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1421

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T33876L Panomifene HCl

EGIS5650 HCl,GYKI 13504 HCl,Panomifene HCl(77599-17-8 Free base),EGIS 5650 HCl

HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Panomifene HCl 是一种选择性抗雌激素化合物,具有抗肿瘤活性,可用于治疗乳腺癌。
T2310L CHIR-99021 HCl

CT99021 HCl,Laduviglusib HCl

GSK-3 PI3K/Akt/mTOR signaling; Stem Cells
CHIR-99021 HCl (Laduviglusib HCl) 是GSK-3α/β的高效选择性抑制剂,IC50值分别为10 nM和6.7 nM。它对GSK-3表现出显著的选择性,对CDC2、ERK2和其他蛋白激酶的选择性超过500倍。此外,CHIR-99021 HCl 是Wnt/β-catenin信号通路的强大激活剂。此外,它在小鼠和人类胚胎干细胞中都表现出增强自我更新的能力。此外,拉杜维格西单盐酸盐诱导自噬[1][2][3]。
T21319L Gimatecan HCl

ST1481 HCL,Gimatecan HCl(292618-32-7 Free base)

Topoisomerase DNA Damage/DNA Repair
Gimatecan HCl (ST1481 HCL) 是一种有效的拓扑异构酶 I (topoisomerase I) 抑制剂。Gimatecan HCl 是一种具有口服活性的喜树碱类似物。具有抗肿瘤活性。
T11227L1 Eravacycline HCl

Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl

Antibiotic Microbiology/Virology
Eravacycline HCl (TP-434 HCl) 是一种具有广谱抗菌活性的强效抗生素。
T13254L UNC10217938A HCl

UNC10217938A HCl(1347749-97-6 Free base),UNC7938 HCl

Others Others
UNC10217938A HCl (UNC7938 HCl) 是具有寡核苷酸 (oligonucleotides) 增强作用的 3-deazapteridine 类似物, 通过调节寡核苷酸在细胞内的运输和从内体中的释放来增强寡核苷酸的作用。UNC10217938A HCl 还增强了 siRN 和反义寡核苷酸的作用。
T80662 CDD0102 HCl

CDD0102A HCl

AChR Neuroscience
CDD0102 HCl 是一种具有选择性和有效的 M1 毒蕈碱 (Muscarinic) 受体激动剂,可用于治疗阿尔兹海默症。
T11497 Ganfeborole HCl

GSK3036656 HCl,GSK656 HCl

Antibacterial Microbiology/Virology
Ganfeborole HCl (GSK3036656 HCl) 是一种具有抗结核活性的小分子化合物,是结核分枝杆菌(Mtb)亮氨酰-tRNA 合成酶(LeuRS;IC50:0.2 μM)的抑制剂。
T30188L Atagabalin HCl

PD-0200390 HCl,Atagabalin HCl(223445-75-8 Free base)

Calcium Channel Membrane transporter/Ion channel; Metabolism
Atagabalin HCl 是一种新型电压依赖性钙通道(VDCC)α2δ亚基(1 和 2)配体,会影响慢波睡眠,可用于治疗失眠。
T33711L Nolomirole HCl

CHF 1035 HCl,CHF 1035,CHF1035,CHF1035 HCl,CHF-1035 HCl,CHF-1035,Nolomirole Hydrochloride

Dopamine Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Nolomirole HCl(CHF 1035) 是一种具有口服活性的新型选择性多巴胺激动剂,对去甲肾上腺素的释放有抑制作用,可用于研究轻度慢性心力衰竭。
T10290L Alpertine HCl

Win 31665 HCl,Alpertine HCl(27076-46-6 Free base)

Others Others
Alpertine HCl 是一种小分子化合物,具有抗神经病作用。
T3465L Vesnarinone HCl

Synonym 2,OPC-8212 HCl,Vesnarinone HCl(81840-15-5 Free base)

Potassium Channel; Calcium Channel; PDE Membrane transporter/Ion channel; Metabolism
Vesnarinone HCl (OPC-8212 HCl) 是一种具有口服活性的 phosphodiesterase 3 (PDE3) 抑制剂。Vesnarinone HCl 可对钙离子和钾离子进行调节, 增加钙通量,减少钾通量。Vesnarinone HCl 是一种新的正性肌力化合物,可增强心肌收缩力,可用于心力衰竭的研究。
T30077L Anisperimus HCl

LF 150195 HCl,Anisperimus HCl(170368-04-4 Free base)

Others Others
Anisperimus HCl (LF 150195 HCl)是一种小分子免疫制剂,可用于研究自身免疫性疾病。
T24797 SK609 HCl

SK-609 HCl,SK609 hydrochloride,SK 609 HCl,SK 609 hydrochloride,SK-609 hydrochloride

SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.
T31221L dBRD9 HCl

dBRD9 HCl(2170679-45-3 Free base)

Epigenetic Reader Domain Chromatin/Epigenetic
dBRD9 HCl 是一种PROTAC,包含cereblon E3连接酶配体与BRD9抑制剂BI 7273。dBRD9 HCl 是有效和选择性的BRD9降解剂,在MOLM-13细胞中IC50的为56.6nM。dBRD9 HCl 在浓度高达5μM 时不会降解BRD4或BRD7。dBRD9 HCl 在人AML 细胞系中显示出抗增殖作用。
T27947L LY339434 HCl

LY339434 HCl(219566-62-8 Free base)

GluR; NMDAR Neuroscience
LY339434 HCl是一种亲和力很低的GluR5红氨酸受体激动剂。LY339434 HCl 主要通过影响 N-甲基-D-天冬氨酸(NMDA)受体来快速的神经元死亡。
T36404L PRLX-93936 HCL

PRLX-93936 hcl(903499-49-0 Free base)

Ferroptosis; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB
PRLX-93936 HCL 是 erastin 的类似物,并显示出与顺铂对非小细胞肺癌 (NSCLC) 细胞的协同作用。
T68050L Dazolicin HCl

Dazolicine HCl,Dazolicine hydrochloride

Others Others
Dazolicin HCl (Dazolicine HCl) 是一种可口服的抗心律失常化合物。
T67956L Litoxetine HCl

litoxetine HCL(86811-09-8 Free base)

5-HT Receptor GPCR/G Protein; Neuroscience
Litoxetine HCl 是一种选择性5-羟色胺(5-HT)再摄取抑制剂(SSRI)和混合5-羟色胺拮抗剂,可用于治疗尿失禁。Litoxetine HCl 在没有抗毒蕈碱特性的浓度下(10 nM-1 microM)引起大鼠离体食道肌肉粘膜的浓度依赖性松弛,使卡巴胆碱张力降低达37%,更高浓度的Litoxetine HCl(3微摩-300微摩)与明显的松弛有关,直至取消卡巴胆碱张力。以前在离体豚鼠肠道中证明的利托西汀的抗心律失常活性,在浓度大于1 microM 时在大鼠离体食道肌肉粘膜中发挥了作用。 Litoxetine HCl 的5-HT 释放作用可以解释利托西汀对未处理的大鼠组织中的5-HT 诱导的松弛的效力,这种效力被pCPA 处理所逆转。
T27342L Flurocitabine HCl

Flurocitabine HCl(37717-21-8 Free base)

Others Others
Flurocitabine HCl 是阿糖胞苷的氟化酸酐类似物,在体内部分水解成两种活性抗肿瘤物质 (阿拉伯糖基-氟尿嘧啶 (ara-FC) 和阿拉伯糖基-氟尿嘧啶 (ara-FU))。Flurocitabine HCl 在急性白血病和实体瘤的 I 期研究中具显示出抗肿瘤活性。
T68151L Tallimustine HCl

Tallimustine HCl(115308-98-0 Free base)

DNA DNA Damage/DNA Repair
Tallimustine HCl 是一种DNA 抑制剂,是二霉素的AT 特异性烷化抗肿瘤衍生物。Tallimustine HCl 可用于成人骨髓性白血病的严重联合免疫缺陷小鼠模型,可用于治疗白血病。
T29067L Upacicalcet HCl

Upacicalcet HCl(1333218-50-0 Free base)

CaSR GPCR/G Protein
Upacicalcet HCl 是一种静脉内拟钙剂,通过直接作用于甲状旁腺细胞膜钙敏感受体来抑制过量的甲状旁腺激素 (PTH) 分泌,从而降低血液中的 PTH 水平。Upacicalcet HCl 可用于治疗血液是一种新型继发性甲状旁腺功能亢进化合物,靶向钙敏感受体的氨基酸结合位点。
T11839L Lesopitron HCl

Lesopitron HCl(132449-89-9 Free base)

5-HT Receptor GPCR/G Protein; Neuroscience
Lesopitron HCl 是一种5-HT1A 受体激动剂,具有抗焦虑化作用,可逆转与小鼠可卡因戒断相关的黑暗回避行为。
T30586L Brefonalol HCl

Brefonalol HCl(103880-26-8 Free base)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Brefonalol HCl 是一种 ADRA 拮抗剂,可用于治疗神经系统疾病和心血管疾病,可用于研究心绞痛、心律失常和高血压。
T68108L Moxilubant HCl

Moxilubant hcl(146978-48-5 Free base)

LTR Immunology/Inflammation
Moxilubant HCl 是一种小分子白三烯 B4 受体 1(LTB4R)拮抗剂,可用于治疗免疫系统疾病、皮肤和肌肉骨骼疾病,可用于研究银屑病和类风湿关节炎。
T27307L Fasnall HCl

Fasnall HCl(929978-58-5 Free base)

Fatty Acid Synthase Metabolism
Fasnall HCl 是一种FASN 选择性抑制剂,通过其辅助因子结合位点起作用。Fasnall HCl 在HER2(+)乳腺癌MMTV-Neu 模型中也显示出强大的抗肿瘤活性,特别是与卡铂联合使用时。
T6960L PU-H71 HCl

PU-H71 HCl(873436-91-0 Free base),Zelavespib HCl

HSP; DNA/RNA Synthesis Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism
PU-H71 HCl (Zelavespib HCl) 是一种新型Hsp90抑制剂,是一种新型嘌呤基类似物,也是一种可能是CIRT的一种有前途的放射增敏剂。PU-H71 HCL 在许多恶性肿瘤临床前模型中显示出抗肿瘤活性。PU-H71 HCL 对 Rad51 和Ku70 的蛋白表达水平有抑制作用,这可能与双链断裂修复的同源重组途径和非同源末端连接途径有关。
T67888L Samidorphan HCl

Samidorphan HCl(852626-89-2 free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Samidorphan HCl 是一种具有口服活性和高效性的 opioid 系统调节剂,可与 μ‐opioid、 κ‐opioid 和 δ‐opioid 受体结合。Samidorphan HCl 是一种新型 μ‐opioid 受体拮抗剂,是 k-opioid 受体和 δ‐opioid 受体的部分激动剂。Samidorphan HCl 可用于预防和治疗精神分裂。
T28145 ND-322 HCl

ND 322 Hydrochloride,ND322 Hydrochloride,ND-322 Hydrochloride,ND322 HCl

MMP Proteases/Proteasome
ND-322 HCl (ND 322 Hydrochloride) 是 MT1-MMP 和 MMP2 的选择性抑制剂,可减少体外黑色素瘤细胞的生长、迁移和侵袭。
T9670L Patamostat HCl

Patamostat HCl(114568-26-2 Free base)

Serine Protease; Protease Proteases/Proteasome
Patamostat HCl 是一种具有高效性和选择性的小分子蛋白酶 (protease) 抑制剂,对胰蛋白酶,纤溶酶和凝血酶有抑制作用,IC50 值分别为 39 nM,950 nM 和 1.9 μM。Patamostat HCl 可用于研究急性胰腺炎。
T26631L Anidoxime HCl

USVP-E142,Anidoxime HCl( 34297-34-2 Free base)

Anidoxime HCl (USVP-E142) 是一种新型可口服的具有抗镇痛活性的化合物。
T27267 ENMD-1068 HCl

ENMD-1068 HCl,ENMD 1068,ENMD-1068,ENMD1068,ENMD-1068 hydrochloride

Protease-activated Receptor GPCR/G Protein
ENMD-1068 HCl (ENMD 1068) 是一种选择性蛋白酶激活受体(PAR-2)拮抗剂,具有抗血管生成和抗炎活性。
T68171L Zabicipril HCl

Zabicipril HCl(83059-56-7 Free base),S 9650,S 10211

Angiotensin-converting Enzyme (ACE) Metabolism
Zabicipril HCl(S 9650) 是一种有效的血管紧张素转换酶抑制剂。
T68114L Nardeterol HCl

Nardeterol HCl(73865-18-6 Free base)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Nardeterol HCl 是一种 β肾上腺素能受体部分激动剂,可用于研究中枢神经系统。
T68135L (Rac)-Sabcomeline HCl

sabcomeline HCl(149156-36-5 Free base)

AChR Neuroscience
Sabcomeline HCl 是一种 M1 receptor 激动剂,可用于研究阿尔茨海默病。
T68182L 3-Hydroxykynurenamine HCl

3-OH-Kynurenamine HCl,3-Hydroxykynurenamine HCl(99362-47-7 Free base)

Others Others
3-Hydroxykynurenamine HCl (3-OH-Kynurenamine HCl) 是一种免疫调节生物胺,是氨基酸分解代谢的中间体,可诱导氧化损伤和促进细胞死亡。
T31931L Gizzerosine HCl

Gizzerosine HCl(89238-78-8 Free base)

Others Others
Gizzerosine HCl 是鱼粉热处理过程中产生的一种物质,可诱导的肉鸡雏鸡组织病理学病变,可提高离体鸡原产鸡的细胞内环腺苷-3',5'-单磷酸水平。
T28453L Propiram fumarate HCl

Propiram fumarate HCl(15686-91-6 Free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Propiram fumarate HCl是一种可口服的Opioid receptors激动剂,具有镇痛活性,可用于研究肌肉骨骼疼痛。
T63351L MS8511 HCl

MS8511 HCl(2866408-21-9 Free base)

Histone Methyltransferase Chromatin/Epigenetic
MS8511 HCl 是一种具有选择性和有效性的 G9a/GLP 共价抑制剂,通过靶向底物结合位点的半胱氨酸残基发挥作用。 MS8511 具有抗癌活性和抗增殖活性,可降低细胞内 H3K9me2 水平。MS8511 可用于研究包括脑癌、乳腺癌、卵巢癌在内的多种癌症。
T4013 SGC2085 HCl

Histone Methyltransferase Chromatin/Epigenetic
SGC2085 HCl 是一种有效的选择性辅激活剂相关的精氨酸甲基转移酶 1 (CARM1) 抑制剂,IC50 为 50 nM,选择性比其他 PRMT 高出数倍。 CARM1 是结直肠癌中 Wnt/β-catenin 转录和肿瘤转化的重要正调节因子,也是雌激素刺激的乳腺癌生长的关键因素,其耗竭导致体内髓性白血病细胞增殖减少。
T72058L CDD-1102 HCl

CDD-1102 HCl(2757619-84-2 Free base)

Epigenetic Reader Domain Chromatin/Epigenetic
CDD-1102 HCl 是一种新型BRDT-BD4 / BRD2-BD1302选择性抑制剂,在体内外实验中显示出非激素避孕潜力。
T68120L Ot-730 HCl

Ot-730 HCl(870809-51-1 Free base)

Others Others
ot-730 HCl 是一种新型选择性β阻滞剂前药,可用于研究眼部疾病。
T26339L XR-11576 HCl

XR-11576 HCl(346689-77-8 Free base)

Topoisomerase DNA Damage/DNA Repair
XR-11576 HCl 是一种新型口服活性拓扑异构酶I 和II 双重抑制剂,具有抗肿瘤活性。
T23288L (S)-3,4-DCPG HCl

(S)-3,4-Dicarboxyphenylglycine HCl,(S)-3,4-DCPG HCl(201730-11-2 Free base)

GluR Neuroscience
(S)-3,4-DCPG HCl ((S)-3,4-Dicarboxyphenylglycine HCl) 是一种具有选择性的代谢型谷氨酸受体 8a (mGluR8a) 激动剂,对表达人类 mGluR8 的 AV12-664 细胞有一种作用,其 EC50 为 31 nM。
T68067L Etilefrine pivalate HCl

Etilefrine pivalate HCl(100696-30-8 Free base)

Etilefrine pivalate HCl 是一种具有口服活性的化合物,可用于治疗偏头痛。
T30188L1 (Iso)-Atagabalin HCl

(Iso)-Atagabalin HCl((Iso)-223445-75-8)

Others Others
(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) 是一种可用于治疗非恢复性睡眠的α -2- δ配体。
T28273L OT-551 HCl

OT-551 HCl(627085-11-4 Free base)

NF-κB NF-κB
OT-551 HCl 是一种 NF-Κb 抑制剂,是一种具有抗氧化特性的二取代羟胺可用于治疗白内障和老年性黄斑变性和地域性萎缩 (GA)。
T11402L GKI-1 HCl

GKI-1 HCl( 2444764-03-6 Free base)

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
GKI-1 HCl 是 Greatwall (GWL)激酶抑制剂,对hGWLFL 和hGWL-KinDom 有抑制作用。GKI-1 HCl 对 ROCK1抑制作用较为显著。
T68037L CBS-1114 HCl

N-Phenylbenzamidrazone hydrochloride,cbs-1114 HCl(46721-85-1 Free base)

Lipoxygenase Metabolism
CBS-1114 HCl (N-Phenylbenzamidrazone hydrochloride) 是一种5-脂氧合酶抑制剂,是一种良好眼睛渗透型号的抗炎化合物。CBS-1114 HCl 可以保持和改善心脏功能,减轻心功能障碍,以及减少患有心血管疾病的受试者的心外膜脂肪组织和/或心包脂肪组织。
T90597 SSR504734 HCl

SSR504734 是一种具有口服活性、选择性和可逆性的 GlyT1抑制剂 (hGlyT1,rGlyT1,mGlyT1IC50分别为 18、15 和 38 nM)。SSR504734 在精神分裂症、焦虑症和抑郁症模型中表现出活性。
T68103L Mk-6186 HCl

Mk-6186 HCl(1034474-19-5 Free base)

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
MK-6186 HCl,一种新型非核苷类逆转录酶抑制剂,具有抗病毒活性,可用于研究HIV。

化合物

Panomifene HCl
Cat.No: T33876L
Synonym: EGIS5650 HCl,GYKI 13504 HCl,Panomifene HCl(77599-17-8 Free base),EGIS 5650 HCl
Target: HER
CHIR-99021 HCl
Cat.No: T2310L
Synonym: CT99021 HCl,Laduviglusib HCl
Target: GSK-3
Gimatecan HCl
Cat.No: T21319L
Synonym: ST1481 HCL,Gimatecan HCl(292618-32-7 Free base)
Target: Topoisomerase
Eravacycline HCl
Cat.No: T11227L1
Synonym: Eravacycline HCL(1207283-85-9 Free bse),TP-434 HCl
Target: Antibiotic
UNC10217938A HCl
Cat.No: T13254L
Synonym: UNC10217938A HCl(1347749-97-6 Free base),UNC7938 HCl
Target: Others
CDD0102 HCl
Cat.No: T80662
Synonym: CDD0102A HCl
Target: AChR
Ganfeborole HCl
Cat.No: T11497
Synonym: GSK3036656 HCl,GSK656 HCl
Target: Antibacterial
Atagabalin HCl
Cat.No: T30188L
Synonym: PD-0200390 HCl,Atagabalin HCl(223445-75-8 Free base)
Target: Calcium Channel
Nolomirole HCl
Cat.No: T33711L
Synonym: CHF 1035 HCl,CHF 1035,CHF1035,CHF1035 HCl,CHF-1035 HCl,CHF-1035,Nolomirole Hydrochloride
Target: Dopamine Receptor, Norepinephrine
Alpertine HCl
Cat.No: T10290L
Synonym: Win 31665 HCl,Alpertine HCl(27076-46-6 Free base)
Target: Others
Vesnarinone HCl
Cat.No: T3465L
Synonym: Synonym 2,OPC-8212 HCl,Vesnarinone HCl(81840-15-5 Free base)
Target: Potassium Channel, Calcium Channel, PDE
Anisperimus HCl
Cat.No: T30077L
Synonym: LF 150195 HCl,Anisperimus HCl(170368-04-4 Free base)
Target: Others
SK609 HCl
Cat.No: T24797
Synonym: SK-609 HCl,SK609 hydrochloride,SK 609 HCl,SK 609 hydrochloride,SK-609 hydrochloride
Target:
dBRD9 HCl
Cat.No: T31221L
Synonym: dBRD9 HCl(2170679-45-3 Free base)
Target: Epigenetic Reader Domain
LY339434 HCl
Cat.No: T27947L
Synonym: LY339434 HCl(219566-62-8 Free base)
Target: GluR, NMDAR
PRLX-93936 HCL
Cat.No: T36404L
Synonym: PRLX-93936 hcl(903499-49-0 Free base)
Target: Ferroptosis, Reactive Oxygen Species
Dazolicin HCl
Cat.No: T68050L
Synonym: Dazolicine HCl,Dazolicine hydrochloride
Target: Others
Litoxetine HCl
Cat.No: T67956L
Synonym: litoxetine HCL(86811-09-8 Free base)
Target: 5-HT Receptor
Flurocitabine HCl
Cat.No: T27342L
Synonym: Flurocitabine HCl(37717-21-8 Free base)
Target: Others
Tallimustine HCl
Cat.No: T68151L
Synonym: Tallimustine HCl(115308-98-0 Free base)
Target: DNA
Upacicalcet HCl
Cat.No: T29067L
Synonym: Upacicalcet HCl(1333218-50-0 Free base)
Target: CaSR
Lesopitron HCl
Cat.No: T11839L
Synonym: Lesopitron HCl(132449-89-9 Free base)
Target: 5-HT Receptor
Brefonalol HCl
Cat.No: T30586L
Synonym: Brefonalol HCl(103880-26-8 Free base)
Target: Adrenergic Receptor
Moxilubant HCl
Cat.No: T68108L
Synonym: Moxilubant hcl(146978-48-5 Free base)
Target: LTR
Fasnall HCl
Cat.No: T27307L
Synonym: Fasnall HCl(929978-58-5 Free base)
Target: Fatty Acid Synthase
PU-H71 HCl
Cat.No: T6960L
Synonym: PU-H71 HCl(873436-91-0 Free base),Zelavespib HCl
Target: HSP, DNA/RNA Synthesis
Samidorphan HCl
Cat.No: T67888L
Synonym: Samidorphan HCl(852626-89-2 free base)
Target: Opioid Receptor
ND-322 HCl
Cat.No: T28145
Synonym: ND 322 Hydrochloride,ND322 Hydrochloride,ND-322 Hydrochloride,ND322 HCl
Target: MMP
Patamostat HCl
Cat.No: T9670L
Synonym: Patamostat HCl(114568-26-2 Free base)
Target: Serine Protease, Protease
Anidoxime HCl
Cat.No: T26631L
Synonym: USVP-E142,Anidoxime HCl( 34297-34-2 Free base)
Target:
ENMD-1068 HCl
Cat.No: T27267
Synonym: ENMD-1068 HCl,ENMD 1068,ENMD-1068,ENMD1068,ENMD-1068 hydrochloride
Target: Protease-activated Receptor
Zabicipril HCl
Cat.No: T68171L
Synonym: Zabicipril HCl(83059-56-7 Free base),S 9650,S 10211
Target: Angiotensin-converting Enzyme (ACE)
Nardeterol HCl
Cat.No: T68114L
Synonym: Nardeterol HCl(73865-18-6 Free base)
Target: Adrenergic Receptor
(Rac)-Sabcomeline HCl
Cat.No: T68135L
Synonym: sabcomeline HCl(149156-36-5 Free base)
Target: AChR
3-Hydroxykynurenamine HCl
Cat.No: T68182L
Synonym: 3-OH-Kynurenamine HCl,3-Hydroxykynurenamine HCl(99362-47-7 Free base)
Target: Others
Gizzerosine HCl
Cat.No: T31931L
Synonym: Gizzerosine HCl(89238-78-8 Free base)
Target: Others
Propiram fumarate HCl
Cat.No: T28453L
Synonym: Propiram fumarate HCl(15686-91-6 Free base)
Target: Opioid Receptor
MS8511 HCl
Cat.No: T63351L
Synonym: MS8511 HCl(2866408-21-9 Free base)
Target: Histone Methyltransferase
SGC2085 HCl
Cat.No: T4013
Synonym:
Target: Histone Methyltransferase
CDD-1102 HCl
Cat.No: T72058L
Synonym: CDD-1102 HCl(2757619-84-2 Free base)
Target: Epigenetic Reader Domain
Ot-730 HCl
Cat.No: T68120L
Synonym: Ot-730 HCl(870809-51-1 Free base)
Target: Others
XR-11576 HCl
Cat.No: T26339L
Synonym: XR-11576 HCl(346689-77-8 Free base)
Target: Topoisomerase
(S)-3,4-DCPG HCl
Cat.No: T23288L
Synonym: (S)-3,4-Dicarboxyphenylglycine HCl,(S)-3,4-DCPG HCl(201730-11-2 Free base)
Target: GluR
Etilefrine pivalate HCl
Cat.No: T68067L
Synonym: Etilefrine pivalate HCl(100696-30-8 Free base)
Target:
(Iso)-Atagabalin HCl
Cat.No: T30188L1
Synonym: (Iso)-Atagabalin HCl((Iso)-223445-75-8)
Target: Others
OT-551 HCl
Cat.No: T28273L
Synonym: OT-551 HCl(627085-11-4 Free base)
Target: NF-κB
GKI-1 HCl
Cat.No: T11402L
Synonym: GKI-1 HCl( 2444764-03-6 Free base)
Target: ROCK
CBS-1114 HCl
Cat.No: T68037L
Synonym: N-Phenylbenzamidrazone hydrochloride,cbs-1114 HCl(46721-85-1 Free base)
Target: Lipoxygenase
SSR504734 HCl
Cat.No: T90597
Synonym:
Target:
Mk-6186 HCl
Cat.No: T68103L
Synonym: Mk-6186 HCl(1034474-19-5 Free base)
Target: HIV Protease, Reverse Transcriptase
Cat. No. Product Name Target Signaling Pathways
T4866 H-Trp-NH2.HCl

L-Tryptophanamide hydrochloride,L-色氨酰胺盐酸盐,(2S)-2-amino-3-(1H-indol-3-yl)propanamide hydrochloride

Others; Endogenous Metabolite Metabolism; Others
H-Trp-NH2.HCl ((2S)-2-amino-3-(1H-indol-3-yl)propanamide hydrochloride) 是一种内源性代谢产物,已在多种生物体液中检测到,如尿液和血液。
T0415 Guanidine hydrochloride

Guanidine HCl,Aminoformamidine HCl,盐酸胍,Aminoformamidine Hydrochloride,Guanidinium chloride

Others; Arginase; DNA/RNA Synthesis; Endogenous Metabolite; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Others
Guanidine hydrochloride (Aminoformamidine Hydrochloride) 是一种强离液剂和一种蛋白质的强变性剂。
T64911 Blasticidin S HCl

Antibiotic Microbiology/Virology
Blasticidin S HCl 是从 Streptomyces griseochromogenes 中分离的肽基核苷类抗生素 (antibiotic),主要通过干扰核糖体中肽键的形成从而抑制原核细胞和真核细胞蛋白的合成。
T0804 Pilocarpine Hydrochloride

NSC 5746 HCl,盐酸毛果芸香碱,Pilocarpine HCl,(+)-Pilocarpine hydrochloride

AChR Neuroscience
Pilocarpine Hydrochloride (NSC 5746 HCl) 是一种 M3 型毒蕈碱乙酰胆碱受体激动剂,用于制作癫痫实验模型
T2953 Ligustrazine hydrochloride

Tetramethylpyrazine hydrochloride,Tetramethylpyrazine HCl,Chuanxiongzine hydrochloride,Tetrapyrazine HCl,盐酸川芎嗪

Others Others
Ligustrazine hydrochloride (Chuanxiongzine hydrochloride) 是一种天然产物。
T6004 Tetrahydropapaverine hydrochloride

Tetrahydropapaverine HCl,Norlaudanosine HCl,Tetrahydroalkali hydrochloride,四氢罂粟碱盐酸盐

Hydroxylase Metabolism
Tetrahydropapaverine hydrochloride (Norlaudanosine HCl) 是一种四氢异喹啉类药物。它对多巴胺神经元有神经毒性作用。
T0783 Mianserin hydrochloride

Mianserin HCl,Org GB 94,盐酸米安色林,ORG GB-94 HCl

Dopamine Receptor; 5-HT Receptor; Opioid Receptor; Adrenergic Receptor; Histamine Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mianserin hydrochloride (Org GB 94) 是一种有抗抑郁活性的 H1 受体反向激动剂。
T0486 Irinotecan hydrochloride trihydrate

Irinotecan HCl Trihydrate,CPT-11 HCl Trihydrate,盐酸伊立替康三水合物

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan hydrochloride trihydrate (CPT-11 HCl Trihydrate) 通过抑制拓扑异构酶 1 来防止 DNA 展开,可研究结肠癌和直肠癌。
T4291 (+)-Isocorydine hydrochloride

盐酸异可利定,Isocorydine HCl

Serine/threonin kinase; Tyrosinase Cell Cycle/Checkpoint; Metabolism; Proteases/Proteasome
(+)-Isocorydine hydrochloride (Isocorydine HCl) 是一种真核生物蛋白激酶抑制剂。
T1174 Topotecan hydrochloride

SKF 104864A,SKFS 104864A,NSC609699,Nogitecan HCl,NSC 609669,盐酸拓扑替康,Topotecan HCl

Apoptosis; Topoisomerase; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair
Topotecan hydrochloride (NSC609699) 是一种具有抗癌活性的拓扑异构酶I 抑制剂。
T3232 Higenamine hydrochloride

Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Higenamine hydrochloride (norcoclaurine HCl) 是一种 β2-AR 激动剂,是用于心力衰竭相关研究的中药乌头的关键成分,具有抗凋亡活性。
T0832 Vancomycin hydrochloride

盐酸万古霉素,Vancomycin HCl

Cell wall; Antibacterial; Antibiotic; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology
Vancomycin hydrochloride (Vancomycin HCl) 是Vancomycin 的盐酸盐,是一种支链三环糖基化肽,对大多数生物体具有杀菌活性,对肠球菌具有抑菌作用。
T1591 Ancitabine hydrochloride

NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C

Others; DNA/RNA Synthesis; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。
T0896 Furaltadone hydrochloride

Furaltadone HCl,盐酸呋喃它酮

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Furaltadone hydrochloride (Furaltadone HCl) 是硝基呋喃药,可研究肠沙门氏菌感染,治疗球虫病。Furaltadone 具有体外抑制葡萄球菌作用。
T2142 Yohimbine hydrochloride

盐酸育亨宾,Antagonil,Yohimbine HCl

Adrenergic Receptor GPCR/G Protein; Neuroscience
Yohimbine hydrochloride (Antagonil) 是一种植物生物碱,具有 α-2-肾上腺素能阻断活性。它被用作散瞳药和治疗勃起功能障碍。
TN4882 Quinine HCl

奎宁树

Adrenergic Receptor GPCR/G Protein; Neuroscience
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
T1549 Raloxifene hydrochloride

LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl

Estrogen Receptor/ERR; Others; MAO; Estrogen/progestogen Receptor; Autophagy Autophagy; Endocrinology/Hormones; Metabolism; Neuroscience; Others
Raloxifene hydrochloride (LY156758 hydrochloride) 是一种选择性且可口服的雌激素受体调节剂,用于预防绝经后妇女的骨质疏松症。它对骨骼和胆固醇代谢具有雌激素激动作用,但对乳腺和子宫组织具有完全的雌激素拮抗作用。
T0912 Tetracycline hydrochloride

NCI-c55561,盐酸四环素,Tetracycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Tetracycline hydrochloride (NCI-c55561) 是一种广谱抗生素,抑制多种革兰氏阳性和革兰氏阴性细菌。
T2941 Glucosamine hydrochloride

Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride

Reactive Oxygen Species; HIF/HIF Prolyl-Hydroxylase; Endogenous Metabolite; Autophagy Autophagy; Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB
Glucosamine hydrochloride (Chitosamine hydrochloride) 是软骨基质和滑液中糖胺聚糖的天然成分,常用作骨关节炎的治疗方法。它也是一种氨基糖,是糖基化蛋白和脂质生化合成的突出前体,用作膳食补充剂。
T2209 Serotonin hydrochloride

5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride

5-HT Receptor; Endogenous Metabolite; Transferase GPCR/G Protein; Metabolism; Neuroscience
Serotonin hydrochloride (Serotonin HCl) 是一种内源性 5-HT 受体激动剂、CNS 中的单胺神经递质和儿茶酚 O-甲基转移酶 (COMT) 抑制剂,Ki 值为 44 μM。
T0330 Diphenhydramine hydrochloride

盐酸苯海拉明,Diphenhydramine HCl,DPH

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Diphenhydramine hydrochloride (DPH) 是一种组胺 H1 拮抗剂,用作镇咳药和止吐药。它还用于治疗瘙痒和皮肤病、过敏反应、抗帕金森病、催眠药和普通感冒制剂的成分。
T1644 Dopamine hydrochloride

盐酸多巴胺,Dopamine HCl,ASL279

Ferroptosis; Dopamine Receptor; 5-HT Receptor; Endogenous Metabolite Apoptosis; GPCR/G Protein; Metabolism; Neuroscience
Dopamine hydrochloride (ASL279) 是在脑黑质、脑腹侧被盖区和下丘脑中产生的一种天然儿茶酚胺,由二羟基苯丙氨酸脱羧形成,是去甲肾上腺素和肾上腺素的前体。它通过 D2 多巴胺受体来诱导 VEGFR2 的内吞作用,有促进血管生成活性。
T4592 TOMATIDINE HYDROCHLORIDE

Tomatidine,Tomatidine HCl,盐酸番茄碱

Others; NF-κB; JNK; Autophagy Autophagy; MAPK; NF-κB; Others
Tomatidine hydrochloride (Tomatidine HCl) 是一种甾体生物碱,可防止肌肉萎缩并促进肌肉生长。它通过阻断 NF-κB 和JNK 信号发挥抗炎作用,可激活哺乳动物细胞或秀丽隐杆线虫中的自噬。
T1304 Chlortetracycline hydrochloride

Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Chlortetracycline hydrochloride (Isphamycin) 是一种特异性钙离子载体抗生素, 抑制氨酰 tRNA 结合到核糖体。
T6688 Synephrine hydrochloride

辛弗林盐酸盐,Oxedrine hydrochloride,Synephrine HCl

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Synephrine hydrochloride (Oxedrine hydrochloride) 是一种来自Citrus aurantium 的α-adrenergic 和β-adrenergic 激动剂的生物碱,也是一种拟交感神经化合物,能够用于减肥。
T4614 Ellipticine hydrochloride

Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐

Topoisomerase DNA Damage/DNA Repair
Ellipticine hydrochloride (NSC-71795 (hydrochloride)) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 的活性。
T4080 Leonurine hydrochloride

盐酸益母草碱,SCM-198 hydrochloride,SCM-198 HCl

TLR; Autophagy Autophagy; Immunology/Inflammation
Leonurine hydrochloride (SCM-198 hydrochloride) 是从益母草中分离的一种生物碱,具有抗氧化和抗炎活性。
T1511 Daunorubicin hydrochloride

Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin

Apoptosis; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Daunorubicin hydrochloride (Rubidomycin hydrochloride) 是一种蒽环类氨基糖苷类抗肿瘤药物,可抑制 DNA 复制和修复以及 RNA 和蛋白质合成。
T6225 Adenine hydrochloride

Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Adenine hydrochloride (6-Aminopurine hydrochloride) 是一种嘌呤,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T1400 Demeclocycline hydrochloride

地美环素,Declomycin,Clortetrin,盐酸地美环素,Detravis,Demeclocycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Demeclocycline hydrochloride (Declomycin) 是四环素类抗生素,可治疗粉刺,莱姆病和支气管炎。
T0551 D-Ornithine hydrochloride

D-Ornithine HCl,D-鸟氨酸盐酸盐,D-Ornithine monohydrochloride

Others; Endogenous Metabolite Metabolism; Others
D-Ornithine hydrochloride (D-Ornithine HCl) 是内源性代谢产物的一种。
T1156 Palonosetron hydrochloride

盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259

5-HT Receptor GPCR/G Protein; Neuroscience
Palonosetron hydrochloride (RS 25259) 是一种 5-HT3 拮抗剂,用于预防和治疗化疗引起的恶心和呕吐。
T0453 Phenylephrine hydrochloride

NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride

Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Phenylephrine hydrochloride (NCI-c55641) 是选择性的α1-肾上腺素能受体激动剂,对α1A,α1B 和α1D 受体的pKis 分为4.70,4.87和5.86。
T6631 Quinine hydrochloride dihydrate

奎宁单盐酸盐二水合物,Quinine HCl Dihydrate,奎宁盐酸盐二水合物

Potassium Channel; Parasite Membrane transporter/Ion channel; Microbiology/Virology
Quinine hydrochloride dihydrate (Quinine HCl Dihydrate) 是一种白色结晶 K+ 通道阻滞剂,用于治疗疟疾,具有退热,抗疟,止痛,抗炎等特性。
T0518 Methacycline hydrochloride

Rondomycin,盐酸甲烯土霉素,盐酸美他环素,Methacycline HCl

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Methacycline hydrochloride (Rondomycin) 是四环素抗生素,可抑制细菌蛋白质的合成。它是上皮-间质转化 (EMT) 抑制剂。它在体外可阻断 EMT,体内抑制纤维发生,不会直接影响 TGF-β1 Smad 信号传导。它是抗菌剂,有潜力研究肺纤维化。
T2917 Tetrahydropalmatine hydrochloride

延胡索乙素盐酸盐,1-Tetrahydropalmitine HCl,Gindarine hydrochloride,盐酸延胡乙素

Others; Dopamine Receptor GPCR/G Protein; Neuroscience; Others
Tetrahydropalmatine hydrochloride (Gindarine hydrochloride) 通过抑制大鼠杏仁核的多巴胺释放来抑制癫痫发作,可用于缓解疼痛的研究。
T6475 (±)-Carnitine chloride

Monocamin,DL-Carnitine HCl,Bicarnesine,混旋肉碱盐酸盐,DL-Carnitine chloride

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
(±)-Carnitine chloride (Monocamin) 有D 和L 两种异构体。其中 L-carnitine 在脂肪酸的 β-氧化中起重要作用,也具有抗氧化作用和抗炎活性。
T0469 Octopamine hydrochloride

章鱼胺盐酸盐,(±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl,章胺盐酸盐

Dopamine Receptor; Endogenous Metabolite; Adrenergic Receptor GPCR/G Protein; Metabolism; Neuroscience
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) 是一种与去甲肾上腺素结构相关的生物单胺类物质,在无脊椎动物中起着神经调节剂、神经激素和神经递质的作用。它对转染人 alpha2-肾上腺素受体(ARs)的中国仓鼠卵巢细胞 α2-ARs 有刺激作用。它提高糖原分解、糖酵解、糖异生、摄氧量和门脉灌注压。
T3999 D(+)-Galactosamine hydrochloride

D-半乳糖胺盐酸盐,D-氨基半乳糖盐酸盐,D-Galactosamine HCl

Others Others
D(+)-Galactosamine hydrochloride (D-Galactosamine HCl) 是一种被证实的实验毒素,它能够产生自由基及UTP 核苷酸的消耗导致肝损伤,中毒剂量会造成肾功能不全,而肾功能衰竭通常和终末期肝损伤有关。脂多糖/D-Galactosamine 诱导的急性肝损伤是一种已知的暴发性肝衰竭动物模型。
T8141 L-Cysteine hydrochloride

L-Cysteine HCl,L-半胱氨酸盐酸盐,L-半胱氨酸盐酸盐(无水物)

Others; Endogenous Metabolite Metabolism; Others
L-Cysteine hydrochloride (L-Cysteine HCl) 是一种条件必需氨基酸,是硫化氢 (H2S)、牛磺酸谷胱甘肽和等生物特性分子的前体。它能抑制胃饥饿素,抑制啮齿动物和人类的食欲。
T21430 Oxytetracycline Hydrochloride

Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin

Antiviral; Endogenous Metabolite; Antibacterial; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology
Oxytetracycline Hydrochloride (Dalimycin) 是由 Streptomyces rimosus 生产的,一种具有抗菌活性的四环素衍生物。它干扰氨酰-tRNA 与 mRNA-核糖体复合物的结合,从而阻止肽延伸并抑制蛋白质合成。
T1411 Terbinafine hydrochloride

KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Terbinafine hydrochloride (KWD 2019) 具有抗真菌感染活性。它是念珠菌属的角鲨烯环氧化酶的非竞争性抑制剂,Ki 值为 30 nM。它还对某些革兰氏阳性和革兰氏阴性细菌具有抗菌活性。
TN7045 N-phenethylbenzamide

N-(2-Phenylethyl)benzamide,Solina New Impurity 21,N-苯乙基-苯甲酰胺,4-(DICHLOROMETHYL)PYRIDINE HCL

Others Others
N-phenethylbenzamide (Solina New Impurity 21) 是一种天然产物。
T1680 Tolazoline hydrochloride

Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)

Adrenergic Receptor GPCR/G Protein; Neuroscience
Tolazoline hydrochloride (NSC35110(hydrochloride)) 是一种 α 肾上腺素受体抑制剂。
T0670 L-Arginine hydrochloride

(S)-(+)-Arginine hydrochloride,左旋精氨酸单盐酸盐,L-Arginine HCl (L-Arg),L-arginine monohydrochloride

Amino Acids and Derivatives; Endogenous Metabolite; NO Synthase Immunology/Inflammation; Metabolism
L-Arginine hydrochloride 为合成一氧化氮的氮供体,是血管扩张剂。
T1020 Doxorubicin hydrochloride

Adriamycin,Doxorubicin (Adriamycin) HCl,Hydroxydaunorubicin hydrochloride,盐酸多柔比星,盐酸阿霉素,NSC 123127

Apoptosis; Mitophagy; HBV; HIV Protease; Topoisomerase; Antibacterial; Antibiotic; AMPK; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Doxorubicin hydrochloride (Adriamycin) 属于蒽环类抗生素,是人类 DNA 拓扑异构酶 I/II 抑制剂 (IC50=0.8/2.67 μM)。Doxorubicin hydrochloride 具有细胞毒性和抗肿瘤活性。Doxorubicin hydrochloride 可降低 AMPK 及其下游靶蛋白乙酰辅酶 A 羧化酶的磷酸化,还可诱导凋亡和自噬。
T0973L Pyridoxine hydrochloride

Pyridoxine HCl,吡哆醇盐酸盐,Pyridoxol (hydrochloride),吡哆醇盐酸盐(维生素B6),Vitamin B6 (hydrochloride),Vitamin B6

Nrf2; Endogenous Metabolite Immunology/Inflammation; Metabolism
Pyridoxine hydrochloride (Vitamin B6) 是一种吡啶衍生物。在于阿尔茨海默病细胞模型中,通过 Nrf-2/HO-1 途径发挥抗氧化作用。
T0894 Thiamine hydrochloride

盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride

Apoptosis; HBV; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology
Thiamine hydrochloride (Vitamin B1) 是一种必需的微量营养素,是许多中枢代谢酶的辅因子。
T6460 Cysteamine hydrochloride

2-Mercaptoethylamine Hydrochloride,β-Mercaptoethylamine Hydrochloride,半胱胺盐酸盐,Thioethanolamine Hydrochloride,2-Aminoethanethiol Hydrochloride,Cysteamine HCl,Bekaptan

Apoptosis; Others; Reactive Oxygen Species; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB; Others
Cysteamine hydrochloride (Thioethanolamine Hydrochloride) 是一种可口服的,用于肾病型胱胺酸症的小分子药物,也可作为抗氧化剂。
T1662 5-Aminolevulinic acid hydrochloride

氨基酮戊酸,Hydrangin,5-ALA,5-Aminolevulinic acid HCl,5-氨基乙酰丙酸盐酸盐,ALA hydrochloride

Apoptosis; Mitophagy; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism
5-Aminolevulinic acid hydrochloride (5-ALA) 是体内血红素生物合成的中间体,也是四吡咯的通用前体。
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天然产物

H-Trp-NH2.HCl
Cat.No: T4866
Synonym: L-Tryptophanamide hydrochloride,L-色氨酰胺盐酸盐,(2S)-2-amino-3-(1H-indol-3-yl)propanamide hydrochloride
Target: Others, Endogenous Metabolite
Guanidine hydrochloride
Cat.No: T0415
Synonym: Guanidine HCl,Aminoformamidine HCl,盐酸胍,Aminoformamidine Hydrochloride,Guanidinium chloride
Target: Others, Arginase, DNA/RNA Synthesis, Endogenous Metabolite, Autophagy
Blasticidin S HCl
Cat.No: T64911
Synonym:
Target: Antibiotic
Pilocarpine Hydrochloride
Cat.No: T0804
Synonym: NSC 5746 HCl,盐酸毛果芸香碱,Pilocarpine HCl,(+)-Pilocarpine hydrochloride
Target: AChR
Ligustrazine hydrochloride
Cat.No: T2953
Synonym: Tetramethylpyrazine hydrochloride,Tetramethylpyrazine HCl,Chuanxiongzine hydrochloride,Tetrapyrazine HCl,盐酸川芎嗪
Target: Others
Tetrahydropapaverine hydrochloride
Cat.No: T6004
Synonym: Tetrahydropapaverine HCl,Norlaudanosine HCl,Tetrahydroalkali hydrochloride,四氢罂粟碱盐酸盐
Target: Hydroxylase
Mianserin hydrochloride
Cat.No: T0783
Synonym: Mianserin HCl,Org GB 94,盐酸米安色林,ORG GB-94 HCl
Target: Dopamine Receptor, 5-HT Receptor, Opioid Receptor, Adrenergic Receptor, Histamine Receptor
Irinotecan hydrochloride trihydrate
Cat.No: T0486
Synonym: Irinotecan HCl Trihydrate,CPT-11 HCl Trihydrate,盐酸伊立替康三水合物
Target: Topoisomerase, Autophagy
(+)-Isocorydine hydrochloride
Cat.No: T4291
Synonym: 盐酸异可利定,Isocorydine HCl
Target: Serine/threonin kinase, Tyrosinase
Topotecan hydrochloride
Cat.No: T1174
Synonym: SKF 104864A,SKFS 104864A,NSC609699,Nogitecan HCl,NSC 609669,盐酸拓扑替康,Topotecan HCl
Target: Apoptosis, Topoisomerase, Autophagy
Higenamine hydrochloride
Cat.No: T3232
Synonym: Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride
Target: Adrenergic Receptor
Vancomycin hydrochloride
Cat.No: T0832
Synonym: 盐酸万古霉素,Vancomycin HCl
Target: Cell wall, Antibacterial, Antibiotic, Autophagy
Ancitabine hydrochloride
Cat.No: T1591
Synonym: NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C
Target: Others, DNA/RNA Synthesis, Autophagy
Furaltadone hydrochloride
Cat.No: T0896
Synonym: Furaltadone HCl,盐酸呋喃它酮
Target: Antibacterial, Antibiotic, Parasite
Yohimbine hydrochloride
Cat.No: T2142
Synonym: 盐酸育亨宾,Antagonil,Yohimbine HCl
Target: Adrenergic Receptor
Quinine HCl
Cat.No: TN4882
Synonym: 奎宁树
Target: Adrenergic Receptor
Raloxifene hydrochloride
Cat.No: T1549
Synonym: LY156758 hydrochloride,盐酸雷洛昔芬,Raloxifene HCl,LY139481 hydrochloride,Keoxifene hydrochloride,LY156758 (Keoxifene) HCl
Target: Estrogen Receptor/ERR, Others, MAO, Estrogen/progestogen Receptor, Autophagy
Tetracycline hydrochloride
Cat.No: T0912
Synonym: NCI-c55561,盐酸四环素,Tetracycline HCl
Target: ribosome, Antibacterial, Antibiotic
Glucosamine hydrochloride
Cat.No: T2941
Synonym: Chitosamine hydrochloride,盐酸氨基葡萄糖,2-Amino-2-deoxy-glucose HCl,Chitosamine HCl,D-(+)-Glucosamine hydrochloride
Target: Reactive Oxygen Species, HIF/HIF Prolyl-Hydroxylase, Endogenous Metabolite, Autophagy
Serotonin hydrochloride
Cat.No: T2209
Synonym: 5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride
Target: 5-HT Receptor, Endogenous Metabolite, Transferase
Diphenhydramine hydrochloride
Cat.No: T0330
Synonym: 盐酸苯海拉明,Diphenhydramine HCl,DPH
Target: Histamine Receptor
Dopamine hydrochloride
Cat.No: T1644
Synonym: 盐酸多巴胺,Dopamine HCl,ASL279
Target: Ferroptosis, Dopamine Receptor, 5-HT Receptor, Endogenous Metabolite
TOMATIDINE HYDROCHLORIDE
Cat.No: T4592
Synonym: Tomatidine,Tomatidine HCl,盐酸番茄碱
Target: Others, NF-κB, JNK, Autophagy
Chlortetracycline hydrochloride
Cat.No: T1304
Synonym: Isphamycin,Chlortetracycline HCl,7-Chlorotetracycline hydrochloride,盐酸金霉素
Target: ribosome, Antibacterial, Antibiotic
Synephrine hydrochloride
Cat.No: T6688
Synonym: 辛弗林盐酸盐,Oxedrine hydrochloride,Synephrine HCl
Target: Endogenous Metabolite, Adrenergic Receptor
Ellipticine hydrochloride
Cat.No: T4614
Synonym: Ellipticine HCl,NSC 71795 (hydrochloride),玫瑰树碱盐酸盐
Target: Topoisomerase
Leonurine hydrochloride
Cat.No: T4080
Synonym: 盐酸益母草碱,SCM-198 hydrochloride,SCM-198 HCl
Target: TLR, Autophagy
Daunorubicin hydrochloride
Cat.No: T1511
Synonym: Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin
Target: Apoptosis, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic, Autophagy
Adenine hydrochloride
Cat.No: T6225
Synonym: Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride
Target: DNA/RNA Synthesis, Endogenous Metabolite
Demeclocycline hydrochloride
Cat.No: T1400
Synonym: 地美环素,Declomycin,Clortetrin,盐酸地美环素,Detravis,Demeclocycline HCl
Target: ribosome, Antibacterial, Antibiotic
D-Ornithine hydrochloride
Cat.No: T0551
Synonym: D-Ornithine HCl,D-鸟氨酸盐酸盐,D-Ornithine monohydrochloride
Target: Others, Endogenous Metabolite
Palonosetron hydrochloride
Cat.No: T1156
Synonym: 盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259
Target: 5-HT Receptor
Phenylephrine hydrochloride
Cat.No: T0453
Synonym: NCI-c55641,Phenylephrine HCl,盐酸去氧肾上腺素,(R)-(-)-Phenylephrine hydrochloride
Target: Endogenous Metabolite, Adrenergic Receptor
Quinine hydrochloride dihydrate
Cat.No: T6631
Synonym: 奎宁单盐酸盐二水合物,Quinine HCl Dihydrate,奎宁盐酸盐二水合物
Target: Potassium Channel, Parasite
Methacycline hydrochloride
Cat.No: T0518
Synonym: Rondomycin,盐酸甲烯土霉素,盐酸美他环素,Methacycline HCl
Target: ribosome, Antibacterial, Antibiotic
Tetrahydropalmatine hydrochloride
Cat.No: T2917
Synonym: 延胡索乙素盐酸盐,1-Tetrahydropalmitine HCl,Gindarine hydrochloride,盐酸延胡乙素
Target: Others, Dopamine Receptor
(±)-Carnitine chloride
Cat.No: T6475
Synonym: Monocamin,DL-Carnitine HCl,Bicarnesine,混旋肉碱盐酸盐,DL-Carnitine chloride
Target: Reactive Oxygen Species
Octopamine hydrochloride
Cat.No: T0469
Synonym: 章鱼胺盐酸盐,(±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl,章胺盐酸盐
Target: Dopamine Receptor, Endogenous Metabolite, Adrenergic Receptor
D(+)-Galactosamine hydrochloride
Cat.No: T3999
Synonym: D-半乳糖胺盐酸盐,D-氨基半乳糖盐酸盐,D-Galactosamine HCl
Target: Others
L-Cysteine hydrochloride
Cat.No: T8141
Synonym: L-Cysteine HCl,L-半胱氨酸盐酸盐,L-半胱氨酸盐酸盐(无水物)
Target: Others, Endogenous Metabolite
Oxytetracycline Hydrochloride
Cat.No: T21430
Synonym: Biosolvomycin,盐酸土霉素,Oxytetracycline HCl,Oxytetracycline.HCl,Dalimycin,Oxytetracycline, Sodium Salt,Dalinmycin
Target: Antiviral, Endogenous Metabolite, Antibacterial, HSV
Terbinafine hydrochloride
Cat.No: T1411
Synonym: KWD 2019,盐酸特比萘芬,Terbinafine HCl,TDT 067 hydrochloride
Target: Antibacterial, Antibiotic, Antifungal
N-phenethylbenzamide
Cat.No: TN7045
Synonym: N-(2-Phenylethyl)benzamide,Solina New Impurity 21,N-苯乙基-苯甲酰胺,4-(DICHLOROMETHYL)PYRIDINE HCL
Target: Others
Tolazoline hydrochloride
Cat.No: T1680
Synonym: Imidaline hydrochloride,苯甲唑啉盐酸盐,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)
Target: Adrenergic Receptor
L-Arginine hydrochloride
Cat.No: T0670
Synonym: (S)-(+)-Arginine hydrochloride,左旋精氨酸单盐酸盐,L-Arginine HCl (L-Arg),L-arginine monohydrochloride
Target: Amino Acids and Derivatives, Endogenous Metabolite, NO Synthase
Doxorubicin hydrochloride
Cat.No: T1020
Synonym: Adriamycin,Doxorubicin (Adriamycin) HCl,Hydroxydaunorubicin hydrochloride,盐酸多柔比星,盐酸阿霉素,NSC 123127
Target: Apoptosis, Mitophagy, HBV, HIV Protease, Topoisomerase, Antibacterial, Antibiotic, AMPK, Autophagy
Pyridoxine hydrochloride
Cat.No: T0973L
Synonym: Pyridoxine HCl,吡哆醇盐酸盐,Pyridoxol (hydrochloride),吡哆醇盐酸盐(维生素B6),Vitamin B6 (hydrochloride),Vitamin B6
Target: Nrf2, Endogenous Metabolite
Thiamine hydrochloride
Cat.No: T0894
Synonym: 盐酸硫胺素,Vitamin B1,Vitamin B1 hydrochloride,Thiamine HCl,盐酸硫胺(维生素B1),Thiamine chloride hydrochloride
Target: Apoptosis, HBV, Endogenous Metabolite
Cysteamine hydrochloride
Cat.No: T6460
Synonym: 2-Mercaptoethylamine Hydrochloride,β-Mercaptoethylamine Hydrochloride,半胱胺盐酸盐,Thioethanolamine Hydrochloride,2-Aminoethanethiol Hydrochloride,Cysteamine HCl,Bekaptan
Target: Apoptosis, Others, Reactive Oxygen Species, Endogenous Metabolite, Autophagy
5-Aminolevulinic acid hydrochloride
Cat.No: T1662
Synonym: 氨基酮戊酸,Hydrangin,5-ALA,5-Aminolevulinic acid HCl,5-氨基乙酰丙酸盐酸盐,ALA hydrochloride
Target: Apoptosis, Mitophagy, Endogenous Metabolite, Autophagy
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