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245

抑制剂 & 化合物

49

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6792 BQ-123

BQ123

Endothelin Receptor GPCR/G Protein
BQ-123 是高效的内皮素 A(ETA)受体选择性拮抗剂,其IC50=7.3 nM,Ki=25 nM。它能够降低高血压大鼠血压,抑制内皮素-1 介导的人肺动脉平滑肌细胞增殖。
T11831 LDN-27219

Others Others
LDN-27219 是一种人组织型转谷氨酰胺酶抑制剂(IC50:600 nM)。
T8405 Vardenafil hydrochloride

伐地那非,盐酸伐地那非

PDE Metabolism
Vardenafil hydrochloride 是口服具有活性的、高效的、选择性的磷酸二酯酶 5抑制剂。它对 PDE1 (180 nM),PDE6 (11 nM),PDE2,PDE3,PDE4 (>1000 nM) 具有选择性。它能够非竞争性地抑制环磷酸鸟苷水解,提高 cGMP 水平。它可用于勃起功能障碍的研究。
T0145 Felodipine

非洛地平,CGH-869

Calcium Channel; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Felodipine (CGH-869) 是一种长效的 1, 4-二氢吡啶钙通道抑制剂,可跨越血脑屏障,可诱导自噬,具有抗高血压活性。它通过选择性作用于血管平滑肌,尤其是阻力血管来降低血压。
T22459 Xanthinol Nicotinate

Angioamin,烟酸占替诺,Complamin

Others Others
Xanthinol Nicotinate (Complamin) 是血管扩张剂,可直接作用于小动脉和毛细血管的平滑肌,能够扩大血管,改善血液流变学并降低外周血管阻力。
T5458 Darusentan

Lu-135252,达卢生坦

Endothelin Receptor GPCR/G Protein
Darusentan (Lu-135252) 是内皮素受体 A (ET-A) 受体选择性拮抗剂,能够作用于 ET-A 受体(Ki:1.4 nM)及ET-B 受体(Ki:184 nM),对 ETA 受体的选择性大于 ETB 受体的100以上。它在大鼠主动脉血管平滑肌细胞膜中竞争结合放射性标记的内皮素(Ki:13 nM)。
T7764 CCG-222740

ROCK; Rho; Ras Cell Cycle/Checkpoint; Cytoskeletal Signaling; GPCR/G Protein; MAPK; Stem Cells
CCG-222740 是一种口服有效的选择性Rho/MRTF 途径抑制剂。它也是 α-平滑肌的肌动蛋白表达抑制剂,可减少皮肤纤维化并阻止黑色素瘤转移。
T7133 Anagliptin

SK-0403,阿拉格列汀

Proteasome; DPP-4 Proteases/Proteasome; Ubiquitination
Anagliptin (SK-0403) 是一种选择性的二肽酰肽酶 4 抑制剂,IC50=3.8 nM,对 DPP-8/9 的选择性相对较弱,IC50分别为 68 和 60 nM。
T8976 PD-089828

EGFR; FGFR; PDGFR; Src Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
PD-089828 是受体酪氨酸激酶 FGFR1、PDGFRβ 和 EGFR 的竞争性抑制剂,IC50分别为0.15、1.76 和 5.47 µM。它也是非受体酪氨酸激酶 c-Src 的非竞争性抑制剂,IC50 为 0.18 µM。
T3461 Losartan Carboxylic Acid

EXP-3174,E-3174

RAAS Endocrinology/Hormones
Losartan Carboxylic Acid (E-3174) 是 Losartan 的活性羧酸代谢产物,是血管紧张素Ⅱ受体 1 型(AT1)拮抗剂。它能够阻断血管紧张素 II 诱导的血管平滑肌细胞反应,可以提高血浆肾素活性,降低平均动脉压。
T0096 Vardenafil

伐地那非,Vivanza,Levitra,Vardenafil hydrochloride

PDE Metabolism
Vardenafil (Vivanza) 是选择性、高效的、具有口服活性的磷酸二酯酶5抑制剂,IC50=0.7 nM。它能够非竞争性地抑制环磷酸鸟苷水解,从而提高 cGMP 水平。它对 PDE1 (180 nM),PDE6 (11 nM),PDE2,PDE3,PDE4 (>1000 nM) 具有选择性。它可用于研究勃起功能障碍。
T1083L Theophylline monohydrate

Quibron,茶碱一水合物

HDAC; PDE; Adenosine Receptor Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience
Theophylline monohydrate (Quibron) 似乎抑制磷酸二酯酶和前列腺素的产生,调节钙通量和细胞内钙分布,并拮抗腺苷。茶碱是黄嘌呤的天然生物碱衍生物,从植物山茶花和小粒咖啡中分离出来。在生理上,该药剂可放松支气管平滑肌,产生血管舒张(脑血管除外),刺激中枢神经系统,刺激心肌,利尿,增加胃酸分泌;它还可以抑制炎症并改善横膈膜的收缩性。
T1487 Fluvastatin sodium

XU 62320 sodium,XU-62-320,氟伐他汀钠,Fluvastatin sodium salt

Ferroptosis; HMG-CoA Reductase; Autophagy Apoptosis; Autophagy; Metabolism
Fluvastatin sodium (Fluvastatin sodium salt) salt 是羟甲基戊二酰辅酶 A 还原酶的竞争性抑制剂,IC50为 8 nM。它通过依赖 Nrf2 的抗氧化通路保护血管平滑肌细胞免受氧化应激,是一种常用的降胆固醇剂。
T4097 Vardenafil hydrochloride trihydrate

Vardenafil HCl Trihydrate,BAY38-9456,盐酸瓦地那非三水合物

PDE Metabolism
Vardenafil hydrochloride trihydrate (BAY38-9456) 是一种新型 PDE 抑制剂,对 PDE5 和 PDE1 的 IC50 分别为 0.7 和 180 nM。
T4480 Vardenafil dihydrochloride

Levitra,Vardenafil Hydrochloride,二盐酸伐地那非

PDE Metabolism
Vardenafil dihydrochloride (Levitra) 是一种新型 PDE 抑制剂,对 PDE5 和 PDE1 的 IC50 分别为 0.7 和 180 nM。
T3996 Dapiprazole Hydrochloride

盐酸达哌唑,Glamidolo Hydrochloride,Reversil Hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Dapiprazole Hydrochloride (Glamidolo Hydrochloride) 是 α-adrenergic 阻断剂的药物。
T0504 Cyclandelate

安脉生,BS 572,环扁桃酯,3,5,5-Trimethylcyclohexyl mandelate

Acyltransferase Metabolism
Cyclandelate (BS 572) 是直接作用的平滑肌松弛剂,用于扩张血管。
T14021 20-HETE

20-hydroxy Arachidonic Acid

Others Others
20-HETE (20-hydroxy Arachidonic Acid) is a CYP450 metabolite and a potent vasoconstrictor and it is an endogenous inhibitor of the large-conductance Ca2+-activated K+ channel in renal arterioles. 20-HETE increases NADPH oxidase, ROS, and NF-κB activity, a
T67911 (Iso)-Dehydroemetine

Dehydroisoemetine, (+/-)-,Dehydroisoemetine

Others Others
(Iso)-Dehydroemetine (Dehydroisoemetine, (+/-)-) 是具有平滑肌解痉作用的化合物。
T25719 Lidamidine

Lidamidina,Lidamidinum,利达脒

Others Others
Lidamidine (Lidamidinum) 是一种临床有效的止泻化合物,可抑制肠道分泌,减少肠道转运,并抑制平滑肌收缩。
T34280 Regrelor disodium

INS-50589,INS50589,Regrelor sodium,Regrelor,INS 50589

P2Y Receptor GPCR/G Protein; Neuroscience
Regrelor disodium (INS 50589) 是一种 p2y12 受体拮抗剂,可预防血栓形成,可有效抑制血管平滑肌细胞收缩,抑制细胞增殖,减少炎症。
T7575L1 [Sar1, Ile8]-Angiotensin II acetate

RAAS Endocrinology/Hormones
[Sar1, Ile8]-Angiotensin II acetate 可激活 NADPH 和 NADH 氧化酶,并刺激血管平滑肌细胞中超氧阴离子的形成。 [Sar1, Ile8]-Angiotensin II acetate 对血管平滑肌有多种作用,包括正常动脉的收缩和培养细胞或病变血管的肥大或增生。
T0324 Isoxsuprine hydrochloride

Duvadilan,Isolait,盐酸异克舒令,盐酸苯氧丙酚胺

Adrenergic Receptor; iGluR GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Isoxsuprine hydrochloride (Isolait) 是 β 肾上腺素受体激动剂和NMDA 受体拮抗剂,对子宫肌层和胎盘的 β 肾上腺素受体的Ki 值分别为 13.65 和 3.48 μM。
T1613 Hydralazine hydrochloride

Hydralazine HCl,Apresoline,盐酸肼屈嗪

MAO; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism; Neuroscience
Hydralazine hydrochloride (Apresoline) 是一种直接作用的血管舒张剂,可抗高血压。
T21478 Cromakalim

BRL-34915,BRL 34915,(±)-Cromakalim,BRL34915

Cromakalim, a potassium channel-opening vasodilator, acts on ATP-sensitive potassium channels and so causes membrane hyperpolarization, it can be used to treat hypertension as it will relax vascular smooth muscle to lower blood pressure. The active isomer
T1115 Doxylamine succinate

琥珀酸多西拉敏,Decapryn

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Doxylamine succinate (Decapryn) 是一种吡啶衍生物组胺 H1 拮抗剂,具有明显的镇静特性。它竞争性阻断组胺 H1 受体并限制典型的过敏和过敏反应,可防止组胺引起的皮肤和粘膜疼痛和瘙痒。
T0343 Nimodipine

尼莫地平,BAY-e 9736

Glucocorticoid Receptor; AhR; Calcium Channel; Autophagy Autophagy; Endocrinology/Hormones; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Nimodipine (BAY-e 9736) 是一种具有口服活性,耐受性良好的光敏二氢吡啶钙拮抗剂。它可研究脑血管疾病。
TNU0266 9-(β-D-Xylofuranosyl)adenine

Xylosyladenine,Adenine xyloside

Nucleoside Antimetabolite/Analog Cell Cycle/Checkpoint; DNA Damage/DNA Repair
9-(β-D-Xylofuranosyl)adenine (Adenine xyloside) 是一种腺嘌呤核苷类似物,是一种潜在的平滑肌血管扩张剂。9-(β-D-Xylofuranosyl)adenine 具有抗癌活性。
T13684 Equilin

7-Dehydroestrone

Calcium Channel Membrane transporter/Ion channel; Metabolism
Equilin (7-Dehydroestrone) 是神经营养性雌激素类固醇,具有血管扩张活性,通过 NF-κB 信号传导增加单核细胞-内皮粘附。Equilin 通过阻断Ca(2+)进入平滑肌来同样放松肠系膜动脉的阻力。
T67951 JB061

Myosin Cytoskeletal Signaling
JB061是一种非肌肉肌球蛋白II抑制剂,针对心肌肌球蛋白、骨骼肌肌球蛋白和平滑肌肌球蛋白II的IC50分别为4.4 μM、9.1 μM和>100 μM。其对ATP酶活性的抑制作用较弱(IC50>200 μM)。此外,JB061对COS-7细胞显示出细胞毒性,IC50值为39 μM。
T11986L Mebeverine acid hydrochloride

Mebeverine acid hydrochloride 是一种有效的、可口服的、可直接作用于胃肠道平滑肌解除痉挛症状的化合物。
T2441 TAS-301

TAS 301

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
TAS-301 是一种平滑肌迁移和增殖抑制剂,能够抑制 PDGF 诱导的 PKC 的活化,可抑制大鼠颈动脉球囊损伤后的内膜增厚。
TP2075L Bombinakinin M acetate

Bombinakinin M acetate(509151-65-9 free base)

Bradykinin Receptor GPCR/G Protein
Bombinakinin M acetate 是一种有效的缓激肽受体激动剂,对哺乳动物动脉平滑肌缓激肽受体具有高度选择性,其效力比缓激肽高约 50 倍。
T28972 Tiaramide hydrochloride

FK-1160,NTA-194,FK 1160,FK1160,tiaramide

Others Others
Tiaramide hydrochloride (FK-1160) 是一种抗炎药,可抑制肥大细胞释放的介质的作用,并具有直接的平滑肌松弛特性。
T7575L [Sar1, Ile8]-Angiotensin II 3TFA

[Sar1, Ile8]-Angiotensin II 3TFA(37827-06-8(free base))

Others Others
[Sar1, Ile8]-Angiotensin II 3TFA ([Sar1, Ile8]-Angiotensin II 3TFA (37827-06-8(free base))) 是一种对血管平滑肌具有多种作用的肽。
T12255 NS19504

Potassium Channel Membrane transporter/Ion channel
NS19504 是 Ca2+激活的 K+通道激活剂 (EC50=11.0 µM),对膀胱平滑肌自发性相位收缩具有松弛作用。
T71746 Pincainide

Others Others
Pincainide 是一种新型β-氨基苯胺,以剂量依赖的方式抑制去甲肾上腺素血管平滑肌功能异常引起的疾病。
T34541 SB-209670

SB 209670

Endothelin Receptor GPCR/G Protein
SB-209670是一种选择性内皮素受体拮抗剂,能够抑制大鼠血管内皮和血管平滑肌中ET(B)受体的活性。
T6968 Riociguat

利奥西呱,BAY 632521

Guanylate cyclase GPCR/G Protein
Riociguat (BAY 632521) 是一种鸟苷酸环化酶的刺激剂,可导致血管平滑肌松弛,用于治疗严重的肺动脉高压。
T25984 Prenalterol

H80/62,H-80/62,H 80/62

Prenalterol 是一种选择性的β1- 肾上腺素能受体激动剂,不影响肠道平滑肌的收缩活动。Prenalterol 具有心血管疾病的研究潜力。
T3194 Ro 46-2005

Endothelin Receptor GPCR/G Protein
Ro 46-2005是新型非肽类内皮素拮抗剂,能够抑制人血管平滑肌细胞(ETA 受体)(IC50:220 nM)。
T1006 Propantheline bromide

Neopepulsan,溴丙胺太林,Pro-Banthine,Neometantyl

AChR Neuroscience
Propantheline bromide (Pro-Banthine) 是一种抗毒蕈碱剂,用于研究多汗症,遗尿,胃肠和膀胱痉挛。
T15049 Daltroban

BM-13505,SKF 96148

PPAR DNA Damage/DNA Repair; Metabolism
Daltroban (SKF 96148) (BM-13505) 是选择性和特异性的血栓素 A2 (TXA2) 受体拮抗剂。Daltroban 可以增加血管平滑肌细胞内钙。Daltroban 显示对再灌注损伤的保护作用。
T0999 Clevidipine

Clevidipine butyrate,丁酸氯维地平,氯维地平,Cleviprex

Calcium Channel; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience
Clevidipine (Clevidipine butyrate) butyrate 是一种二氢吡啶 L 型钙通道阻滞剂,IC50为7.1 nM。它对血管平滑肌有选择性,可用于降低血压。
T5195 Alrestatin

阿瑞司他丁,AY-22284

Reductase Endocrinology/Hormones; Metabolism
Alrestatin (AY-22284) 是醛糖还原酶的特异性抑制剂,能够在体外减弱大鼠血管平滑肌中葡萄糖诱导的血管紧张素 II 的产生。
T67952 JB062

Myosin Cytoskeletal Signaling
JB062是一种针对非肌肉肌球蛋白(nonmusclemyosin)的抑制剂,其IC50值对骨骼肌肌球蛋白为1.6μM、心肌肌球蛋白为5.4μM,而对平滑肌肌球蛋白II大于100μM。此化合物对人类癌细胞显示出细胞毒性,对正常细胞则无此作用。JB062在肌肉痉挛、慢性肌肉骨骼疼痛及肥厚型心肌病研究中有潜在应用价值。
T16564 PPADS tetrasodium

P2X Receptor; Na+/Ca2+ Exchanger Membrane transporter/Ion channel; Neuroscience
PPADS tetrasodiuma 是一种有效的 P2X 受体拮抗剂,也是是豚鼠气道平滑肌 Na/Ca²⁺ 交换逆模式的抑制剂,对谷氨酸/NMDA毒性有神经保护作用。PPADS tetrasodiuma 抑制 P2X1、P2X-2、P2X-3 和 P2X-5。
T27554 HS38

HS 38,HS-38

DAPK Apoptosis
HS38 是一种特异性的 ATP 竞争性 DAPK 抑制剂,对 DAPK1、PIM3 和 ZIPK 的 Kds 分别为 300 nM、200 nM 和 280 nM。 HS38 可用于平滑肌相关疾病的研究。
T21405 Fluvastatin

Canef,XU-62320,Vastin,Cranoc,Lescol

HMG-CoA Reductase Metabolism
Fluvastatin (XU-62320) 是一种具有高效性和竞争性的 HMG-CoA 还原酶抑制剂(IC50 :8 nM),可通过依赖 Nrf2 通路抑制血管平滑肌细胞免受氧化应激,用于降低血浆胆固醇水平和预防心血管疾病。
T1439 Lacidipine

SN-305,拉西地平,GX-1048,GR-43659X

Apoptosis; Calcium Channel; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB
Lacidipine (SN-305) 是一种L 型钙离子通道阻断剂。

化合物

BQ-123
Cat.No: T6792
Synonym: BQ123
Target: Endothelin Receptor
LDN-27219
Cat.No: T11831
Synonym:
Target: Others
Vardenafil hydrochloride
Cat.No: T8405
Synonym: 伐地那非,盐酸伐地那非
Target: PDE
Felodipine
Cat.No: T0145
Synonym: 非洛地平,CGH-869
Target: Calcium Channel, Autophagy
Xanthinol Nicotinate
Cat.No: T22459
Synonym: Angioamin,烟酸占替诺,Complamin
Target: Others
Darusentan
Cat.No: T5458
Synonym: Lu-135252,达卢生坦
Target: Endothelin Receptor
CCG-222740
Cat.No: T7764
Synonym:
Target: ROCK, Rho, Ras
Anagliptin
Cat.No: T7133
Synonym: SK-0403,阿拉格列汀
Target: Proteasome, DPP-4
PD-089828
Cat.No: T8976
Synonym:
Target: EGFR, FGFR, PDGFR, Src
Losartan Carboxylic Acid
Cat.No: T3461
Synonym: EXP-3174,E-3174
Target: RAAS
Vardenafil
Cat.No: T0096
Synonym: 伐地那非,Vivanza,Levitra,Vardenafil hydrochloride
Target: PDE
Theophylline monohydrate
Cat.No: T1083L
Synonym: Quibron,茶碱一水合物
Target: HDAC, PDE, Adenosine Receptor
Fluvastatin sodium
Cat.No: T1487
Synonym: XU 62320 sodium,XU-62-320,氟伐他汀钠,Fluvastatin sodium salt
Target: Ferroptosis, HMG-CoA Reductase, Autophagy
Vardenafil hydrochloride trihydrate
Cat.No: T4097
Synonym: Vardenafil HCl Trihydrate,BAY38-9456,盐酸瓦地那非三水合物
Target: PDE
Vardenafil dihydrochloride
Cat.No: T4480
Synonym: Levitra,Vardenafil Hydrochloride,二盐酸伐地那非
Target: PDE
Dapiprazole Hydrochloride
Cat.No: T3996
Synonym: 盐酸达哌唑,Glamidolo Hydrochloride,Reversil Hydrochloride
Target: Adrenergic Receptor
Cyclandelate
Cat.No: T0504
Synonym: 安脉生,BS 572,环扁桃酯,3,5,5-Trimethylcyclohexyl mandelate
Target: Acyltransferase
20-HETE
Cat.No: T14021
Synonym: 20-hydroxy Arachidonic Acid
Target: Others
(Iso)-Dehydroemetine
Cat.No: T67911
Synonym: Dehydroisoemetine, (+/-)-,Dehydroisoemetine
Target: Others
Lidamidine
Cat.No: T25719
Synonym: Lidamidina,Lidamidinum,利达脒
Target: Others
Regrelor disodium
Cat.No: T34280
Synonym: INS-50589,INS50589,Regrelor sodium,Regrelor,INS 50589
Target: P2Y Receptor
[Sar1, Ile8]-Angiotensin II acetate
Cat.No: T7575L1
Synonym:
Target: RAAS
Isoxsuprine hydrochloride
Cat.No: T0324
Synonym: Duvadilan,Isolait,盐酸异克舒令,盐酸苯氧丙酚胺
Target: Adrenergic Receptor, iGluR
Hydralazine hydrochloride
Cat.No: T1613
Synonym: Hydralazine HCl,Apresoline,盐酸肼屈嗪
Target: MAO, HIF/HIF Prolyl-Hydroxylase
Cromakalim
Cat.No: T21478
Synonym: BRL-34915,BRL 34915,(±)-Cromakalim,BRL34915
Target:
Doxylamine succinate
Cat.No: T1115
Synonym: 琥珀酸多西拉敏,Decapryn
Target: Histamine Receptor
Nimodipine
Cat.No: T0343
Synonym: 尼莫地平,BAY-e 9736
Target: Glucocorticoid Receptor, AhR, Calcium Channel, Autophagy
9-(β-D-Xylofuranosyl)adenine
Cat.No: TNU0266
Synonym: Xylosyladenine,Adenine xyloside
Target: Nucleoside Antimetabolite/Analog
Equilin
Cat.No: T13684
Synonym: 7-Dehydroestrone
Target: Calcium Channel
JB061
Cat.No: T67951
Synonym:
Target: Myosin
Mebeverine acid hydrochloride
Cat.No: T11986L
Synonym:
Target:
TAS-301
Cat.No: T2441
Synonym: TAS 301
Target: PKC
Bombinakinin M acetate
Cat.No: TP2075L
Synonym: Bombinakinin M acetate(509151-65-9 free base)
Target: Bradykinin Receptor
Tiaramide hydrochloride
Cat.No: T28972
Synonym: FK-1160,NTA-194,FK 1160,FK1160,tiaramide
Target: Others
[Sar1, Ile8]-Angiotensin II 3TFA
Cat.No: T7575L
Synonym: [Sar1, Ile8]-Angiotensin II 3TFA(37827-06-8(free base))
Target: Others
NS19504
Cat.No: T12255
Synonym:
Target: Potassium Channel
Pincainide
Cat.No: T71746
Synonym:
Target: Others
SB-209670
Cat.No: T34541
Synonym: SB 209670
Target: Endothelin Receptor
Riociguat
Cat.No: T6968
Synonym: 利奥西呱,BAY 632521
Target: Guanylate cyclase
Prenalterol
Cat.No: T25984
Synonym: H80/62,H-80/62,H 80/62
Target:
Ro 46-2005
Cat.No: T3194
Synonym:
Target: Endothelin Receptor
Propantheline bromide
Cat.No: T1006
Synonym: Neopepulsan,溴丙胺太林,Pro-Banthine,Neometantyl
Target: AChR
Daltroban
Cat.No: T15049
Synonym: BM-13505,SKF 96148
Target: PPAR
Clevidipine
Cat.No: T0999
Synonym: Clevidipine butyrate,丁酸氯维地平,氯维地平,Cleviprex
Target: Calcium Channel, AChR
Alrestatin
Cat.No: T5195
Synonym: 阿瑞司他丁,AY-22284
Target: Reductase
JB062
Cat.No: T67952
Synonym:
Target: Myosin
PPADS tetrasodium
Cat.No: T16564
Synonym:
Target: P2X Receptor, Na+/Ca2+ Exchanger
HS38
Cat.No: T27554
Synonym: HS 38,HS-38
Target: DAPK
Fluvastatin
Cat.No: T21405
Synonym: Canef,XU-62320,Vastin,Cranoc,Lescol
Target: HMG-CoA Reductase
Lacidipine
Cat.No: T1439
Synonym: SN-305,拉西地平,GX-1048,GR-43659X
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species
Cat. No. Product Name Target Signaling Pathways
T8198 Visnagin

Others Others
Visnagin 是一种抗氧化剂呋喃香豆素衍生物。它具有预防Cerulein 诱导的急性胰腺炎的潜力。它在血管平滑肌中具有良好的血管扩张作用。它具有抗炎作用,可用于缓解疼痛的研究。
T1431 Khellin

凯林,Amicardine,Methafrone,Visammin

EGFR; Others Angiogenesis; JAK/STAT signaling; Others; Tyrosine Kinase/Adaptors
Khellin (Methafrone) 是从阿米芹中提取得到的一种呋喃并色酮,是EGFR 抑制剂,IC50为 0.15 µM。它体外具有抗增殖活性,还具有抗痉挛和冠状动脉舒张作用。
T3S0364 L-Arginine

L-精氨酸,L-Arg,(S)-(+)-Arginine

IL Receptor; Endogenous Metabolite; NO Synthase Immunology/Inflammation; Metabolism
L-Arginine (L-Arg) 是内皮型一氧化氮合酶(eNOS) 的底物。L-Arginine 通过阳离子氨基酸转运体家族转运到血管平滑肌细胞,并被代谢成一氧化氮、多胺或 L-脯氨酸。
T1083 Theophylline

Theo-24,1,3-Dimethylxanthine,茶碱

Endogenous Metabolite; HDAC; PDE; Adenosine Receptor; Autophagy Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; Neuroscience
Theophylline (1,3-Dimethylxanthine) 是茶中的甲基黄嘌呤衍生物,具有利尿、平滑肌松弛、支气管扩张、心脏和中枢神经系统兴奋作用。
T8288 14-Deoxyandrographolide

去氧穿心莲内酯,14-去氧穿心莲内酯

Apoptosis; Others Apoptosis; Others
14-Deoxyandrographolide 是穿心莲中的一种天然产物,是一种钙通道阻断剂,具有保肝功效。它通过诱导 TNFRSF1A 的释放,使肝细胞对 TNF-α 介导的凋亡脱敏。
T8178 Acetagastrodin

乙酰天麻素,Acegastrodine

Others Others
Acetagastrodin (Acegastrodine) 是一种抗氧化剂,也是合成 DBPG 的中间体。
T2520 Desloratadine

Sch34117,地氯雷他定,NSC 675447

Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Desloratadine (Sch34117) 是非镇静H1抗组胺药 Loratadine 的主要口服代谢物,可减少对支气管平滑肌、毛细血管和胃肠道平滑肌中 H1 受体的典型组胺能作用,包括血管舒张、支气管收缩、血管通透性增加、疼痛、瘙痒和胃肠道平滑肌的痉挛性收缩。它是一种选择性H1受体拮抗剂,具有抗过敏和抗炎活性。
TN1683 Gentisin

龙胆根素,龍膽根素

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Gentisin 是一种提取于 Gentianae radix (Gentianaceae) 的天然化合物,具有诱变活性。
TN1248 3-Epioleanolic acid

AChR Neuroscience
3-Epioleanolic acid 是一种分离自马鞭草的有效成分,具有抗炎作用。
TN3243 7-O-Methyleriodictyol

AChR Neuroscience
7-O-Methyleriodictyol 是一种从单乳蒿中分离出的黄烷酮,对大鼠分离的平滑肌有生物学作用。
T3805 Prim-O-glucosylcimifugin

升麻苷,Cimifugin beta-D-glucopyranoside,Cimifugin 7-glucoside

TNF; COX; JAK; NO Synthase Angiogenesis; Apoptosis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; Stem Cells
Prim-O-glucosylcimifugin (Cimifugin 7-glucoside) 具有强效的抗炎作用。通过调节 JAK2/STAT3 信号传导可抑制iNOS 和COX-2表达。
T0892 Diphylline

二羟丙茶碱,Dyphylline,Diprophylline

PDE; Adenosine Receptor GPCR/G Protein; Metabolism; Neuroscience
Diphylline (Diprophylline) 是一种A1/A2腺苷受体拮抗剂,也是环状核苷酸磷酸二酯酶抑制剂。它是一种黄嘌呤衍生物,具有支气管扩张和血管扩张作用,有用于治疗慢性支气管炎和肺气肿的潜力。
T6S2025 8-​O-​Acetylharpagide

8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide

Antibacterial Microbiology/Virology
8-O-Acetylharpagide 是从 Ajuga reptans 中分离得到的一种环烯醚萜,有抗肿瘤、抗病毒、抗菌和抗炎作用。它对豚鼠的离体平滑肌有生物活性。
T6S1418 Praeruptorin C

Antioxidant; Calcium Channel Membrane transporter/Ion channel; Metabolism; oxidation-reduction
Praeruptorin C 是白花前胡中的一种主要成分,是钙拮抗剂,pD2′值为 5.7。
T5014 Prostaglandin E2

地诺前列酮,前列腺素 E2,PGE2,Dinoprostone,Prostaglandin E2 (PGE2)

Endogenous Metabolite; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
Prostaglandin E2 (PGE2) 是一种天然激素,参与人体内的各种生理过程,包括平滑肌收缩和放松、调节血管扩张和收缩、调节血压和炎症调节。
T20604L Litorin acetate(55749-97-8 Free base)

Bombesin Receptor GPCR/G Protein
Litorin acetate 是一种两栖类铃蟾肽衍生物,是一种铃蟾肽受体激动剂。它刺激平滑肌收缩,刺激胃泌素、胃酸和胰腺分泌,抑制体内营养。
T0965 Histamine

Ergamine,组胺

5-HT Receptor; Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine (Ergamine) 是通过组胺的酶促脱羧衍生的胺。它是一种强大的胃分泌兴奋剂、支气管平滑肌的收缩剂、血管扩张剂以及中枢作用的神经递质。
T6534 Histamine dihydrochloride

组胺二盐酸盐,peremin,Ceplene,Histamine 2HCl

Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine dihydrochloride (Ceplene) 是 Histamine 的二盐酸形式。Histamine 是一种有机氮化合物,是一种强效的胃分泌兴奋剂,支气管平滑肌收缩剂,血管舒张剂,也是一种中枢作用的神经递质。
T6102 2'-acetylacteoside

Antioxidant; Reductase Endocrinology/Hormones; Metabolism; oxidation-reduction
2'-Acetylacteoside 是一种苯乙醇苷类化合物,分离自来江藤中,可抑制自由基诱导的红细胞溶血,具有清除自由基的作用。
T4S1102 Liensinine diperchlorate

莲心碱高氯酸盐,莲心碱二高氯酸盐,Liensinine-Perchlorate

Mitophagy; Others; Autophagy Autophagy; Others
Liensinine Diperchlorate 是从芙蕖种子胚中提取的一种异喹啉生物碱。它通过阻断自噬小体-溶酶体融合来抑制晚期自噬,具有抗心律不齐、抗高血压、抗肺纤维化和血管平滑肌松弛等生物学活性。
T3427 Polydatin

Piceid,虎杖苷,Polydotin Peceid

Apoptosis; Mitophagy; NF-κB; Autophagy Apoptosis; Autophagy; NF-κB
Polydatin (Piceid) 是从传统中药虎杖根中提取的一种天然产物,在多个实验模型中具有抗炎作用。它可抑制 G6PD,并诱导氧化和内质网应激。
T4S0998 Trifolirhizin

红车轴草根甙/三叶豆紫檀苷,三叶豆紫檀苷

TNF; Tyrosinase Apoptosis; Proteases/Proteasome
Trifolirhizin 是一种从苦参根中分离出的 pterocarpan 黄酮类化合物。它具有酪氨酸酶高抑制活性,IC50=506 μM。它具有抗炎和抗癌的潜能。
T1626 Prostaglandin E1

前列地尔,PGE1,列腺素E1,Alprostadil

Endogenous Metabolite; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
Prostaglandin E1 (Alprostadil) 是一种前列腺素受体配体,对小鼠 EP1、EP2、EP3、EP4和 IP 的 Ki 值分别为 36、10、1.1、2.1 和 33 nM。它诱导血管舒张并抑制血小板聚集,可作为血管扩张剂用于外周血管疾病的研究。
T37709 2,2,2-Trichloroethanol

Potassium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
2,2,2-Trichloroethanol 是非经典的 K2P 通道 TREK-1和 TRAAK 的激动剂。
T4S1619 L-Hyoscyamine sulfate

Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate,硫酸天仙子胺水合物,L-莨菪碱硫酸盐

AChR Neuroscience
L-Hyoscyamine sulfate (Levsin Sulfate) 是来自山莨菪的一种托烷生物碱,是竞争性的毒蕈碱受体拮抗剂。它是 Atropine 的左旋异构体。
T0962 L-Hyoscyamine

Daturine,Hyoscyamine,L-莨菪碱,L-天仙子胺

AChR Neuroscience
L-Hyoscyamine (Daturine) 是从山莨菪中提取的一种托烷生物碱,是竞争性的毒蕈碱受体拮抗剂。它是 Atropine 的左旋异构体。
T5065 GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD

Monosodium-GMP,cGMP sodium salt,鸟苷-3',5'-环磷酸一钠盐,Cyclic GMP

PKA Tyrosine Kinase/Adaptors
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD (cGMP sodium salt) 也称为 cGMP,是一种细胞调节剂,被描述为第二信使。它的水平随着各种激素的增加而增加,包括乙酰胆碱、胰岛素和催产素。 cGMP 激活蛋白激酶 G(PKG) 并调节离子通道电导,信号传导影响多种过程,包括平滑肌松弛和增殖、光转导和能量稳态。
T6429 Caffeic Acid Phenethyl Ester

Phenylethyl Caffeate,咖啡酸苯乙酯,CAPE

Apoptosis; NF-κB Apoptosis; NF-κB
Caffeic Acid Phenethyl Ester (Phenylethyl Caffeate) 是咖啡酸的苯乙醇酯,是蜂巢蜂胶的生物活性成分。它抑制核转录因子 NF-kappa B 的激活,具有抗肿瘤、细胞保护和免疫调节活性。它抑制 PDGF 诱导的血管平滑肌细胞增殖。
T3229 Cytochalasin D

ATPase; p38 MAPK; Calcium Channel; Akt; PI3K Cytoskeletal Signaling; MAPK; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling
Cytochalasin D is an actin inhibitor, the removal of actin stress fibers is crucial for the chondrogenic differentiation. It may be an inhibitor of some fertilization processes such as sperm penetration or sperm head decondensation. Cytochalasin D inhibit
T3123 Allicin

ERK; IL Receptor; Others; IκB/IKK; p38 MAPK; TNF; ROS; Caspase; Antifection Apoptosis; Immunology/Inflammation; MAPK; Microbiology/Virology; NF-κB; Others; Proteases/Proteasome
Allicin 具有抗氧化、杀菌、抗癌、抗炎活性,对肠上皮细胞具有抑制性免疫调节作用。 Allicin 能显着抑制胰岛素诱导的血管平滑肌细胞的增殖和迁移,这可能与抑制 ERK 信号通路的激活有关。 Allicin 有利于降低高胆固醇血症大鼠的血液胆固醇、甘油三酯水平和收缩压,它可能有益于影响动脉粥样硬化的两个危险因素——高脂血症和高血压。
T5S0106 Peimisine

贝母辛,Ebeiensine

RAAS; AChR Endocrinology/Hormones; Neuroscience
Peimisine (Ebeiensine) 非竞争性拮抗气管平滑肌 M 受体,抑制 Ach 引起的平滑肌收缩。它兴奋 β 受体和拮抗内钙释放,促进一氧化氮释放,可舒张气管平滑肌,有平喘作用。
T3794 Pentagalloylglucose

Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose,1,2,3,4,6-五没食子酰葡萄糖

Influenza Virus Microbiology/Virology
1,2,3,4,6-O-Pentagalloylglucose (Penta-O-galloyl-β-D-glucose) 存在于多种植物中,具有重要的药理作用。Pentagalloylglucose 表现出显著的抗狂犬病病毒 (RABV) 活性。
T20604 Litorin

Litorin, an amphibian bombesin peptide derivative, is found to suppress the nutriment, to stimulate the contraction of smooth muscle, to stimulate gastrin, gastric acid, and pancreatic secretion.
TN1338 7Beta-Hydroxycholesterol

LDL; Calcium Channel; MAPK MAPK; Membrane transporter/Ion channel; Metabolism
7beta-Hydroxycholesterol, a major cytotoxin in oxidized LDL, induces Ca(2+) oscillations, MAP kinase activation and apoptosis in human aortic smooth muscle cells.
TN4051 Fargesone B

cAMP; Calcium Channel GPCR/G Protein; Membrane transporter/Ion channel; Metabolism
Fargesone B inhibits the vascular smooth muscle contraction by suppressing the voltage- and receptor-activated calcium influxes in a nonselective manner.
TN5341 Pterosin Z

Pterosin Z has smooth muscle relaxant activity, is approximately equipotent with that of the related fungal pterosin (EC50 of 2.9 +/- 1.6 x 10(-6) M).
TN5608 Paspalinine

Paspalinine can inhibit binding of [125I]charybdotoxin (ChTX) to maxi-K channels in bovine aortic smooth muscle sarcolemmal membranes. Paspalinine shows tremorgenic action, which may be due in part to their inhibition of GABAA receptor function.
TN5234 Vindorosine

Calcium Channel; Sodium Channel Membrane transporter/Ion channel; Metabolism
Vindorosine has blood vessel relaxation effect, possible underlying mechanisms involving the inhibition of Ca(2+) entry via L-type Ca(2+) channels in vascular smooth muscles.
TN2075 Pimaric acid

MMP; p38 MAPK; NF-κB MAPK; NF-κB; Proteases/Proteasome
Pimaric acid has potent anti-atherosclerotic activity with inhibitory action on matrix metalloproteinase-9 production and cell migration in TNF-α±-induced human aortic smooth muscle cells.
TN1985 Neoprzewaquinone A

ROCK; Pim; STAT Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Stem Cells
Neoprzewaquinone A (NEO) 是 S. miltiorrhiza 的活性成分,通过靶向 PIM1 阻断 ROCK2/STAT3 通路来抑制乳腺癌细胞迁移并促进平滑肌松弛。
TN3319 9-Hydroxycanthin-6-one

Potassium Channel; GSK-3; Calcium Channel; Wnt/beta-catenin Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling; Stem Cells
9-Hydroxycanthin-6-one might be the active component that contributed to the aphrodisiac effect of E. longifolia by antagonizing the smooth muscle tone of CC as well as SV probably through interfering with Ca2+ mobilization.9-Hydroxycanthin-6-one inhibits Wnt signaling through the activation of GSK3β independent of CK1α.
T83454 13-Hydroxylupanine hydrochloride

Hydroxylupanine hydrochloride

13-Hydroxylupanine是甜羽扇豆中一种典型的生物碱。它具有阻断神经节传递、降低心肌收缩力以及收缩子宫平滑肌的作用。
TN1875 Liriodenine

鹅掌揪碱

BCL; Caspase; p53 Apoptosis; Proteases/Proteasome
Liriodenine is a potent inhibitor of topoisomerase II (EC 5.99.1.3) both in vivo and in vitro, it has antitumor, antibacterial and antifungal activities, it can suppress ventricular arrhythmias induced by myocardial ischaemia reperfusion, through inhibiti
TN5330 Lacinilene C

3,10-Dihydroxy-1,3,5,7-cadinatetraen-9-one

Lacinilene C, lacinilene C 7-methyl ether, scopoletin, 2-hydroxy-7-methoxycadalene and 2,7-dihydroxycadalene are 5 induced phytoalexins in cotton leaves. Lacinilene C methyl ether elicits contraction of TSM by enhancing the movement of calcium through pot
T25687 Leukotriene C4

白三烯C4,LTC4,Leukotriene C

Leukotriene C4 is the conjugation product of Leukotriene A4 and glutathione. It is the major arachidonic acid metabolite in human mast cells, macrophages, and antigen-sensitized lung tissue. It stimulates mucus secretion in the lung and produces contracti
T74193 (R)-IDHP

(R)-IDHP为IDHP异构体,属于丹参代谢物。该化合物能通过抑制血管平滑肌细胞电压依赖性钙通道与受体操作钙通道的Ca2+释放和Ca2+内流,发挥血管松弛作用,适用于心脑血管疾病研究。
TN5186 Triptoquinone A

IL Receptor; NOS Immunology/Inflammation
Triptoquinone A may be a useful candidate for the development of a drug as a potent inhibitor of iNOS gene over-expression. Triptoquinone A has anti-inflammatory activity, it prevents ndotoxin-or interleukin-1 beta-promoted induction of nitric oxide synth
TN1690 Glabrene

Others; Estrogen/progestogen Receptor; Tyrosinase Endocrinology/Hormones; Others; Proteases/Proteasome
Glabrene, Liquiritin apioside, neolicuroside, and 18α²-glycyrrhetic acid are the predominant phenolic derivatives partitioning at the interface and most likely the major contributors to the notable synergistic antioxidant activity when coupled with pea pr
T72152 Eicosapentaenoic Acid sodium

二十碳五烯酸钠盐,Timnodonic acid sodium,EPA sodium

Eicosapentaenoic Acid (EPA) sodium 为口服活性 ω-3 长链多不饱和脂肪酸 (ω-3 LC-PUFAs)。其通过DNA去甲基化,促进肿瘤抑制基因CCAAT/增强子结合蛋白δ (C/EBPδ)的重新表达,并通过H-RAS内含子1 CpG岛的去甲基化,激活U937白血病细胞中RAS/ERK/C/EBPβ途径。此外,该化合物能够促进血管平滑肌细胞松弛和血管舒张。

天然产物

Visnagin
Cat.No: T8198
Synonym:
Target: Others
Khellin
Cat.No: T1431
Synonym: 凯林,Amicardine,Methafrone,Visammin
Target: EGFR, Others
L-Arginine
Cat.No: T3S0364
Synonym: L-精氨酸,L-Arg,(S)-(+)-Arginine
Target: IL Receptor, Endogenous Metabolite, NO Synthase
Theophylline
Cat.No: T1083
Synonym: Theo-24,1,3-Dimethylxanthine,茶碱
Target: Endogenous Metabolite, HDAC, PDE, Adenosine Receptor, Autophagy
14-Deoxyandrographolide
Cat.No: T8288
Synonym: 去氧穿心莲内酯,14-去氧穿心莲内酯
Target: Apoptosis, Others
Acetagastrodin
Cat.No: T8178
Synonym: 乙酰天麻素,Acegastrodine
Target: Others
Desloratadine
Cat.No: T2520
Synonym: Sch34117,地氯雷他定,NSC 675447
Target: Endogenous Metabolite, Histamine Receptor
Gentisin
Cat.No: TN1683
Synonym: 龙胆根素,龍膽根素
Target: DNA/RNA Synthesis
3-Epioleanolic acid
Cat.No: TN1248
Synonym:
Target: AChR
7-O-Methyleriodictyol
Cat.No: TN3243
Synonym:
Target: AChR
Prim-O-glucosylcimifugin
Cat.No: T3805
Synonym: 升麻苷,Cimifugin beta-D-glucopyranoside,Cimifugin 7-glucoside
Target: TNF, COX, JAK, NO Synthase
Diphylline
Cat.No: T0892
Synonym: 二羟丙茶碱,Dyphylline,Diprophylline
Target: PDE, Adenosine Receptor
8-​O-​Acetylharpagide
Cat.No: T6S2025
Synonym: 8-O-乙酰哈巴苷,8-Acetylharpagide,3-Acetylharpagide,Acetylharpagide,8-O-Acetylharpagide
Target: Antibacterial
Praeruptorin C
Cat.No: T6S1418
Synonym:
Target: Antioxidant, Calcium Channel
Prostaglandin E2
Cat.No: T5014
Synonym: 地诺前列酮,前列腺素 E2,PGE2,Dinoprostone,Prostaglandin E2 (PGE2)
Target: Endogenous Metabolite, Prostaglandin Receptor
Litorin acetate(55749-97-8 Free base)
Cat.No: T20604L
Synonym:
Target: Bombesin Receptor
Histamine
Cat.No: T0965
Synonym: Ergamine,组胺
Target: 5-HT Receptor, Endogenous Metabolite, Histamine Receptor
Histamine dihydrochloride
Cat.No: T6534
Synonym: 组胺二盐酸盐,peremin,Ceplene,Histamine 2HCl
Target: Endogenous Metabolite, Histamine Receptor
2'-acetylacteoside
Cat.No: T6102
Synonym:
Target: Antioxidant, Reductase
Liensinine diperchlorate
Cat.No: T4S1102
Synonym: 莲心碱高氯酸盐,莲心碱二高氯酸盐,Liensinine-Perchlorate
Target: Mitophagy, Others, Autophagy
Polydatin
Cat.No: T3427
Synonym: Piceid,虎杖苷,Polydotin Peceid
Target: Apoptosis, Mitophagy, NF-κB, Autophagy
Trifolirhizin
Cat.No: T4S0998
Synonym: 红车轴草根甙/三叶豆紫檀苷,三叶豆紫檀苷
Target: TNF, Tyrosinase
Prostaglandin E1
Cat.No: T1626
Synonym: 前列地尔,PGE1,列腺素E1,Alprostadil
Target: Endogenous Metabolite, Prostaglandin Receptor
2,2,2-Trichloroethanol
Cat.No: T37709
Synonym:
Target: Potassium Channel, Endogenous Metabolite
L-Hyoscyamine sulfate
Cat.No: T4S1619
Synonym: Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate,硫酸天仙子胺水合物,L-莨菪碱硫酸盐
Target: AChR
L-Hyoscyamine
Cat.No: T0962
Synonym: Daturine,Hyoscyamine,L-莨菪碱,L-天仙子胺
Target: AChR
GUANOSINE 3':5'-CYCLIC MONOPHOSPHATE SOD
Cat.No: T5065
Synonym: Monosodium-GMP,cGMP sodium salt,鸟苷-3',5'-环磷酸一钠盐,Cyclic GMP
Target: PKA
Caffeic Acid Phenethyl Ester
Cat.No: T6429
Synonym: Phenylethyl Caffeate,咖啡酸苯乙酯,CAPE
Target: Apoptosis, NF-κB
Cytochalasin D
Cat.No: T3229
Synonym:
Target: ATPase, p38 MAPK, Calcium Channel, Akt, PI3K
Allicin
Cat.No: T3123
Synonym:
Target: ERK, IL Receptor, Others, IκB/IKK, p38 MAPK, TNF, ROS, Caspase, Antifection
Peimisine
Cat.No: T5S0106
Synonym: 贝母辛,Ebeiensine
Target: RAAS, AChR
Pentagalloylglucose
Cat.No: T3794
Synonym: Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose,1,2,3,4,6-五没食子酰葡萄糖
Target: Influenza Virus
Litorin
Cat.No: T20604
Synonym:
Target:
7Beta-Hydroxycholesterol
Cat.No: TN1338
Synonym:
Target: LDL, Calcium Channel, MAPK
Fargesone B
Cat.No: TN4051
Synonym:
Target: cAMP, Calcium Channel
Pterosin Z
Cat.No: TN5341
Synonym:
Target:
Paspalinine
Cat.No: TN5608
Synonym:
Target:
Vindorosine
Cat.No: TN5234
Synonym:
Target: Calcium Channel, Sodium Channel
Pimaric acid
Cat.No: TN2075
Synonym:
Target: MMP, p38 MAPK, NF-κB
Neoprzewaquinone A
Cat.No: TN1985
Synonym:
Target: ROCK, Pim, STAT
9-Hydroxycanthin-6-one
Cat.No: TN3319
Synonym:
Target: Potassium Channel, GSK-3, Calcium Channel, Wnt/beta-catenin
13-Hydroxylupanine hydrochloride
Cat.No: T83454
Synonym: Hydroxylupanine hydrochloride
Target:
Liriodenine
Cat.No: TN1875
Synonym: 鹅掌揪碱
Target: BCL, Caspase, p53
Lacinilene C
Cat.No: TN5330
Synonym: 3,10-Dihydroxy-1,3,5,7-cadinatetraen-9-one
Target:
Leukotriene C4
Cat.No: T25687
Synonym: 白三烯C4,LTC4,Leukotriene C
Target:
(R)-IDHP
Cat.No: T74193
Synonym:
Target:
Triptoquinone A
Cat.No: TN5186
Synonym:
Target: IL Receptor, NOS
Glabrene
Cat.No: TN1690
Synonym:
Target: Others, Estrogen/progestogen Receptor, Tyrosinase
Eicosapentaenoic Acid sodium
Cat.No: T72152
Synonym: 二十碳五烯酸钠盐,Timnodonic acid sodium,EPA sodium
Target:
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