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117

抑制剂 & 化合物

55

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Cat. No. Product Name Target Signaling Pathways
T21729 (±)-Lisofylline

Others Others
(±)-Lisofylline 是一种对映异构体特异性、烷基取代的甲基黄嘌呤,在下调白细胞活化方面具有特异性和有效的活性。它是一种抗炎剂。
T38361 GSK717

IL Receptor; NOD Immunology/Inflammation; NF-κB
GSK717 是 NOD2(核苷酸结合寡聚结构域 2) 的选择性抑制剂。它抑制壁酰二肽 (MDP) 诱导的 NOD2 介导的信号转导,抑制 MDP 刺激的 HEK293/hNOD2 细胞分泌 IL-8 (IC50为 400 nM)。
T8233 BRD3308

Apoptosis; HIV Protease; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
BRD3308 是一种高选择性的HDAC3抑制剂,IC50为 54 nM。它可激活HIV-1转录并破坏HIV-1潜伏期。它抑制由炎性细胞因子或糖脂毒性应激诱导的胰腺 β 细胞凋亡,并增加功能性胰岛素释放。
T6716 Valsartan

Diovan,缬沙坦,Tareg,CGP 48933

RAAS Endocrinology/Hormones
Valsartan (CGP 48933) 是一种血管紧张素 II 受体拮抗剂,有用于高血压和心力衰竭的研究潜力。
T2036 6-OAU

GTPL5846

GPR Endocrinology/Hormones; GPCR/G Protein
6-OAU (GTPL5846) 是 GPR84 的替代激动剂,在 Gqi5 嵌合体存在的情况下,在 HEK293 细胞中激活人 GPR84,在 PI 测定中 EC50 为 105 nM。
T0446 Naphazoline hydrochloride

盐酸萘甲唑啉,Albalon,Rhinantin,Naphazoline HCl

Adrenergic Receptor GPCR/G Protein; Neuroscience
Naphazoline hydrochloride (Naphazoline HCl) 是一种咪唑啉衍生物,是一种眼血管收缩剂。
T21445 Naphazoline

AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林

Adrenergic Receptor GPCR/G Protein; Neuroscience
Naphazoline (Naphcon-a) 是一种具有显着 α 肾上腺素能活性的拟交感神经化合物。 萘甲唑啉可用作血管收缩剂,当应用于粘膜时可快速减少肿胀。
T38423 CL097

CL097

Reactive Oxygen Species; TLR Immunology/Inflammation; Metabolism; NF-κB
CL097 是 TLR7 和 TLR8 的有效激动剂。 CL097 诱导巨噬细胞中的促炎细胞因子和 NADPH 氧化酶引发,从而增加 fMLF 刺激的 ROS 产生。
T4982 Benznidazol

苄哒唑,苄硝唑,Radanil,Benznidazole,Ro 71051,Ro 07-1051

Antibiotic; Parasite Microbiology/Virology
Benznidazol (Benznidazole) 是一种抗寄生虫药物,对哥伦比亚 T. cruzi 菌株的 IC50值为 20.35 μM,有潜力研究美洲锥虫病。
T27034 CL075

3M002,CL-075

NF-κB; TLR; MyD88 Immunology/Inflammation; NF-κB
CL075 (3M002) 是一种选择性TLR8 激动剂。CL075具有免疫调节活性,通过触发 MyD88 依赖性信号通路,激活 NF-κB 和 IRF7 引发炎症性细胞因子和 I 型干扰素 (IFN) 的产生。
T9543 Syk Inhibitor II hydrochloride

Others Others
Syk Inhibitor II hydrochloride 信号传导的影响在狼疮中可能很突出。
T20763 Betamethasone disodium phosphate

Vista-Methasone,NSC90616,Betamethasone 21-phosphate disodium salt,NSC-90616

Others Others
Betamethasone disodium phosphate (Betamethasone 21-phosphate disodium salt) 是一种具有抗炎活性的皮质类固醇,通过减少促炎细胞因子的分泌促进 M1 至 M2 巨噬细胞极化,可用于研究瘢痕疙瘩和类风湿性关节炎。
T6964 Resiquimod

R848,雷西莫特,S28463

HCV Protease; TLR Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Resiquimod (R848) 是一种 Toll 样受体7/8的激动剂,可诱导细胞因子上调。
T7872 Monolaurin

Others Others
Monolaurin 是椰子油中的一种表面活性剂和乳化剂。它抑制葡萄球菌、链球菌、加德纳菌、念珠菌和嗜血杆菌的生长,并减少促炎细胞因子的产生。
T6914 Oclacitinib maleate

PF-03394197 maleate,奥拉替尼马来酸盐,PF-03394197

Tyrosine Kinases; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Oclacitinib maleate (PF-03394197 maleate) 是一种新型JAK 抑制剂,有效抑制JAK1,IC50为 10 nM。
T30231 AVP-13358

Others Others
AVP-13358是一种CD23拮抗剂(免疫球蛋白ε-Fc 受体拮抗剂),一种免疫球蛋白E 抑制剂。AVP-13358对IgE、细胞因子和CD23有强效活性 ,可用于治疗免疫系统疾病、感染和耳鼻喉科疾病。
T81135 Sodium caseinates

Sodium caseinates,作为主要乳蛋白,能诱导粒细胞增殖与活化,同时提高关键细胞因子GM-CSF与G-CSF的血清浓度。该化合物还可引起小鼠粒细胞的生成。
T36310 AKT-IN-6

INCB-047775

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
AKT-IN-6 (INCB-047775)对ATK 有抑制作用。Akt 是对生长因子、细胞因子和其他细胞刺激的细胞信号传导的重要组成部分。Akt 的异常激活与2型糖尿病和癌症的发生密切相关。
T33535 MW01-2-151SRM

MW 151,MW-151,MW012151SRM,MW151,MW01 2 151SRM

Others Others
MW01-2-151SRM 是一种新型可穿过血脑屏障的小分子小胶质细胞活化抑制剂,具有抗神经炎作用,可减弱神经炎症模型中的神经胶质细胞因子上调,可用研究创伤性脑损伤、阿尔茨海默病和海藻氨酸毒性。
T0468 Lidocaine

Lignocaine,Alphacaine,Xylocaine,利多卡因

Apoptosis; ERK; NF-κB; MEK; Sodium Channel; Histamine Receptor Apoptosis; GPCR/G Protein; Immunology/Inflammation; MAPK; Membrane transporter/Ion channel; Neuroscience; NF-κB
Lidocaine (Alphacaine) 是一种酰胺衍生物,抑制涉及复杂电压和依赖性的钠通道,可用于研究室性心律失常。它通过调节 miR-145 表达和进一步抑制 MEK/ERK 和 NF-κB 信号通路来减少胃癌细胞的生长,迁移和侵袭。
T79600 Zharp2-1

RIP kinase Apoptosis; NF-κB
Zharp2-1是一种 RIPK2 抑制剂,抑制了 MDP 诱导或单核细胞增生李斯特菌感染诱导的炎症细胞因子的转录,缓解MDP诱导的小鼠腹膜炎症状,可用于研究炎症性肠病 (IBD)。
T2401 Alogliptin Benzoate

苯甲酸阿格列汀,SYR 322,Alogliptin(SYR-322)benzoate

Ferroptosis; Proteasome; DPP-4 Apoptosis; Proteases/Proteasome; Ubiquitination
Alogliptin Benzoate (SYR 322) 是一种有效且特异性的 DPP-4 抑制剂 ,IC50值小于 10 nM,其选择性比 DPP-8/9 高 10,000 倍以上,可用于研究 2 型糖尿病。
T6273 Vadimezan

DMXAA,伐地美生,5,6-Dimethylxanthenone-4-acetic Acid,NSC 640488,ASA-404

Influenza Virus; VDA; STING; IFNAR Angiogenesis; Immunology/Inflammation; Microbiology/Virology
Vadimezan (DMXAA) 是一种血管破坏剂,一种鼠 STING 激动剂,也是一种细胞因子如 I 型 IFN 的诱导剂。Vadimezan 具有抗肿瘤活性,可以诱导肿瘤中的血流快速停止,但不影响正常组织中的血流。
TP1592L C-Reactive Protein (CRP) 174-185 acetate

C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base)

Others Others
C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base) 是一种急性期血清蛋白,可响应炎性细胞因子而合成,在动物中产生抗肿瘤作用。片段 CRP (174-185) (RS-83277) 通过显着增强体外人单核细胞和肺泡巨噬细胞的杀肿瘤活性显示出相似的活性。
T67896 CB2R/FAAH modulator-1

Cannabinoid Receptor; FAAH GPCR/G Protein; Metabolism; Neuroscience
CB2R/FAAH modulator-1是一种大麻素2型受体(CB2R)激动剂,同时也是脂肪酸酰胺水解酶(FAAH)抑制剂(IC50=4 μM),可减少促炎和增加抗炎细胞因子的产生,常用于炎症研究。对 CB2R 和 CB1R 的Kis 分别为14.8 nM 和241.3 nM。
T76781 Itolizumab

EQ-001

Others Others
Itolizumab (Anti-Human CD6 Recombinant Antibody) 是一种人源化针对 CD6 的细胞外 SRCR 远端结构域 1的重组 抗 CD6 单克隆抗体。Itolizumab 可减缓 T 细胞增殖并抑制促炎细胞因子的产生。Itolizumab 可用于研究银屑病、类风湿性关节炎 (RA)和 COVID-19 疾病等多种疾病。
T38362 Guselkumab

CNTO 1959

IL Receptor Immunology/Inflammation
Guselkumab (CNTO 1959) 是一种针对IL-23p19亚基的重组人IgG1单克隆抗体。Guselkumab 与人和食蟹猴IL-23结合,Kd 值分别为3.3和1.9 pmol/L。Guselkumab 对IL-23信号通路下游细胞因子的产生具有抑制作用,可用于银屑病关节炎的研究。
T15017 CU-T12-9

TLR Immunology/Inflammation
CU-T12-9 是特异性 TLR1/2激动剂,可激活先天免疫系统和适应性免疫系统。它选择性激活 TLR1/2 异二聚体,可通过促进 TLR1 和 TLR2 二聚而激活 NF-κB 信号,引起下游 TNF-α、IL-10 和 iNOS 增加。
T67924 ABzOH

ABzOH 是一种苯甲酸衍生物,结构类似于阿司匹林等非甾体抗炎药,具有抗炎、抗肿瘤和抗增殖作用。ABzOH 不仅可以抑制肿瘤坏死因子- α (TNF-a)、白细胞介素-1β (IL-1β)和白细胞介素-6 (IL-6)等促炎细胞因子的表达还对乳腺癌、肺癌和胰腺癌具有抑制作用。
T12848 SB-657510

Others; Neurotensin Receptor GPCR/G Protein; Others
SB-657510 是 urotensin II (UII) receptor (UT) 拮抗剂。 对于人,猴,猫,大鼠和小鼠的UT 的 Ki 值分别为 61、17、30、65 和 56 nM。SB-657510 通过抑制 UII 诱导的人类血管内皮细胞中炎性介质,如粘附分子,使细胞因子和组织因子上调从而发挥抗炎作用。SB 657510对糖尿病小鼠模型中糖尿病相关动脉粥样硬化疾病具有治疗作用。
T61025 GSK-1482160

P2X Receptor Membrane transporter/Ion channel; Neuroscience
GSK-1482160是一种CNS-渗透的P2X7受体负变构调节剂,具有口服活性。P2X7受体参与中枢和外周免疫细胞产生促炎细胞因子,因此GSK-1482160具有研究炎症性疾病的潜力。GSK-1482160具有出色的体外效价(在包括人类在内的多种物种的重组和初始P2X7受体的功能和电生理测试中)和交叉靶标选择性。
T15096 Delgocitinib

JTE-052,迪高替尼,Corectim(Delgocitinib)

Tyrosine Kinases; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Delgocitinib (Corectim(Delgocitinib)) 是一种有效的、有特异性的 JAK 抑制剂,对 JAK1, JAK2, JAK3 和 Tyk2 具有抑制作用,其 IC50 值分别为 2.8,2.6,13 和 58 nM。Delgocitinib 通过JAK-依赖性细胞因子参与多种炎症和自身免疫性疾病,可广泛用于治疗各种炎症性疾病,是全球首款治疗特应性皮炎的JAK 局部外用化合物。
T2548 Diflorasone

Glucocorticoid Receptor Endocrinology/Hormones
Diflorasone 是一种皮质类固醇激素受体激动剂,具有抗炎和免疫抑制作用。它可通过细胞膜扩散进入细胞,并与细胞质中的糖皮质激素受体结合。它用于研究湿疹、牛皮癣等皮肤病。
T41142 EM 163

IL Receptor; p38 MAPK; MyD88 Immunology/Inflammation; MAPK
EM 163是一种 TIR-TIR 相互作用抑制剂,它是MyD88蛋白的TIR(Toll/白细胞介素-1受体)结构域拟态。EM 163针对IL-1受体中的TIR 结构域,阻断与MyD88的相互作用。EM 163抑制葡萄球菌肠毒素B(SEB)引起的体内炎症细胞因子的产生。EM 163能保护小鼠免受SEB 冲击引起的死亡。在体外的大鼠海马神经元中,EM 163阻断p38的激活和IL-1β对化学诱导的长期电位(LTP)引发的蛋白质合成的抑制作用。
T25453 Glaspimod

F 107647,SK&,F-107647,F107647

Glaspimod is a synthetic hematoregulatory peptide. It shares biological and/or modulatory activities with natural hematopoetic cytokines.
T31018 CP 115953

CP115953,Cp-115,953,CP-115953

CP 115953 stimulated the production of cytokines by lymphocytes. CP 115953 inhibits the activity of topoisomerase II by interacting with the enzyme.
T16570 Pralnacasan

VX-740,HMR 3480

Others Others
Pralnacasan inhibits proinflammatory cytokines IL-18, IL-1β , and IFN-γ. Pralnacasan is an effective, non-peptide, and orally active interleukin-1β converting enzyme inhibitor (Ki: 1.4 nM). Pralnacasan has the potential for osteoarthritis and rheumatoid a
T71711 ST029248

ST029248 is a potent mast cell (MC) activator, promoting de novo synthesis of cytokines and inducing the release of eicosanoids from human and mouse MCs.
T70484 AD-35

AD-35 is a neuroprotectant for treating Alzheimer’s diseases by significantly inhibiting the production and release of proinflammatory cytokines TNF-α and IL-1β.
T7503L Upadacitinib tartrate

ABT 494,ABT-494,ABT494

Upadacitinib is a potent and selective JAK inhibitor. Upadacitinib is approximately 74 fold selective for Jak1 over Jak2 in cellular assays dependent on specific, relevant cytokines. Upadacitinib demonstrates efficacy in rat arthritis models.
T71814 ST026567

ST026567 is a potent mast cell (MC) activator which promotes de novo synthesis of cytokines and induces the release of eicosanoids from human and mouse MCs.
T10366 Arg-Gly-Asp-Ser

Fibronectin tetrapeptide,RGDS peptide

Others Others
Arg-Gly-Asp-Ser is an integrin-binding sequence that inhibits integrin receptor function. It decreases systemic inflammation via inhibition of collagen-triggered activation of leukocytes and attenuates expression of inflammatory cytokines, MMP-9, and iNOS
T30831 Cgp 43182

Cgp-43182,Cgp43182

CGP 43182 is an effective inhibitor of group IIA secretory phospholipase A2 (Group IIA sPLA2) activity in vitro, which can be used to prevent the synergistic effect of pro-inflammatory genes stimulated by cytokines mediated by NFkappaB.
T70001 Pyrazinib

Pyrazinib is a novel inhibitor of angiogenesis and metabolism of oesophageal adenocarcinoma (oac) radioresistance, significantly inhibiting the secretion of il-6, il-4, il-8 and il-13 cytokines from in oac radioresistant cells
T72223 Anti-inflammatory agent 7

Anti-inflammatory agent 7 通过阻断 LPS 处理的 RAW 264.7 细胞和小鼠的 NF-κB/MAPK 信号通路抑制促炎细胞因子。
T26776 Berteroin

OR-009512,KB-47947,LP-088984,KB47947,LP088984

Berteroin is an erucin homolog and potential antioxidant. It is present in cruciferous vegetables, including rucola salad leaves, Chinese cabbage and mustard oil. It decreases the release of pro-inflammatory cytokines in LPS-stimulated macrophages. It als
T70367 SNU-BP

SNU-BP is an agonist of PPAR-gamma, inhibiting lipopolysaccharide (LPS)-induced NO production and pro-inflammatory cytokines. SNU-BP potentiates interleukin-4-induced arginase-1 expression, and promotes microglial polarization toward an M2 anti-inflammatory phenotype.
T70015 GSK563

GSK563 is a potent GVIA iPLA2 inhibitor (XI(50) 0.0000021, IC50 1 nM). GSK563 is 22 000 times more active against GVIA iPLA2 than GIVA cPLA2. It was found to reduce β-cell apoptosis induced by proinflammatory cytokines, raising the possibility that it can be beneficial in countering autoimmune diseases, such as type 1 diabetes.
TP2035 FSL-1

FSL 1

TLR2/6 agonist (also a putative TLR10 ligand). Activates NF-κB. Induces pro-inflammatory cytokines including IL-8, IL-1β, CCL20 and TNF-α in vitro. Synergizes with IFNγ to induce CXCL10 release from melanoma cells.
T60517 CL097 hydrochloride

CL097 hydrochloride 是一种有效的 TLR7和 TLR8激动剂。CL097 hydrochloride 可在巨噬细胞中诱导促炎细胞因子和 NADPH 氧化酶启动活性,从而增加 fMLF 刺激的ROS 产生。

化合物

(±)-Lisofylline
Cat.No: T21729
Synonym:
Target: Others
GSK717
Cat.No: T38361
Synonym:
Target: IL Receptor, NOD
BRD3308
Cat.No: T8233
Synonym:
Target: Apoptosis, HIV Protease, HDAC
Valsartan
Cat.No: T6716
Synonym: Diovan,缬沙坦,Tareg,CGP 48933
Target: RAAS
6-OAU
Cat.No: T2036
Synonym: GTPL5846
Target: GPR
Naphazoline hydrochloride
Cat.No: T0446
Synonym: 盐酸萘甲唑啉,Albalon,Rhinantin,Naphazoline HCl
Target: Adrenergic Receptor
Naphazoline
Cat.No: T21445
Synonym: AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林
Target: Adrenergic Receptor
CL097
Cat.No: T38423
Synonym: CL097
Target: Reactive Oxygen Species, TLR
Benznidazol
Cat.No: T4982
Synonym: 苄哒唑,苄硝唑,Radanil,Benznidazole,Ro 71051,Ro 07-1051
Target: Antibiotic, Parasite
CL075
Cat.No: T27034
Synonym: 3M002,CL-075
Target: NF-κB, TLR, MyD88
Syk Inhibitor II hydrochloride
Cat.No: T9543
Synonym:
Target: Others
Betamethasone disodium phosphate
Cat.No: T20763
Synonym: Vista-Methasone,NSC90616,Betamethasone 21-phosphate disodium salt,NSC-90616
Target: Others
Resiquimod
Cat.No: T6964
Synonym: R848,雷西莫特,S28463
Target: HCV Protease, TLR
Monolaurin
Cat.No: T7872
Synonym:
Target: Others
Oclacitinib maleate
Cat.No: T6914
Synonym: PF-03394197 maleate,奥拉替尼马来酸盐,PF-03394197
Target: Tyrosine Kinases, JAK
AVP-13358
Cat.No: T30231
Synonym:
Target: Others
Sodium caseinates
Cat.No: T81135
Synonym:
Target:
AKT-IN-6
Cat.No: T36310
Synonym: INCB-047775
Target: Akt
MW01-2-151SRM
Cat.No: T33535
Synonym: MW 151,MW-151,MW012151SRM,MW151,MW01 2 151SRM
Target: Others
Lidocaine
Cat.No: T0468
Synonym: Lignocaine,Alphacaine,Xylocaine,利多卡因
Target: Apoptosis, ERK, NF-κB, MEK, Sodium Channel, Histamine Receptor
Zharp2-1
Cat.No: T79600
Synonym:
Target: RIP kinase
Alogliptin Benzoate
Cat.No: T2401
Synonym: 苯甲酸阿格列汀,SYR 322,Alogliptin(SYR-322)benzoate
Target: Ferroptosis, Proteasome, DPP-4
Vadimezan
Cat.No: T6273
Synonym: DMXAA,伐地美生,5,6-Dimethylxanthenone-4-acetic Acid,NSC 640488,ASA-404
Target: Influenza Virus, VDA, STING, IFNAR
C-Reactive Protein (CRP) 174-185 acetate
Cat.No: TP1592L
Synonym: C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base)
Target: Others
CB2R/FAAH modulator-1
Cat.No: T67896
Synonym:
Target: Cannabinoid Receptor, FAAH
Itolizumab
Cat.No: T76781
Synonym: EQ-001
Target: Others
Guselkumab
Cat.No: T38362
Synonym: CNTO 1959
Target: IL Receptor
CU-T12-9
Cat.No: T15017
Synonym:
Target: TLR
ABzOH
Cat.No: T67924
Synonym:
Target:
SB-657510
Cat.No: T12848
Synonym:
Target: Others, Neurotensin Receptor
GSK-1482160
Cat.No: T61025
Synonym:
Target: P2X Receptor
Delgocitinib
Cat.No: T15096
Synonym: JTE-052,迪高替尼,Corectim(Delgocitinib)
Target: Tyrosine Kinases, JAK
Diflorasone
Cat.No: T2548
Synonym:
Target: Glucocorticoid Receptor
EM 163
Cat.No: T41142
Synonym:
Target: IL Receptor, p38 MAPK, MyD88
Glaspimod
Cat.No: T25453
Synonym: F 107647,SK&,F-107647,F107647
Target:
CP 115953
Cat.No: T31018
Synonym: CP115953,Cp-115,953,CP-115953
Target:
Pralnacasan
Cat.No: T16570
Synonym: VX-740,HMR 3480
Target: Others
ST029248
Cat.No: T71711
Synonym:
Target:
AD-35
Cat.No: T70484
Synonym:
Target:
Upadacitinib tartrate
Cat.No: T7503L
Synonym: ABT 494,ABT-494,ABT494
Target:
ST026567
Cat.No: T71814
Synonym:
Target:
Arg-Gly-Asp-Ser
Cat.No: T10366
Synonym: Fibronectin tetrapeptide,RGDS peptide
Target: Others
Cgp 43182
Cat.No: T30831
Synonym: Cgp-43182,Cgp43182
Target:
Pyrazinib
Cat.No: T70001
Synonym:
Target:
Anti-inflammatory agent 7
Cat.No: T72223
Synonym:
Target:
Berteroin
Cat.No: T26776
Synonym: OR-009512,KB-47947,LP-088984,KB47947,LP088984
Target:
SNU-BP
Cat.No: T70367
Synonym:
Target:
GSK563
Cat.No: T70015
Synonym:
Target:
FSL-1
Cat.No: TP2035
Synonym: FSL 1
Target:
CL097 hydrochloride
Cat.No: T60517
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T3S2312 Poncirin

枸橘苷,Isosakuranetin-7-neohesperidoside

Apoptosis; Others Apoptosis; Others
Poncirin (Isosakuranetin-7-neohesperidoside) 是从三叶草中分离出来的一种天然产物,具有抗炎活性。 它防止脂肪生成,增强间充质干细胞中的成骨细胞分化,增加骨矿物质密度,改善小梁微结构,可能反映 GIO 小鼠的骨形成增加和骨吸收减少。
TN1721 Gypenoside L

ERK; p38 MAPK; Calcium Channel; NF-κB; ROS Immunology/Inflammation; MAPK; Membrane transporter/Ion channel; Metabolism; NF-κB
Gypenoside L 是存在于绞股蓝中的一种皂苷,可增加 SA-β-半乳糖苷酶活性,促进衰老相关分泌细胞因子的产生。它还可以激活p38和ERK MAPK 通路和NF-κB 通路以诱导衰老,具有抗肿瘤和抗炎活性。
T9862 Pseudocoptisine chloride

盐酸异黄连碱,Isocoptisine chloride

AChE Neuroscience
Pseudocoptisine chloride (Isocoptisine chloride) 是从 Corydalis Tuber 中分离出来的,具有抗炎和抗健忘的作用。 Pseudocoptisine chloride 抑制乙酰胆碱酯酶 (AChE) 活性 (IC50 = 12.8 μM)。
TN6722 Terminolic acid

2α,6β,23-trihydroxyl oleanolic acid

Antibacterial Microbiology/Virology
Terminolic acid (2α,6β,23-trihydroxyl oleanolic acid) 是一种从 Combretum racemosum 中分离得到的五环三萜糖苷,可通过与 IL-1β 和 IL-6 的受体活性位点结合抑制促炎细胞因子,并通过与 IL-4 受体结合位点结合增强抗炎细胞因子。它还表现出适度的抗菌活性。
TN6796 2'-FUCOSYLLACTOSE

2'-Fucosyl-D-lactose,2'-岩藻糖基乳糖

Others Others
2'-FUCOSYLLACTOSE (2'-Fucosyl-D-lactose) 是一种含岩藻糖的寡糖。
TN1291 7,3',4'-Tri-O-methylluteolin

5-Hydroxy-3',4',7-trimethoxyflavone,木犀草素-7,3',4'-三甲醚

TNF; COX; Interleukin Apoptosis; Immunology/Inflammation; Neuroscience
7,3',4'-Tri-O-methylluteolin (5-Hydroxy-3',4',7-trimethoxyflavone) 是来自草药马鞭草科的一种类黄酮,具有抗炎,解热,镇咳,抗糖尿病、抗癌和抗黑素生成特性。它以浓度依赖方式明显抑制促炎细胞因子,可显著降低在转录水平的诱导型一氧化氮合酶和环加氧酶-2 的 mRNA 表达。
T34295 Resiniferatoxin

RTX,[3H]resiniferatoxin,树脂毒素

IL Receptor Immunology/Inflammation
Resiniferatoxin ([3H]resiniferatoxin) 抑制 Th1 细胞因子的产生,有助于防御 T.spiralis 感染,并可用于免疫反应调节剂的研究。
T14149 AICAR phosphate

AICA Riboside phosphate,Acadesine phosphate

Mitophagy; NOS; YAP; AMPK Autophagy; Chromatin/Epigenetic; Immunology/Inflammation; PI3K/Akt/mTOR signaling; Stem Cells
AICAR phosphate (Acadesine phosphate) 是 AMPK 激活剂且是自噬、YAP 和 mitophagy 抑制剂,也是一种腺苷类似物, 可调节糖代谢和脂代谢,抑制促炎细胞因子和 iNOS 的产生。
T10689 Cauloside D

Others Others
Cauloside D 是一种分离自 Caulophyllum robustumMax 中的三萜苷类化合物。它能够阻碍 iNOS 和促炎细胞因子的表达,具有抗炎活性。
T6S0107 Peimine

贝母素甲,Wanpeinine A,Dihydroisoimperialine,Verticine,贝母甲素

Others Others
Peimine (Wanpeinine A) 是一种天然化合物,具有很好抗炎症活性。
T5660 Menthone

IL Receptor; TNF; NF-κB; Parasite Apoptosis; Immunology/Inflammation; Microbiology/Virology; NF-κB
Menthone 是一种从植物和薄荷油中提取的单萜,是精油的主要挥发性成分,具有抗炎和抗氧化特性。
T3829 Ginsenoside F3

人参皂苷F3

Others; IFNAR; Interleukin Immunology/Inflammation; Others
Ginsenoside F3 是一种皂苷,提取自Panax ginseng 叶片。它能够调节1 型 (IL-2, IFN-γ) 及 2 型细胞因子(IL-4 and IL-10) 的产生和表达,有免疫增强的作用。
T3826 Polygalasaponin F

异牡荆苷,瓜子金皂苷己

NF-κB; TLR; Akt; PI3K Cytoskeletal Signaling; Immunology/Inflammation; NF-κB; PI3K/Akt/mTOR signaling
Polygalasaponin F 是从瓜子金中提取的齐墩果烷型三萜皂苷,可通过调节TLR4-PI3K/AKT-NF-kB 信号通路减少神经炎症细胞因子的分泌,能降低炎性细胞因子肿瘤坏死因子 α 的释放。
T5S0167 Atractylenolide I

白术内酯 I,白术内酯I;苍术内酯I

IL Receptor; TNF; TLR; JAK; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Stem Cells
Atractylenolide I 是从白术根中得到的一种倍半萜烯,具有神经保护、抗过敏、抗炎和抗癌等多种生物活性。它是一种TLR4拮抗剂,在 A375 细胞中,能够降低JAK2和STAT3的磷酸化水平。
TN2091 Polygalacin D

Apoptosis; IAP Apoptosis
Polygalacin D 是从桔梗中分离的一种天然产物,具有抗癌和抗增殖特性。它通过 PI3K/Akt 途径诱导凋亡。它抑制 IAP 蛋白家族的表达,并通过抑制 GSK3β,Akt 的磷酸化和 PI3K 的表达来阻断 PI3K/Akt 途径。
T5S1895 Norisoboldine

Laurelliptine,去甲异波尔定,(+)-Laurelliptine

MAPK; Adenosine Receptor GPCR/G Protein; MAPK; Neuroscience
Norisoboldine ((+)-Laurelliptine) 是一种可口服的芳基烃受体激动剂,是乌药中主要的异喹啉类生物碱,可用于类风湿性关节炎和溃疡性结肠炎的研究。
TN1410 Asperulosidic acid

ASPA,车叶草苷酸

ERK; NF-κB MAPK; NF-κB
Asperulosidic acid (ASPA) 是从白花蛇舌草药中提取的一种环烯醚萜苷,具有抗肿瘤、抗氧化和抗炎作用。它通过抑制 NF-κB 和丝裂原活化蛋白激酶信号通路抑制炎性细胞因子释放发挥抗炎作用。
T3426 Bacoside A

MMP; Others; TNF; Dopamine Receptor; NOS; ROS Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience; Others; Proteases/Proteasome
Bacoside A has a possible anticancer activity that could be inducing cell cycle arrest and apoptosis through Notch pathway in GBM in vitro. It exerts cytoprotective efficacy by attenuation of ROS generated through oxidative stress by an increase in the concentration of antioxidant enzymes and sustain membrane integrity which leads to restoring the damage caused by tBHP. Bacoside A can able to inhibit the progression of Experimental Autoimmune Encephalomyelitis (EAE) may be by the inhibition of i...
T2S2362 Dehydrocorydaline nitrate

去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱

BCL; Others; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Others; Proteases/Proteasome
Dehydrocorydaline nitrate 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达,激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌、抗疟疾等功效。
T2S2173 (E)-Naringenin chalcone

Isosalipurpol,柚皮苷查尔酮,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone,柚皮素查耳酮

Others Others
Naringenin chalcone (Isosalipurpol) 是一种黄酮醇生物合成的中间体,在查耳酮异构酶的作用下,自发代谢成柚皮素。它具有抗炎和抗过敏活性。
T5S0045 Isofraxidin

6,8-Dimethoxyumbelliferone,异秦皮啶,Phytodolor,异嗪皮啶

MMP; ERK; p38 MAPK; TLR; COX Immunology/Inflammation; MAPK; Neuroscience; Proteases/Proteasome
Isofraxidin (Phytodolor) 是来自刺五加的香豆素成分,抑制MMP-7表达和人肝癌细胞侵袭。它作用于肝癌细胞,抑制ERK1/2磷酸化。它减弱iNOS 和COX-2表达,还抑制TLR4/髓样分化蛋白 2 复合物的形成。
T6S0139 Neobavaisoflavone

Apoptosis; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Neobavaisoflavone 是一种从Psoralea corylifolia 的种子中分离出来的类黄酮。它具有抗炎,抗癌和抗氧化的作用。它在中至高浓度下可抑制 DNA 聚合酶,也可抑制血小板聚集。
TN1448 (-)-Bornyl acetate

L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯

p38 MAPK; NF-κB; JNK; Antifungal MAPK; Microbiology/Virology; NF-κB
(-)-Bornyl acetate (L-(-)-Bornyl acetate) 是存在于牛膝草油中的一种具有抗真菌活性的 (+)-Bornyl acetate 低活性异构体。
T3877 Esculentoside A

NF-κB; COX Immunology/Inflammation; Neuroscience; NF-κB
Esculentoside A 是一种三萜皂苷,从商陆根部分离得到。它在具有抗炎活性,对环氧合酶-2 具有选择性抑制活性。它通过抑制NF-κB 和丝裂原活化蛋白激酶信号通路抑制 LPS 诱导的急性肺损伤中的炎症反应。
T3779 Crocin II

Crocin 2,西红花苷II,Crocetin gentiobiosylglucosyl ester,藏红花,Tricrocin,Crocin B

Caspase; COX; NO Synthase Apoptosis; Immunology/Inflammation; Neuroscience; Proteases/Proteasome
Crocin II (Crocetin gentiobiosylglucosyl ester) 是从栀子果实中分离出来的一种天然产物,具有抗氧化、抗癌和抗抑郁活性。它抑制 iNOS 和 COX-2的蛋白质和 m-RNA 的表达,还抑制NO 产生,IC50值为 31.1 μM。
T9113 Myristicin

Myristicine,肉豆蔻醚

IL Receptor; Anti-infection; BCL; P450; PARP; 5-HT Receptor; Caspase; GABA Receptor; NO Synthase Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Myristicin (Myristicine) 是一种在香料和伞形植物中发现的天然产物。肉豆蔻素具有抗胆碱能、抗菌和肝保护作用,还具有抗炎作用,其通过钙途径抑制dsrna 刺激的巨噬细胞中的NO、细胞因子、趋化因子和生长因子。Myristicin 可以诱导细胞凋亡,其特征是改变线粒体膜电位、细胞色素c 释放、Caspase-3激活、parp 切割和DNA 断裂。
T4S0878 Prunetin

樱黄素,Prunusetin

ERK; Dehydrogenase; NF-κB MAPK; Metabolism; NF-κB
Prunetin (Prunusetin) 是一种O-甲基化异黄酮,具有抗炎的作用。它是人醛脱氢酶的有效抑制剂。
TN1831 Macranthoside A

Kalopanaxsaponin H

Antioxidant oxidation-reduction
Macranthoside A (Kalopanaxsaponin H) 是一种从地黄中提取的三萜糖苷,属于环烯醚萜类化合。Macranthoside A 具有抗炎、抗氧化、抗菌和神经保护活性,抑制促炎细胞因子的产生和抑制炎症信号通路的激活,有助于中和有害的自由基,保护细胞免受氧化损伤,可以促进神经元的存活和生长,并防止氧化应激或神经毒性化合物引起的神经元细胞死亡,具有治疗神经退行性疾病、心血管疾病和肝损伤的潜力。
T2S2264 Linalool

Linalol,(±)-Linalool,Phantol,沉香醇

Apoptosis; IL Receptor; TNF; Endogenous Metabolite; iGluR Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Linalool (Linalol) 是存在芫荽等植物中的单萜类天然产物,是竞争性NMDA 受体拮抗剂,具有抗肿瘤和抗心脏毒性的作用。它通过激活 Nrf2 诱导抗氧化防御和通过抑制 NF-κB 减少炎症反应来保护其免受 LPS/GalN 诱导的肝损伤,具有镇痛、抗菌和抗炎的特性。
T2563 Acetyl-L-carnitine hydrochloride

Acetyl L-carnitine hydrochloride,O-Acetylcarnitine,乙酰-L-肉(毒)碱盐酸盐,O-acetyl-L-carnitine,O-Acetyl-L-carnitine hydrochloride

Others; Endogenous Metabolite Metabolism; Others
Acetyl-L-carnitine hydrochloride (Acetyl L-carnitine hydrochloride) 是一种由内源性左旋肉碱的乙酰化形式的盐酸盐组成的营养补充剂,具有潜在的神经保护、认知增强、抗抑郁和免疫调节活性。还可缓解化疗、糖尿病或其他疾病引起的周围神经病变。此外,乙酰左旋肉碱可能通过增加T淋巴细胞成熟来调节免疫反应,并可能下调促炎细胞因子对病毒(如SARS-CoV-2)的反应。它还可能破坏ACE2信号通路并抑制活性氧(ROS)的产生。
T4S0797 Berberine

小檗碱,Berberin,Umbellatine,黄连素

Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic; Autophagy Autophagy; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Berberine (Umbellatine) 是从中草药黄连中分离出来的一种生物碱抗生素。它诱导活性氧生成并抑制 DNA 拓扑异构酶,具有抗肿瘤特性。
T3S2259 Methyl eugenol

4-allylveratrole,eugenyl methyl ether,O-methyleugenol,Eugenol Methyl ether,丁香酚甲醚,丁子香酚甲醚

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Methyl eugenol (4-allylveratrole) 是一种苯丙类化合物,存在于植物叶子、果实、根茎中,当植物相应的部位因食草动物进食而受损时,就会释放。它可用于消灭雄性东方果蝇。
T6677 Sophocarpine

ERK; p38 MAPK; NF-κB; TLR; COX; HER; JNK; STAT Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; MAPK; Neuroscience; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Sophocarpine 是一种从传统草药苦参中提取的重要生物碱。苦参具有抗病毒、抗肿瘤和抗炎等多种药理作用。它通过多种机制显著抑制癌细胞的生长,具有抗肿瘤活性。
TN1485 Chicanine

Others; NF-κB; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; NF-κB; Others
Chicanine has anti-inflammatory activity in macrophages by down-regulating LPS-induced inflammatory cytokines in IκBα±/MAPK/ERK signaling pathways.
TN6566 Licoflavanone

Licoflavanone exhibits antioxidant and anti-inflammatory activities,it markedly decreases pro-inflammatory cytokines and cyclooxygenase 2/inducible nitric oxide synthase (COX-2/iNOS) expression levels.
TMA2576 Episappanol

IL Receptor; TNF Apoptosis; Immunology/Inflammation
Episappanol has anti-inflammatory activity , it can significantly inhibit the secretion of the pro-inflammatory cytokines interleukin (IL-6) and tumor necrosis factor-alpha (TNF-α).
T14877 Cauloside C

Others Others
Cauloside C, a triterpene glycoside isolated from Caulophyllum robustum Max, exerts anti-inflammatory effects through the inhibition of expression of iNOS and proinflammatory cytokines.
TN1504 Citreorosein

羟基大黄素

cAMP; NF-κB; PI3K GPCR/G Protein; NF-κB; PI3K/Akt/mTOR signaling
Citreorosein is a cAMP phosphodiesterase inhibitor, it has anti-inflammatory effect, inhibits proinflammatory cytokines production through the inhibition of both MAPKs and AKT-mediated IκB kinase (IKK) phosphorylation and subsequent inhibition of transcription factor NF-κB activation.
TN6366 Lupinalbin A

鲁冰花

Lupinalbin A as the most potent estrogen receptor α- and aryl hydrocarbon receptor agonist in Eriosema laurentii de Wild. (Leguminosae). It exerts anti-inflammatory effects via the inhibition of pro-inflammatory cytokines and blocking of IFN-β/STAT1 pathw
TN4879 Questinol

IL Receptor; TNF; COX; Prostaglandin Receptor Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Questinol exhibits significant anti-obesity activity. It shows anti-inflammatory effect in lipopolysaccharide (LPS)-stimulated RAW 264.7 cells, it can inhibit the production of pro-inflammatory cytokines, including TNF-α, IL-1β, and IL-6 and inhibit NO an
T38838 QS-21

Stimulon,QS-21

QS-21, an immunostimulatory saponin, is a powerful vaccine adjuvant that stimulates both Th2 humoral and Th1 cell-mediated immune responses by interacting with antigen presenting cells (APCs) and T cells. Additionally, QS-21 activates the NLRP3 inflammasome, leading to the release of cytokines IL-1β and IL-18, which are dependent on caspase-1.
TN4013 Esculentic acid

IL Receptor; TNF; COX Apoptosis; Immunology/Inflammation; Neuroscience
Esculentic acid has anti-inflammatory effect, it has protective effects against LPS-induced endotoxic shock may be mediated, at least in part, by regulation the release of inflammatory cytokines and mediators, and protein expression of COX-2 in mice.
T5S0313 Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside

Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷

Others; TNF Apoptosis; Others
Liquiritin apioside has antioxidant property by inducing glutathione (GSH) biosynthesis via the inhibition of cytokines and protected lung epithelial cells against cigarette smoke-mediated oxidative stress, might be as protective agent against epithelial
TN5149 Tirotundin

NF-κB; COX; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Tirotundin is a PPARα/γ dual agonist, it exerts anti-diabetic effect through PPARγ pathway. It shows anti-inflammatory activity, it inhibits inhibit the activation of NF-kappa B, thereby, the synthesis of inflammatory mediators such as cytokines and chemo
T81408 Preleoheterin

Preleoheterin(化合物3)为一类从L. japonicus分离得到的拉丹烷二萜。
T38394 PSMα3

PSMα3 is a peptide compound that can be utilized to induce tolerance in dendritic cells (DCs) for DC vaccination strategies. It effectively penetrates and modulates human monocyte-derived DCs by modifying the maturation process induced by TLR2 or TLR4. Additionally, PSMα3 inhibits the production of both pro- and anti-inflammatory cytokines and decreases antigen uptake. Notably, PSMα3 is a significant virulence factor released by the most pathogenic strains of methicillin-resistant Staphylococcus...
TN5474 Bonducellin

Bonducellin has anti-inflammatory activities, it can significantly and dose-dependently inhibit the inflammatory mediators; nitric oxide (NO), and cytokines [tumor necrosis factor (TNF)-alpha and interleukin (IL)-12. Bonducellin shows weak antimalarial ac
T26545 Acanthoic acid

NP1302,NP 1302: NP-1302

Acanthoic acid is a pimaradiene diterpene isolated from Acanthopanax koreanum with anti-inflammatory activities. Acanthoic acid downregulates LPS-induced IL-1β, IL-6 and TNF-α production in BALF, attenuates lung histopathologic changes, and inhibits infla
TN3983 Ergosta-7,22-dien-3-one

NO Synthase; LTR Immunology/Inflammation
Ergosta-7,22-dien-3-one 是一种羊毛甾烷,能够从台湾灵芝的子实体中分离得到。Ergosta-7,22-dien-3-one 具有促炎特性,它能刺激一氧化氮的产生,诱导基因的表达,并诱导 J774A.1 细胞产生 TLRs、细胞因子、趋化因子和细胞粘附分子。
TN2243 Sugiol

10-Deoxoxanthoperol

IL Receptor; TNF; ROS Apoptosis; Immunology/Inflammation
Sugiol (10-Deoxoxanthoperol) 是一种枞烷二萜,可从台湾板栗树 (Calocedrus formosana) 的树皮中分离出来。Sugiol 具有抗炎活性,可有效减少脂多糖 (LPS) 刺激巨噬细胞后的活性氧 (ROS) 产生。
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天然产物

Poncirin
Cat.No: T3S2312
Synonym: 枸橘苷,Isosakuranetin-7-neohesperidoside
Target: Apoptosis, Others
Gypenoside L
Cat.No: TN1721
Synonym:
Target: ERK, p38 MAPK, Calcium Channel, NF-κB, ROS
Pseudocoptisine chloride
Cat.No: T9862
Synonym: 盐酸异黄连碱,Isocoptisine chloride
Target: AChE
Terminolic acid
Cat.No: TN6722
Synonym: 2α,6β,23-trihydroxyl oleanolic acid
Target: Antibacterial
2'-FUCOSYLLACTOSE
Cat.No: TN6796
Synonym: 2'-Fucosyl-D-lactose,2'-岩藻糖基乳糖
Target: Others
7,3',4'-Tri-O-methylluteolin
Cat.No: TN1291
Synonym: 5-Hydroxy-3',4',7-trimethoxyflavone,木犀草素-7,3',4'-三甲醚
Target: TNF, COX, Interleukin
Resiniferatoxin
Cat.No: T34295
Synonym: RTX,[3H]resiniferatoxin,树脂毒素
Target: IL Receptor
AICAR phosphate
Cat.No: T14149
Synonym: AICA Riboside phosphate,Acadesine phosphate
Target: Mitophagy, NOS, YAP, AMPK
Cauloside D
Cat.No: T10689
Synonym:
Target: Others
Peimine
Cat.No: T6S0107
Synonym: 贝母素甲,Wanpeinine A,Dihydroisoimperialine,Verticine,贝母甲素
Target: Others
Menthone
Cat.No: T5660
Synonym:
Target: IL Receptor, TNF, NF-κB, Parasite
Ginsenoside F3
Cat.No: T3829
Synonym: 人参皂苷F3
Target: Others, IFNAR, Interleukin
Polygalasaponin F
Cat.No: T3826
Synonym: 异牡荆苷,瓜子金皂苷己
Target: NF-κB, TLR, Akt, PI3K
Atractylenolide I
Cat.No: T5S0167
Synonym: 白术内酯 I,白术内酯I;苍术内酯I
Target: IL Receptor, TNF, TLR, JAK, STAT
Polygalacin D
Cat.No: TN2091
Synonym:
Target: Apoptosis, IAP
Norisoboldine
Cat.No: T5S1895
Synonym: Laurelliptine,去甲异波尔定,(+)-Laurelliptine
Target: MAPK, Adenosine Receptor
Asperulosidic acid
Cat.No: TN1410
Synonym: ASPA,车叶草苷酸
Target: ERK, NF-κB
Bacoside A
Cat.No: T3426
Synonym:
Target: MMP, Others, TNF, Dopamine Receptor, NOS, ROS
Dehydrocorydaline nitrate
Cat.No: T2S2362
Synonym: 去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱
Target: BCL, Others, PARP, p38 MAPK, Caspase, Parasite, Autophagy
(E)-Naringenin chalcone
Cat.No: T2S2173
Synonym: Isosalipurpol,柚皮苷查尔酮,Chalconaringenin,trans-2'4'6'4-tetrahydroxychalcone,柚皮素查耳酮
Target: Others
Isofraxidin
Cat.No: T5S0045
Synonym: 6,8-Dimethoxyumbelliferone,异秦皮啶,Phytodolor,异嗪皮啶
Target: MMP, ERK, p38 MAPK, TLR, COX
Neobavaisoflavone
Cat.No: T6S0139
Synonym:
Target: Apoptosis, DNA/RNA Synthesis
(-)-Bornyl acetate
Cat.No: TN1448
Synonym: L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯
Target: p38 MAPK, NF-κB, JNK, Antifungal
Esculentoside A
Cat.No: T3877
Synonym:
Target: NF-κB, COX
Crocin II
Cat.No: T3779
Synonym: Crocin 2,西红花苷II,Crocetin gentiobiosylglucosyl ester,藏红花,Tricrocin,Crocin B
Target: Caspase, COX, NO Synthase
Myristicin
Cat.No: T9113
Synonym: Myristicine,肉豆蔻醚
Target: IL Receptor, Anti-infection, BCL, P450, PARP, 5-HT Receptor, Caspase, GABA Receptor, NO Synthase
Prunetin
Cat.No: T4S0878
Synonym: 樱黄素,Prunusetin
Target: ERK, Dehydrogenase, NF-κB
Macranthoside A
Cat.No: TN1831
Synonym: Kalopanaxsaponin H
Target: Antioxidant
Linalool
Cat.No: T2S2264
Synonym: Linalol,(±)-Linalool,Phantol,沉香醇
Target: Apoptosis, IL Receptor, TNF, Endogenous Metabolite, iGluR
Acetyl-L-carnitine hydrochloride
Cat.No: T2563
Synonym: Acetyl L-carnitine hydrochloride,O-Acetylcarnitine,乙酰-L-肉(毒)碱盐酸盐,O-acetyl-L-carnitine,O-Acetyl-L-carnitine hydrochloride
Target: Others, Endogenous Metabolite
Berberine
Cat.No: T4S0797
Synonym: 小檗碱,Berberin,Umbellatine,黄连素
Target: Reactive Oxygen Species, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic, Autophagy
Methyl eugenol
Cat.No: T3S2259
Synonym: 4-allylveratrole,eugenyl methyl ether,O-methyleugenol,Eugenol Methyl ether,丁香酚甲醚,丁子香酚甲醚
Target: GABA Receptor
Sophocarpine
Cat.No: T6677
Synonym:
Target: ERK, p38 MAPK, NF-κB, TLR, COX, HER, JNK, STAT
Chicanine
Cat.No: TN1485
Synonym:
Target: Others, NF-κB, Prostaglandin Receptor
Licoflavanone
Cat.No: TN6566
Synonym:
Target:
Episappanol
Cat.No: TMA2576
Synonym:
Target: IL Receptor, TNF
Cauloside C
Cat.No: T14877
Synonym:
Target: Others
Citreorosein
Cat.No: TN1504
Synonym: 羟基大黄素
Target: cAMP, NF-κB, PI3K
Lupinalbin A
Cat.No: TN6366
Synonym: 鲁冰花
Target:
Questinol
Cat.No: TN4879
Synonym:
Target: IL Receptor, TNF, COX, Prostaglandin Receptor
QS-21
Cat.No: T38838
Synonym: Stimulon,QS-21
Target:
Esculentic acid
Cat.No: TN4013
Synonym:
Target: IL Receptor, TNF, COX
Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside
Cat.No: T5S0313
Synonym: Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷
Target: Others, TNF
Tirotundin
Cat.No: TN5149
Synonym:
Target: NF-κB, COX, PPAR
Preleoheterin
Cat.No: T81408
Synonym:
Target:
PSMα3
Cat.No: T38394
Synonym:
Target:
Bonducellin
Cat.No: TN5474
Synonym:
Target:
Acanthoic acid
Cat.No: T26545
Synonym: NP1302,NP 1302: NP-1302
Target:
Ergosta-7,22-dien-3-one
Cat.No: TN3983
Synonym:
Target: NO Synthase, LTR
Sugiol
Cat.No: TN2243
Synonym: 10-Deoxoxanthoperol
Target: IL Receptor, TNF, ROS
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