autophagy Autophagy; Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB
Glucosamine hydrochloride (Chitosamine hydrochloride) 是软骨基质和滑液中糖胺聚糖的天然成分,常用作骨关节炎的治疗方法。它也是一种氨基糖,是糖基化蛋白和脂质生化合成的突出前体,用作膳食补充剂。
T1304 Chlortetracycline hydrochloride

Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
T2209 Serotonin hydrochloride

5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride

5-HT Receptor; Endogenous Metabolite; Transferase GPCR/G Protein; Metabolism; Neuroscience
Serotonin hydrochloride (Serotonin HCl) 是一种内源性 5-HT 受体激动剂、CNS 中的单胺神经递质和儿茶酚 O-甲基转移酶 (COMT) 抑制剂,Ki 值为 44 μM。
T4753 Imidazoleacetic acid hydrochloride

I4AA,(4-Imidazolyl)acetic acid hydrochloride,4-咪唑乙酸盐酸盐,4-Imidazoleacetic acid hydrochloride

Endogenous Metabolite; Antibiotic Metabolism; Microbiology/Virology
Imidazoleacetic acid hydrochloride (I4AA) 是咪唑衍生物,具有潜在的抗结核性能。它还用于制备β-分泌酶的酰基胍抑制剂。
T4080 Leonurine hydrochloride

盐酸益母草碱,SCM-198 hydrochloride,SCM-198 HCl

TLR; Autophagy Autophagy; Immunology/Inflammation
Leonurine hydrochloride (SCM-198 hydrochloride) 是从益母草中分离的一种生物碱,具有抗氧化和抗炎活性。
T2811 Harmine hydrochloride

telepathine hydrochloride,盐酸哈尔明碱

5-HT Receptor; DYRK; GluR Cell Cycle/Checkpoint; GPCR/G Protein; Neuroscience; Tyrosine Kinase/Adaptors
Harmine hydrochloride (telepathine hydrochloride) 是一种 DYRK 抑制剂,具有抗癌和抗炎活性。它对5-HT2A 血清素受体具有高亲和力,Ki 值为 397 nM。
T0973L Pyridoxine hydrochloride

Pyridoxine HCl,吡哆醇盐酸盐,Pyridoxol (hydrochloride),吡哆醇盐酸盐(维生素B6),Vitamin B6 (hydrochloride),Vitamin B6

Nrf2; Endogenous Metabolite Immunology/Inflammation; Metabolism
Pyridoxine hydrochloride (Vitamin B6) 是一种吡啶衍生物。在于阿尔茨海默病细胞模型中,通过 Nrf-2/HO-1 途径发挥抗氧化作用。
T6688 Synephrine hydrochloride

辛弗林盐酸盐,Oxedrine hydrochloride,Synephrine HCl

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Synephrine hydrochloride (Oxedrine hydrochloride) 是一种来自Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂的生物碱,也是一种拟交感神经化合物,能够用于减肥。
T22327 Ethanolamine hydrochloride

甲基氧氯酸,2-Aminoethanol hydrochloride,乙醇胺盐酸盐

Others Others
Ethanolamine hydrochloride (2-Aminoethanol hydrochloride) 是一种具有氨气味的粘性、吸湿性氨基醇,广泛分布于生物组织中,是卵磷脂的一种成分。
T0894 Thiamine hydrochloride

盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride

Apoptosis; HBV; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology
Thiamine hydrochloride (Vitamin B1) 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。
T3529 Bestatin hydrochloride

盐酸乌苯美司,Ubenimex hydrochloride,苯丁抑制素

Integrin; Aminopeptidase; Antibacterial; Antibiotic Cytoskeletal Signaling; Metabolism; Microbiology/Virology
Bestatin hydrochloride (Ubenimex hydrochloride) 是CD13(Aminopeptidase N)/APN 和leukotriene A4 hydrolase 抑制剂,可研究癌症。
T1511 Daunorubicin hydrochloride

Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin

Apoptosis; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Daunorubicin hydrochloride (Rubidomycin hydrochloride) 是一种蒽环类氨基糖苷类抗肿瘤药物,可抑制 DNA 复制和修复以及 RNA 和蛋白质合成。
T0415 Guanidine hydrochloride

Guanidine HCl,Aminoformamidine HCl,盐酸胍,Aminoformamidine Hydrochloride,Guanidinium chloride

Others; Arginase; DNA/RNA Synthesis; Endogenous Metabolite; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Others
Guanidine hydrochloride (Aminoformamidine Hydrochloride) 是一种强离液剂和一种蛋白质的强变性剂。
T6225 Adenine hydrochloride

Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Adenine hydrochloride (6-Aminopurine hydrochloride) 是一种嘌呤,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T5805 Guvacoline hydrochloride

1,2,5,6-四氢吡啶-3-甲酸甲酯盐酸盐,Norarecoline hydrochloride,去甲槟榔碱

AChR Neuroscience
Guvacoline hydrochloride (Norarecoline hydrochloride) 是从三药槟榔中发现的一种吡啶生物碱,可作为心房和回肠的毒蕈碱激动剂。
T0804 Pilocarpine Hydrochloride

NSC 5746 HCl,盐酸毛果芸香碱,Pilocarpine HCl,(+)-Pilocarpine hydrochloride

AChR Neuroscience
Pilocarpine Hydrochloride (NSC 5746 HCl) 是一种 M3 型毒蕈碱乙酰胆碱受体激动剂,用于制作癫痫实验模型
T4945 Normetanephrine hydrochloride

DL-Normetanephrine hydrochloride,DL-去甲变肾上腺素盐酸盐

Endogenous Metabolite Metabolism
Normetanephrine hydrochloride (DL-Normetanephrine hydrochloride) 是肾上腺素的代谢物。它与肾上腺素一起存在于尿液和某些组织中。
T6004 Tetrahydropapaverine hydrochloride

Tetrahydropapaverine HCl,Norlaudanosine HCl,Tetrahydroalkali hydrochloride,四氢罂粟碱盐酸盐

Hydroxylase Metabolism
Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) 是一种四氢异喹啉类药物。它对多巴胺神经元有神经毒性作用。
T1411 Terbinafine hydrochloride

KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Terbinafine hydrochloride (KWD 2019) 具有抗真菌感染活性。它是念珠菌属的角鲨烯环氧化酶的非竞争性抑制剂,Ki 值为 30 nM。它还对某些革兰氏阳性和革兰氏阴性细菌具有抗菌活性。
T4614 Ellipticine hydrochloride

Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐

Topoisomerase DNA Damage/DNA Repair
Ellipticine hydrochloride (NSC-71795 (hydrochloride)) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 的活性。
T4710 3-Methoxytyramine hydrochloride

3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐

Others; Endogenous Metabolite; Drug Metabolite Metabolism; Others
3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) 是多巴胺的无活性代谢物,能够活化痕量胺相关受体1 。
T2917 Tetrahydropalmatine hydrochloride

延胡索乙素盐酸盐,1-Tetrahydropalmitine HCl,Gindarine hydrochloride,盐酸延胡乙素

Others; Dopamine Receptor GPCR/G Protein; Neuroscience; Others
Tetrahydropalmatine hydrochloride (Gindarine hydrochloride) 通过抑制大鼠杏仁核的多巴胺释放来抑制癫痫发作,可用于缓解疼痛的研究。
T1235 Lincomycin hydrochloride monohydrate

洁霉素盐酸盐,林可霉素,Lincomycin hydrochloride hydrate

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Lincomycin hydrochloride monohydrate (Lincomycin hydrochloride hydrate) 是一种窄谱抗生素, 具有与红霉素相似的效力, 对革兰氏阳性球菌的作用效果很好, 主要抑制细菌细胞蛋白质的合成。
T8071 L-Lysine hydrochloride

赖氨酸盐酸盐,Lysine hydrochloride,L-赖氨酸盐酸盐

Virus Protease Microbiology/Virology
L-Lysine hydrochloride 是一种人类必需氨基酸,能增加钙吸收,减少糖尿病相关疾病和改善肠道健康,可用于疱疹的研究。
T8130 Ciprofloxacin hydrochloride monohydrate

Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan

Antibacterial; Antibiotic Microbiology/Virology
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。
T0453 Phenylephrine hydrochloride

NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Phenylephrine hydrochloride (NCI-c55641) 是选择性的α1-肾上腺素能受体激动剂,对α1A,α1B 和α1D 受体的pKis 分为4.70,4.87和5.86。
T4937 DL-5-Hydroxylysine hydrochloride

5-hydroxylysine hydrochloride,5-羟基-DL-赖氨酸盐酸盐

Others; Endogenous Metabolite Metabolism; Others
DL-5-Hydroxylysine hydrochloride (5-hydroxylysine hydrochloride) 是内源性代谢产物的一种。
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天然产物

Harmaline hydrochloride
Cat.No: T8769
Synonym: Harmidine hydrochloride
Target: Others
Viquidil hydrochloride
Cat.No: T13302
Synonym: Quinotoxine hydrochloride
Target: Others
Lycorine hydrochloride
Cat.No: T2774
Synonym: 石蒜碱,Licorine hydrochloride,Galanthidine hydrochloride,Narcissine hydrochloride,Lycorine chloride,Amarylline hydrochloride,盐酸石蒜碱
Target: Virus Protease, HCV Protease, Antibacterial, Autophagy
Cysteamine hydrochloride
Cat.No: T6460
Synonym: 2-Mercaptoethylamine Hydrochloride,β-Mercaptoethylamine Hydrochloride,半胱胺盐酸盐,Thioethanolamine Hydrochloride,2-Aminoethanethiol Hydrochloride,Cysteamine HCl,Bekaptan
Target: Apoptosis, Others, Reactive Oxygen Species, Endogenous Metabolite, Autophagy
(-)-Coclaurine hydrochloride
Cat.No: TN1519L
Synonym: (-)-Coclaurine hydrochloride (486-39-5 Free base)
Target: AChR
Harmalol hydrochloride
Cat.No: TN1724
Synonym: Harmidol hydrochloride
Target: P450, Antioxidant
Higenamine hydrochloride
Cat.No: T3232
Synonym: Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride
Target: Adrenergic Receptor
Sinomenine hydrochloride
Cat.No: T2921
Synonym: 盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride
Target: Apoptosis, NF-κB, Opioid Receptor, Autophagy
Tolazoline hydrochloride
Cat.No: T1680
Synonym: Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)
Target: Adrenergic Receptor
Raloxifene hydrochloride
Cat.No: T1549
Synonym: LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl
Target: Estrogen Receptor/ERR, Others, MAO, Estrogen/progestogen Receptor, Autophagy
Rauwolscine hydrochloride
Cat.No: T4429
Synonym: Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
Ligustrazine hydrochloride
Cat.No: T2953
Synonym: Tetramethylpyrazine hydrochloride,Tetramethylpyrazine HCl,Chuanxiongzine hydrochloride,Tetrapyrazine HCl,盐酸川芎嗪
Target: Others
Lobeline hydrochloride
Cat.No: T0268
Synonym: 盐酸洛贝林,α-Lobeline hydrochloride,L-Lobeline hydrochloride
Target: AChR
β-N-methylamino-L-alanine hydrochloride
Cat.No: T22911
Synonym: L-BMAA hydrochloride
Target: Others
D-Carnitine hydrochloride
Cat.No: T2203
Synonym: (S)-Carnitine Hydrochloride,L-Carnitine hydrochloride
Target: Others, Endogenous Metabolite
Irinotecan Hydrochloride
Cat.No: T0486L
Synonym: 盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride
Target: Topoisomerase, Autophagy
Gatifloxacin hydrochloride
Cat.No: T8384
Synonym: AM-1155 (hydrochloride),BMS-206584 (hydrochloride),PD135432 (hydrochloride),加替沙星盐酸盐
Target: Topoisomerase, Antibacterial, Antibiotic
N-Noratherosperminine hydrochloride
Cat.No: TN6787L
Synonym: N-Noratherosperminine hydrochloride (74606-53-4 free base)
Target: Others
N-Nornuciferine hydrochloride(4846-19-9 free base)
Cat.No: TQ0296L
Synonym: N-Nornuciferine hydrochloride
Target: P450
Ancitabine hydrochloride
Cat.No: T1591
Synonym: NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C
Target: Others, DNA/RNA Synthesis, Autophagy
Vasicine hydrochloride
Cat.No: T8298
Synonym: 鸭嘴花碱盐酸盐,Peganine hydrochloride
Target: Antibacterial, Antibiotic
1-Deoxynojirimycin hydrochloride
Cat.No: T21344
Synonym: Moranoline,去氧野艽霉素盐酸盐,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin
Target: PI3K, Antibacterial, Antibiotic, Glucosidase
Dobutamine hydrochloride
Cat.No: T8149
Synonym: 盐酸多巴酚丁胺,Dobutamine (hydrochloride)
Target: Adrenergic Receptor
Glucosamine hydrochloride
Cat.No: T2941
Synonym: Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride
Target: Reactive Oxygen Species, HIF/HIF Prolyl-Hydroxylase, Endogenous Metabolite, Autophagy
Chlortetracycline hydrochloride
Cat.No: T1304
Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素
Target: ribosome, Antibacterial, Antibiotic
Serotonin hydrochloride
Cat.No: T2209
Synonym: 5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride
Target: 5-HT Receptor, Endogenous Metabolite, Transferase
Imidazoleacetic acid hydrochloride
Cat.No: T4753
Synonym: I4AA,(4-Imidazolyl)acetic acid hydrochloride,4-咪唑乙酸盐酸盐,4-Imidazoleacetic acid hydrochloride
Target: Endogenous Metabolite, Antibiotic
Leonurine hydrochloride
Cat.No: T4080
Synonym: 盐酸益母草碱,SCM-198 hydrochloride,SCM-198 HCl
Target: TLR, Autophagy
Harmine hydrochloride
Cat.No: T2811
Synonym: telepathine hydrochloride,盐酸哈尔明碱
Target: 5-HT Receptor, DYRK, GluR
Pyridoxine hydrochloride
Cat.No: T0973L
Synonym: Pyridoxine HCl,吡哆醇盐酸盐,Pyridoxol (hydrochloride),吡哆醇盐酸盐(维生素B6),Vitamin B6 (hydrochloride),Vitamin B6
Target: Nrf2, Endogenous Metabolite
Synephrine hydrochloride
Cat.No: T6688
Synonym: 辛弗林盐酸盐,Oxedrine hydrochloride,Synephrine HCl
Target: Endogenous Metabolite, Adrenergic Receptor
Ethanolamine hydrochloride
Cat.No: T22327
Synonym: 甲基氧氯酸,2-Aminoethanol hydrochloride,乙醇胺盐酸盐
Target: Others
Thiamine hydrochloride
Cat.No: T0894
Synonym: 盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride
Target: Apoptosis, HBV, Endogenous Metabolite
Bestatin hydrochloride
Cat.No: T3529
Synonym: 盐酸乌苯美司,Ubenimex hydrochloride,苯丁抑制素
Target: Integrin, Aminopeptidase, Antibacterial, Antibiotic
Daunorubicin hydrochloride
Cat.No: T1511
Synonym: Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin
Target: Apoptosis, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic, Autophagy
Guanidine hydrochloride
Cat.No: T0415
Synonym: Guanidine HCl,Aminoformamidine HCl,盐酸胍,Aminoformamidine Hydrochloride,Guanidinium chloride
Target: Others, Arginase, DNA/RNA Synthesis, Endogenous Metabolite, Autophagy
Adenine hydrochloride
Cat.No: T6225
Synonym: Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride
Target: DNA/RNA Synthesis, Endogenous Metabolite
Guvacoline hydrochloride
Cat.No: T5805
Synonym: 1,2,5,6-四氢吡啶-3-甲酸甲酯盐酸盐,Norarecoline hydrochloride,去甲槟榔碱
Target: AChR
Pilocarpine Hydrochloride
Cat.No: T0804
Synonym: NSC 5746 HCl,盐酸毛果芸香碱,Pilocarpine HCl,(+)-Pilocarpine hydrochloride
Target: AChR
Normetanephrine hydrochloride
Cat.No: T4945
Synonym: DL-Normetanephrine hydrochloride,DL-去甲变肾上腺素盐酸盐
Target: Endogenous Metabolite
Tetrahydropapaverine hydrochloride
Cat.No: T6004
Synonym: Tetrahydropapaverine HCl,Norlaudanosine HCl,Tetrahydroalkali hydrochloride,四氢罂粟碱盐酸盐
Target: Hydroxylase
Terbinafine hydrochloride
Cat.No: T1411
Synonym: KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride
Target: Antibacterial, Antibiotic, Antifungal
Ellipticine hydrochloride
Cat.No: T4614
Synonym: Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐
Target: Topoisomerase
3-Methoxytyramine hydrochloride
Cat.No: T4710
Synonym: 3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐
Target: Others, Endogenous Metabolite, Drug Metabolite
Tetrahydropalmatine hydrochloride
Cat.No: T2917
Synonym: 延胡索乙素盐酸盐,1-Tetrahydropalmitine HCl,Gindarine hydrochloride,盐酸延胡乙素
Target: Others, Dopamine Receptor
Lincomycin hydrochloride monohydrate
Cat.No: T1235
Synonym: 洁霉素盐酸盐,林可霉素,Lincomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
L-Lysine hydrochloride
Cat.No: T8071
Synonym: 赖氨酸盐酸盐,Lysine hydrochloride,L-赖氨酸盐酸盐
Target: Virus Protease
Ciprofloxacin hydrochloride monohydrate
Cat.No: T8130
Synonym: Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan
Target: Antibacterial, Antibiotic
Phenylephrine hydrochloride
Cat.No: T0453
Synonym: NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride
Target: Endogenous Metabolite, Adrenergic Receptor
DL-5-Hydroxylysine hydrochloride
Cat.No: T4937
Synonym: 5-hydroxylysine hydrochloride,5-羟基-DL-赖氨酸盐酸盐
Target: Others, Endogenous Metabolite
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