首页 工具
登录
购物车

搜索结果

Search Results for " receptor-1 "

2628

抑制剂 & 化合物

104

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T12910 Sigma-1 receptor antagonist 1

Sigma receptor GPCR/G Protein
Sigma-1 receptor antagonist 1 是一种有效、特异性的 sigma-1 受体拮抗剂。 Sigma-1 receptor antagonist 1 具有抗神经性疼痛活性,可用于治疗神经性疼痛研究。
T15785 LPA1 receptor antagonist 1

LPA1 R antagonist 1

LPA Receptor GPCR/G Protein
LPA1 receptor antagonist 1(LPA1 R antagonist 1) 是一种具有选择性和高效性的溶血磷脂酸 (LPA1) 受体拮抗剂( IC50 : 25 nM),可用于研究特发性肺纤维化。
T4031 S1p receptor agonist 1

S1p-receptor-agonist-1

S1P Receptor; LPL Receptor GPCR/G Protein
S1p receptor agonist 1 (S1p-receptor-agonist-1) 是有口服活性的S1P 受体激动剂,具有诱导 S1P1 内化的活性,EC50为9.83 nM。它有潜力用于关节炎和实验性自身免疫性脑炎)的相关研究。
T10058 A2B receptor antagonist 1

Adenosine Receptor GPCR/G Protein; Neuroscience
A2B receptor antagonist 1 是一个有效的 A2B 腺苷受体 (A2B adenosine receptor) 拮抗剂。
T10307 AMPA receptor modulator-1

iGluR Membrane transporter/Ion channel; Neuroscience
AMPA receptor modulator-1可被谷氨酸激活,从而调节离子通道。
T5829 H4 Receptor antagonist 1

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
H4 Receptor antagonist 1 是选择性组胺 H4受体反向激动剂,其IC50值为19 nM。
T37908 Glucocorticoid receptor agonist-1

Glucocorticoid Receptor Endocrinology/Hormones
Glucocorticoid receptor agonist-1是一种强效糖皮质激素受体激动剂,其 IC50 值为 2.8 nM。
T10499 H3 receptor-MO-1

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
H3 receptor-MO-1 是一种有效的组胺 H3 受体 (histamine H3 receptor) 调节剂,可用于研究神经分裂和认知障碍。
T13736 Interferon receptor inducer-1

IFNAR Immunology/Inflammation
Interferon receptor inducer-1 是一种干扰素(IFN)受体诱导剂,可用于干扰素诱导参与的紊乱性疾病的研究。
T9244 σ1 Receptor antagonist-1

Sigma receptor GPCR/G Protein
σ1 Receptor antagonist-1 是高选择性的 sigma 1受体拮抗剂,pKi 为10.28。它抑制细胞生长,在 G0/G1 期阻滞细胞周期并诱导 MCF-7/ADR 细胞凋亡。
T10250 ADRA1D receptor antagonist 1 HCl

ADRA1D receptor antagonist 1 HCl(1191908-24-3 free base)

Adrenergic Receptor GPCR/G Protein; Neuroscience
ADRA1D receptor antagonist 1 HCl 是一种具有口服活性、高效性和选择性的 α1D 肾上腺素受体拮抗剂(Ki:1.6 nM),具有潜在的抗增殖活性。
T11211 EP4 receptor antagonist 1

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
EP4 receptor antagonist 1 是一种有效的特异性前列腺素 EP4受体拮抗剂,对人和小鼠 EP4受体的 IC50分别为6.1 nM 和16.2 nM。 EP4 receptor antagonist 1 可用于癌症免疫治疗的研究。
T11349 GABAA receptor agent 1

GABA Receptor Membrane transporter/Ion channel; Neuroscience
GABAA receptor agent 1 是GABAA 受体的高亲和力配体,有抗惊厥活性。
T12155 Y1 receptor antagonist 1

H 409-22 isomer

Others Others
Y1 receptor antagonist 1 is an antagonist of neuropeptide Y1 receptor.
T15249 Estrogen receptor modulator 1

Estrogen Receptor/ERR Endocrinology/Hormones
Estrogen receptor modulator 1 是一种有效的、具有口服活性的、选择性雌激素受体(estrogen receptor)调节剂 (SERM),其 pIC50为 0.46。它能够诱导 Tamoxifen 耐药、激素非依赖性异种移植瘤的消退。
T11137 (E)-GABAB receptor antagonist 1

GABA Receptor Membrane transporter/Ion channel; Neuroscience
(E)-GABAB receptor antagonist 1 是 GABAB receptor antagonist 1 的反式结构。(E)-GABAB receptor antagonist 1 降低 GABA 诱导的 IP3 (三磷酸肌醇) 产生,IC50 为 37.9 μM。GABAB receptor antagonist 1是选择性的 GABAB (γ-氨基丁酸) 受体的负变构调节剂。
T12912 Sigma-1 receptor antagonist 3

Sigma receptor; HER Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Sigma-1 receptor antagonist 3 是 Sigma-1受体选择性拮抗剂,Ki 为 1.14 nM。它抑制 hERG,IC50为 1.54μM。它在神经性疼痛方面有研究的价值。
T12911 Sigma-1 receptor antagonist 2

Sigma receptor GPCR/G Protein
Sigma-1 receptor antagonist 2 是有效的sigma 1受体选择性拮抗剂,与 σ1 和 σ2 受体结合的Ki 分别为 3.88 和 1288 nM。
T12404 CCK-A receptor inhibitor 1

cholecystokinin GPCR/G Protein
CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50:340 nM)。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。
T11077 Dopamine D2 receptor antagonist-1

Others Others
Dopamine D2 receptor antagonist-1,一种对多巴胺D2受体(D2R)表现出亚毫摩尔级别亲和力的负变构调节剂(NAM)。
T37792 A2A receptor antagonist 1

CPI-444 analog,A2A receptor antagonist 1

Adenosine Receptor GPCR/G Protein; Neuroscience
A2A receptor antagonist 1 (CPI-444 analog)是腺苷 A2A 和 A1受体的拮抗剂,Ki 值分别为4和264 nM。
T9157 GP130 receptor agonist-1

N-(4-Fluorophenyl)-4-phenyl-2-thiazolami

Interleukin Immunology/Inflammation
GP130 receptor agonist-1 (N-(4-Fluorophenyl)-4-phenyl-2-thiazolami) 是一种有效的、口服有活性的、可透过血脑屏障的 GP130受体激动剂。它对 NMDA 诱导的神经毒性具有神经保护作用。
T38836L Protease-Activated Receptor-1, PAR-1 Agonist acetate

Protease-activated Receptor GPCR/G Protein
Protease-Activated Receptor-1, PAR-1 Agonist acetate 是一种选择性蛋白酶激活受体 1 (PAR-1) 激动剂肽。 它对应于 PAR1 栓系配体,可以选择性地模拟凝血酶通过该受体的作用。
T4521 Edg-2 receptor inhibitor 1

SAR-100842

LPA Receptor GPCR/G Protein
Edg-2 receptor inhibitor 1 (SAR-100842) 是一种提取的 Edg-2 受体抑制剂 (IC50: <0.1 μM)。
T12247 NOT Receptor Modulator 1

2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol

Others Others
NOT Receptor Modulator 1 (2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol) 是核受体 NOT 调节剂。
T9247 Vanilloid receptor antagonist 1

4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile

TRP/TRPV Channel Membrane transporter/Ion channel
Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) 是香草酸受体的有效拮抗剂。
T67915 Succinate/succinate receptor antagonist 1

Others Others
Succinate/succinate receptor antagonist 1 是一种有效的琥珀酸受体拮抗剂。Succinate/succinate receptor antagonist 1 中断牙龈组织中的琥珀酸信号,抑制琥珀酸受体 1 (SucnRl Antagonist 1) 的激活,对琥珀酸受体 1的 IC50 值为 20 μΜ。Succinate/succinate receptor antagonist 1 可用于治疗牙周病。
T9579L GLP-1 receptor agonist 9 citrate

GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base)

Glucagon Receptor GPCR/G Protein
GLP-1 receptor agonist 9 citrate 是 GLP-1 的激动剂。
T38836 Protease-Activated Receptor-1, PAR-1 Agonist

Protease-Activated Receptor-1 (PAR-1) Agonist, a selective peptide, activates the PAR-1 receptor by mimicking the specific actions of thrombin. It corresponds to the PAR1 tethered ligand, facilitating selective activation of this receptor.
T11408 Orforglipron

LY3502970,GLP-1 receptor agonist 1

Glucagon Receptor GPCR/G Protein
Orforglipron (LY3502970; GLP-1 receptor agonist 1) 是一种可口服的胰高血糖素样肽 (GLP-1) 受体激动剂,可用于研究成人肥胖和1型糖尿病。
T11236 Giredestrant tartrate

Estrogen receptor antagonist 1

Estrogen Receptor/ERR; Others Endocrinology/Hormones; Others
Giredestrant tartrate (Estrogen receptor antagonist 1) 是一种新型的、具有口服活性的、有选择性的、有效的的非甾体雌激素受体拮抗剂。Giredestrant tartrate 与 ER 强效结合,导致 ER 无法激活靶向基因的转录,并促使 ER 蛋白降解。Giredestrant tartrate 可用于治疗肿瘤疾病。
T39694 GluN2B receptor modulator-1

GluN2B receptor modulator-1

GluN2B receptor modulator-1 is a potent and selective allosteric modulator of the GluN2B receptor. It demonstrates negative modulation, inhibiting receptor activity, and exhibits high selectivity towards the GluN2B subunit, with an impressive IC50 value of 31 nM.
T36288 Protease-Activated Receptor-1, PAR-1 Agonist TFA

Protease-Activated Receptor-1 (PAR-1) Agonist TFA is a selective peptide that acts as an agonist for the proteinase-activated receptor-1 (PAR-1). Corresponding to the tethered ligand of PAR-1, this compound mimics the actions of thrombin through the PAR-1 receptor[1][2].
T10911 H3 receptor antagonist 1

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor antagonist.
T40307 Adenosine receptor antagonist 1

Adenosine receptor antagonist 1 is a highly selective antagonist for the A2aR adenosine receptor, exhibiting an IC50 value of 0.29 nM. It demonstrates a remarkable 14-fold selectivity towards the A2aR receptor in comparison to the A2bR receptor.
T11413 Glucagon receptor antagonists-1

Others Others
Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.
T40808 Glucocorticoids receptor agonist 1

Glucocorticoids receptor agonist 1 (GRA-1) is a highly effective arylpyrazole-based compound that acts as an agonist for the glucocorticoid receptor. GRA-1 exhibits strong anti-inflammatory properties while maintaining insulin secretion function.
T11350 GABAB receptor antagonist 1

GABA Receptor Membrane transporter/Ion channel; Neuroscience
(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB receptor antagonist 1 is a selective and negative allosteric modulator of GABAB (γ-Aminobutyric acid) receptors.
T10320 Androgen receptor antagonist 1

Others Others
Androgen receptor antagonist 1 is an orally available full androgen receptor antagonist (IC50: 59 nM). It can be used in the synthesis of PROTAC AR degraders, which results in 24% and 47 % AR protein degradation in LNCaP cells at 1 μM and 10 μM, respectively.
T12314 Opioid receptor modulator 1

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Opioid receptor modulator 1 is a modulator of opioid receptor.
T39813 APJ receptor agonist 1

APJ receptor agonist 1, a potent biphenyl acid derivative, acts as an agonist (EC50 of 0.093 nM and 0.12 nM for human and rat APJ receptors, respectively) for the APJ receptor (APJ-R). It exhibits significant in vitro potency towards apelin-13, the endogenous peptidic ligand for the APJ receptor. APJ receptor agonist 1 holds promise for heart failure research.
T38287 C3a Receptor Agonist

C3a receptor agonist 1,C3a受体激动剂,Complement 3a Receptor Agonist

Complement System Immunology/Inflammation
C3a Receptor Agonist (C3a receptor agonist 1) 结合免疫系统补体途径中的G 蛋白偶联C3a 受体(C3aRs)。在肠缺血再灌注损伤模型中,C3aR 的激活可防止中性粒细胞动员。C3aRs 在成年小鼠的神经祖细胞和未成熟神经元上表达。C3a 在体外刺激神经祖细胞的分化。
T16883 Sigma-2 receptor antagonist 1

Others Others
Sigma-2 receptor antagonist 1 is an antagonist of the sigma-2 (σ-2) receptor.
T13261 CCK-B Receptor Antagonist 1

Others Others
CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
T38634 Histamine H4 receptor antagonist-1

Histamine H4 receptor antagonist-1

Histamine H4 receptor antagonist-1 is a potent antagonist of the histamine H4 receptor.
T67742 EX-A5386

Glucocorticoid receptor modulator-1

Glucocorticoid Receptor Endocrinology/Hormones
EX-A5386 (Glucocorticoid receptor modulator-1)是一种有效的糖皮质激素受体调节剂,IC50/EC50<100nM。
T12821 S1PR1 modulator 1

LPL Receptor GPCR/G Protein
S1PR1 modulator 1 是 S1PR1 的特异性抑制剂,pIC50 为 7.6。
T11407 GLP-1 receptor agonist 2

Others Others
GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.
T9579 GLP-1 receptor agonist 9

Glucagon Receptor GPCR/G Protein
1H-Benzimidazole-6-carboxylic acid 是GLP-1 receptor 激动剂。
T10121 Substance P Receptor Antagonist 1

Others Others
Substance P Receptor Antagonist 1 has the potential function in gastrointestinal disorders, inflammatory diseases, respiratory, and central nervous system disorders.

化合物

Sigma-1 receptor antagonist 1
Cat.No: T12910
Synonym:
Target: Sigma receptor
LPA1 receptor antagonist 1
Cat.No: T15785
Synonym: LPA1 R antagonist 1
Target: LPA Receptor
S1p receptor agonist 1
Cat.No: T4031
Synonym: S1p-receptor-agonist-1
Target: S1P Receptor, LPL Receptor
A2B receptor antagonist 1
Cat.No: T10058
Synonym:
Target: Adenosine Receptor
AMPA receptor modulator-1
Cat.No: T10307
Synonym:
Target: iGluR
H4 Receptor antagonist 1
Cat.No: T5829
Synonym:
Target: Histamine Receptor
Glucocorticoid receptor agonist-1
Cat.No: T37908
Synonym:
Target: Glucocorticoid Receptor
H3 receptor-MO-1
Cat.No: T10499
Synonym:
Target: Histamine Receptor
Interferon receptor inducer-1
Cat.No: T13736
Synonym:
Target: IFNAR
σ1 Receptor antagonist-1
Cat.No: T9244
Synonym:
Target: Sigma receptor
ADRA1D receptor antagonist 1 HCl
Cat.No: T10250
Synonym: ADRA1D receptor antagonist 1 HCl(1191908-24-3 free base)
Target: Adrenergic Receptor
EP4 receptor antagonist 1
Cat.No: T11211
Synonym:
Target: Prostaglandin Receptor
GABAA receptor agent 1
Cat.No: T11349
Synonym:
Target: GABA Receptor
Y1 receptor antagonist 1
Cat.No: T12155
Synonym: H 409-22 isomer
Target: Others
Estrogen receptor modulator 1
Cat.No: T15249
Synonym:
Target: Estrogen Receptor/ERR
(E)-GABAB receptor antagonist 1
Cat.No: T11137
Synonym:
Target: GABA Receptor
Sigma-1 receptor antagonist 3
Cat.No: T12912
Synonym:
Target: Sigma receptor, HER
Sigma-1 receptor antagonist 2
Cat.No: T12911
Synonym:
Target: Sigma receptor
CCK-A receptor inhibitor 1
Cat.No: T12404
Synonym:
Target: cholecystokinin
Dopamine D2 receptor antagonist-1
Cat.No: T11077
Synonym:
Target: Others
A2A receptor antagonist 1
Cat.No: T37792
Synonym: CPI-444 analog,A2A receptor antagonist 1
Target: Adenosine Receptor
GP130 receptor agonist-1
Cat.No: T9157
Synonym: N-(4-Fluorophenyl)-4-phenyl-2-thiazolami
Target: Interleukin
Protease-Activated Receptor-1, PAR-1 Agonist acetate
Cat.No: T38836L
Synonym:
Target: Protease-activated Receptor
Edg-2 receptor inhibitor 1
Cat.No: T4521
Synonym: SAR-100842
Target: LPA Receptor
NOT Receptor Modulator 1
Cat.No: T12247
Synonym: 2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol
Target: Others
Vanilloid receptor antagonist 1
Cat.No: T9247
Synonym: 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
Target: TRP/TRPV Channel
Succinate/succinate receptor antagonist 1
Cat.No: T67915
Synonym:
Target: Others
GLP-1 receptor agonist 9 citrate
Cat.No: T9579L
Synonym: GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base)
Target: Glucagon Receptor
Protease-Activated Receptor-1, PAR-1 Agonist
Cat.No: T38836
Synonym:
Target:
Orforglipron
Cat.No: T11408
Synonym: LY3502970,GLP-1 receptor agonist 1
Target: Glucagon Receptor
Giredestrant tartrate
Cat.No: T11236
Synonym: Estrogen receptor antagonist 1
Target: Estrogen Receptor/ERR, Others
GluN2B receptor modulator-1
Cat.No: T39694
Synonym: GluN2B receptor modulator-1
Target:
Protease-Activated Receptor-1, PAR-1 Agonist TFA
Cat.No: T36288
Synonym:
Target:
H3 receptor antagonist 1
Cat.No: T10911
Synonym:
Target: Histamine Receptor
Adenosine receptor antagonist 1
Cat.No: T40307
Synonym:
Target:
Glucagon receptor antagonists-1
Cat.No: T11413
Synonym:
Target: Others
Glucocorticoids receptor agonist 1
Cat.No: T40808
Synonym:
Target:
GABAB receptor antagonist 1
Cat.No: T11350
Synonym:
Target: GABA Receptor
Androgen receptor antagonist 1
Cat.No: T10320
Synonym:
Target: Others
Opioid receptor modulator 1
Cat.No: T12314
Synonym:
Target: Opioid Receptor
APJ receptor agonist 1
Cat.No: T39813
Synonym:
Target:
C3a Receptor Agonist
Cat.No: T38287
Synonym: C3a receptor agonist 1,C3a受体激动剂,Complement 3a Receptor Agonist
Target: Complement System
Sigma-2 receptor antagonist 1
Cat.No: T16883
Synonym:
Target: Others
CCK-B Receptor Antagonist 1
Cat.No: T13261
Synonym:
Target: Others
Histamine H4 receptor antagonist-1
Cat.No: T38634
Synonym: Histamine H4 receptor antagonist-1
Target:
EX-A5386
Cat.No: T67742
Synonym: Glucocorticoid receptor modulator-1
Target: Glucocorticoid Receptor
S1PR1 modulator 1
Cat.No: T12821
Synonym:
Target: LPL Receptor
GLP-1 receptor agonist 2
Cat.No: T11407
Synonym:
Target: Others
GLP-1 receptor agonist 9
Cat.No: T9579
Synonym:
Target: Glucagon Receptor
Substance P Receptor Antagonist 1
Cat.No: T10121
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T1009 Estrone

Oestrone,雌酮,Fluoroethyl,Aquacrine

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Estrone (Aquacrine) 是内源性雌激素的主要代表,由多种组织产生,尤其是脂肪组织。它是脂肪细胞中雄烯二酮芳构化过程的结果。
T1626 Prostaglandin E1

前列地尔,PGE1,列腺素E1,Alprostadil

Endogenous Metabolite; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism
Prostaglandin E1 (Alprostadil) 是一种前列腺素受体配体,对小鼠 EP1、EP2、EP3、EP4和 IP 的 Ki 值分别为 36、10、1.1、2.1 和 33 nM。它诱导血管舒张并抑制血小板聚集,可作为血管扩张剂用于外周血管疾病的研究。
TQ0205 Procyanidin B1

原花青素B1,原花青素 B1

TLR Immunology/Inflammation
Procyanidin B1 是水果中常见的多酚类黄酮,能够与TLR4/MD-2复合体结合,具有抗炎活性。
T2917 Tetrahydropalmatine hydrochloride

延胡索乙素盐酸盐,1-Tetrahydropalmitine HCl,Gindarine hydrochloride,盐酸延胡乙素

Others; Dopamine Receptor GPCR/G Protein; Neuroscience; Others
Tetrahydropalmatine hydrochloride (Gindarine hydrochloride) 通过抑制大鼠杏仁核的多巴胺释放来抑制癫痫发作,可用于缓解疼痛的研究。
T22974 Methyl 2,5-dihydroxycinnamate

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Methyl 2,5-dihydroxycinnamate 是 erbstatin 类似物,是一种高效、稳定的 EGF 受体相关酪氨酸激酶的抑制剂。
T3870 Cyasterone

杯苋甾酮,Cyasteron

Apoptosis; EGFR Angiogenesis; Apoptosis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Cyasterone (Cyasteron) 是主要分离自金疮小草的一种天然 EGFR 抑制剂。它通过诱导细胞凋亡和细胞周期阻滞表现出抗增殖作用,可用于抗人类肿瘤的相关研究。
T2S0271 Voacamine

老刺木胺,Voacanginine

Cannabinoid Receptor; P-gp GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Voacamine (Voacanginine) 是非洲马铃果中的一种吲哚生物碱,可抑制多药耐药肿瘤细胞中的 P-糖蛋白作用,具有强效的大麻素 CB1受体拮抗活性。
T2932 Ginsenoside Rh1

Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1

IL Receptor; TNF; Endogenous Metabolite; PPAR; Interleukin Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism
Ginsenoside Rh1 (Sanchinoside B2) 是人参的一种主要成分,具有抗炎作用,抑制PPAR-γ,TNF-α,IL-6和IL-1β的表达。
T5077 Deoxycholic acid sodium salt

脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid sodium salt (Sodium deoxycholate) 是 G 蛋白偶联胆汁酸受体TGR5的激活剂。
T1431 Khellin

凯林,Amicardine,Methafrone,Visammin

EGFR; Others Angiogenesis; JAK/STAT signaling; Others; Tyrosine Kinase/Adaptors
Khellin (Methafrone) 是从阿米芹中提取得到的一种呋喃并色酮,是EGFR 抑制剂,IC50为 0.15 µM。它体外具有抗增殖活性,还具有抗痉挛和冠状动脉舒张作用。
TL0016 Sulforaphene

油菜

Apoptosis; ERK; EGFR; NF-κB Angiogenesis; Apoptosis; JAK/STAT signaling; MAPK; NF-κB; Tyrosine Kinase/Adaptors
Sulforaphene 是从萝卜种子中分离出来的天然产物,对鹿茸幼苗的 ED50 约为 2 x 10 -4 M。它通过抑制 EGFR、p-ERK1/2、NF-κB 和其他信号促进癌细胞凋亡并抑制迁移。
T3896 Shanzhiside methyl ester

三栀子甙甲酯,山芝皂苷甲酯

Glucagon Receptor GPCR/G Protein
Shanzhiside methyl ester 是一种小分子胰高血糖素样肽 1 受体激动剂,分离自轮状乳杆菌,能够诱导抗异常性痛觉耐受。
T2965 Deoxycholic acid

Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。
T16442 PCO371

2,4-Imidazolidinedione, 1-(3,5-dimethyl-4-(2-((4-oxo-2-(4-(trifluoromethoxy)phenyl)-1,3,8-triazaspiro(4.5)dec-1-en-8-yl)sulfonyl)ethyl)phenyl)-5,5-dimethyl-

Thyroid hormone receptor(THR) Endocrinology/Hormones
PCO371 (2,4-Imidazolidinedione, 1-(3,5-dimethyl-4-(2-((4-oxo-2-(4-(trifluoromethoxy)phenyl)-1,3,8-triazaspiro(4.5)dec-1-en-8-yl)sulfonyl)ethyl)phenyl)-5,5-dimethyl-) 是口服具有活性的甲状旁腺激素受体 1 的完全激动剂,对 PTHR2 无作用
T0700 Ursodeoxycholic acid

熊去氧胆酸,UDCA,Ursodiol

Potassium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
Ursodeoxycholic acid (UDCA)是一种有效的肝脏特异性脂肪酸转运蛋白 5 (FATP5) 抑制剂,通过 FATP5 依赖性方式抑制原代肝细胞摄取长链脂肪酸。Ursodeoxycholic acid 能够抑制胆固醇的吸收,用于溶解胆结石,并具有研究与肥胖相关的脂肪肝疾病的潜力。
T2995 Chrysophanol

大黄酚,3-Methylchrysazin,Chrysophanic Acid,Turkey Rhubarb

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Chrysophanol (Turkey Rhubarb) 是掌叶大黄中的一种蒽醌类天然产物,可抑制EGF-诱导的EGFR 磷酸化,且抑制AKT 和mTOR/p70S6K 激活。
T0760 Cholesterol

Cholesterin,Cholesteryl alcohol,胆固醇

Estrogen Receptor/ERR; MRP; Endogenous Metabolite; ROR Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Cholesterol (Cholesteryl alcohol) 属于天然产物,是哺乳动物中的主要固醇,是一种雌激素相关受体 α (ERRα) 的激动剂。Cholesterol 广泛存在于动物的细胞膜,也是合成几种重要荷尔蒙及胆酸的材料。
T2968 Hyodeoxycholic acid

NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA

FXR; Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Hyodeoxycholic acid (NSC 60672) 是由肠道菌群在小肠中形成的次级胆汁酸,是TGR5(GPCR19)的激动剂, CHO 细胞中的EC50=31.6 µM。它已用于研究高胆固醇血症的治疗。
T1737 Genistein

NPI 031L,三叶草,染料木素,金雀异黄酮

Apoptosis; EGFR; Endogenous Metabolite; Autophagy Angiogenesis; Apoptosis; Autophagy; JAK/STAT signaling; Metabolism; Tyrosine Kinase/Adaptors
Genistein (NPI 031L) 是一种大豆异黄酮,是一种多重的酪氨酸激酶抑制剂,通过改变细胞凋亡,细胞周期和血管生成以及抑制转移对多种癌症有化疗作用。
T2822 Ginsenoside Rb1

Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III

ATPase; Mitophagy; IRAK; NF-κB; Autophagy; HSV Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Ginsenoside Rb1 (Gypenoside Ⅲ) 是中药人参的成分,可能具有抑制或阻止肿瘤生长的特性。
T6427 Butein

2’,3,4,4’-tetrahydroxy Chalcone,紫铆因

Apoptosis; EGFR; Others; PDE; Autophagy Angiogenesis; Apoptosis; Autophagy; JAK/STAT signaling; Metabolism; Others; Tyrosine Kinase/Adaptors
Butein (2’,3,4,4’-tetrahydroxy Chalcone) 是一种 cAMP 特异性PDE 抑制剂,也是蛋白酪氨酸激酶抑制剂,还是一种SIRT1激活剂。它通过 AKT 和 ERK/p38 MAPK 通路,靶向 FoxO3a 使 HeLa 细胞对 Cisplatin 敏感。
T1181 Gefitinib

ZD1839,吉非替尼

EGFR; Tyrosine Kinases; Autophagy Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Gefitinib (ZD1839) 是一种 EGFR 一代抑制剂,具有口服活性,抑制 EGFR 19 Del 和 L858R 突变。Gefitinib 具有抗肿瘤活性,用于治疗 EGFR 突变的非小细胞肺癌。Gefitinib 用药会产生 EGFR C797S 耐药突变。
T1205 Chloramphenicol

Chlornitromycin,Levomycetin,Chloromycetin,氯霉素

ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
T2851 Daphnetin

7,8-Dihydroxycoumarin,Daphnetol,瑞香素

EGFR; PKA; PKC; Parasite; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物,有抗氧化、抗炎、抗疟疾和解热作用,可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。
TN1440 Beta-Hydroxyisovalerylshikonin

EGFR; Tyrosine Kinases; Prostaglandin Receptor; Src; AMPK; Fatty Acid Synthase Angiogenesis; Chromatin/Epigenetic; GPCR/G Protein; Immunology/Inflammation; JAK/STAT signaling; Metabolism; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Beta-hydroxyisovalerylshikonin 是分离自Lithospermium radix 的天然产物,具有抑制PTK 的作用, 对 EGFR 和 v-Src 受体作用的IC50分别为 0.7 μM 和 1 μM。它对多种肿瘤细胞系均有抑制作用,可以高效诱导 NCI-H522 和 DMS114 细胞的死亡。
T4183 lavendustin A

RG-14355,NSC 678027,薰草菌素

EGFR; Tyrosinase Angiogenesis; JAK/STAT signaling; Proteases/Proteasome; Tyrosine Kinase/Adaptors
lavendustin A (RG-14355) 是从链霉菌中分离得到的一种天然产物,是细胞渗透性表皮生长因子受体 (EGFR) 酪氨酸激酶抑制剂,能抑制血管内皮生长因子诱导的血管生成,阻断 LTPGABA-A 的诱导。
T29078 Ursodeoxycholic acid sodium

UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,熊去氧胆酸钠盐,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium

FXR; Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) 是一种天然存在的次级胆汁酸,具有抗炎和细胞保护活性。Ursodeoxycholic acid sodium 作为信号分子,通过与胆汁酸激活受体相互作用发挥其作用,包括 G 蛋白偶联胆汁酸受体 5 (TGR5) 和法尼醇 X 受体 (FXR)。
T8789 N-Acetyl-L-tryptophan

N-acetyltryptophan,N-乙酰-L-色氨酸

Endogenous Metabolite; Neurokinin receptor GPCR/G Protein; Metabolism; Neuroscience
N-Acetyl-L-tryptophan (N-acetyltryptophan) 是内源性代谢产物的一种。
T4429 Rauwolscine hydrochloride

Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) 是一种高选择性的 α2 adrenergic 受体拮抗剂,Ki=12 nM。
TP2167 β-CGRP, human acetate

β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate

CGRP Receptor GPCR/G Protein; Neuroscience
β-CGRP, human acetate 是降钙素肽之一,通过受体活性修饰蛋白 (RAMP) 和降钙素受体样受体 (CRLR) 的复合物发挥作用(对于 CRLR/RAMP1 和 CRLR,IC50:1 nM 和 300 nM /RAMP2 在单元格中)。
T2S1992 Perillartine

Perilla sugar,Peryllartine,紫苏葶,DL-Perillartine

Others; Endogenous Metabolite Metabolism; Others
Perillartine (DL-Perillartine) 是甜味剂,能够激活味觉受体 1 型成员 2 。
T2766 Arctiin

Arctigenin-4-glucoside,Arctii,NSC 315527,牛蒡子苷

Adiponectin receptor GPCR/G Protein
Arctiin (Arctigenin-4-glucoside) 是一种从牛蒡种子中提取的植物木酚素,具有抗癌作用。
TL0006 Cichoric Acid

菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。
T7060 Amantadine

1-Aminoadamantane,1-金刚烷胺,金刚烷胺,1-Adamantanamine,1-Adamantylamine

Others Others
Amantadine (1-Aminoadamantane) 是抗病毒药物,也是是 NMDA 型谷氨酸受体的弱拮抗剂,能促进高多巴胺的释放,并阻断多巴胺的再摄取。
T1168 Desonide

Tridesilon,地索奈德,Locapred,Prednacinolone

Glucocorticoid Receptor Endocrinology/Hormones
Desonide (Prednacinolone) 是一种非氟化皮质类固醇抗炎剂,能够作用于糖皮质激素受体。
T6S0109 Sipeimine

Kashmirine,西贝母碱,Imperialine,西贝碱

Others Others
Sipeimine (Kashmirine) 是一种天然产物,从平贝母中分离得到。
TN1377 α-Spinasterol

Α-波菜甾醇,alpha-Spinasterol,菠甾醇

COX; Antibacterial; TRP/TRPV Channel Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
α-Spinasterol 是一种从Spinacia oleracea 分离的瞬时受体电位香草酸 1 拮抗剂,具有抗菌、抗炎、抗抑郁、抗氧化和抗伤害作用。它抑制COX-1和COX-2活性,IC50值分别为 16.17 μM 和 7.76 μM。
T4S0295 Apigenin 7-glucoside

波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Apigenin 7-glucoside (Cosmosiin) 是一种 ROS 清除剂,具有抗增殖、抗氧化作用。
TN3575 (±)-Cannabichromene

Cannabichromene,大麻色原烯,Cannabichrome

Cannabinoid Receptor GPCR/G Protein
(±)-Cannabichromene 是一种发现于大麻的 2,2-dimethyl-2H-chromene 衍生物。
T3385 Gypenoside XVII

GP-17,Gynosaponin S,七叶胆苷XVII

Estrogen Receptor/ERR; GSK-3; Endogenous Metabolite Endocrinology/Hormones; Metabolism; PI3K/Akt/mTOR signaling; Stem Cells
Gypenoside XVII (Gynosaponin S) 是一种绞股蓝皂甙类的新型植物雌激素,能够激活雌激素受体。
TN5131 Tetrahydrocannabivarin

THCV,delta9-Tetrahydrocannabivarin,CRM,Tetrahydrocannavarin

Cannabinoid Receptor GPCR/G Protein
Tetrahydrocannabivarin (CRM) 是 cannabinoid type 1 receptor 的中性拮抗剂,对 2 型糖尿病有潜在治疗价值。
T8689 Chloroquine

CQ,氯喹

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine 是一种 Toll 样受体抑制剂,可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性,广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。
T4710 3-Methoxytyramine hydrochloride

3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐

Others; Endogenous Metabolite; Drug Metabolite Metabolism; Others
3-Methoxytyramine hydrochloride (3-O-methyl Dopamine hydrochloride) 是多巴胺的无活性代谢物,能够活化痕量胺相关受体1
TN1677 Gartanin

1,3,5,8-四羟基-2,4-双(3-甲基-2-丁烯基)-9H-氧杂蒽-9-酮,藤黄苷

BCL; Caspase; JNK Apoptosis; MAPK; Proteases/Proteasome
Gartanin 是山竹果中的一种天然黄酮,具有抗氧化、抗真菌、抗炎、神经保护和抗肿瘤活性。它能够诱导人脑胶质瘤细胞的细胞周期阻滞和自噬,抑制其迁移。
TN6694 5,6-Benzoflavone

β-Naphthoflavone,beta-NF

Antioxidant oxidation-reduction
5,6-Benzoflavone (β-Naphthoflavone) 是芳烃受体的外源配体,可破坏人肝癌 HepG2 细胞中的锌稳态。5,6-Benzoflavone (β-Naphthoflavone) 具有抗炎和抗氧化活性,抑制通过 AKT/Nrf-2/HO-1-NF-kappaB 信号转导轴,抑制 LPS 诱导的炎症,抑制TNF-α诱导的ICAM-1和VCAM-1表达,可用于研究神经退行性疾病。
TN1567 Delphinidin chloride

Estrogen Receptor/ERR; VEGFR Angiogenesis; Endocrinology/Hormones; Tyrosine Kinase/Adaptors
Delphinidin chloride 是一种花青素,是一种可从浆果和红酒中分离得到的天然植物色素,是某些花青素的前体。Delphinidin chloride 诱导血管内皮释放一氧化氮,引起血管松弛。在1 ~ 40 μM 剂量下,对上皮生长因子受体的信号传导和雌激素受体α的表达有抑制作用,与细胞凋亡和自噬有关。Delphinidin chloride 能调节 JAK/STAT3 和 MAPKinase 信号传导。Delphinidin 还能抑制 p300/CBP 的组蛋白乙酰转移酶活性(IC50 在约为30 μM)
T3369 Nuciferine

(-)-Nuciferine,VLT 049,荷叶碱,Sanjoinine E

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Nuciferine ((-)-Nuciferine) 是一种在埃及蓝睡莲和水芙蓉中发现的生物碱,是5-HT2A、5-HT2B 和5-HT2C 拮抗剂,IC50分别为 478 nM、1 μM 和 131 nM。它也是5-HT7的反向激动剂,IC50为 150 nM。
T2915 Bardoxolone

RTA 401,齐墩果烷三萜化合物,CDDO

Others; Nrf2 Immunology/Inflammation; Others
Bardoxolone (CDDO) 是新型核调节因子激活剂。
T2768 Saikosaponin A

柴胡皂苷A,柴胡皂苷 A

NF-κB; Antibacterial; Liver X Receptor Metabolism; Microbiology/Virology; NF-κB
Saikosaponin A 是银柴胡中的主要活性成分,有抗炎活性,可上调 LXRα的表达。
T4973 Paraxanthine

1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE

Endogenous Metabolite Metabolism
Paraxanthine (1,7-dimethylxanthine) 是一种 caffeine 的代谢物,能够刺激Ryanodine 受体通道来抑制多巴胺能细胞的死亡。
------------------------ 更多 ------------------------

天然产物

Estrone
Cat.No: T1009
Synonym: Oestrone,雌酮,Fluoroethyl,Aquacrine
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Prostaglandin E1
Cat.No: T1626
Synonym: 前列地尔,PGE1,列腺素E1,Alprostadil
Target: Endogenous Metabolite, Prostaglandin Receptor
Procyanidin B1
Cat.No: TQ0205
Synonym: 原花青素B1,原花青素 B1
Target: TLR
Tetrahydropalmatine hydrochloride
Cat.No: T2917
Synonym: 延胡索乙素盐酸盐,1-Tetrahydropalmitine HCl,Gindarine hydrochloride,盐酸延胡乙素
Target: Others, Dopamine Receptor
Methyl 2,5-dihydroxycinnamate
Cat.No: T22974
Synonym:
Target: EGFR
Cyasterone
Cat.No: T3870
Synonym: 杯苋甾酮,Cyasteron
Target: Apoptosis, EGFR
Voacamine
Cat.No: T2S0271
Synonym: 老刺木胺,Voacanginine
Target: Cannabinoid Receptor, P-gp
Ginsenoside Rh1
Cat.No: T2932
Synonym: Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1
Target: IL Receptor, TNF, Endogenous Metabolite, PPAR, Interleukin
Deoxycholic acid sodium salt
Cat.No: T5077
Synonym: 脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate
Target: Endogenous Metabolite, GPCR19
Khellin
Cat.No: T1431
Synonym: 凯林,Amicardine,Methafrone,Visammin
Target: EGFR, Others
Sulforaphene
Cat.No: TL0016
Synonym: 油菜
Target: Apoptosis, ERK, EGFR, NF-κB
Shanzhiside methyl ester
Cat.No: T3896
Synonym: 三栀子甙甲酯,山芝皂苷甲酯
Target: Glucagon Receptor
Deoxycholic acid
Cat.No: T2965
Synonym: Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
PCO371
Cat.No: T16442
Synonym: 2,4-Imidazolidinedione, 1-(3,5-dimethyl-4-(2-((4-oxo-2-(4-(trifluoromethoxy)phenyl)-1,3,8-triazaspiro(4.5)dec-1-en-8-yl)sulfonyl)ethyl)phenyl)-5,5-dimethyl-
Target: Thyroid hormone receptor(THR)
Ursodeoxycholic acid
Cat.No: T0700
Synonym: 熊去氧胆酸,UDCA,Ursodiol
Target: Potassium Channel, Endogenous Metabolite
Chrysophanol
Cat.No: T2995
Synonym: 大黄酚,3-Methylchrysazin,Chrysophanic Acid,Turkey Rhubarb
Target: EGFR
Cholesterol
Cat.No: T0760
Synonym: Cholesterin,Cholesteryl alcohol,胆固醇
Target: Estrogen Receptor/ERR, MRP, Endogenous Metabolite, ROR
Hyodeoxycholic acid
Cat.No: T2968
Synonym: NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA
Target: FXR, Endogenous Metabolite, GPCR19
Genistein
Cat.No: T1737
Synonym: NPI 031L,三叶草,染料木素,金雀异黄酮
Target: Apoptosis, EGFR, Endogenous Metabolite, Autophagy
Ginsenoside Rb1
Cat.No: T2822
Synonym: Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III
Target: ATPase, Mitophagy, IRAK, NF-κB, Autophagy, HSV
Butein
Cat.No: T6427
Synonym: 2’,3,4,4’-tetrahydroxy Chalcone,紫铆因
Target: Apoptosis, EGFR, Others, PDE, Autophagy
Gefitinib
Cat.No: T1181
Synonym: ZD1839,吉非替尼
Target: EGFR, Tyrosine Kinases, Autophagy
Chloramphenicol
Cat.No: T1205
Synonym: Chlornitromycin,Levomycetin,Chloromycetin,氯霉素
Target: ribosome, HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
Daphnetin
Cat.No: T2851
Synonym: 7,8-Dihydroxycoumarin,Daphnetol,瑞香素
Target: EGFR, PKA, PKC, Parasite, Autophagy
Beta-Hydroxyisovalerylshikonin
Cat.No: TN1440
Synonym:
Target: EGFR, Tyrosine Kinases, Prostaglandin Receptor, Src, AMPK, Fatty Acid Synthase
lavendustin A
Cat.No: T4183
Synonym: RG-14355,NSC 678027,薰草菌素
Target: EGFR, Tyrosinase
Ursodeoxycholic acid sodium
Cat.No: T29078
Synonym: UDCA Na,UDCA sodium,Sodium Ursodeoxycholate,熊去氧胆酸钠盐,Ursodiol sodium,Ursodeoxycholic Acid (sodium salt),Ursodeoxycholate sodium
Target: FXR, Endogenous Metabolite, GPCR19
N-Acetyl-L-tryptophan
Cat.No: T8789
Synonym: N-acetyltryptophan,N-乙酰-L-色氨酸
Target: Endogenous Metabolite, Neurokinin receptor
Rauwolscine hydrochloride
Cat.No: T4429
Synonym: Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
β-CGRP, human acetate
Cat.No: TP2167
Synonym: β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate
Target: CGRP Receptor
Perillartine
Cat.No: T2S1992
Synonym: Perilla sugar,Peryllartine,紫苏葶,DL-Perillartine
Target: Others, Endogenous Metabolite
Arctiin
Cat.No: T2766
Synonym: Arctigenin-4-glucoside,Arctii,NSC 315527,牛蒡子苷
Target: Adiponectin receptor
Cichoric Acid
Cat.No: TL0006
Synonym: 菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid
Target: Reactive Oxygen Species, HIV Protease
Amantadine
Cat.No: T7060
Synonym: 1-Aminoadamantane,1-金刚烷胺,金刚烷胺,1-Adamantanamine,1-Adamantylamine
Target: Others
Desonide
Cat.No: T1168
Synonym: Tridesilon,地索奈德,Locapred,Prednacinolone
Target: Glucocorticoid Receptor
Sipeimine
Cat.No: T6S0109
Synonym: Kashmirine,西贝母碱,Imperialine,西贝碱
Target: Others
α-Spinasterol
Cat.No: TN1377
Synonym: Α-波菜甾醇,alpha-Spinasterol,菠甾醇
Target: COX, Antibacterial, TRP/TRPV Channel
Apigenin 7-glucoside
Cat.No: T4S0295
Synonym: 波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin
Target: Reactive Oxygen Species, HIV Protease
(±)-Cannabichromene
Cat.No: TN3575
Synonym: Cannabichromene,大麻色原烯,Cannabichrome
Target: Cannabinoid Receptor
Gypenoside XVII
Cat.No: T3385
Synonym: GP-17,Gynosaponin S,七叶胆苷XVII
Target: Estrogen Receptor/ERR, GSK-3, Endogenous Metabolite
Tetrahydrocannabivarin
Cat.No: TN5131
Synonym: THCV,delta9-Tetrahydrocannabivarin,CRM,Tetrahydrocannavarin
Target: Cannabinoid Receptor
Chloroquine
Cat.No: T8689
Synonym: CQ,氯喹
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
3-Methoxytyramine hydrochloride
Cat.No: T4710
Synonym: 3-O-methyl Dopamine hydrochloride,3-O-methyl Dopamine hydrochloride),3-O-甲基多巴胺盐酸盐
Target: Others, Endogenous Metabolite, Drug Metabolite
Gartanin
Cat.No: TN1677
Synonym: 1,3,5,8-四羟基-2,4-双(3-甲基-2-丁烯基)-9H-氧杂蒽-9-酮,藤黄苷
Target: BCL, Caspase, JNK
5,6-Benzoflavone
Cat.No: TN6694
Synonym: β-Naphthoflavone,beta-NF
Target: Antioxidant
Delphinidin chloride
Cat.No: TN1567
Synonym:
Target: Estrogen Receptor/ERR, VEGFR
Nuciferine
Cat.No: T3369
Synonym: (-)-Nuciferine,VLT 049,荷叶碱,Sanjoinine E
Target: Dopamine Receptor, 5-HT Receptor
Bardoxolone
Cat.No: T2915
Synonym: RTA 401,齐墩果烷三萜化合物,CDDO
Target: Others, Nrf2
Saikosaponin A
Cat.No: T2768
Synonym: 柴胡皂苷A,柴胡皂苷 A
Target: NF-κB, Antibacterial, Liver X Receptor
Paraxanthine
Cat.No: T4973
Synonym: 1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE
Target: Endogenous Metabolite
--------- 更多 ---------
共2628条,每页50条 1 2 3 4 5 ... 53
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼