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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T28869 Streptomyces A-Factor

A-Factor (Lactone)

Streptomyces A-Factor is a microbial hormone found in Streptomyces griseus. A-factor triggers streptomycin biosynthesis and cell differentiation by binding a repressor-type receptor protein (ArpA) and dissociating it from DNA.
T31742 Factor 390 A

F390-A,F390A,P-5-(S)-N-(N-(1-Oxo-2-(phosphonooxy)propyl)-L-gamma-glutamyl)-L-glutamate,F390 A

Factor 390 A is a phosphodiester between AMP & methanogen factor 420.
TP1106L α-Factor Mating Pheromone, yeast acetate

Mating Factor α acetate,α-Factor Mating Pheromone, yeast acetate(59401-28-4 free base)

Others Others
α-Factor Mating Pheromone, yeast acetate (Mating Factor α acetate)(59401-28-4 free base) 是由酿酒酵母α细胞分泌的13个氨基酸的肽。
T11373 GCN2-IN-1

A-92

Others Others
GCN2-IN-1 (A-92) 是一种有效的一般性调控阻遏蛋白激酶 2 抑制剂,可作为化疗药物用于癌症治疗的研究。
T2098 A 77-01

A77-01

ALK; TGF-beta/Smad Angiogenesis; Stem Cells; Tyrosine Kinase/Adaptors
A 77-01 是 TGF-βI 型受体家族 ALK5抑制剂(IC50:25 nM)。
T3031 A 83-01

ALK5 Inhibitor IV,A8301

ALK; TGF-beta/Smad Angiogenesis; Stem Cells; Tyrosine Kinase/Adaptors
A 83-01 (ALK5 Inhibitor IV) 是一种 TGF-βI 型受体 ALK5、ALK4 和 ALK7 的抑制剂 (IC50=12/45/7.5 nM)。A 83-01 可促进小鼠成纤维细胞重编程为 iPSCs。A 83-01 可用于类器官培养。
T4288 hVEGF-IN-1

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
hVEGF-IN-1 是一种喹唑啉衍生物,可以特异性结合内部核糖体进入位点 A 中富含 G 的序列,并会使 G-四链体结构不稳定。在 SPR 实验中,它与 IRES-A (WT) 结合的Kd 值为 0.928 μM。它能够抑制VEGF-A 蛋白表达,阻止肿瘤细胞迁移,抑制肿瘤生长。
T21445 Naphazoline

AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林

Adrenergic Receptor GPCR/G Protein; Neuroscience
Naphazoline (Naphcon-a) 是一种具有显着 α 肾上腺素能活性的拟交感神经化合物。 萘甲唑啉可用作血管收缩剂,当应用于粘膜时可快速减少肿胀。
T2479 Tyrphostin A9

Malonoben,Tyrphostin 9,SF 6847,AG 17,RG-50872

EGFR; VEGFR; Influenza Virus; PDGFR Angiogenesis; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Tyrphostin A9 (SF 6847) 是一种线粒体分裂诱导剂,是 PDGFR 抑制剂,具有抗流感病毒的活性。
TP1106 α-Factor Mating Pheromone, yeast

Mating Factor α

Alpha factor mating pheromone is a peptide of 13 amino acids secreted by Saccharomyces cerevisiae α cells.
T4637 R-7050

TNF-α Antagonist III

TNF Apoptosis
R-7050 (TNF-α Antagonist III) 是一种肿瘤坏死因子受体拮抗剂,对 TNFα具有更高选择性。
T2063 Tyrphostin 23

RG-50810,TX 825,Tyrphostin A23,AG18

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Tyrphostin 23 (AG18) 是一种EGFR 抑制剂,IC50值为35 μM。
TP1105 α-Factor Mating Pheromone, yeast (TFA)

α-Factor Mating Pheromone, yeast (TFA)(59401-28-4,FREE),Mating Factor α (TFA)

The alpha factor pheromone arrests yeast in the G1 phase of their cell cycle. Alpha Factor Mating Pheromone induces the expression of mating genes, changes in nuclear architecture, and polarzes growth toward the mating partner.
T76360 a-Helical Corticotropin Releasing Factor (12-41)

a-Helical Corticotropin Releasing Factor (12-41),一种含有30个氨基酸的α螺旋促肾上腺皮质激素释放因子/激素类似物。作为下丘脑激素的促肾上腺皮质激素释放因子 (CRF) 能促进肾上腺皮质激素 (ACTH) 分泌,而a-Helical Corticotropin Releasing Factor (12-41) 则抑制该刺激效应。
T76204 a-Helical Corticotropin Releasing Factor (9-41)

α-Helical Corticotropin Releasing Factor (9-41) 为corticotropin releasing factor (CRF)的拮抗剂,具有降低体内血浆生长激素(GH)水平的功能。
T7361 Verucerfont

NBI77860,3-(4-甲氧基-2-甲基苯基)-2,5-二甲基-N-[(1S)-1-(3-甲基-1,2,4-恶二唑-5-基)丙基]吡唑并[1,5-A]嘧啶-7-胺,GSK561679

CRFR GPCR/G Protein
Verucerfont (NBI77860) 是促肾上腺皮质激素释放因子受体 1 (CRF1) 拮抗剂,作用于 CRF1(IC50:6.1 nM),CRF2 (IC50>1000 nM)和 CRF-BP (IC50>1000 nM)。
T6146 Dorsomorphin dihydrochloride

BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride

AMPK; Autophagy; TGF-beta/Smad Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Stem Cells
Dorsomorphin dihydrochloride (BML-275 2HCl) 是一种选择性和 ATP 竞争性的AMPK 抑制剂,Ki 为 109 nM。它诱导自噬,通过靶向抑制 I 型受体ALK2,ALK3和ALK6来抑制 BMP 途径。
T27102 CV-6209

CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.
T15401 GNE-371

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
GNE-371 是一种选择性人类转录起始因子 TFIID 亚基 1 和转录起始因子 TFIID 亚基 1-like 第二溴结构域的探针。
T27257 EMD-503982

EMD503982,EMD 503982

Factor Xa Metabolism
EMD-503982 是潜在的因子Xa和因子VIIa抑制剂,具有潜在的抗癌抗肿瘤活性,可用于研究血栓栓塞性疾病和神经系统疾病。
T2160 Suramin Sodium Salt

苏拉明钠,BAY-205,Suramin hexasodium salt,苏拉明钠盐,NF-060

Apoptosis; Phosphatase; SARS-CoV; Sirtuin; Reverse Transcriptase; Topoisomerase; Parasite Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
Suramin Sodium Salt (BAY-205) 是可逆的竞争性蛋白酪氨酸磷酸酶抑制剂。它抑制 IP5K,是抗寄生虫,抗肿瘤和抗血管生成剂。它是sirtuins 的有效抑制剂,也是 SARS-CoV-2 RNA 依赖性 RNA 聚合酶抑制剂。
T4508 Glycyl-L-Histidyl-L-Lysine

Others Others
Glycyl-L-Histidyl-L-Lysine 是一种肝细胞生长因子和一种合成的肝营养剂,可刺激肝红细胞生成因子的产生。
T14905 CCT251236

HSP Cytoskeletal Signaling; Metabolism
CCT251236 is an orally available Pirin ligand obtained from a heat shock transcription factor 1 (hsf1) phenotypic screen. It inhibits HSF1-mediated HSP72 induction (IC50: 19 nM).
T77457 Emicizumab

ACE 910,RO 5534262

Others Others
Emicizumab(ACE 910) 是一种人源化单克隆抗体,桥接活化因子 IX 和激活因子 X,以模拟活化因子 VIII 的功能。Emicizumab 可用于预防和治疗血友病 A
T5475 ZD-4190

EGFR; VEGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
ZD-4190 是血管内皮细胞生长因子受体 2 (VEGFR2) 和表皮生长因子受体 (EGFR) 信号传导的抑制剂,用于治疗癌症。
T28607 Rocepafant

LAU 8080,LAU8080,BN 50730,LAU-8080,BN50730,BN-50730

Platelet aggregation Others
Rocepafant (LAU8080) 是一种血小板活化因子(PAF)拮抗剂,可减轻新生大鼠缺氧缺血性脑损伤。Rocepafant 抑制肿瘤坏死因子-Afa 介导的小鼠 L929 肿瘤细胞的细胞毒性。
T28740 SDZ-62-434

SDZ 62 434,SDZ62434

Platelet aggregation Others
SDZ-62-434 是一种血小板活化因子抑制剂,具有抗肿瘤活性,抑制静止的瑞士 3T3 细胞中 bombesin 和血小板衍生生长因子诱导的 DNA 合成,可用于研究白血病、人异种移植结直肠癌和肺癌。
T60064 WAY-270360

N-[4-(1H-benzimidazol-2-yl)phenyl]-2,4-dimethoxybenzamide

EGFR; Sirtuin Angiogenesis; Chromatin/Epigenetic; DNA Damage/DNA Repair; JAK/STAT signaling; Tyrosine Kinase/Adaptors
WAY-270360 (N-[4-(1H-benzimidazol-2-yl)phenyl]-2,4-dimethoxybenzamide) 是一种 Sirtuin 调节剂和一种表皮生长因子受体 (EGFR) 抑制剂。
T8460 Olmutinib

HM61713,BI1482694

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Olmutinib (BI1482694) 是一种新型表皮生长因子受体酪氨酸激酶抑制剂。
T20454 4-Chlorophenylurea

NSC12971,NSC 12971,NSC-12971,4-氯苯基脲

Factor Xa Metabolism
4-Chlorophenylurea (NSC-12971) 是一种新型口服生物可利用的 Xa 因子抑制剂。
T24804 SM27

SM-27,NSC-37204,SM 27,NSC37204

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
SM27 是一种成纤维细胞生长因子 2(FGF2) 抑制剂,具有抗血管生成活性,可用于研究肿瘤。
T3469 PCI-27483

PCI27483

Others Others
PCI-27483 是一种FVIIa/tissue factor 抑制剂,具有抗肿瘤的作用。
T67853 Rivaroxaban Impurity

Rivaroxaban-10

Factor Xa Metabolism
Rivaroxaban Impurity (Rivaroxaban-10) 是一种强效凝血因子Xa 抑制剂,IC50=66 nM。
TP1820L Osteogenic Growth Peptide, OGP acetate

Osteogenic Growth Peptide, OGP acetate(132996-61-3 free base)

Others Others
Osteogenic Growth Peptide, OGP acetate(132996-61-3 free base) 是一种短的、天然存在的 14 聚体生长因子肽,存在于血清中,浓度为 μM。成骨生长肽 OGP 是局部骨髓损伤全身成骨反应机制的关键因素。
T24612 Pentachloropseudilin

PClP

Pentachloropseudilin is a selective inhibitor of Myosin-1. In target cells, It acts by suppressing transforming growth factor-β activity by accelerating cell-surface type II TGF-β receptor turnover.
T9189 Iptacopan hydrochloride

Iptacopan HCl,LNP023 hydrochloride

Complement System Immunology/Inflammation
Iptacopan hydrochloride (LNP023 hydrochloride) 是一种可口服、高效和高选择性的因子 B 抑制剂,IC50 为 10 nM。 LNP023 显示与人因子 B 的直接、可逆和高亲和力结合,KD 为 7.9 nM。
T19584L TNF-α (31-45), human acetate

TNF-α (31-45), human acetate(144796-71-4 free base)

Others Others
TNF-α (31-45), human acetate(144796-71-4 free base) 是一种肿瘤坏死因子-α 的肽。
T27318 Fidexaban

CI-1031,BX-807834,PD-200022,CI1031,BX807834,ZK-807834

Factor Xa Metabolism
Fidexaban (CI1031) 是一种新型、强效、选择性和口服活性 Xa 因子抑制剂,在多种测定中均显示出抗血栓活性。
T8151 Mobocertinib

tak788

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Mobocertinib (tak788) 是可口服的EGFR 和HER2突变的抑制剂,具有抗肿瘤活性。
T3721 Avitinib maleate

艾维替尼马来酸盐,艾维替尼

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Avitinib maleate 是基于吡咯并嘧啶的不可逆的表皮生长因子受体抑制剂,IC50值为7.68 nM。
T14007 PAF-AN-1

PAFR GPCR/G Protein
PAF-AN-1是一种新型有效的血小板激活因子受体 (PAF) 拮抗剂,参与研究过敏性死亡。
TQ0137 A-484954

A 484954

CaMK; Parasite; Autophagy Autophagy; Microbiology/Virology; Neuroscience
A-484954 (A 484954) 是一种高度特异性的真核延伸因子-2 抑制剂,其 IC50值为 280 nM。
T11561 HIF-2α-IN-2

HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Chromatin/Epigenetic; Metabolism
HIF-2α-IN-2 是低氧诱导因子抑制剂,IC50=16 nM。
T9927 Panitumumab

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Panitumumab 是一种重组全人源 IgG2 单克隆抗体,可与表皮生长因子(EGFR)结合,具有抗肿瘤活性。
T22592 ATPγS tetralithium salt

ATP-gamma-S tetralithium salt

PERK Apoptosis
ATPγS tetralithium salt 是真核生物翻译起始因子 eIF4A 的核苷酸水解和RNA解链活性的底物,与 p97 突变体和朊病毒相关。
T10174 5-R-Rivaroxaban

Factor Xa Metabolism
5-R-Rivaroxaban 是一种 Rivaroxaban 的 R 型对映体。其中 Rivaroxaban 是选择性的Factor Xa(FXa) 抑制剂。
TP1155L Human growth hormone-releasing factor acetate

GHSR GPCR/G Protein
Human growth hormone-releasing factor acetate 是一种下丘脑多肽,通过与垂体前叶细胞上的 GHRH 受体 (GHRHR) 结合来刺激 GH 的产生和释放。
T4397 DIM-C-pPhOCH3

C-DIM5

Others Others
DIM-C-pPhOCH3 (C-DIM5) 是 Nur77 激动剂。其中 Nur77 是孤儿核受体。
T31095 Crinecerfont

SSR125543,SSR 125543,SSR-125543,SSR125543A,SSR 125543A,SSR-125543A

CRFR GPCR/G Protein
Crinecerfont (SSR-125543) 是促肾上腺皮质激素释放因子 1 受体 (CRF1) 的特异性拮抗剂,可用于经典先天性肾上腺增生的研究。
T6894 ML264

CID-51003603

DNA/RNA Synthesis; KLF Cell Cycle/Checkpoint; DNA Damage/DNA Repair; MAPK
ML264 (CID-51003603) 是抗肿瘤剂,能够特异性地抑制 Krüppel 样因子 5 表达。

化合物

Streptomyces A-Factor
Cat.No: T28869
Synonym: A-Factor (Lactone)
Target:
Factor 390 A
Cat.No: T31742
Synonym: F390-A,F390A,P-5-(S)-N-(N-(1-Oxo-2-(phosphonooxy)propyl)-L-gamma-glutamyl)-L-glutamate,F390 A
Target:
α-Factor Mating Pheromone, yeast acetate
Cat.No: TP1106L
Synonym: Mating Factor α acetate,α-Factor Mating Pheromone, yeast acetate(59401-28-4 free base)
Target: Others
GCN2-IN-1
Cat.No: T11373
Synonym: A-92
Target: Others
A 77-01
Cat.No: T2098
Synonym: A77-01
Target: ALK, TGF-beta/Smad
A 83-01
Cat.No: T3031
Synonym: ALK5 Inhibitor IV,A8301
Target: ALK, TGF-beta/Smad
hVEGF-IN-1
Cat.No: T4288
Synonym:
Target: VEGFR
Naphazoline
Cat.No: T21445
Synonym: AK-Con,Naphcon-a,Clear Eyes,All Clear,萘甲唑林
Target: Adrenergic Receptor
Tyrphostin A9
Cat.No: T2479
Synonym: Malonoben,Tyrphostin 9,SF 6847,AG 17,RG-50872
Target: EGFR, VEGFR, Influenza Virus, PDGFR
α-Factor Mating Pheromone, yeast
Cat.No: TP1106
Synonym: Mating Factor α
Target:
R-7050
Cat.No: T4637
Synonym: TNF-α Antagonist III
Target: TNF
Tyrphostin 23
Cat.No: T2063
Synonym: RG-50810,TX 825,Tyrphostin A23,AG18
Target: EGFR
α-Factor Mating Pheromone, yeast (TFA)
Cat.No: TP1105
Synonym: α-Factor Mating Pheromone, yeast (TFA)(59401-28-4,FREE),Mating Factor α (TFA)
Target:
a-Helical Corticotropin Releasing Factor (12-41)
Cat.No: T76360
Synonym:
Target:
a-Helical Corticotropin Releasing Factor (9-41)
Cat.No: T76204
Synonym:
Target:
Verucerfont
Cat.No: T7361
Synonym: NBI77860,3-(4-甲氧基-2-甲基苯基)-2,5-二甲基-N-[(1S)-1-(3-甲基-1,2,4-恶二唑-5-基)丙基]吡唑并[1,5-A]嘧啶-7-胺,GSK561679
Target: CRFR
Dorsomorphin dihydrochloride
Cat.No: T6146
Synonym: BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride
Target: AMPK, Autophagy, TGF-beta/Smad
CV-6209
Cat.No: T27102
Synonym:
Target:
GNE-371
Cat.No: T15401
Synonym:
Target: DNA/RNA Synthesis
EMD-503982
Cat.No: T27257
Synonym: EMD503982,EMD 503982
Target: Factor Xa
Suramin Sodium Salt
Cat.No: T2160
Synonym: 苏拉明钠,BAY-205,Suramin hexasodium salt,苏拉明钠盐,NF-060
Target: Apoptosis, Phosphatase, SARS-CoV, Sirtuin, Reverse Transcriptase, Topoisomerase, Parasite
Glycyl-L-Histidyl-L-Lysine
Cat.No: T4508
Synonym:
Target: Others
CCT251236
Cat.No: T14905
Synonym:
Target: HSP
Emicizumab
Cat.No: T77457
Synonym: ACE 910,RO 5534262
Target: Others
ZD-4190
Cat.No: T5475
Synonym:
Target: EGFR, VEGFR
Rocepafant
Cat.No: T28607
Synonym: LAU 8080,LAU8080,BN 50730,LAU-8080,BN50730,BN-50730
Target: Platelet aggregation
SDZ-62-434
Cat.No: T28740
Synonym: SDZ 62 434,SDZ62434
Target: Platelet aggregation
WAY-270360
Cat.No: T60064
Synonym: N-[4-(1H-benzimidazol-2-yl)phenyl]-2,4-dimethoxybenzamide
Target: EGFR, Sirtuin
Olmutinib
Cat.No: T8460
Synonym: HM61713,BI1482694
Target: EGFR
4-Chlorophenylurea
Cat.No: T20454
Synonym: NSC12971,NSC 12971,NSC-12971,4-氯苯基脲
Target: Factor Xa
SM27
Cat.No: T24804
Synonym: SM-27,NSC-37204,SM 27,NSC37204
Target: FGFR
PCI-27483
Cat.No: T3469
Synonym: PCI27483
Target: Others
Rivaroxaban Impurity
Cat.No: T67853
Synonym: Rivaroxaban-10
Target: Factor Xa
Osteogenic Growth Peptide, OGP acetate
Cat.No: TP1820L
Synonym: Osteogenic Growth Peptide, OGP acetate(132996-61-3 free base)
Target: Others
Pentachloropseudilin
Cat.No: T24612
Synonym: PClP
Target:
Iptacopan hydrochloride
Cat.No: T9189
Synonym: Iptacopan HCl,LNP023 hydrochloride
Target: Complement System
TNF-α (31-45), human acetate
Cat.No: T19584L
Synonym: TNF-α (31-45), human acetate(144796-71-4 free base)
Target: Others
Fidexaban
Cat.No: T27318
Synonym: CI-1031,BX-807834,PD-200022,CI1031,BX807834,ZK-807834
Target: Factor Xa
Mobocertinib
Cat.No: T8151
Synonym: tak788
Target: EGFR
Avitinib maleate
Cat.No: T3721
Synonym: 艾维替尼马来酸盐,艾维替尼
Target: EGFR
PAF-AN-1
Cat.No: T14007
Synonym:
Target: PAFR
A-484954
Cat.No: TQ0137
Synonym: A 484954
Target: CaMK, Parasite, Autophagy
HIF-2α-IN-2
Cat.No: T11561
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase, HIF
Panitumumab
Cat.No: T9927
Synonym:
Target: EGFR
ATPγS tetralithium salt
Cat.No: T22592
Synonym: ATP-gamma-S tetralithium salt
Target: PERK
5-R-Rivaroxaban
Cat.No: T10174
Synonym:
Target: Factor Xa
Human growth hormone-releasing factor acetate
Cat.No: TP1155L
Synonym:
Target: GHSR
DIM-C-pPhOCH3
Cat.No: T4397
Synonym: C-DIM5
Target: Others
Crinecerfont
Cat.No: T31095
Synonym: SSR125543,SSR 125543,SSR-125543,SSR125543A,SSR 125543A,SSR-125543A
Target: CRFR
ML264
Cat.No: T6894
Synonym: CID-51003603
Target: DNA/RNA Synthesis, KLF
Cat. No. Product Name Target Signaling Pathways
TQ0131 Rocaglamide

Rocaglamide A,楝酰胺,Roc-A

HSP; NF-κB; PERK Apoptosis; Cytoskeletal Signaling; Metabolism; NF-κB
Rocaglamide (Roc-A) 是从米仔兰中分离出来的一种天然产物,具有抗癌特性,可用于咳嗽,受伤,哮喘和炎症性皮肤病。它是一种有效的选择性热休克因子 1 活化抑制剂,IC50约为 50 nM。它是 T 细胞中 NF-κB 活化的有效抑制剂,还抑制翻译起始因子eIF4A 的功能。
T5687 WITHAFERIN A

醉茄素 A,醉茄素A

Ferroptosis; NF-κB Apoptosis; NF-κB
Withaferin A 是从南非醉茄中分离到的一种甾体内酯,是内皮蛋白 C 受体脱落抑制剂,可以抑制NF-kB 的活性,具有抗炎,抗肿瘤等作用。它是一种新型 NFkappaB 抑制剂,有望成为治疗各种炎症性疾病和癌症的新型抗炎药。
T3877 Esculentoside A

NF-κB; COX Immunology/Inflammation; Neuroscience; NF-κB
Esculentoside A 是一种三萜皂苷,从商陆根部分离得到。它在具有抗炎活性,对环氧合酶-2 具有选择性抑制活性。它通过抑制NF-κB 和丝裂原活化蛋白激酶信号通路抑制 LPS 诱导的急性肺损伤中的炎症反应。
T3777 Praeruptorin A

(+)-Praeruptorin A,白花前胡甲素

CaMK; NF-κB Neuroscience; NF-κB
Praeruptorin A ((+)-Praeruptorin A) 是一种白花前胡的主要生物活性成分。它能够抑制 NF-κB 活化,发挥抗炎作用。
T6S1966 Curculigoside

Curculigoside A,仙茅苷

Antioxidant; NF-κB; JAK; STAT Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; NF-κB; oxidation-reduction; Stem Cells
Curculigoside (Curculigoside A) 是仙茅中的主要皂苷,具有显著的抗氧化、抗骨质疏松、抗抑郁和神经保护作用。它通过调节JAK/STAT/NF-κB 信号传导途径,具有抗关节炎作用。
T6S1597 Mulberroside A

桑皮苷 A,桑皮苷A

TNF; Tyrosinase; Interleukin Apoptosis; Immunology/Inflammation; Proteases/Proteasome
Mulberroside A 是桑中的一种主要活性成分,可降低TNF-α、IL-1β和IL-6的表达,抑制 NALP3、caspase-1 和 NF-κB 的激活以及 ERK、JNK 和 p38 的磷酸化 。它抑制蘑菇酪氨酸酶,具有抗炎和抗细胞凋亡作用。
T2913 Schisantherin A

五味子酯甲,Schisanwilsonin H,Gomisin-C,Wuweizi ester-A,Schizantherin-A,Arisanschinin K

NF-κB NF-κB
Schisantherin A (Wuweizi ester-A) 是一种利用 IκBα 降解,抑制p65-NF-κB 易位进入细胞核的木脂素。
TN2081 Maohuoside A

MAPK MAPK
Maohuoside A 是从 E. koreanum 中分离出的单一化合物,具有促进成骨作用。它能够利用 MAPK 信号通路骨及形态发生蛋白 (BMP) ,促进骨髓间充质干细胞的成骨作用。
T2921 Sinomenine hydrochloride

盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride

Apoptosis; NF-κB; Opioid Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; GPCR/G Protein; Neuroscience; NF-κB
Sinomenine hydrochloride (Kukoline hydrochloride) 是来自汉防己的一种生物碱,是NF-κB 活化的阻断剂。Sinomenine 也是一种 μ 阿片受体激活剂。
T2801 Aristolochic acid A

马兜铃酸,TR 1736,Aristolochin,Aristolochine,Aristolochic Acid I,Aristolochic Acid

Others; NF-κB NF-κB; Others
Aristolochic acid A (TR 1736) 是植物提取物 Aristolochic acids 的主要成分,主要存在于 AristolochiaAsarum 草本植物中。它降低人细胞中膀胱癌相关BLCAP 基因表达。它显著降低激活蛋白1 (AP-1) 和NF-κB 活性。
T2777 Ginsenoside Rg1

Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2

Apoptosis; Beta Amyloid; NF-κB Apoptosis; Neuroscience; NF-κB
Ginsenoside Rg1 (Panaxoside Rg1) 是人参的主要活性成分之一,可减少NF-κB 核易位。它改善认知功能受损,通过降低大脑Aβ水平来发挥作用。
T78500 α-Factor Mating Pheromone, yeast TFA

Mating Factor α TFA

α-Factor Mating Pheromone, yeast (TFA)为一来自S. cerevisiae的α细胞分泌的十三肽,通过Ste2p受体发挥作用。
T0200 α-Lipoic Acid

Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid,α-硫辛酸,硫辛酸

Apoptosis; NF-κB; HIV Protease; Mitochondrial Metabolism; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
α-Lipoic Acid (DL-α-Lipoic acid) 是线粒体酶复合物的重要辅助因子,是一种抗氧化剂,可抑制NF-κB 依赖性的HIV-1LTR 活化。它还可诱导内质网应激介导的肝癌细胞凋亡。
TN1694 Gliotoxin

Apoptosis; NF-κB; Wnt/beta-catenin; COX; PKA; Antibacterial; Antifection Apoptosis; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Neuroscience; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Gliotoxin 是一种次生代谢产物,由A. fumigatus 分泌,可以抑制巨噬细胞的吞噬作用和其他免疫细胞的免疫功能。它通过阻止 IκB 降解来抑制诱导型NF-κB 活性,从而诱导宿主细胞凋亡。它可以激活PKA 并增加细胞内 cAMP 浓度,调节肌动蛋白细胞骨架重排以促进A. fumigatus 内化到肺上皮细胞。
T2932 Ginsenoside Rh1

Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1

IL Receptor; TNF; Endogenous Metabolite; PPAR; Interleukin Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism
Ginsenoside Rh1 (Sanchinoside B2) 是人参的一种主要成分,具有抗炎作用,抑制PPAR-γ,TNF-α,IL-6和IL-1β的表达。
TWA2417 Sodium taurocholate

牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium

Others Others
Sodium taurocholate (Taurocholate Sodium) hydrate 具有显著的生物学效应,例如通过上调 VEGF-A 的表达抑制肝动脉结扎所致的胆道损伤。对免疫系统具有一定的调节作用。
T2851 Daphnetin

7,8-Dihydroxycoumarin,Daphnetol,瑞香素

EGFR; PKA; PKC; Parasite; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物,有抗氧化、抗炎、抗疟疾和解热作用,可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。
T4183 lavendustin A

RG-14355,NSC 678027,薰草菌素

EGFR; Tyrosinase Angiogenesis; JAK/STAT signaling; Proteases/Proteasome; Tyrosine Kinase/Adaptors
lavendustin A (RG-14355) 是从链霉菌中分离得到的一种天然产物,是细胞渗透性表皮生长因子受体 (EGFR) 酪氨酸激酶抑制剂,能抑制血管内皮生长因子诱导的血管生成,阻断 LTPGABA-A 的诱导。
T6943 Picropodophyllin

AXL1717,苦鬼臼脂素,Picropodophyllin (PPP),Picropodophyllotoxin,PPP,苦鬼臼毒素

Apoptosis; IGF-1R Apoptosis; Tyrosine Kinase/Adaptors
Picropodophyllin (Picropodophyllin (PPP)) 是一种选择性的胰岛素样生长因子-1受体抑制剂,IC50为1 nM。
TN1635 Euphorbia factor L8

Others Others
Euphorbia factor L8 是大戟种子中的二萜。
TN1634 Euphorbia factor L7b

千金子素L7B

Others Others
Euphorbia factor L7b 是从大戟属植物大戟中提取的天然产物。
T125211 Deoxy euphorbia factor L1

Others Others
Deoxy euphorbia factor L1是一种天然产物,存在于植物续随子 Euphorbia lathyris L 的种子中。
T5789 XYLOTRIOSE

Others Others
Xylotriose 是双歧杆菌促生因子,是天然的低聚木糖。
T4S2014 5,15-Diacetyl-3-benzoyllathyrol

,大戟因子L3,二乙酰基苯甲酰基香豌豆醇,5,15-二乙酰基-3-苯甲酰千金子二萜醇;千金二萜醇二乙酰苯甲酰酯,Euphorbia factor L3

Others Others
5,15-Diacetyl-3-benzoyllathyrol (Euphorbia factor L3) 是一种具有抗癌作用的萜类化合物。
T10233 Acetylarenobufagin

HIF Angiogenesis; Chromatin/Epigenetic
Acetylarenobufagin 是一种类固醇缺氧诱导因子-1 (HIF-I) 调节剂。
T4779 4-Methylcatechol

p-Methylcatechol,3,4-二羟基甲苯,Homocatechol,4-methylbenzene-1,2-diol,3,4-Dihydroxytoluene

Others; Endogenous Metabolite Metabolism; Others
4-Methylcatechol (3,4-Dihydroxytoluene) 是 p-toluate 的代谢物,它是 Catechol 2,3-Dioxygenase 的自杀性底物抑制剂。
T3S0027 Picropodophyllotoxin

AXL 1717,Picropodophyllin,苦鬼臼毒素

IGF-1R Tyrosine Kinase/Adaptors
Picropodophyllotoxin (AXL 1717) 是一种环木脂素生物碱,存在于五月树(Podophyllum peltatum) 中,是一种具有潜在抗肿瘤活性的胰岛素样生长因子 1 受体 (IGF1R) 的小分子抑制剂。它特异性抑制 IGF1R 的活性并下调细胞表达,而不干扰其他生长因子受体的活性,例如胰岛素受体、表皮生长因子、血小板衍生生长因子、成纤维细胞生长因子和肥大/干细胞生长因子 (KIT) )。该药剂在抑制肿瘤细胞增殖和诱导肿瘤细胞凋亡方面显示出有效的活性。 IGF1R 是一种在多种人类癌症中过度表达的受体酪氨酸激酶,在多种癌细胞的生长和存活中起关键作用。
TN4662 Nonanal

Others Others
Nonanal 是木材腐烂真菌的生长因子。 Nonanal 是松梢甲虫的潜在引诱剂。
T2984 Scopoletin

Chrysatropic acid,东莨菪内酯,Esculetin 6-methyl ether,Gelseminic acid,6-Methylesculetin

Apoptosis; AChR; AChE Apoptosis; Neuroscience
Scopoletin (Esculetin 6-methyl ether) 是一种源自东莨菪根的植物生长因子,可抑制乙酰胆碱酯酶。
TQ0099 20-O-Acetylingenol-3-angelate

巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1

Others Others
20-O-Acetylingenol-3-angelate (Euphorbia factor Pe1) 是一种天然化合物,存在于植物英加的叶子和茎中。它具有多种生物活性,包括抑制肿瘤生长、抗炎、抗真菌和抗氧化作用。
TQ0280 Feretoside

HSP Cytoskeletal Signaling; Metabolism
Feretoside 是分离自杜仲树皮的一种酚类化合物。它是 HSP 诱导剂,可作为细胞保护剂。
T3007 Spermine

Gerontine,Musculamine,精胺,4,9-Diaza-1,12-dodecanediamine,NSC 268508,Neuridine

Influenza Virus; Endogenous Metabolite Metabolism; Microbiology/Virology
Spermine (Neuridine) 作为一个直接的自由基清除剂,具有抗病毒作用,能够保护 DNA 免受自由基的攻击。
T13108 Pamufetinib

H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115

VEGFR; c-Met/HGFR Angiogenesis; Tyrosine Kinase/Adaptors
Pamufetinib (TAS-115) 是VEGFR 和c-Met/HGFR 抑制剂,能够抑制 rVEGFR2 (IC50:30 nM)和 rMET (IC50:32 nM)的活性。
T7203 Oglufanide

奥谷法奈,L-Glutamyl-L-tryptophan,H-Glu-Trp-OH

VEGFR; HCV Protease; Endogenous Metabolite Angiogenesis; Metabolism; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Oglufanide (H-Glu-Trp-OH) 是一种从小牛胸腺中分离出来的二肽免疫调节剂,可抑制血管内皮生长因子,可刺激细胞内细菌感染和对丙型肝炎病毒的免疫反应。
TN1163 2'-Hydroxychalcone

Others Others
2'-Hydroxychalcone 是一种药物合成中间体,可用于合成黄酮类化合物。负载在纳米乳液中的2'-Hydroxychalcone 在Danio rerio 模型对副球孢子菌显示出杀真菌活性。2'-Hydroxychalcone 通过负载脂质的Hepg2细胞中的氧化应激诱导细胞毒性。2'-Hydroxychalcone 抑制通过逆转录聚合酶链反应确定的肿瘤坏死因子-α诱导ICAM-1,VCAM-1和E-选择素的稳态转录水平,因此可能会干扰其基因的转录。
T3843 Pinosylvin

银松素,3,5-stilbenediol,5-Styrylresorcinol

Apoptosis; Others; Antibacterial; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Others
Pinosylvin (5-Styrylresorcinol) 是从Pinus spp 的心材中分离出来的一种白藜芦醇类似物,可诱导白血病细胞凋亡和自噬。它是一种感染前的类苯乙烯类毒素,具有抗菌活性。
T13502 3-Oxo-5β-cholanoic acid

3-氧代-5β-胆烷酸,Dehydrolithocholic acid

ROR Metabolism
3-Oxo-5β-cholanoic acid (Dehydrolithocholic acid) 是胆汁酸的一种代谢产物。3-Oxo-5β-cholanoic acid 直接与关键转录因子RORγt(Kd=1.13 μM) 结合抑制TH17细胞分化。
T2S0843 Negletein

黄芩素-7-甲醚,7-O-Methylbaicalein,Baicalein-7-methylether

IL Receptor; TNF; NOS; Interleukin Apoptosis; Immunology/Inflammation
Negletein (7-O-Methylbaicalein) 一种神经保护剂,可增强神经生长因子的作用并诱导 PC12 细胞中的神经突生长。它通过抑制TNF-α和IL-1β表现出抗炎活性,其 IC50值分别为 16.4 和 10.8 μM。它还具有抗菌、抗缺氧和抗阿尔茨海默病活性。
TN2259 Taurocholic acid

N-Choloyltaurine

TNF; PI3K Apoptosis; PI3K/Akt/mTOR signaling
Taurocholic acid (N-Choloyltaurine) 是一种胆汁酸,参与脂肪的乳化。Taurocholic acid 具有细胞保护作用,可通过 PI3K 介导的途径防止肿瘤坏死因子-α 诱导的胆管细胞损伤。
T2745 18α-Glycyrrhetinic acid

18-α-甘草次酸,甘草次酸,Enoxolone,Glycyrrhetinic acid

Apoptosis; NF-κB; Proteasome Apoptosis; NF-κB; Proteases/Proteasome; Ubiquitination
18α-Glycyrrhetinic acid (Enoxolone) 是 NF-kB 的抑制剂和蛋白酶体的激活剂,在多细胞生物中起到促进长寿和抗聚集因子的作用。它诱导细胞凋亡。
T0131 Cepharanthine

NSC-623442,千金藤碱,千金藤素

Apoptosis; TNF; HIV Protease; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Cepharanthine (NSC-623442) 是从Stephania cepharanthaHayata 中提取的一种生物碱,具有抗炎、抗氧化作用。它可抑制肿瘤坏死因子 (TNF)-α 介导的 NFκB 刺激、质膜脂质过氧化和血小板聚集,并抑制细胞因子的产生。
T9715 Aplidine

SARS-CoV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Aplidine 是有效的eEF1A2(KD=80 nM) 靶向的抗癌药物。Aplidine 具有抗病毒活性,抑制SARS-CoV-2的 IC90为 0.88 nM。Aplidine 在多发性骨髓瘤,晚期癌症及 COVID-19 领域有研究的价值。
T6429 Caffeic Acid Phenethyl Ester

Phenylethyl Caffeate,咖啡酸苯乙酯,CAPE

Apoptosis; NF-κB Apoptosis; NF-κB
Caffeic Acid Phenethyl Ester (Phenylethyl Caffeate) 是咖啡酸的苯乙醇酯,是蜂巢蜂胶的生物活性成分。它抑制核转录因子 NF-kappa B 的激活,具有抗肿瘤、细胞保护和免疫调节活性。它抑制 PDGF 诱导的血管平滑肌细胞增殖。
T4A2462 Telocinobufagin

Telobufotoxin,远华蟾蜍精,Telocinobufogenin

Others Others
Telocinobufagin (Telobufotoxin) 是一种从蟾酥中分离提取获得的组份。
TN6393 fulvotomentoside A

Others Others
fulvotomentoside A 可降低肠道中 IL-6 和 IL-17A 的过表达,并显着增加调节性 T 细胞特异性转录因子 Foxp3 的表达。这可能是Ful 改善肠道炎症的机制之一。
T0465 Ellagic acid

鞣花酸,Gallogen,Elagostasine

Hedgehog/Smoothened; Casein Kinase; Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; PKA; Syk; PKC; Carbonic Anhydrase Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Ellagic acid (Gallogen) 是从 Eucalyptus maculata Hook 和 E. Hemipholia F. Muell 的 kino 中分离出来的稠合四环天然产物,是一种有效的,ATP 竞争性的CK2抑制剂,IC50和Ki 值分别为 40 nM 和 20 nM。
T3902 Atractylenolide III

白术内酯 III,ICodonolactone,8β-Hydroxyasterolide

Apoptosis Apoptosis
Atractylenolide III (ICodonolactone) 是白术根茎主要成分,通过诱导细胞色素 c 的释放、上调 Bax 的表达和易位凋亡诱导因子,是治疗人肺癌的潜力。
TN2322 Yangambin

Calcium Channel; PAFR GPCR/G Protein; Membrane transporter/Ion channel; Metabolism
Yangambin 是从诸如番荔枝科植物中分离出来的呋喃木脂素,是选择性PAF 受体拮抗剂,通过调控Ca2+通道抑制 Ca2+流入,导致 [Ca2+]i 在血管平滑肌细胞和随后的外周血管舒张中减少,具有降压作用。
T5530 Mithramycin A

Plicamycin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Mithramycin A (Plicamycin) 是一种dna 结合的抗肿瘤抗生素,选择性特异性蛋白1 (Sp1)抑制剂,通过降低Sp1蛋白抑制多种肿瘤的生长。特异性蛋白1 (Sp1)是一种锌指转录因子,调节多种细胞功能,促进肿瘤进展。
T2787 Picroside I

6'-Cinnamoylcatalpol,胡黄连苦苷I

MMP; STAT JAK/STAT signaling; Proteases/Proteasome; Stem Cells
Picroside I (6'-Cinnamoylcatalpol) 是胡黄连的一种天然产物,是有肝脏保护作用的代谢成分,可用于哮喘研究,有减轻炎症作用,还下调 pSTAT6 和 GATA3 表达。
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天然产物

Rocaglamide
Cat.No: TQ0131
Synonym: Rocaglamide A,楝酰胺,Roc-A
Target: HSP, NF-κB, PERK
WITHAFERIN A
Cat.No: T5687
Synonym: 醉茄素 A,醉茄素A
Target: Ferroptosis, NF-κB
Esculentoside A
Cat.No: T3877
Synonym:
Target: NF-κB, COX
Praeruptorin A
Cat.No: T3777
Synonym: (+)-Praeruptorin A,白花前胡甲素
Target: CaMK, NF-κB
Curculigoside
Cat.No: T6S1966
Synonym: Curculigoside A,仙茅苷
Target: Antioxidant, NF-κB, JAK, STAT
Mulberroside A
Cat.No: T6S1597
Synonym: 桑皮苷 A,桑皮苷A
Target: TNF, Tyrosinase, Interleukin
Schisantherin A
Cat.No: T2913
Synonym: 五味子酯甲,Schisanwilsonin H,Gomisin-C,Wuweizi ester-A,Schizantherin-A,Arisanschinin K
Target: NF-κB
Maohuoside A
Cat.No: TN2081
Synonym:
Target: MAPK
Sinomenine hydrochloride
Cat.No: T2921
Synonym: 盐酸青藤碱,Sabianine A hydrochloride,Cucoline hydrochloride,Kukoline hydrochloride
Target: Apoptosis, NF-κB, Opioid Receptor, Autophagy
Aristolochic acid A
Cat.No: T2801
Synonym: 马兜铃酸,TR 1736,Aristolochin,Aristolochine,Aristolochic Acid I,Aristolochic Acid
Target: Others, NF-κB
Ginsenoside Rg1
Cat.No: T2777
Synonym: Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2
Target: Apoptosis, Beta Amyloid, NF-κB
α-Factor Mating Pheromone, yeast TFA
Cat.No: T78500
Synonym: Mating Factor α TFA
Target:
α-Lipoic Acid
Cat.No: T0200
Synonym: Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid,α-硫辛酸,硫辛酸
Target: Apoptosis, NF-κB, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite
Gliotoxin
Cat.No: TN1694
Synonym:
Target: Apoptosis, NF-κB, Wnt/beta-catenin, COX, PKA, Antibacterial, Antifection
Ginsenoside Rh1
Cat.No: T2932
Synonym: Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1
Target: IL Receptor, TNF, Endogenous Metabolite, PPAR, Interleukin
Sodium taurocholate
Cat.No: TWA2417
Synonym: 牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium
Target: Others
Daphnetin
Cat.No: T2851
Synonym: 7,8-Dihydroxycoumarin,Daphnetol,瑞香素
Target: EGFR, PKA, PKC, Parasite, Autophagy
lavendustin A
Cat.No: T4183
Synonym: RG-14355,NSC 678027,薰草菌素
Target: EGFR, Tyrosinase
Picropodophyllin
Cat.No: T6943
Synonym: AXL1717,苦鬼臼脂素,Picropodophyllin (PPP),Picropodophyllotoxin,PPP,苦鬼臼毒素
Target: Apoptosis, IGF-1R
Euphorbia factor L8
Cat.No: TN1635
Synonym:
Target: Others
Euphorbia factor L7b
Cat.No: TN1634
Synonym: 千金子素L7B
Target: Others
Deoxy euphorbia factor L1
Cat.No: T125211
Synonym:
Target: Others
XYLOTRIOSE
Cat.No: T5789
Synonym:
Target: Others
5,15-Diacetyl-3-benzoyllathyrol
Cat.No: T4S2014
Synonym: ,大戟因子L3,二乙酰基苯甲酰基香豌豆醇,5,15-二乙酰基-3-苯甲酰千金子二萜醇;千金二萜醇二乙酰苯甲酰酯,Euphorbia factor L3
Target: Others
Acetylarenobufagin
Cat.No: T10233
Synonym:
Target: HIF
4-Methylcatechol
Cat.No: T4779
Synonym: p-Methylcatechol,3,4-二羟基甲苯,Homocatechol,4-methylbenzene-1,2-diol,3,4-Dihydroxytoluene
Target: Others, Endogenous Metabolite
Picropodophyllotoxin
Cat.No: T3S0027
Synonym: AXL 1717,Picropodophyllin,苦鬼臼毒素
Target: IGF-1R
Nonanal
Cat.No: TN4662
Synonym:
Target: Others
Scopoletin
Cat.No: T2984
Synonym: Chrysatropic acid,东莨菪内酯,Esculetin 6-methyl ether,Gelseminic acid,6-Methylesculetin
Target: Apoptosis, AChR, AChE
20-O-Acetylingenol-3-angelate
Cat.No: TQ0099
Synonym: 巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1
Target: Others
Feretoside
Cat.No: TQ0280
Synonym:
Target: HSP
Spermine
Cat.No: T3007
Synonym: Gerontine,Musculamine,精胺,4,9-Diaza-1,12-dodecanediamine,NSC 268508,Neuridine
Target: Influenza Virus, Endogenous Metabolite
Pamufetinib
Cat.No: T13108
Synonym: H2OL3Q4XRD,4-(2-Fluoro-4-(3-(2-phenylacetyl)thioureido)phenoxy)-7-methoxy-N-methylquinoline-6-carboxamide,TAS-115
Target: VEGFR, c-Met/HGFR
Oglufanide
Cat.No: T7203
Synonym: 奥谷法奈,L-Glutamyl-L-tryptophan,H-Glu-Trp-OH
Target: VEGFR, HCV Protease, Endogenous Metabolite
2'-Hydroxychalcone
Cat.No: TN1163
Synonym:
Target: Others
Pinosylvin
Cat.No: T3843
Synonym: 银松素,3,5-stilbenediol,5-Styrylresorcinol
Target: Apoptosis, Others, Antibacterial, Autophagy
3-Oxo-5β-cholanoic acid
Cat.No: T13502
Synonym: 3-氧代-5β-胆烷酸,Dehydrolithocholic acid
Target: ROR
Negletein
Cat.No: T2S0843
Synonym: 黄芩素-7-甲醚,7-O-Methylbaicalein,Baicalein-7-methylether
Target: IL Receptor, TNF, NOS, Interleukin
Taurocholic acid
Cat.No: TN2259
Synonym: N-Choloyltaurine
Target: TNF, PI3K
18α-Glycyrrhetinic acid
Cat.No: T2745
Synonym: 18-α-甘草次酸,甘草次酸,Enoxolone,Glycyrrhetinic acid
Target: Apoptosis, NF-κB, Proteasome
Cepharanthine
Cat.No: T0131
Synonym: NSC-623442,千金藤碱,千金藤素
Target: Apoptosis, TNF, HIV Protease, Autophagy
Aplidine
Cat.No: T9715
Synonym:
Target: SARS-CoV, DNA/RNA Synthesis
Caffeic Acid Phenethyl Ester
Cat.No: T6429
Synonym: Phenylethyl Caffeate,咖啡酸苯乙酯,CAPE
Target: Apoptosis, NF-κB
Telocinobufagin
Cat.No: T4A2462
Synonym: Telobufotoxin,远华蟾蜍精,Telocinobufogenin
Target: Others
fulvotomentoside A
Cat.No: TN6393
Synonym:
Target: Others
Ellagic acid
Cat.No: T0465
Synonym: 鞣花酸,Gallogen,Elagostasine
Target: Hedgehog/Smoothened, Casein Kinase, Reactive Oxygen Species, Topoisomerase, Endogenous Metabolite, PKA, Syk, PKC, Carbonic Anhydrase
Atractylenolide III
Cat.No: T3902
Synonym: 白术内酯 III,ICodonolactone,8β-Hydroxyasterolide
Target: Apoptosis
Yangambin
Cat.No: TN2322
Synonym:
Target: Calcium Channel, PAFR
Mithramycin A
Cat.No: T5530
Synonym: Plicamycin
Target: DNA/RNA Synthesis
Picroside I
Cat.No: T2787
Synonym: 6'-Cinnamoylcatalpol,胡黄连苦苷I
Target: MMP, STAT
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