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Targets Recommended: Nucleoside Antimetabolite/Analog Drug Metabolite Endogenous Metabolite Oxytocin Receptor

266

抑制剂 & 化合物

54

天然产物

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化合物库

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Cat. No. Product Name
L7840 高溶解性卤化片段化合物库

796 compounds
高溶解性卤化片段库包含796 个卤化片段化合物。
L7810 高溶解性多官能团片段化合物库

1159 compounds
高溶解性多官能团片段库包含1159 种片段分子
L6001 Mini真菌代谢天然产物筛选库

Inquiry
L7800 高溶解性片段库

2728 compounds
2728 种片段分子合集,数量适中,是 FBDD 方法新药筛选的有力工具。
L7850 高溶解性3D结构多样性片段化合物库

1079 compounds
高溶解性3D 结构多样性片段库包含1079 个化合物。
L2500 人内源代谢化合物库

499 compounds
499 种内源性生物活性化合物的独特集合,用于高通量、高内涵筛选;
L2540 肠道微生物代谢化合物库

614 compounds
614 种肠道微生物代谢物的集合,可以用于高通量和高内涵筛选;
L7830 高溶解性片段药效团化合物库

985 compounds
高溶解性片段药效团库包含985 个片段小分子。
L6200 瑶药化合物库

221 compounds
221 种瑶药来源的天然产物分子集合,可以用于高通量和高内涵筛选;
L2530 小鼠代谢化合物库

218 compounds
218 种小鼠代谢化合物的集合,可用于高通量筛选和高内涵筛选;
L5800 药物代谢杂质库

197 compounds
197 种药物异构体/代谢产物的特有集合,可用于高通量、高内涵筛选;
L7820 高溶解性微型片段化合物库

1081 compounds
高溶解性微型片段化合物库由 1081 个低分子量片段组成。
L7870 可溶性羧酸片段化合物库

1806 compounds
可溶性羧酸片段库包含 1806 个化合物
L2570 人代谢物化合物库

4454 compounds
4454 种人代谢物的独特集合,用于高通量、高内涵筛选;
L2501 人内源代谢化合物库 Plus

1283 compounds
1283种内源性生物活性化合物的独特集合,用于高通量、高内涵筛选。

化合物库

高溶解性卤化片段化合物库
Cat.No: L7840
Compounds: 796
高溶解性多官能团片段化合物库
Cat.No: L7810
Compounds: 1159
Mini真菌代谢天然产物筛选库
Cat.No: L6001
Compounds: Inquiry
高溶解性片段库
Cat.No: L7800
Compounds: 2728
高溶解性3D结构多样性片段化合物库
Cat.No: L7850
Compounds: 1079
人内源代谢化合物库
Cat.No: L2500
Compounds: 499
肠道微生物代谢化合物库
Cat.No: L2540
Compounds: 614
高溶解性片段药效团化合物库
Cat.No: L7830
Compounds: 985
瑶药化合物库
Cat.No: L6200
Compounds: 221
小鼠代谢化合物库
Cat.No: L2530
Compounds: 218
药物代谢杂质库
Cat.No: L5800
Compounds: 197
高溶解性微型片段化合物库
Cat.No: L7820
Compounds: 1081
可溶性羧酸片段化合物库
Cat.No: L7870
Compounds: 1806
人代谢物化合物库
Cat.No: L2570
Compounds: 4454
人内源代谢化合物库 Plus
Cat.No: L2501
Compounds: 1283
Cat. No. Product Name Target Signaling Pathways
T11857 LIT-001

Oxytocin Receptor Endocrinology/Hormones; GPCR/G Protein
LIT-001 是非肽类催产素受体激动剂,EC50为55 nM,Ki 为226 nM。它可改善孤独症小鼠模型的社交互动。
T5207 LIT927

LIT 927,LIT-927

CXCR Autophagy; GPCR/G Protein; Immunology/Inflammation
LIT927 (LIT-927) 是一种具有口服活性的 CXCL12 中性配体(对于 CXCL12 与 CXCR4 的结合,Ki:267 nM)。
T11856 LIT-001 free base

Others Others
LIT-001 free base improves social interaction in a mouse model of autism. LIT-001 free base is the first nonpeptide oxytocin receptor (OT-R) agonist (EC50=55 nM; Ki=226 nM).
T12309 Omeprazole metabolite Omeprazole sulfone

Omeprazole sulphone,Omeprazole sulfone

Others Others
Omeprazole metabolite Omeprazole sulfone 是Omeprazole 的代谢物,能够抑制质子泵。
T38404 MJ33 lithium salt

ROS Immunology/Inflammation
MJ33 lithium salt 是 NADPH 氧化酶 2 型介导的 ROS 生成抑制剂,是一种氟化磷脂类似物,可抑制过氧化物还蛋白 6 (Prdx6) 的磷脂酶 A2 (PLA2) 活性,可用于研究急性肺损伤。
TQ0210 Savolitinib

AZD-6094,Volitinib,沃利替尼,赛沃替尼,HMPL-504

c-Met/HGFR Tyrosine Kinase/Adaptors
Savolitinib (Volitinib) 是一种高效选择性、口服生物利用度c-Met 抑制剂,能够抑制 c-Met (IC50:5 nM)和 p-Met (IC50:3 nM)。它以 ATP 竞争的方式选择性结合并抑制 c-Met 的激活,破坏 c-Met 信号转导途径,具有抗肿瘤作用。
T6719 Varlitinib

ASLAN001,ARRY-334543

HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Varlitinib (ASLAN001) 是有效,可逆的泛 EGFR 小分子抑制剂,对 HER1,HER2 和 HER4 的 IC50 值分别为7,2,4 nM。
T6678 Splitomicin

1-Naphthalenepropanoic Acid,斯普利特麻一辛

Sirtuin; HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
Splitomicin (1-Naphthalenepropanoic Acid) 是 NAD(+) 依赖性组蛋白去乙酰化酶 Sir2p 的特异性抑制剂,可抑制酵母提取物中 HDAC,IC50为 60 μM。
T15581 Inolitazone

RS5444,Efatutazone,CS-7017,伊诺他酮

PPAR DNA Damage/DNA Repair; Metabolism
Inolitazone (RS5444) 是一种高亲和力PPARγ激动剂。在体外,Inotazone 显示生长抑制的IC50约为0.8 nM。
T4274 Melitracen hydrochloride

盐酸美利曲辛,盐酸美力他欣,Thymeol hydrochloride,Melixeran

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Melitracen hydrochloride (Thymeol hydrochloride) 是一种可口服的双相抗抑郁药和抗焦虑药。它可以通过突触前膜抑制去甲肾上腺素和5-羟色胺(5-HT)的吸收,从而诱导突触空间中单胺递质的增加。
T20864 7-Troc-paclitaxel

Others Others
7-Troc-paclitaxel 是紫杉醇的前体,紫杉醇具有抗肿瘤活性。
T1829 Ruxolitinib

芦可替尼,INCB018424,鲁索替尼,(R)-Ruxolitinib

Apoptosis; Mitophagy; Tyrosine Kinases; JAK; Autophagy Angiogenesis; Apoptosis; Autophagy; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Ruxolitinib (INCB018424) 是一种 JAK1/2 抑制剂 (IC50=3.3/2.8 nM),具有有效性和选择性。Ruxolitinib 具有抗肿瘤活性,可以诱导细胞自噬和凋亡。
T36522 Isoallolithocholic acid

Alloisolithocholic Acid,AILCA,3β-Hydroxy-5α-cholanic acid

Others Others
Isoallolithocholic acid (3β-Hydroxy-5α-cholanic acid) 是一种 T 细胞调节剂,是一种胆汁酸代谢物,具有抗炎活性,与人类免疫稳态有关。
T4235 Roblitinib

FGF-401

FGFR Angiogenesis; Tyrosine Kinase/Adaptors
Roblitinib (FGF-401) 是一种口服有效的,高选择性的FGFR4抑制剂(IC50:1.9 nM),具有抗癌作用。
T10738 Abemaciclib metabolite M20

CDK4/6-IN-4,LSN3106726

CDK Cell Cycle/Checkpoint
Abemaciclib metabolite M20 (CDK4/6-IN-4) 是 Abemaciclib 的活性代谢物。 Abemaciclib metabolite M20 是一种特异性 CDK4/6 抑制剂,可用于癌症治疗的相关研究。
T16045 Methotrexate metabolite

DAMPA,甲喋呤杂质E

Antifolate; Drug Metabolite Cell Cycle/Checkpoint; Metabolism
Methotrexate metabolite (DAMPA) (DAMPA)是 Methotrexate 的活性代谢物。Methotrexate 具有拮抗叶酸 (folic acid) 的作用,被用作免疫抑制剂。
T15567 Imiglitazar

TAK-559

PPAR DNA Damage/DNA Repair; Metabolism
Imiglitazar (TAK559)是有效的 PPAR-β/δ受体激动剂,具有降血糖作用。
T125575 Isourolithin A

Isourolithin A 是一种天然存在的化合物,存在于各种植物中,包括欧芹、芹菜和洋甘菊。Isourolithin A 是类黄酮家族的一员,以其抗氧化和抗炎特性而闻名。
T67956 Litoxetine

5-HT Receptor GPCR/G Protein; Neuroscience
Litoxetine 是一种选择性的5-HT 摄取抑制剂,是具有5-HT3受体拮抗剂。Litoxetine 可作为一种抗抑郁剂,在雪貂身上显示出止吐特性。Litoxetine (1和10毫克/公斤静脉注射)剂量依赖性地减少了反胃和呕吐的次数,延迟了呕吐的发生。Litoxetine 对大脑5HT3受体有亲和力(Ki = 85 nM)。
T3170 Troglitazone

CS-045,Romozin,Rezulin,Romglizone,Noscal,Prelay,曲格列酮

Apoptosis; Ferroptosis; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism
Troglitazone (Romglizone) 是一种 PPARγ 激动剂,具有抗炎和抗肿瘤活性。
T0214L Pioglitazone hydrochloride

U-72107E,AD 4833,U 72107A,Pioglitazone HCl,匹格列酮盐酸盐

Ferroptosis; PPAR Apoptosis; DNA Damage/DNA Repair; Metabolism
Pioglitazone hydrochloride (AD 4833) 是一种选择性PPARγ激动剂,高亲和力结合到 PPARγ 配体结合域。作用于人和鼠 PPARγ,EC50分别为 0.93 和 0.99 μM。它是一种口服活性噻唑烷二酮的盐酸盐,具有抗糖尿病特性和潜在的抗肿瘤活性。
T18886 3,6-Dichlorotrimellitic anhydride

Others Others
3,6-Dichlorotrimellitic anhydride 是一种能够制备多种二氯化荧光素和罗丹明 (如TET 和HEX) 的关键性前体试剂,其中氯化荧光素和罗丹明普遍用于寡核苷酸和DNA 测序的标记。
T21059 Ticagrelor metabolite M5

Ticagrelor metabolite M5,,T437700,替格瑞洛杂质H,AR-C133913XX

P2Y Receptor GPCR/G Protein; Neuroscience
Ticagrelor metabolite M5 (T437700) 是 Ticagrelor 的代谢物,是 P2Y12 受体的第一个可逆口服拮抗剂。与氯吡格雷相比,替格瑞洛对 ADP 受体具有更快和更一致的抑制作用。替格瑞洛用于治疗急性冠状动脉综合征(ACS)。
T10814 Cinacalcet metabolite M4

3-三氟甲基苯丙胺,Rarechem AL BW 1078

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cinacalcet metabolite M4 (Rarechem AL BW 1078) 是 Cinacalcet 的代谢物。Cinacalcet 是具有活性的 Ca receptor 激动剂,可用于心血管疾病。
T36624L α-Hydroxyglutaric Acid Lithium

α-Hydroxyglutaric Acid Lithium(2889-31-8 Free base)

Decarboxylase; Endogenous Metabolite; mTOR Metabolism; Others; PI3K/Akt/mTOR signaling
α-Hydroxyglutaric Acid Lithium 在微生物和动物体内有谷氨酸转化而来,是 α-酮戊二酸依赖性双加氧酶和 5-甲基胞嘧啶羟化酶抑制剂,对 ATP 合酶和 mTOR 信号传导有抑制作用。
T12834 Saroglitazar Magnesium

Others Others
Saroglitazar Magnesium 是一种新型过氧化物酶体增殖物激活受体(PPAR)激动剂,对PPARα (EC50 0.65pM)具有显著的激活活性以及对PPARγ(EC50 3 nM)有中等的激活活性。
T2327 Pelitinib

培利替尼,EKB-569,WAY-EKB 569

EGFR; Raf; MEK; Src Angiogenesis; JAK/STAT signaling; MAPK; Tyrosine Kinase/Adaptors
Pelitinib (EKB-569) 是一种可逆的EGFR 抑制剂,IC50值为38.5 nM。它也抑制Src、MEK/ERK 和 ErbB2,IC50值分别为282、800 和 1255 nM。
T15790 Lucifer Yellow CH dilithium salt

Lucifer Yellow CH dilithium salt 是一种荧光染料,可常用于选择性染色和研究光动力破坏真核细胞和亚细胞结构。
T12400 Peliglitazar racemate

(Rac)-Peliglitazar,(Rac)-BMS 426707-01,BMS 426707-01 racemate

PPAR DNA Damage/DNA Repair; Metabolism
Peliglitazar racemate(BMS 426707-01 racemate) 是 Peliglitazar 的外消旋体。Peliglitazar racemate 可作为潜在的抗糖尿病和抗肥胖剂。
T15575 Indeglitazar

PPM 204

PPAR DNA Damage/DNA Repair; Metabolism
Indeglitazar (PPM 204) 是 PPAR 的泛激动剂,包括亚型 alpha (α)、delta (δ) 和 gamma (γ)。
T14336 Allitinib

AST-1306,ALS 1306

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Allitinib (AST-1306) 是可口服的 EGFR 和 ErbB2不可逆抑制剂,IC50分别为 0.5 和 3 nM。它具有抗癌活性,抑制 ErbB4,IC50为 0.8 nM。
T17044 Tesaglitazar

PPAR DNA Damage/DNA Repair; Metabolism
Tesaglitazar 是一种有效且具有选择性的过氧化物 PPAR α / γ受体双重激动剂,对 PPARγ的亲和力比 PPARα更有效,对大鼠PPARα和人PPARα的EC50分别为13.4 μM 和3.6 μM,对大鼠PPARγ和人类 PPARγ的EC50都是0.2 μM。Tesaglitazar 诱导大鼠皮下组织间质间充质细胞DNA 合成和纤维肉瘤形成。
T22708 Darglitazone

CP-86325

PPAR DNA Damage/DNA Repair; Metabolism
Darglitazone (CP-86325) 是一种噻唑烷二酮,是口服有效的PPAR-γ选择性激动剂。Darglitazone 可以有效控制血糖和脂质代谢,在 II 型糖尿病中有研究价值。
T14176 Aleglitazar

RO0728804,R1439

PPAR DNA Damage/DNA Repair; Metabolism
Aleglitazar (R1439) 是一种高效的 PPARα/γ 双重激动剂,对人 PPARα 和 PPARγ 作用的 IC50 分别为 38 nM 和 19 nM。Aleglitazar 可用于 II 型糖尿病的研究。
T1622 Rosiglitazone maleate

BRL 49653C,BRL 49653,马来酸罗格列酮

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone maleate (BRL 49653) 是一种选择性PPARγ激活剂,具有抗糖尿病特性和潜在抗肿瘤活性。它也是TRP 通道调节剂,可抑制 TRPM2、TRPM3 的活性,激活 TRPC5。
T28743 Seglitide acetate

MK 678,MK678,MK-678

Somatostatin GPCR/G Protein
Seglitide acetate (MK-678) 是一种选择性的 sst2生长抑素受体激动剂。
T28501 Ragaglitazar

NNC61-0029,NN-622,(-)-DRF-2725,NNC-61-0029,NN 622,NNC 61-0029

PPAR DNA Damage/DNA Repair; Metabolism
Ragaglitazar(NNC-61-0029) 是一种有效的 PPARα和 PPARγ双重激动剂,在动物模型中显示出有效的降脂和胰岛素增敏作用。Ragaglitazar 可用于研究 2 型糖尿病。
T2331 Solithromycin

索利霉素,OP-1068,CEM-101

Antibacterial; Antibiotic Microbiology/Virology
Solithromycin (OP-1068) 是口服可生物利用的抗菌剂,抑制肺炎链球菌、葡萄球菌、金黄色葡萄球菌和流感嗜血杆菌的细胞活力、蛋白质合成和生长速率, IC50 值分别为 7.5 ng/mL、40 ng/mL 和 125 ng/mL。它可与核糖体的大 50S 亚基结合抑制蛋白质生物合成。
T20018 Barium lithol red

HSDB 5523,立索尔大红,PR-258,Barium lithol,1883 red

Others Others
Barium lithol red (HSDB 5523) 是一种透明的蓝色调红色颜料,主要应用于印墨着色。
T33647L Nesosteine Lithium

Nesosteine Lithium(84233-61-4 Free baes)

Nesosteine Lithium 是一种新型的粘液调节剂,对豚鼠 Herxheimer 微休克具有抑制作用且抑制卵清蛋白诱导的组胺在致敏动物气管中的释放。Nesosteine Lithium 能够保护致敏动物免受卵清蛋白诱导的支气管痉挛但对组胺和乙酰胆碱诱导的支气管痉挛无效。
T14979 Clavulanate lithium

Clavulanic acid lithium,克拉维酸锂

Antibacterial Microbiology/Virology
Clavulanate lithium (Clavulanic acid lithium) 是一种β-lactamase 的高效抑制剂,可作抗生素。
T27841 Lobeglitazone Sulfate

CKD501 Sulfate,CKD501,CKD-501 Sulfate,CKD 501 Sulfate,CKD 501,CKD-501,Lobeglitazone Sulfate. trade name Duvie, Chong Kun Dang

NOD Immunology/Inflammation; NF-κB
Lobeglitazone Sulfate(CKD-501 Sulfate) 是一种新型噻唑烷二酮,具有抗炎活性,抑制LPS诱导的NLRP3炎症小体活化和肝脏炎症,可用于研究 2 型糖尿病 (T2DM)。
T7435 Selitrectinib

LOXO-195

Trk receptor Tyrosine Kinase/Adaptors
Selitrectinib (LOXO-195) 是二代原肌凝蛋白相关激酶(TRK)抑制剂,能够作用于 TRKA (IC50:0.6 nM) 和 TRKC (IC50<2.5 nM)。
T22592 ATPγS tetralithium salt

ATP-gamma-S tetralithium salt

PERK Apoptosis
ATPγS tetralithium salt 是真核生物翻译起始因子 eIF4A 的核苷酸水解和RNA解链活性的底物,与 p97 突变体和朊病毒相关。
T0334 Rosiglitazone

BRL49653,罗格列酮

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone (BRL49653) 是一种 PPARγ 激动剂、TRPC5 激活剂和 TRPM3 抑制剂,具有口服活性。Rosiglitazone 也是一种降糖剂,是噻唑烷二酮类胰岛素增敏剂。
T12835 Saroglitazar

Lipaglyn

PPAR DNA Damage/DNA Repair; Metabolism
Saroglitazar (Lipaglyn) 是 PPAR 的激动剂,对 PPARα 和 PPARγ 的 EC50 值为 0.65 pM 和 3 nM。
T4639 Azemiglitazone

MSDC 0602

Mitochondrial Metabolism; mTOR Metabolism; PI3K/Akt/mTOR signaling
Azemiglitazone (MSDC 0602) 是一种 PPARγ 保留的噻唑烷二酮类药物 (TZD),与能够线粒体丙酮酸载体 (MPC) 相互作用并抑制其活性,降低 pparγ 介导的副作用的风险,有用于 2 型糖尿病研究的潜能。
T64334 Glycolithocholic acid, sodium salt

Others Others
Glycolithocholic acid, sodium salt 是 Glycolithocholic acid 的钠盐。Glycolithocholic acid 是一种甘氨酸结合的次级胆汁酸。Glycolithocholic acid 可用于诊断溃疡性结肠炎 (UC),非酒精性脂肪性肝炎 (NASH0) 和原发性硬化性胆管炎 (PSC)。
T26986 Cevoglitazar

LBM-642,LBM 642,LBM642

PPAR DNA Damage/DNA Repair; Metabolism
Cevoglitazar (LBM-642) 是一种 PPARɑ 激动剂和 PPARγ激动剂。Cevoglitazar 能有效减少肥胖小鼠和猴的食物摄入量和体重。
TP1299L1 Melittin Acetate

Melittin Acetate(20449-79-0 Free base),Forapin Acetate

Phospholipase Metabolism
Melittin Acetate (Forapin Acetate) 是一种PLA2激活剂。Melittin Acetate 低分子量 PLA2 的活性具有刺激,而不会增加高分子量 PLA2 的活性。

化合物

LIT-001
Cat.No: T11857
Synonym:
Target: Oxytocin Receptor
LIT927
Cat.No: T5207
Synonym: LIT 927,LIT-927
Target: CXCR
LIT-001 free base
Cat.No: T11856
Synonym:
Target: Others
Omeprazole metabolite Omeprazole sulfone
Cat.No: T12309
Synonym: Omeprazole sulphone,Omeprazole sulfone
Target: Others
MJ33 lithium salt
Cat.No: T38404
Synonym:
Target: ROS
Savolitinib
Cat.No: TQ0210
Synonym: AZD-6094,Volitinib,沃利替尼,赛沃替尼,HMPL-504
Target: c-Met/HGFR
Varlitinib
Cat.No: T6719
Synonym: ASLAN001,ARRY-334543
Target: HER
Splitomicin
Cat.No: T6678
Synonym: 1-Naphthalenepropanoic Acid,斯普利特麻一辛
Target: Sirtuin, HDAC
Inolitazone
Cat.No: T15581
Synonym: RS5444,Efatutazone,CS-7017,伊诺他酮
Target: PPAR
Melitracen hydrochloride
Cat.No: T4274
Synonym: 盐酸美利曲辛,盐酸美力他欣,Thymeol hydrochloride,Melixeran
Target: Dopamine Receptor, 5-HT Receptor
7-Troc-paclitaxel
Cat.No: T20864
Synonym:
Target: Others
Ruxolitinib
Cat.No: T1829
Synonym: 芦可替尼,INCB018424,鲁索替尼,(R)-Ruxolitinib
Target: Apoptosis, Mitophagy, Tyrosine Kinases, JAK, Autophagy
Isoallolithocholic acid
Cat.No: T36522
Synonym: Alloisolithocholic Acid,AILCA,3β-Hydroxy-5α-cholanic acid
Target: Others
Roblitinib
Cat.No: T4235
Synonym: FGF-401
Target: FGFR
Abemaciclib metabolite M20
Cat.No: T10738
Synonym: CDK4/6-IN-4,LSN3106726
Target: CDK
Methotrexate metabolite
Cat.No: T16045
Synonym: DAMPA,甲喋呤杂质E
Target: Antifolate, Drug Metabolite
Imiglitazar
Cat.No: T15567
Synonym: TAK-559
Target: PPAR
Isourolithin A
Cat.No: T125575
Synonym:
Target:
Litoxetine
Cat.No: T67956
Synonym:
Target: 5-HT Receptor
Troglitazone
Cat.No: T3170
Synonym: CS-045,Romozin,Rezulin,Romglizone,Noscal,Prelay,曲格列酮
Target: Apoptosis, Ferroptosis, PPAR, Autophagy
Pioglitazone hydrochloride
Cat.No: T0214L
Synonym: U-72107E,AD 4833,U 72107A,Pioglitazone HCl,匹格列酮盐酸盐
Target: Ferroptosis, PPAR
3,6-Dichlorotrimellitic anhydride
Cat.No: T18886
Synonym:
Target: Others
Ticagrelor metabolite M5
Cat.No: T21059
Synonym: Ticagrelor metabolite M5,,T437700,替格瑞洛杂质H,AR-C133913XX
Target: P2Y Receptor
Cinacalcet metabolite M4
Cat.No: T10814
Synonym: 3-三氟甲基苯丙胺,Rarechem AL BW 1078
Target: Calcium Channel
α-Hydroxyglutaric Acid Lithium
Cat.No: T36624L
Synonym: α-Hydroxyglutaric Acid Lithium(2889-31-8 Free base)
Target: Decarboxylase, Endogenous Metabolite, mTOR
Saroglitazar Magnesium
Cat.No: T12834
Synonym:
Target: Others
Pelitinib
Cat.No: T2327
Synonym: 培利替尼,EKB-569,WAY-EKB 569
Target: EGFR, Raf, MEK, Src
Lucifer Yellow CH dilithium salt
Cat.No: T15790
Synonym:
Target:
Peliglitazar racemate
Cat.No: T12400
Synonym: (Rac)-Peliglitazar,(Rac)-BMS 426707-01,BMS 426707-01 racemate
Target: PPAR
Indeglitazar
Cat.No: T15575
Synonym: PPM 204
Target: PPAR
Allitinib
Cat.No: T14336
Synonym: AST-1306,ALS 1306
Target: EGFR
Tesaglitazar
Cat.No: T17044
Synonym:
Target: PPAR
Darglitazone
Cat.No: T22708
Synonym: CP-86325
Target: PPAR
Aleglitazar
Cat.No: T14176
Synonym: RO0728804,R1439
Target: PPAR
Rosiglitazone maleate
Cat.No: T1622
Synonym: BRL 49653C,BRL 49653,马来酸罗格列酮
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
Seglitide acetate
Cat.No: T28743
Synonym: MK 678,MK678,MK-678
Target: Somatostatin
Ragaglitazar
Cat.No: T28501
Synonym: NNC61-0029,NN-622,(-)-DRF-2725,NNC-61-0029,NN 622,NNC 61-0029
Target: PPAR
Solithromycin
Cat.No: T2331
Synonym: 索利霉素,OP-1068,CEM-101
Target: Antibacterial, Antibiotic
Barium lithol red
Cat.No: T20018
Synonym: HSDB 5523,立索尔大红,PR-258,Barium lithol,1883 red
Target: Others
Nesosteine Lithium
Cat.No: T33647L
Synonym: Nesosteine Lithium(84233-61-4 Free baes)
Target:
Clavulanate lithium
Cat.No: T14979
Synonym: Clavulanic acid lithium,克拉维酸锂
Target: Antibacterial
Lobeglitazone Sulfate
Cat.No: T27841
Synonym: CKD501 Sulfate,CKD501,CKD-501 Sulfate,CKD 501 Sulfate,CKD 501,CKD-501,Lobeglitazone Sulfate. trade name Duvie, Chong Kun Dang
Target: NOD
Selitrectinib
Cat.No: T7435
Synonym: LOXO-195
Target: Trk receptor
ATPγS tetralithium salt
Cat.No: T22592
Synonym: ATP-gamma-S tetralithium salt
Target: PERK
Rosiglitazone
Cat.No: T0334
Synonym: BRL49653,罗格列酮
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
Saroglitazar
Cat.No: T12835
Synonym: Lipaglyn
Target: PPAR
Azemiglitazone
Cat.No: T4639
Synonym: MSDC 0602
Target: Mitochondrial Metabolism, mTOR
Glycolithocholic acid, sodium salt
Cat.No: T64334
Synonym:
Target: Others
Cevoglitazar
Cat.No: T26986
Synonym: LBM-642,LBM 642,LBM642
Target: PPAR
Melittin Acetate
Cat.No: TP1299L1
Synonym: Melittin Acetate(20449-79-0 Free base),Forapin Acetate
Target: Phospholipase
Cat. No. Product Name Target Signaling Pathways
T21165 Pellitorine

AI3-19560,墙草碱,Pellitorin

TRP/TRPV Channel Membrane transporter/Ion channel
Pellitorine (Pellitorin) 是提取自 Piper nigrum 的根的一种化合物。它对 HL60 和 MCT-7 细胞系表现出显著的细胞毒活性。它可用于癌症疾病的研究。
TQ0269 Melittoside

蜜力特苷,美利妥双甙

Antioxidant oxidation-reduction
Melittoside 是一种天然酚苷,存在于梅利藤属的花蜜中。它具有抗氧化、抗炎和抗真菌的活性,以及研究了它在治疗各种疾病中的潜在用途,包括癌症、糖尿病和心血管疾病。
T8299 Dimethyl lithospermate B

丹酚酸B二甲酯,dmLSB

Sodium Channel Membrane transporter/Ion channel
Dimethyl lithospermate B (dmLSB) 是 Na+通道的选择性激动剂,减缓钠电流 (INa) 失活,导致动作电位 (AP) 早期内向电流增加。
TN7030 Heteroclitin G

Others Others
Heteroclitin G 被发现是 KIS 补血活性的潜在生物标志物,定量分析为进一步药理研究提供了研究基础。
T20604L Litorin acetate(55749-97-8 Free base)

Bombesin Receptor GPCR/G Protein
Litorin acetate 是一种两栖类铃蟾肽衍生物,是一种铃蟾肽受体激动剂。它刺激平滑肌收缩,刺激胃泌素、胃酸和胰腺分泌,抑制体内营养。
T0968 Paclitaxel

Taxol,紫杉醇,NSC 125973

Apoptosis; Microtubule Associated; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling
Paclitaxel (Taxol) 属于天然产物,是一种微管聚合物稳定剂。Paclitaxel 具有抗肿瘤活性;通过诱导有丝分裂停滞、细胞凋亡、细胞自噬等,导致细胞死亡。
T3683 lithospermic acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
Lithospermic acid 是一种植物来源的多环酚类羧酸,从丹参中分离得到,对 CCl4诱导的急性和体外肝损伤具有抗氧化和保肝活性。
T5213 Acetyl phosphate(lithium potassium)

乙酰磷酸锂钾盐,Lithium potassium acetyl phosphate,Acetylphosphoric acid

Others; Endogenous Metabolite Metabolism; Others
Acetyl phosphate lithium potassium (Lithium potassium acetyl phosphate) 是内源性代谢产物的一种。
TN1722 Hamamelitannin

Antifection Microbiology/Virology
Hamamelitannin 是分离自 Hamamelis virginiana 树皮的一种多酚,是群体感应抑制剂。它通过影响肽聚糖生物合成和 eDNA 释放增加金黄色葡萄球菌生物膜的抗生素敏感性。
TN1513 Clitorin

碟豆宁,碟豆素

PKC; Antifection Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
Clitorin 是一种山奈酚糖苷,分离自 Acalypha indica 的花和叶,表现出抗氧化活性。
T1529 Miglitol

BAY1099,米格列醇,BAY-m1099

Others Others
Miglitol (BAY1099) 是一种口服抗糖尿病化合物,能够抑制糖复合体分解为葡萄糖。
T13522 7-Ketolithocholic acid

3α-Hydroxy-7-oxo-5β-cholanic acid

Endogenous Metabolite Metabolism
7-Ketolithocholic acid (3α-Hydroxy-7-oxo-5β-cholanic acid) (3α-Hydroxy-7-oxo-5β-cholanic acid) is capable of absorption and serves to suppress the production of endogenous bile acid and the secretion of biliary cholesterol.
T16338 Norgestimate metabolite Norelgestromin

17-Deacetyl norgestimate,17-Deacylnorgestimate,甲基孕酮

Drug Metabolite Metabolism
Norgestimate metabolite Norelgestromin (17-Deacylnorgestimate) 是norgestimate 的一种活性代谢物。它是用于避孕贴片的甾体孕激素,与雌激素乙炔雌二醇结合使用。
T3S1916 Heteroclitin D

异型南五味子丁素,异南五味子丁素;异型南五味子丁素

Calcium Channel Membrane transporter/Ion channel; Metabolism
Heteroclitin D 是异形南五味子中的一种木脂素,可抑制 L 型钙通道,具有抗脂质过氧化作用。
T5749 10-Deacetyl-7-xylosyl paclitaxel

10-Deacetyl-7-xylosyltaxol,10-Deacetyltaxol 7-Xyloside,7-Xylosyl-10-deacetyltaxol,7-木糖甙-10-脱乙酰基紫杉醇,10-Deacetylpaclitaxel 7-Xyloside

Others; Microtubule Associated Cytoskeletal Signaling; Others
10-Deacetyl-7-xylosyl paclitaxel (7-Xylosyl-10-deacetyltaxol) 是一种紫杉醇衍生物,具有改进的药理特性和更高的水溶性,用于治疗癌症。
T0589 Xylitol

木糖醇,Adonitol,Ribitol,Xylite,D-Xylitol,Adonite

Others; Endogenous Metabolite; Autophagy Autophagy; Metabolism; Others
Xylitol (Ribitol) 是一种五碳糖醇,通过还原羰基衍生自木糖。它和蔗糖一样甜,可用作防龋甜味剂。
T30969 Clitocine

Apoptosis; BCL Apoptosis
Clitocine 是一种来从蘑菇中提取的一种腺苷类似物,是一种有效的转录通读剂,是一种无义突变的抑制剂,具有抗癌活性,可诱导携带 p53 无义突变等位基因的细胞产生 p53 蛋白。Clitocine 通过促进 Mcl-1 降解来增强 TRAIL 介导的人结肠癌细胞凋亡。
TN7108 Urolithin C

Apoptosis; Calcium Channel; Reactive Oxygen Species; IGF-1R; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Tyrosine Kinase/Adaptors
Urolithin C 属于多酚类,是鞣花酸的肠道微生物代谢产物,具有胰岛素分泌的葡萄糖依赖性激活活性。Urolithin C 是 L 型 Ca2+通道开放剂,可增强 Ca2+的流入。它通过线粒体介导的途径诱导细胞凋亡,并刺激活性氧的形成。
T5738 7-Epi 10-desacetyl paclitaxel

10-Deacetyl-7-epipaclitaxel,7-Epi-10-deacetyltaxol,7-表-10-去乙酰基云南紫杉宁A

Others Others
7-Epi 10-desacetyl paclitaxel (10-Deacetyl-7-epipaclitaxel) 是紫杉醇衍生物,对 HeLa 细胞具有细胞毒性(IC50:85 μM)。
T35792 Isolithocholic Acid

3-Epilithocholic acid,3β-Hydroxy-5β-cholanic acid,β-Lithocholic acid,isoLCA

Endogenous Metabolite Metabolism
Isolithocholic Acid (3-Epilithocholic acid) (β-Lithocholic acid) 是石胆酸的一种同分异构体。Isolithocholic Acid 是一种胆酸,由 Lithocholic acid 或 Lithocholic acid 3α-sulfate 经微生物代谢形成。
T7174 Urolithin A

尿石素A,3,8-二羟基-6H-二苯并[B,D]吡喃-6-酮

Apoptosis; Reactive Oxygen Species; DNA/RNA Synthesis; Endogenous Metabolite; Autophagy; Drug Metabolite Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; NF-κB
Urolithin A 是一种鞣花酸的肠道微生物代谢产物,可诱导自噬和凋亡,抑制细胞周期进程,抑制DNA 合成,具有抗炎、抗增殖和抗氧化的特性。
TN1855 Laurolitsine

去甲异波尔定,(+)-Norboldine

Others Others
Laurolitsine ((+)-Norboldine) 是一种生物碱,从 Peumus boldusMolina 叶子中分离得到。
T13265 Urolithin B

尿石素B,3-羟基-6H-苯并[C]苯并吡喃-6-酮

ERK; NF-κB; Akt; Endogenous Metabolite; JNK; AMPK Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Urolithin B 是一种 ellagitannins 的肠道微生物代谢产物,具有抗炎和抗氧化作用。它也是骨骼肌质量的调节因子,通过减少 IκBα 的磷酸化和降解来抑制 NF-κB 活性,并抑制 JNK、ERK 和 Akt 的磷酸化,并增强 AMPK 的磷酸化。
T2202 Lithocholic acid

3α-Hydroxy-5β-cholanic acid,石胆酸

Apoptosis; Others; FXR; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism; Others
Lithocholic acid (3α-Hydroxy-5β-cholanic acid) 是由鹅去氧胆酸盐通过细菌作用形成的胆汁酸,通常与甘氨酸或牛磺酸结合,被用作利胆剂。 它作为清洁剂溶解脂肪以供吸收,并且本身被吸收。
T4727 Taurolithocholic acid sodium salt

牛磺石胆酸钠,Sodium taurolithocholate

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
T3756 Allitol

Allodulcit,蒜糖醇,Allodulcitol,d-allitol

Others Others
Allitol (d-allitol) 是一种罕见的可作为甜味剂天然多元醇。它是制备 azasugars 的重要中间体,可用于制备抗癌症、糖尿病及包括艾滋病在内的病毒感染的药物。
T3784 Lithospermoside

Griffonin,紫草氰苷

Others Others
Lithospermoside (Griffonin) 是一种分离自 Ochna schweinfurthiana F.Hoffm 茎皮中的天然产物。
T20793 Magnesium Lithospermate B

丹參酸B鎂,Monomethyl lithospermate B,丹参酸 B 镁,Lithospermate B

Others Others
Magnesium Lithospermate B 是一种咖啡酸四聚体的衍生物,从Salviae miltiorrhizae 中提取得到。它能够抑制神经炎症并减轻神经变性。它被广泛用于心血管疾病的研究,并且可以防止葡萄糖引起的细胞内氧化损伤。
T8878 urolithin M6

尿石素M6,3,8,9,10-tetrahydroxy urolithin

Others Others
urolithin M6 (3,8,9,10-tetrahydroxy urolithin) 是一种由肠道微生物群产生的鞣花单宁代谢物,被确定为推定的没食子黄素模拟物。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
T31964 Glycolithocholic acid

Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine

Others Others
Glycolithocholic acid (Lithocholic acid glycine conjugate) 属于内源性代谢产物,是甘氨酸结合的次级胆汁酸。它可用于诊断非酒精性脂肪性肝炎,溃疡性结肠炎和原发性硬化性胆管炎。
T8207 Evolitrine

Others Others
Evolitrine 是一种来源于Acronychia pedunculata、具有抗炎作用的物质。
TN1028 Militarine

Others Others
Militarine 是一种糖苷化合物,分离自 Bletilla striata,能够抑制植物生长。
TN4742 Patulitrin

Antifection Microbiology/Virology
Patulitrin has antioxidant, anti-inflammatory, and larvicidal activities, oral and topical administration of patuletin and patulitrin inhibited acute inflammation in mice.
TN3323 Monomethyl lithospermate

Lithospermic acid monomethyl ester

Akt; PI3K Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Monomethyl lithospermate (Lithospermic acid monomethyl ester) 具有潜在的抗病毒活性,通过激活PI5K/Akt信号传导,减轻体内大脑中动脉闭塞小鼠缺血性中风损伤,并在体外保护氧葡萄糖剥夺/复氧诱导的SHSY-3Y细胞。Monomethyl lithospermate 能提高 SHSY-5Y 细胞的生存能力,抑制线粒体膜电位 (MMOP) 崩溃,抑制细胞凋亡。Monomethyl lithospermate 还降低中动脉闭塞 (MCAO) 大鼠脑组织中的氧化应激水平,改善缺血性中风 (IS) 大鼠神经损伤。
T73758 Glycolithocholic acid 3-sulfate

Glycolithocholic acid 3-sulfate (SLCG) 为一种胆汁酸衍生物及甘胆酸的代谢产物,具有抑制HIV-1复制的作用。该化合物在HIV感染和胆囊疾病的研究中有潜在应用价值。
T78487 Laurolitsine hydrochloride

(+)-Norboldine hydrochloride

Laurolitsine hydrochloride,从台湾雅楠中分离得到的生物碱型化合物,表现出轻微的抗炎活性。
TN4444 Litseglutine B

Others Others
Litseglutine B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4444,CAS号为 25368-01-8。
T74005 Urolithin D

Urolithin D 是EphA 受体的竞争性可逆拮抗剂。Urolithin D 表现出类内选择性。
TN4639 Neolitsine

Others Others
Neolitsine has anthelmintic activity, it exhibits EC90 values (concentration at which 90% loss of larval motility is observed) of 6.4 microg/mL.Neolitsine and dicentrine have potent vasorelaxing effects on precontracted rat aortic preparations with mean IC 50 values between 0.08 and 2.48 microM.
T38478 Mevalonic acid 5-pyrophosphate tetralithium

Mevalonicacid5-diphosphatetetralithium,Mevalonic acid 5-pyrophosphate tetralithium,5-Diphosphomevalonic acid tetralithium

Mevalonic acid 5-pyrophosphate (also known as 5-Diphosphomevalonic acid) tetralithium is an endogenous metabolite involved in the mevalonate pathway.
T82209 Heteroclitin A

Heteroclitin A为一种可从五味子(Schisandra propinqua)茎部提取的木脂素。
TN3109 5-Epilithospermoside

Others Others
(-)-5-Epilithospermoside is proposed as a potential marker of botanical origin for phacelia honey.
TMA2563 Pedalitin

Tyrosinase Proteases/Proteasome
Pedalitin is a mixed-type inhibitor of tyrosinase. In the assay of α-glucosidase inhibition, rosmarinic acid is a competitive inhibitor, whereas both methyl rosmarinate and Pedalitin are mixed-type inhibitors.
TN1020 Monomelittoside

Danmelittoside,单密力特苷

Others Others
Monomelittoside (Danmelittoside) 是从中国蜜蜂的毒液中提取的一种化合物,属于黄酮类糖苷,已经发现它具有抗炎、抗肿瘤和抗糖尿病的特性,它也被证明对肝脏和肾脏有保护作用。
T4854 Acetoacetic acid lithium salt

LithoTab acetoacetate,Lithium acetoacetate,Lithium 3-Oxobutyrate,乙酰乙酸锂

Others; Endogenous Metabolite Metabolism; Others
Acetoacetic acid lithium salt (Lithium 3-Oxobutyrate) 是内源性代谢产物的一种。
T32799 Lithospermidin B

Lithospermidin B is a minor pigment isolated from the roots of L. erythrorhizon.
TN4207 Heteroclitin B

Others Others
Heteroclitin B是一种天然产物,属于五味子科南五味子属,其产品编号为 TN4207,CAS号为 140461-47-8。Heteroclitin B可用作对照参考。
TN4208 Heteroclitin C

Others Others
Heteroclitin C is a natural product from Kadsura heteroclita.
TN5531 Eupalitin

3,5,4'-Trihydroxy-6,7-dimethoxyflavone

Eupalitin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5531,CAS号为 29536-41-2。
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天然产物

Pellitorine
Cat.No: T21165
Synonym: AI3-19560,墙草碱,Pellitorin
Target: TRP/TRPV Channel
Melittoside
Cat.No: TQ0269
Synonym: 蜜力特苷,美利妥双甙
Target: Antioxidant
Dimethyl lithospermate B
Cat.No: T8299
Synonym: 丹酚酸B二甲酯,dmLSB
Target: Sodium Channel
Heteroclitin G
Cat.No: TN7030
Synonym:
Target: Others
Litorin acetate(55749-97-8 Free base)
Cat.No: T20604L
Synonym:
Target: Bombesin Receptor
Paclitaxel
Cat.No: T0968
Synonym: Taxol,紫杉醇,NSC 125973
Target: Apoptosis, Microtubule Associated, Autophagy
lithospermic acid
Cat.No: T3683
Synonym:
Target: HIV Protease
Acetyl phosphate(lithium potassium)
Cat.No: T5213
Synonym: 乙酰磷酸锂钾盐,Lithium potassium acetyl phosphate,Acetylphosphoric acid
Target: Others, Endogenous Metabolite
Hamamelitannin
Cat.No: TN1722
Synonym:
Target: Antifection
Clitorin
Cat.No: TN1513
Synonym: 碟豆宁,碟豆素
Target: PKC, Antifection
Miglitol
Cat.No: T1529
Synonym: BAY1099,米格列醇,BAY-m1099
Target: Others
7-Ketolithocholic acid
Cat.No: T13522
Synonym: 3α-Hydroxy-7-oxo-5β-cholanic acid
Target: Endogenous Metabolite
Norgestimate metabolite Norelgestromin
Cat.No: T16338
Synonym: 17-Deacetyl norgestimate,17-Deacylnorgestimate,甲基孕酮
Target: Drug Metabolite
Heteroclitin D
Cat.No: T3S1916
Synonym: 异型南五味子丁素,异南五味子丁素;异型南五味子丁素
Target: Calcium Channel
10-Deacetyl-7-xylosyl paclitaxel
Cat.No: T5749
Synonym: 10-Deacetyl-7-xylosyltaxol,10-Deacetyltaxol 7-Xyloside,7-Xylosyl-10-deacetyltaxol,7-木糖甙-10-脱乙酰基紫杉醇,10-Deacetylpaclitaxel 7-Xyloside
Target: Others, Microtubule Associated
Xylitol
Cat.No: T0589
Synonym: 木糖醇,Adonitol,Ribitol,Xylite,D-Xylitol,Adonite
Target: Others, Endogenous Metabolite, Autophagy
Clitocine
Cat.No: T30969
Synonym:
Target: Apoptosis, BCL
Urolithin C
Cat.No: TN7108
Synonym:
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species, IGF-1R, Endogenous Metabolite
7-Epi 10-desacetyl paclitaxel
Cat.No: T5738
Synonym: 10-Deacetyl-7-epipaclitaxel,7-Epi-10-deacetyltaxol,7-表-10-去乙酰基云南紫杉宁A
Target: Others
Isolithocholic Acid
Cat.No: T35792
Synonym: 3-Epilithocholic acid,3β-Hydroxy-5β-cholanic acid,β-Lithocholic acid,isoLCA
Target: Endogenous Metabolite
Urolithin A
Cat.No: T7174
Synonym: 尿石素A,3,8-二羟基-6H-二苯并[B,D]吡喃-6-酮
Target: Apoptosis, Reactive Oxygen Species, DNA/RNA Synthesis, Endogenous Metabolite, Autophagy, Drug Metabolite
Laurolitsine
Cat.No: TN1855
Synonym: 去甲异波尔定,(+)-Norboldine
Target: Others
Urolithin B
Cat.No: T13265
Synonym: 尿石素B,3-羟基-6H-苯并[C]苯并吡喃-6-酮
Target: ERK, NF-κB, Akt, Endogenous Metabolite, JNK, AMPK
Lithocholic acid
Cat.No: T2202
Synonym: 3α-Hydroxy-5β-cholanic acid,石胆酸
Target: Apoptosis, Others, FXR, Endogenous Metabolite, Autophagy
Taurolithocholic acid sodium salt
Cat.No: T4727
Synonym: 牛磺石胆酸钠,Sodium taurolithocholate
Target: Others, Calcium Channel
Allitol
Cat.No: T3756
Synonym: Allodulcit,蒜糖醇,Allodulcitol,d-allitol
Target: Others
Lithospermoside
Cat.No: T3784
Synonym: Griffonin,紫草氰苷
Target: Others
Magnesium Lithospermate B
Cat.No: T20793
Synonym: 丹參酸B鎂,Monomethyl lithospermate B,丹参酸 B 镁,Lithospermate B
Target: Others
urolithin M6
Cat.No: T8878
Synonym: 尿石素M6,3,8,9,10-tetrahydroxy urolithin
Target: Others
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Glycolithocholic acid
Cat.No: T31964
Synonym: Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine
Target: Others
Evolitrine
Cat.No: T8207
Synonym:
Target: Others
Militarine
Cat.No: TN1028
Synonym:
Target: Others
Patulitrin
Cat.No: TN4742
Synonym:
Target: Antifection
Monomethyl lithospermate
Cat.No: TN3323
Synonym: Lithospermic acid monomethyl ester
Target: Akt, PI3K
Glycolithocholic acid 3-sulfate
Cat.No: T73758
Synonym:
Target:
Laurolitsine hydrochloride
Cat.No: T78487
Synonym: (+)-Norboldine hydrochloride
Target:
Litseglutine B
Cat.No: TN4444
Synonym:
Target: Others
Urolithin D
Cat.No: T74005
Synonym:
Target:
Neolitsine
Cat.No: TN4639
Synonym:
Target: Others
Mevalonic acid 5-pyrophosphate tetralithium
Cat.No: T38478
Synonym: Mevalonicacid5-diphosphatetetralithium,Mevalonic acid 5-pyrophosphate tetralithium,5-Diphosphomevalonic acid tetralithium
Target:
Heteroclitin A
Cat.No: T82209
Synonym:
Target:
5-Epilithospermoside
Cat.No: TN3109
Synonym:
Target: Others
Pedalitin
Cat.No: TMA2563
Synonym:
Target: Tyrosinase
Monomelittoside
Cat.No: TN1020
Synonym: Danmelittoside,单密力特苷
Target: Others
Acetoacetic acid lithium salt
Cat.No: T4854
Synonym: LithoTab acetoacetate,Lithium acetoacetate,Lithium 3-Oxobutyrate,乙酰乙酸锂
Target: Others, Endogenous Metabolite
Lithospermidin B
Cat.No: T32799
Synonym:
Target:
Heteroclitin B
Cat.No: TN4207
Synonym:
Target: Others
Heteroclitin C
Cat.No: TN4208
Synonym:
Target: Others
Eupalitin
Cat.No: TN5531
Synonym: 3,5,4'-Trihydroxy-6,7-dimethoxyflavone
Target:
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Cat. No. Product Name Species Expression System
TMPY-04722 DcR1/TRAILR3 Protein, Human, Recombinant (His)

TRAILR3,TRID,DCR1,TRAIL-R3,CD263,DCR1-TNFR,tumor necrosis fa...

Human HEK293 Cells
TNFRSF10C CNV in patients with CRC is associated with distant metastatic disease. A high frequency of CGI methylation in the TNFRSF10C promoter results in inactivation of the gene and enhancement of tumor growth in most PC cell lines (except CFPAC-1). Inactivation of TNFRSF10C by CpG island (CGI) hypermethylation can play an important role in PC progression and be potentially useful as a diagnostic marker and a new therapeutic approach for PC.
TMPY-03058 SLITL2/VASN Protein, Human, Recombinant (His)

SLITL2,vasorin

Human HEK293 Cells
Vasorin is a typical type I membrane protein. It contains 1 EGF-like domain, 1 fibronectin type-III domain, 10 LRR (leucine-rich) repeats, 1 LRRCT domain and 1 LRRNT domain. Vasorin is predominantly expressed in vascular smooth muscle cells, and that its expression is developmentally regulated. vasorin It directly binds to transforming growth factor (TGF)-β and attenuates TGF-β signaling in vitro. This suggests that down-regulation of vasorin expression contributes to neointimal formation after ...
TMPH-03716 Invasin Protein, Yersinia enterocolitica, Recombinant (His & SUMO)

Yersinia enterocolitica E. coli
Invasin is a protein that allows enteric bacteria to penetrate cultured mammalian cells. The entry of invasin in the cell is mediated by binding several beta-1 chain integrins.
TMPY-00922 SLITRK1 Protein, Human, Recombinant (His & hFc)

KIAA0918,KIAA1910,SLIT and NTRK like family member ...

Human HEK293 Cells
SLITRK1 Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 95 kDa and the accession number is Q96PX8.
TMPH-03720 YscM Protein, Yersinia enterocolitica, Recombinant (His & SUMO)

Yersinia enterocolitica E. coli
Belongs to an operon involved in the translocation of Yop proteins across the bacterial membranes or in the specific control of this function.
TMPY-00923 SLITRK1 Protein, Human, Recombinant (His)

TTM,FLJ54428,LRRC12,RP11-395N17.1,KIAA0918,SLITRK1,...

Human HEK293 Cells
SLITRK1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 105-115 kDa and the accession number is Q96PX8.
TMPH-03715 Y-STB Protein, Yersinia enterocolitica, Recombinant (His & SUMO)

Yersinia enterocolitica E. coli
Toxin which activates the particulate form of guanylate cyclase and increases cyclic GMP levels within the host intestinal epithelial cells. Could play an important role in pathogenesis.
TMPY-03063 SLITRK6 Protein, Human, Recombinant (His)

SLIT and NTRK like family member 6,SLITRK6...

Human HEK293 Cells
SLITRK6 belongs to the SLITRK family. Members of this family share two conserved leucine-rich repeat domains in the extracellular domain. SLITRK6 contains 11 LRR (leucine-rich) repeats, 2 LRRCT domains and 2 LRRNT domains. Expression of SlITRK proteins is highly restricted to neural and brain tumor tissues, but varies within the protein family. SLITRK6 is highly expressed in putamen with no expression in cerebral cortex. It also can be detected in adult and fetal lung and fetal liver. It can sup...
TMPY-02484 SLITRK4 Protein, Human, Recombinant (His)

DKFZp547M2010,SLIT and NTRK like family member 4

Human HEK293 Cells
SLIT and NTRK-like family proteins 4 is a member of the SLIT and NTRK-like family. This protein is characterized as an integral membrane protein that has two leucine-rich repeat (LRR) domains and a carboxy-terminal domain that is partially similar to SLIT protein and TRK Neurotrophin There are six members in this family: SLITRK1, SLITRK2, SLITRK3, SLITRK4, SLITRK5, and SLITRK6. Their expression was detected mainly in the brain, but the expression profile of each SLITRK was unique. Each of these ...
TMPH-03719 YopH Protein, Yersinia enterocolitica, Recombinant (His & Myc)

Yersinia enterocolitica E. coli
Essential virulence determinant. This protein is a protein tyrosine phosphatase. The essential function of YopH in Yersinia pathogenesis is host-protein dephosphorylation. It contributes to the ability of the bacteria to resist phagocytosis by peritoneal macrophages.
TMPH-03718 YopB Protein, Yersinia enterocolitica, Recombinant (His)

Yersinia enterocolitica E. coli
Plays a role in virulence.
TMPH-02364 Japanese encephalitis virus Genome polyprotein (His & SUMO)

JEV E. coli
Japanese encephalitis virus Genome polyprotein (His & SUMO) is expressed in E. coli.
TMPY-04234 Influenza A H17N10 (A/little yellow-shouldered bat/Guatemala/164/2009) Hemagglutinin/HA1 Protein (His)

Harvey rat sarcoma viral oncogene homolog

H17N10 HEK293 Cells
Influenza A H17N10 (A/little yellow-shouldered bat/Guatemala/164/2009) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.7 kDa and the accession number is H6QM73.
TMPH-02763 Lithostathine-1/Reg1 Protein, Mouse, Recombinant (His & SUMO)

Mouse E. coli
Lithostathine-1/Reg1 Protein, Mouse, Recombinant (His & SUMO) is expressed in E. coli.
TMPY-04652 Influenza A H17N10 (A/little yellow-shouldered bat/Guatemala/164/2009) Hemagglutinin/HA Protein (His)

Harvey rat sarcoma viral oncogene homolog

H17N10 Baculovirus Insect Cells
Influenza A H17N10 (A/little yellow-shouldered bat/Guatemala/164/2009) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 59 kDa and the accession number is H6QM73.
TMPH-03717 YopE Protein, Yersinia enterocolitica, Recombinant (His)

Yersinia enterocolitica E. coli
Essential virulence determinant; cytotoxic effector, involved in resistance to phagocytosis.

重组蛋白

DcR1/TRAILR3 Protein, Human, Recombinant (His)
Cat.No: TMPY-04722
Species: Human
Expression System: HEK293 Cells
SLITL2/VASN Protein, Human, Recombinant (His)
Cat.No: TMPY-03058
Species: Human
Expression System: HEK293 Cells
Invasin Protein, Yersinia enterocolitica, Recombinant (His & SUMO)
Cat.No: TMPH-03716
Species: Yersinia enterocolitica
Expression System: E. coli
SLITRK1 Protein, Human, Recombinant (His & hFc)
Cat.No: TMPY-00922
Species: Human
Expression System: HEK293 Cells
YscM Protein, Yersinia enterocolitica, Recombinant (His & SUMO)
Cat.No: TMPH-03720
Species: Yersinia enterocolitica
Expression System: E. coli
SLITRK1 Protein, Human, Recombinant (His)
Cat.No: TMPY-00923
Species: Human
Expression System: HEK293 Cells
Y-STB Protein, Yersinia enterocolitica, Recombinant (His & SUMO)
Cat.No: TMPH-03715
Species: Yersinia enterocolitica
Expression System: E. coli
SLITRK6 Protein, Human, Recombinant (His)
Cat.No: TMPY-03063
Species: Human
Expression System: HEK293 Cells
SLITRK4 Protein, Human, Recombinant (His)
Cat.No: TMPY-02484
Species: Human
Expression System: HEK293 Cells
YopH Protein, Yersinia enterocolitica, Recombinant (His & Myc)
Cat.No: TMPH-03719
Species: Yersinia enterocolitica
Expression System: E. coli
YopB Protein, Yersinia enterocolitica, Recombinant (His)
Cat.No: TMPH-03718
Species: Yersinia enterocolitica
Expression System: E. coli
Japanese encephalitis virus Genome polyprotein (His & SUMO)
Cat.No: TMPH-02364
Species: JEV
Expression System: E. coli
Influenza A H17N10 (A/little yellow-shouldered bat/Guatemala/164/2009) Hemagglutinin/HA1 Protein (His)
Cat.No: TMPY-04234
Species: H17N10
Expression System: HEK293 Cells
Lithostathine-1/Reg1 Protein, Mouse, Recombinant (His & SUMO)
Cat.No: TMPH-02763
Species: Mouse
Expression System: E. coli
Influenza A H17N10 (A/little yellow-shouldered bat/Guatemala/164/2009) Hemagglutinin/HA Protein (His)
Cat.No: TMPY-04652
Species: H17N10
Expression System: Baculovirus Insect Cells
YopE Protein, Yersinia enterocolitica, Recombinant (His)
Cat.No: TMPH-03717
Species: Yersinia enterocolitica
Expression System: E. coli
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