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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TP2198 Platelet Membrane Glycoprotein IIB Peptide (296-306)

Others Others
GPllb is composed of a 125 Kd heavy chain that is disulfide-linked to a 23 Kd light chain. Hydropathicity analysis of the cDNA sequence indicates that GPllb is anchored to the platelet through a single transmembrane domain located within 20 amino acids of
T81824 Membrane-Permeable Sequence, MPS

Membrane-Permeable Sequence(MPS)是一种CPP,常用于研究跨膜机制。
T80209 Human membrane-bound PD-L1 polypeptide

PD-1/PD-L1 Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation
Human membrane-bound PD-L1 polypeptide 作为抗原,可诱导生成相应的PD-L1抗体。
T9423 Alkyne tyramide

Others Others
Alkyne tyramide 是抗坏血酸过氧化物酶 2 探针。它有助于鉴定 APEX 标记位点,明确线粒体蛋白的膜拓扑的分配。它显著提高了完整酵母细胞的 APEX 标记效率,比 APEX2 底物生物素苯酚具有更大的细胞壁渗透性。
T83737 LRRKtide TFA

Moesin (550-564),Membrane-organizing Extension Spike Protein (550-564)

LRRKtide是一个针对富含亮氨酸重复激酶2 (LRRK2)的肽基底物,LRRK2是在帕金森病患者中频繁发生突变的酶,对应于膜组织扩展刺突蛋白(moesin)的550-564氨基酸。该化合物用于识别LRRK2的抑制剂。
T21992 Vacuolin-1

PI3K; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Vacuolin-1 是一种细胞渗透性抑制剂,可抑制 Ca2+ 依赖性溶酶体与细胞膜的融合。它通过抑制溶酶体内容物的释放起作用。它是一种有效的选择性 PIKfyve 抑制剂,通过损害溶酶体成熟来抑制晚期自噬。
T83705 BING TFA

Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria

BING是一种来源于日本稻田鱼(O. laptipes)的抗菌肽,由液泡蛋白质分选相关蛋白13D样(Vps13D)衍生而来。对包括耐甲氧西林的金黄色葡萄球菌(MRSA; MICs = 4-64 µg/ml)在内的各种革兰氏阴性和革兰氏阳性细菌都有活性。与氨苄西林、阿莫西林和新霉素共同使用时,对抗铜绿假单胞菌(P. aeruginosa)表现出协同效应,并能抑制大肠杆菌(E. coli)对卡那霉素和氨苄西林的抗药性发展。在体内,BING提高了被鳗弧菌(E. tarda)感染的O. laptipes的生存率。
T11520 GW806742X

MLK; VEGFR Angiogenesis; MAPK; Tyrosine Kinase/Adaptors
GW806742X 是ATP 模拟物,是MLKL 抑制剂,可结合 MLKL 假激酶结构域,Kd 值为 9.3μM。它对VEGFR2的IC50为 2 nM,延缓 MLKL 膜移位并抑制坏死。
T8995 NCGC00262650

Others; Src Angiogenesis; Others; Tyrosine Kinase/Adaptors
NCGC00262650 是 AMA1-RON2 相互作用和 c-Src 酪氨酸激酶活性的抑制剂。
T8946 Indophagolin

P2X Receptor; 5-HT Receptor; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Indophagolin 是一种有效的含有二氢吲哚的自噬抑制剂,IC50 为 140 nM。它拮抗 Gq 蛋白偶联的 P2Y4、P2Y6和 P2Y11受体。它还拮抗嘌呤能受体 P2X4 以及 P2X1 和 P2X3,IC50 分别为 2.71、2.40 和 3.49 μM。
T8851 I3MT-3

HMPSNE

Hippo pathway Stem Cells
I3MT-3 (HMPSNE) 是一种有效的、具有细胞膜渗透性的、选择性的 3-巯基丙酮酸硫转移酶 (3MST)的抑制剂,IC50值为2.7 μM,对其他硫化氢/磺胺制硫酶没有活性。它靶向位于 3MST 活性位点的过硫半胱氨酸残基。
T9915 Eculizumab

Complement System Immunology/Inflammation
Eculizumab 是针对补体 C5 的长效人源化单克隆抗体。它对 C5 裂解为 C5a 和 C5b 具有抑制作用,并抑制了末端补体系统的部署,其中包括膜攻击复合物的形成。它可用于溶血的研究。
T14984 CLP257

Potassium Channel Membrane transporter/Ion channel
CLP257 是有效的 K+-Cl- 协同转运蛋白 KCC2 选择性激活剂 (EC50: 616 nM)。它可减轻神经性疼痛大鼠的超敏反应,并在翻译后调节质膜 KCC2 蛋白周转。它在 KCC2 活性降低的神经元中恢复受损的 Cl- 转运。
T5827 BI-6C9

Apoptosis; Others; Mitochondrial Metabolism Apoptosis; Metabolism; Others
BI-6C9 是一种高特异性的 BH3 相互作用结构域抑制剂,可阻止线粒体外膜电位和线粒体分裂,并保护细胞免受线粒体凋亡诱导因子释放和不依赖 caspase 的细胞死亡。
T10952 Dabuzalgron

达布扎琼,Ro 115-1240

Apoptosis; Adrenergic Receptor Apoptosis; GPCR/G Protein; Neuroscience
Dabuzalgron (Ro 115-1240) 是一种口服活性选择性 α-1A 肾上腺素受体激动剂,用于治疗尿失禁。它通过维持线粒体功能来预防多柔比星引起的心脏毒性。
T11282 FGTI-2734

Transferase Metabolism
FGTI-2734 是 有效的RAS C-末端法尼基转移酶 (FT) 和香叶烯基转移酶-1 (GGT-1) 抑制剂,IC50s 分别为 250 nM 和 520 nM。 它可以阻断 KRAS 的膜定位,从而解决 KRAS 耐药性问题,并抑制突变的 KRAS 胰腺肿瘤。
T2298 ML204

TRP/TRPV Channel Membrane transporter/Ion channel
ML204 是有效的TRPC4/TRPC5通道选择性抑制剂,相比于 TRPC6 ,对TRPC4/TRPC5通道的选择性高出 19 倍,不影响其他的 TRP 通道和电压门控的钠、钾或 Ca2+通道。
T40996 Coppersensor 1

Coppersensor 1,CS1

Others Others
Coppersensor 1 (CS1) 是一种基于硼二吡咯亚甲基的荧光传感器,用于选择性和灵敏地检测生物样品中的铜 (I) 离子 (Cu + )。 Coppersensor 1 可以使用任何类型的荧光显微镜进行成像,包括落射荧光、共焦和多光子。
T19729 Dodecylphosphocholine

FOS-维生素B-12,DPC,n C12PC,Foscholine-12,DDPPC,nC12PC,n-C12PC

Others Others
Dodecylphosphocholine (DPC) 是一种去污剂,普遍用于膜蛋白核磁共振的研究。
T17217 Vamorolone

地塞米松EP杂质E,VBP15

Glucocorticoid Receptor; NF-κB Endocrinology/Hormones; NF-κB
Vamorolone (VBP15) 是一种首创的,具有口服活性的解离性类固醇 (dissociative steroidal) 抗炎药和膜稳定剂。它抑制 (NF-κB) 抑制作用,并降低了激素的影响。它改善肌营养不良,无副作用。
T6658 SB-408124

N-(6,8-二氟-2-甲基-4-喹啉)- N-[4-(二甲氨基)苯基]尿素

OX Receptor GPCR/G Protein; Neuroscience
SB408124 是一种 OX1 受体的非肽拮抗剂,在全细胞和膜中的 Ki 值分别为 57 和 27 nM,其选择性是 OX2 受体的 50 倍。
T1000L Chlorhexidine diacetate

醋酸氯己定,Hibitane diacetate,Chlorhexidine Acetate,Bactigras

CAT; Antibacterial; Antibiotic; Antifection Microbiology/Virology; oxidation-reduction
Chlorhexidine diacetate (Bactigras) 是一种双胍类杀菌剂,能快速消灭革兰氏阳性菌和革兰氏阴性菌。它也用作漱口水以防止口腔菌斑。
T22665 PD 128042

CI 976

Acyltransferase Metabolism
PD 128042 (CI 976) 是口服有效的ACAT (酰基辅酶 A: 胆固醇酰基转移酶)选择性抑制剂。它也是LPAT(溶血磷脂酰基转移酶) 抑制剂。它抑制高尔基体相关 LPAT 活性 (IC50=15 μM)。它抑制多种膜运输步骤,包括在内吞和分泌途径中发现的步骤。
T20843 Aplodan

Nergize,Creatinolfosfate,磷酸肌肉醇,creatinol-O-phosphate,Creatinolfosfate, Creatinol Phosphate

Others Others
Aplodan (creatinol-O-phosphate) 表现出抗缺血和抗心律失常的能力以及对细胞膜的保护作用。 Aplodan 可用于缺血性心脏病或伴有持续性室性早搏的缺血性心脏病的研究。
T8978 DD1

3,3'-Diamino-4'-methoxyflavone,HUN85111

Proteasome Proteases/Proteasome; Ubiquitination
DD1 (HUN85111) 是一种蛋白酶体抑制剂,可诱导人髓系肿瘤选择性凋亡。
T18893 5(6)-Carboxyfluorescein

5(6)-羧基荧光素,5-(and-6)-Carboxyfluorescein mixed isomers,5(6)-FAM

Others Others
5(6)-Carboxyfluorescein (5-(and-6)-Carboxyfluorescein mixed isomers) 是一种胺反应性 pH 敏感的绿色荧光标记物,能够标记蛋白质、多肽和氨基酸,可用于体内实验检测肿瘤位置。
T1460 Dicyclomine hydrochloride

AChR Neuroscience
Dicyclomine hydrochloride 是口服活性毒蕈碱胆碱能受体拮抗剂。它是一种抗痉挛试剂,在体内可缓解胃肠道平滑肌痉挛。它对 M1 受体亚型和 M2 受体亚型,Ki 分别为5.1和54.6nM,在刷状缘膜和基底质膜中均表现出较高的亲和力。
T14490 Talipexole dihydrochloride

Domnin,盐酸他利克索,B-HT 920 dihydrochloride

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Talipexole dihydrochloride (Domnin) 是一种多巴胺 D2 受体激动剂、α2-肾上腺素受体激动剂和 5-HT3 受体拮抗剂,有抗帕金森病活性。
T11217 Eplivanserin

依利色林,SR-46349

5-HT Receptor GPCR/G Protein; Neuroscience
Eplivanserin (SR-46349) 是一种有效和特异性的 5-HT2A 受体拮抗剂,Kd 值为 1.14 nM,在大鼠皮质膜中 IC50 值为 5.8 nM。
T6063 LY-411575

LY411575

Apoptosis; Gamma-secretase Apoptosis; Neuroscience; Proteases/Proteasome; Stem Cells
LY-411575 是一种高效的γ-secretase 抑制剂,能够抑制 Aβ40 蛋白的产生,在膜中的 IC50 为 0.078 nM,在细胞中为 0.082 nM。 它还抑制 Notch 切割,IC50 为 0.39 nM。
T0386L Ropivacaine

LEA-103 HCl,罗哌卡因

Potassium Channel; Sodium Channel Membrane transporter/Ion channel
Ropivacaine (LEA-103 HCl) 是有效的钠通道阻断剂,通过可逆地抑制钠离子内流从而引起神经纤维脉冲传导阻滞。Ropivacaine 也是一种 K2P(双孔钾通道)TREK-1的抑制剂,在 COS-7 细胞膜上的 IC50值为 402.7 μM。Ropivacaine 可以用于神经性疼痛的缓解的相关研究。
T15947 MAC13243 HCl

Antibacterial Microbiology/Virology
MAC13243 HCl 是一种将脂蛋白从内膜运输到外膜的周质伴侣LolA的抑制剂,是一种具有特异性的抗菌剂,对革兰氏阴性菌抑制作用显著。
T9293 SSAA09E3

SARS-CoV Microbiology/Virology
SSAA09E3 是一种新型 SARS-CoV 复制抑制剂,通过阻止病毒膜与宿主细胞膜融合而起作用。
T0030 Bupivacaine hydrochloride

Vivacaine,Bupivacaine HCl,盐酸布比卡因

Sodium Channel Membrane transporter/Ion channel
Bupivacaine hydrochloride (Vivacaine) 是NMDA 受体抑制剂,可用于慢性疼痛的研究。它可阻断钠、L-钙和钾通道,还阻断SCN5A 通道,IC50为 69.5 μM。
T6645 Ropivacaine hydrochloride monohydrate

Ropivacaine HCl,Ropivacaine HCl monohydrate,LEA 103,盐酸罗哌卡因,盐酸罗哌卡因一水合物,LEA-103 HCl

Potassium Channel; Sodium Channel Membrane transporter/Ion channel
Ropivacaine hydrochloride monohydrate (LEA-103 HCl) 是钠通道阻断剂,通过可逆地抑制钠离子内流从而引起神经纤维脉冲传导阻滞。Ropivacaine HCl monohydrate 也是 K2P(双孔钾通道)TREK-1的抑制剂。在动物实验模型中,Ropivacaine HCl monohydrate 可用于神经性疼痛的缓解。
T20642 Laurdan

6-十二酰基-N,N-二甲基-2-萘胺,6-Dodecanoyl-2-dimethylaminonaphthalene

Others Others
Laurdan (6-Dodecanoyl-2-dimethylaminonaphthalene) 是膜透性荧光探针。它的广义极化 (GP) 定量可用于磷脂相的鉴定,对与之结合的细胞膜磷脂相具有光谱敏感性。
T20992 MEGA-9

Nonanoyl-N-Methylglucamide

Serine Protease Proteases/Proteasome
MEGA-9 (Nonanoyl-N-Methylglucamide) 可溶解膜蛋白,可用作非离子去污剂。
T38651 Lauryl maltose neopentyl glycol

LMNG

Lauryl maltose neopentyl glycol (LMNG) 是一种能溶解和稳定膜蛋白的洗涤剂。Lauryl maltose neopentyl glycol 能从膜上提取完整的膜蛋白,从而改善G 蛋白偶联受体和呼吸系统复合物等膜蛋白的稳定性。Lauryl maltose neopentyl glycol 具有增溶作用。
T26829 Bitertanol

KWG-0599,联苯三唑醇,KWG0599,Baycor,Biloxazol,KWG 0599,Sibutol

Antifungal Microbiology/Virology
Bitertanol (KWG 0599) 是一种三唑类杀菌剂。 Bitertanol 抑制去甲基化,破坏膜功能,并阻止甾醇合成。
T19060 SPQ

Others Others
SPQ 可用于测量膜氯化物传输机制。
T83657 CCD Lipid01

LP-01

Others Others
CCD Lipid01 (LP-01) 是一种脂质膜,可用于输送生物活性制剂 。
T19068 TMA-DPH

Others Others
TMA-DPH 是疏水性荧光膜探针 (Ex=355 nm; Em=430 nm)。
T12608 QX-314 chloride

Sodium Channel Membrane transporter/Ion channel
QX-314 chloride 是钠离子通道电荷阻滞剂,具有膜不渗透性。
T83656 DLIN-MC4-DMA

Others Others
DLIN-MC4-DMA 是一种脂质膜,是一种潜在的核酸载体。
T3934 Isavuconazonium sulfate

Antifungal Microbiology/Virology
Isavuconazonium sulfate 是一种口服活性抗真菌药,是活性三唑类抗真菌药物 Isavuconazole 的前药,可用于侵袭性曲霉菌病和毛霉菌病。
T22714 Decynium 22

Others Others
Decynium 22 是有机阳离子转运蛋白和单胺转运蛋白的抑制剂,具有抗抑郁作用。
T64345 4-(Dimethylamino)phenol

Others Others
4-(Dimethylamino)phenol enhances extracellular lactate dehydrogenase (LDH) levels without significant effects on gluconeogenesis. Only when the membrane becomes permeable to LDH does 4-(Dimethylamino)phenol reduce ATP content.
T1290 Oxiconazole nitrate

硝酸奥昔康唑,Ro 13-8996

Others; Antibiotic; Antifection; Antifungal Microbiology/Virology; Others
Oxiconazole nitrate (Ro 13-8996) 是广谱抗真菌药物,抑制T. tonsurans 和T.rubrum 的生长,MIC90值分别为 0.25 和 0.5 μg/mL。
T0502 Zinc pyrithione

吡硫锌,OM-1563,吡啶硫酮锌

Proton pump; Antibacterial; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Zinc pyrithione (OM-1563) 通过阻断质子泵破坏膜转运,具有抗真菌和细菌作用。
T83654 Dilinoleyl Ketone

Bis(linoleyl) ketone

Others Others
Dilinoleyl Ketone (Bis(linoleyl) ketone) 是一种脂质膜,是一种潜在的核酸载体。

化合物

Platelet Membrane Glycoprotein IIB Peptide (296-306)
Cat.No: TP2198
Synonym:
Target: Others
Membrane-Permeable Sequence, MPS
Cat.No: T81824
Synonym:
Target:
Human membrane-bound PD-L1 polypeptide
Cat.No: T80209
Synonym:
Target: PD-1/PD-L1
Alkyne tyramide
Cat.No: T9423
Synonym:
Target: Others
LRRKtide TFA
Cat.No: T83737
Synonym: Moesin (550-564),Membrane-organizing Extension Spike Protein (550-564)
Target:
Vacuolin-1
Cat.No: T21992
Synonym:
Target: PI3K, Autophagy
BING TFA
Cat.No: T83705
Synonym: Blocker of Inter-membrane Stress Responses of Gram-negative Bacteria
Target:
GW806742X
Cat.No: T11520
Synonym:
Target: MLK, VEGFR
NCGC00262650
Cat.No: T8995
Synonym:
Target: Others, Src
Indophagolin
Cat.No: T8946
Synonym:
Target: P2X Receptor, 5-HT Receptor, Autophagy
I3MT-3
Cat.No: T8851
Synonym: HMPSNE
Target: Hippo pathway
Eculizumab
Cat.No: T9915
Synonym:
Target: Complement System
CLP257
Cat.No: T14984
Synonym:
Target: Potassium Channel
BI-6C9
Cat.No: T5827
Synonym:
Target: Apoptosis, Others, Mitochondrial Metabolism
Dabuzalgron
Cat.No: T10952
Synonym: 达布扎琼,Ro 115-1240
Target: Apoptosis, Adrenergic Receptor
FGTI-2734
Cat.No: T11282
Synonym:
Target: Transferase
ML204
Cat.No: T2298
Synonym:
Target: TRP/TRPV Channel
Coppersensor 1
Cat.No: T40996
Synonym: Coppersensor 1,CS1
Target: Others
Dodecylphosphocholine
Cat.No: T19729
Synonym: FOS-维生素B-12,DPC,n C12PC,Foscholine-12,DDPPC,nC12PC,n-C12PC
Target: Others
Vamorolone
Cat.No: T17217
Synonym: 地塞米松EP杂质E,VBP15
Target: Glucocorticoid Receptor, NF-κB
SB-408124
Cat.No: T6658
Synonym: N-(6,8-二氟-2-甲基-4-喹啉)- N-[4-(二甲氨基)苯基]尿素
Target: OX Receptor
Chlorhexidine diacetate
Cat.No: T1000L
Synonym: 醋酸氯己定,Hibitane diacetate,Chlorhexidine Acetate,Bactigras
Target: CAT, Antibacterial, Antibiotic, Antifection
PD 128042
Cat.No: T22665
Synonym: CI 976
Target: Acyltransferase
Aplodan
Cat.No: T20843
Synonym: Nergize,Creatinolfosfate,磷酸肌肉醇,creatinol-O-phosphate,Creatinolfosfate, Creatinol Phosphate
Target: Others
DD1
Cat.No: T8978
Synonym: 3,3'-Diamino-4'-methoxyflavone,HUN85111
Target: Proteasome
5(6)-Carboxyfluorescein
Cat.No: T18893
Synonym: 5(6)-羧基荧光素,5-(and-6)-Carboxyfluorescein mixed isomers,5(6)-FAM
Target: Others
Dicyclomine hydrochloride
Cat.No: T1460
Synonym:
Target: AChR
Talipexole dihydrochloride
Cat.No: T14490
Synonym: Domnin,盐酸他利克索,B-HT 920 dihydrochloride
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Eplivanserin
Cat.No: T11217
Synonym: 依利色林,SR-46349
Target: 5-HT Receptor
LY-411575
Cat.No: T6063
Synonym: LY411575
Target: Apoptosis, Gamma-secretase
Ropivacaine
Cat.No: T0386L
Synonym: LEA-103 HCl,罗哌卡因
Target: Potassium Channel, Sodium Channel
MAC13243 HCl
Cat.No: T15947
Synonym:
Target: Antibacterial
SSAA09E3
Cat.No: T9293
Synonym:
Target: SARS-CoV
Bupivacaine hydrochloride
Cat.No: T0030
Synonym: Vivacaine,Bupivacaine HCl,盐酸布比卡因
Target: Sodium Channel
Ropivacaine hydrochloride monohydrate
Cat.No: T6645
Synonym: Ropivacaine HCl,Ropivacaine HCl monohydrate,LEA 103,盐酸罗哌卡因,盐酸罗哌卡因一水合物,LEA-103 HCl
Target: Potassium Channel, Sodium Channel
Laurdan
Cat.No: T20642
Synonym: 6-十二酰基-N,N-二甲基-2-萘胺,6-Dodecanoyl-2-dimethylaminonaphthalene
Target: Others
MEGA-9
Cat.No: T20992
Synonym: Nonanoyl-N-Methylglucamide
Target: Serine Protease
Lauryl maltose neopentyl glycol
Cat.No: T38651
Synonym: LMNG
Target:
Bitertanol
Cat.No: T26829
Synonym: KWG-0599,联苯三唑醇,KWG0599,Baycor,Biloxazol,KWG 0599,Sibutol
Target: Antifungal
SPQ
Cat.No: T19060
Synonym:
Target: Others
CCD Lipid01
Cat.No: T83657
Synonym: LP-01
Target: Others
TMA-DPH
Cat.No: T19068
Synonym:
Target: Others
QX-314 chloride
Cat.No: T12608
Synonym:
Target: Sodium Channel
DLIN-MC4-DMA
Cat.No: T83656
Synonym:
Target: Others
Isavuconazonium sulfate
Cat.No: T3934
Synonym:
Target: Antifungal
Decynium 22
Cat.No: T22714
Synonym:
Target: Others
4-(Dimethylamino)phenol
Cat.No: T64345
Synonym:
Target: Others
Oxiconazole nitrate
Cat.No: T1290
Synonym: 硝酸奥昔康唑,Ro 13-8996
Target: Others, Antibiotic, Antifection, Antifungal
Zinc pyrithione
Cat.No: T0502
Synonym: 吡硫锌,OM-1563,吡啶硫酮锌
Target: Proton pump, Antibacterial, Antifungal
Dilinoleyl Ketone
Cat.No: T83654
Synonym: Bis(linoleyl) ketone
Target: Others
Cat. No. Product Name Target Signaling Pathways
T21164 Sulfentrazone

甲磺草胺,FP-846

Others Others
Sulfentrazone (FP-846) 是苯基三唑啉酮除草剂,能够抑制原卟啉原氧化酶,导致脂质细胞膜破裂,可用于控制某些阔叶和禾本科杂草。
T4947 3-Hydroxybutyric acid

Butanoic acid,3-羟基丁酸

Endogenous Metabolite Metabolism
3-Hydroxybutyric acid (Butanoic acid) 是一种人内源性代谢物,在 I 型糖尿病中升高。它能够调节膜脂的性质。
T4893 Spermidine

N-(3-Aminopropyl)-1,4-diaminobutane,亚精胺,N-(4-Aminobutyl)-1,3-diaminopropane

Endogenous Metabolite Metabolism
Spermidine (N-(3-Aminopropyl)-1,4-diaminobutane) 能够维持细胞膜稳定性,提高抗氧化酶活性,改善光系统 II 以及相关基因表达。它结合并激活 NMDA,并已显示以浓度依赖性方式增强 NMDA 诱导的电流。
T5080 Spermidine trihydrochloride

Spermidine hydrochloride,4-Azaoctamethylenediamine trihydrochloride,三盐酸亚精胺,亚精胺盐酸盐

NMDAR; Autophagy Autophagy; Neuroscience
Spermidine trihydrochloride (4-Azaoctamethylenediamine trihydrochloride) 能够维持细胞膜稳定性,提高抗氧化酶特性,改善光系统 II (PSII) 以及相关基因表达,也能够显著抑制 H2O2和 O2.-含量。
T16075 (Rac)-Idroxioleic acid

2-Hydroxyoleic acid,2-OHOA,2-羟基乳清酸,Minerval

Apoptosis Apoptosis
(Rac)-Idroxioleic acid (2-Hydroxyoleic acid) 是一种具有抗肿瘤作用的脂肪酸酰胺水解酶抑制剂。 它与质膜结合并改变脂质组织。
T5239 Cholesteryl sulfate sodium

Cholesterol 3-Sulfate Sodium Salt,胆固醇硫酸酯钠盐,Sodium Cholesteryl Sulfate

Endogenous Metabolite; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism
Cholesteryl sulfate sodium (Sodium Cholesteryl Sulfate) 是内源性代谢产物的一种。
TF0083 POPE

POPE 是从大肠杆菌中发现的化合物,是细胞膜的一部分,可用来研究改变细胞膜通透性。
TN2349 Taurodeoxycholate sodium salt

Sodium taurodeoxylate,牛磺脱氧胆酸钠

Endogenous Metabolite Metabolism
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
TN7022 Cymen-ar-ol

Antibacterial Microbiology/Virology
Cymen-ar-ol 是一种广谱高效的杀菌剂,可接触黏膜。
TN4675 Nortrachelogenin

(-)-Wikstromol,(-)-Nortrachelogenin

Apoptosis; Antifungal Apoptosis; Microbiology/Virology
Nortrachelogenin ((-)-Wikstromol) 可从 Partrinia scabiosaefolia 提取得到,具有抗真菌活性,可诱导膜破坏和半胱天冬酶依赖性细胞凋亡.
T4889 2,6-Diaminoheptanedioic acid

Others; Endogenous Metabolite Metabolism; Others
2,6-Diaminoheptanedioic acid 是内源性代谢产物的一种。
T3S0289 Araloside X

Calcium Channel Membrane transporter/Ion channel; Metabolism
Aralosides possess protective effect against experimental myocardial ischemia and infarction, the mechanism of myocardial protection may be attributed to the amelioration of FFA metabolic deterioration and membrane peroxidation induced by oxygen free radi
T35951 Alkaline Phosphatase

Others Others
Alkaline phosphatase 是一种膜结合糖蛋白,在碱性条件下可催化磷酸单酯的水解。它可用于分子生物学和酶免分析。
T38141 Glycerophospholipids, cephalins

Phosphatidylethanolamines (egg)

Glycerophospholipids, cephalins (Phosphatidylethanolamines (egg)) 是一种从鸡蛋中分离出来的磷脂酰乙醇胺的混合物,在 sn-1和 sn-2位置有各种脂肪酰基。Glycerophospholipids, cephalins 完全水解可得到1mol 的甘油、磷酸、乙醇胺和2mol 的脂肪酸。Phosphatidylethanolamines 在膜融合和细胞分裂过程中收缩环的拆卸中起作用,可调节膜的弯曲度。Phosphatidylethanolamines 能够在没有任何蛋白质或核酸的帮助下传播传染性朊病毒。Phosphatidylethanolamines 在细菌膜中的主要作用之一是分散由阴离子膜磷脂引起的负电荷。
T3237 Lecithin

Phospholutein,卵磷脂,L-α-磷脂酰胆碱,L-α-Phosphatidylcholine,Phosphatidylcholines

Others; Endogenous Metabolite Metabolism; Others
Lecithin (L-α-Phosphatidylcholine) 被认为是安全的常规磷脂源。磷脂能够改变动物细胞膜的脂肪酸组成和微观结构。
T13701 Genistein 8-c-glucoside

G8CG

Mitochondrial Metabolism Metabolism
Genistein 8-c-glucoside (G8CG) 诱导线粒体膜去极化从而导致细胞凋亡。Genistein 8-c-glucoside 是一种来源于 Lupinus luteus L.花中的天然葡萄糖苷。
T12451 Phosphoenolpyruvic acid tricyclohexylammoniu​m salt

PEP 3 CHA,phosphoenolpyruvic-acid-tricyclohexylammonium-salt,phosphoenolpyruvic-acid-tricyclohexylammoniu-m-salt,磷酸烯醇丙酮酸三(环已胺)盐

Others Others
Phosphoenolpyruvic acid tricyclohexylammoniu​m salt (PEP 3 CHA) 是一种能够透过细胞膜的糖酵解代谢物,含有高能磷酸基团,具有细胞保护和抗氧化作用。
T0146 Tioconazole

UK-20349,Vagistat,噻康唑

Antibiotic; Antifection; Antifungal Microbiology/Virology
Tioconazole (Vagistat) 是一种广谱性的抗真菌咪唑衍生物。它抑制几种皮肤真菌和几种酵母菌的 MIC50分别小于 3.12 mg/L 和 9 mg/L。
T6323 Oligomycin A

MCH 32,寡霉素A

ATPase; Antibiotic; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Oligomycin A (MCH 32) 是从链霉菌属中得到的一种线粒体F0F1-ATPase 抑制剂,抑制氧化磷酸化和线粒体偶联膜上发生的所有 ATP 依赖性过程。
T3771 Methyl protodioscin

山药,Smilax saponin B,NSC-698790

Apoptosis Apoptosis
Methyl protodioscin (Smilax saponin B) 是一种甾二糖苷,能诱导细胞周期阻滞,具有抗肿瘤活性。
TN2158 Robinetin

3,3',4',5',7-Pentahydroxyflavone,洋槐黄素

Anti-infection; HIV Protease; Antibacterial Microbiology/Virology; Proteases/Proteasome
Robinetin (3,3',4',5',7-Pentahydroxyflavone) 是一种天然黄酮,具有显著的“两种颜色”固有荧光特性。它具有抗真菌、抗病毒、抗菌、抗突变、抗氧化和抗自由基活性,高效抑制 EYPC 膜脂质过氧化和 HbA 糖基化。
T19554 L-Aspartic aicd sodium

L-Aspartic acid sodium,Sodium L-aspartate

Others; Sodium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
L-Aspartic aicd sodium (Sodium L-aspartate) 是一种氨基酸,是一种结肠特异性活性分子输送的前体活性分子,可促进大鼠前脑膜囊泡的 Na+外排。
T3S0156 Atractyloside potassium salt

Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐

Others Others
Atractyloside potassium salt (Atractyloside Dipotassium Salt) 是一种从苍术果实中分离出得到的二萜苷类化合物,具有毒性。它能抑制大鼠心脏线粒体膜的氯离子通道。它是高效、特异性的线粒体 ADP/ATP 转运 (ADP/ATP transport) 抑制剂。
T0131 Cepharanthine

NSC-623442,千金藤碱,千金藤素

Apoptosis; TNF; HIV Protease; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Cepharanthine (NSC-623442) 是从Stephania cepharanthaHayata 中提取的一种生物碱,具有抗炎、抗氧化作用。它可抑制肿瘤坏死因子 (TNF)-α 介导的 NFκB 刺激、质膜脂质过氧化和血小板聚集,并抑制细胞因子的产生。
T21437 DSPS

Phosphatidylserine(36:0),磷脂酰丝氨酸,Dioctadecanoylphosphatidylserine,Distearoyl phosphatidylserine

Others Others
DSPS (Dioctadecanoylphosphatidylserine) 是一种甘油磷脂,是重要的磷脂膜成分,在细胞周期信号传导中起关键作用。DSPS 可以调节细胞活性,介导细胞凋亡。DSPS 被广泛用作营养补充剂。
T41078 Lipopolysaccharides, Escherichiacoli (11C)

LPS E. coli O55:B5,Lipopolysaccharide, E. coli O111:B4

Others Others
Lipopolysaccharides, Escherichiacoli (11C) (LPS E. coli O55:B5)是革兰阴性菌外膜的大分子成分,由脂质a、寡糖核心和o -特异性多糖(O-antigen) 3个区域组成。
T3232 Higenamine hydrochloride

Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Higenamine hydrochloride (norcoclaurine HCl) 是一种 β2-AR 激动剂,是用于心力衰竭相关研究的中药乌头的关键成分,具有抗凋亡活性。
T4852 Trimyristin

Trimyristoylglycerol,Tritetradecanoin,三肉豆蔻酸甘油酯,Glyceryl trimyristate,甘油三肉豆蔻酸酯,1,2,3-Tritetradecanoylglycerol

Phosphatase; Endogenous Metabolite; AChE Metabolism; Neuroscience
Trimyristin (Tritetradecanoin) 是一种 Myristica fragransHoutt 的有效成分,能够显著抑制乙酰胆碱酯酶 (AChE),酸性和碱性磷酸酶 (ACP/ALP) 特性。它对 AChE,ACP 和 ALP 的 IC50分别为 0.11、0.16 和 0.18 mM。
T3S1319 (+)-Magnoflorine

Escholin,Magnoflorine,Thalictrin,Escholine,木兰花碱

Others; Antifungal Microbiology/Virology; Others
(+)-Magnoflorine (Thalictrin) 是从 Acoruscalamus 中分到的一种阿朴啡生物碱,可以减少 C. albicans 生物膜的形成,具有抗真菌、抗氧化、抗糖尿病、镇静和抗焦虑的作用。
T6702 Terbinafine

Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Terbinafine (TDT 067) 是念珠菌属的角鲨烯环氧化酶有效的非竞争性抑制剂,Ki 值为 30 nM。它具有抗真菌感染活性。
T11855 Lipopolysaccharides

脂多糖,LPS

Others Others
Lipopolysaccharides (LPS) 属于天然产物,是一种来源于革兰氏阴性菌外膜外叶的内毒素。Lipopolysaccharides 是一种高免疫原性抗原,可以增强免疫反应,可以用于炎症模型构建。
T6564 Leupeptin Hemisulfate

亮肽素

Serine Protease; Cysteine Protease Proteases/Proteasome
Leupeptin hemisulfate 是一种蛋白酶抑制剂,具有细胞膜渗透性、可逆性、竞争性和口服活性。Leupeptin hemisulfate 可以抑制 Cathepsin B、Cathepsin H、Cathepsin L 的活性,阻断两性溶酶体的融合。Leupeptin hemisulfate 还具有抗炎活性。
T5238 1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine

1,2-Dipalmitoyl-sn-glycero-3-PE,L-磷脂酰乙醇胺,1,2-Dipalmitoyl-sn-glycerol-3-Phosphoethanolamine,1,2-DPPE

Others; Endogenous Metabolite Metabolism; Others
1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine (DPPE) 是内源性代谢产物的一种。
T2732 (-)-Epicatechin gallate

表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG

Virus Protease; COX; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience
(-)-Epicatechin gallate ((-)-Epicatechin 3-O-gallate) 抑制环加氧酶-1 的IC50值为 7.5 μM。
TN1624 Ethyl cinnamate

Calcium Channel; ROS; NO Synthase Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Ethyl cinnamate 是食品香料和化妆品添加剂,也是哺乳动物组织的优良清除剂。
TN2160 Roemerine

(-)-Roemerine

Antibiotic Microbiology/Virology
Roemerine ((-)-Roemerine) 是一种来自塞内加尔番荔枝的卟啉生物碱,具有抗真菌和抗癌活性,通过抑制 Bmr 来防止小檗碱外排。Roemerine 以浓度依赖性方式增加细胞膜通透性,可用于研究真菌感染和前列腺癌。
T13708 Glycol chitosan

羟乙基脱乙酰壳多糖,乙二醇壳聚糖

Antibacterial Microbiology/Virology
Glycol chitosan 是具有亲水性乙二醇支链的壳聚糖衍生物。它抑制大肠杆菌,金黄色葡萄球菌和肠炎链球菌的生长,MIC 值分别为 4 μg/mL,32 μg/m L 和 <0.5 μg/mL。它可增强 Glycine max Harosoy 63W 细胞的膜通透性和渗漏。
T2P2806 Hederacolchiside A1

黑海常春藤苷A1,革叶常春藤皂苷 A1,Raddeanoside R13

Apoptosis; ERK; MEK; Akt; PI3K; Parasite; mTOR Apoptosis; Cytoskeletal Signaling; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling
Hederacolchiside A1 (Raddeanoside R13) 是从白头翁中分离的一种有抗利什曼原虫和抗肿瘤增殖活性的天然产物。
T8183 Deslanoside

洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C

ATPase; Drug Metabolite Membrane transporter/Ion channel; Metabolism
Deslanoside (Desacetyllanatoside C) 是一种快速作用的强心苷,可抑制Na-K-ATPase 膜泵,导致细胞内钠和钙浓度增加。它用于研究充血性心力衰竭和因折返机制引起的室上性心律失常,并在研究慢性心房颤动时控制心室率。
T3426 Bacoside A

MMP; Others; TNF; Dopamine Receptor; NOS; ROS Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience; Others; Proteases/Proteasome
Bacoside A has a possible anticancer activity that could be inducing cell cycle arrest and apoptosis through Notch pathway in GBM in vitro. It exerts cytoprotective efficacy by attenuation of ROS generated through oxidative stress by an increase in the concentration of antioxidant enzymes and sustain membrane integrity which leads to restoring the damage caused by tBHP. Bacoside A can able to inhibit the progression of Experimental Autoimmune Encephalomyelitis (EAE) may be by the inhibition of i...
T0034 Cortisone acetate

醋酸可的松,Cortisone 21-acetate,NSC 49420

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Cortisone acetate (NSC-49420) 是 Cortisol(一种糖皮质激素)的氧化代谢产物。它在高浓度下能够部分干预 Glucocorticoid 与Glucocorticoid-receptor 的结合。它具有免疫抑制和消炎的作用。
T5214 Cholesteryl linoleate

CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯

Others; Endogenous Metabolite Metabolism; Others
Cholesteryl linoleate (Linoleic Acid cholesteryl ester) 是低密度脂蛋白和动脉粥样硬化病变中主要的胆固醇酯。它存在于 LDL 中的胆固醇酯,利用 LDL 受体相关蛋白转移到表达 15-脂氧合酶的巨噬细胞和 CHO 细胞的质膜,被氧化形成胆固醇亚油酸氢过氧化物。
T0884 1-Docosanol

Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol

Antifection; HSV Microbiology/Virology
1-Docosanol (Behenic alcohol) 是一种具有抗病毒活性的饱和 22 碳脂肪醇,局部用于治疗复发性单纯性唇疱疹发作并缓解相关疼痛并可能有助于更快地治愈疮。
T5004 Hyaluronic acid sodium

透明质酸钠,Sodium Hyaluronate

Others Others
Hyaluronic acid sodium (Sodium Hyaluronate) 是一种生物聚合物,由二糖的重复单元组成,应用领域广泛。
T3388 Calycosin-7-O-β-D-glucoside

毛蕊异黄酮苷,calycosin-7-O-beta-D-glucopyranoside,Calycosin-7-O-beta-D-glucoside

MMP; Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB; Proteases/Proteasome
Calycosin-7-O-β-D-glucoside (calycosin-7-O-beta-D-glucopyranoside) 是一种异黄酮,从黄芪中分离得到。它具有多种生物活性,包括心脏保护、神经保护、抗炎和抗氧化作用。
T4S0800 Demethyleneberberine

P450; NOS; NF-κB; HIF; AMPK Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Demethyleneberberine 是从黄连中提取的一种天然产物,是线粒体靶向抗氧化剂。它也可作为AMPK 激活剂,用于非酒精性脂肪性肝病的研究。它通过抑制NF-κB 通路和调节 Th 细胞的平衡来减轻小鼠结肠炎并抑制炎症反应。
TN1853 Lariciresinol

(+)-落叶松树脂醇

VEGFR; Antifection Angiogenesis; Microbiology/Virology; Tyrosine Kinase/Adaptors
Lariciresinol 是一种肠木脂素前体,它通过破坏真菌质膜具有杀真菌活性,并具有作为治疗人类真菌感染性疾病的新型抗真菌剂的治疗潜力。膳食 lariciresinol 可以减缓乳腺肿瘤的生长并降低人 MCF-7 乳腺癌异种移植物和致癌物诱导的大鼠乳腺肿瘤的血管密度。
T2S2362 Dehydrocorydaline nitrate

去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱

BCL; Others; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Others; Proteases/Proteasome
Dehydrocorydaline nitrate 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达,激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌、抗疟疾等功效。
T5S1097 Neferine

(R)-1,2-Dimethoxyaporphine,(-)-Neferine,甲基莲心碱

Apoptosis; NF-κB; Autophagy Apoptosis; Autophagy; NF-κB
Neferine ((-)-Neferine) 是一种双苄基异喹啉类生物碱,可强效抑制NF-κB 激活,具有抗肿瘤活性。
T3926 Echinatin

刺甘草查尔酮,Retrochalcone

Free radical scavengers oxidation-reduction
Echinatin (Retrochalcone) 是分离自中草药甘草中,具有保肝和抗炎活性。在大鼠中,它可以被快速吸收和消除,并广泛分布,绝对生物利用度约为 6.81%。
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天然产物

Sulfentrazone
Cat.No: T21164
Synonym: 甲磺草胺,FP-846
Target: Others
3-Hydroxybutyric acid
Cat.No: T4947
Synonym: Butanoic acid,3-羟基丁酸
Target: Endogenous Metabolite
Spermidine
Cat.No: T4893
Synonym: N-(3-Aminopropyl)-1,4-diaminobutane,亚精胺,N-(4-Aminobutyl)-1,3-diaminopropane
Target: Endogenous Metabolite
Spermidine trihydrochloride
Cat.No: T5080
Synonym: Spermidine hydrochloride,4-Azaoctamethylenediamine trihydrochloride,三盐酸亚精胺,亚精胺盐酸盐
Target: NMDAR, Autophagy
(Rac)-Idroxioleic acid
Cat.No: T16075
Synonym: 2-Hydroxyoleic acid,2-OHOA,2-羟基乳清酸,Minerval
Target: Apoptosis
Cholesteryl sulfate sodium
Cat.No: T5239
Synonym: Cholesterol 3-Sulfate Sodium Salt,胆固醇硫酸酯钠盐,Sodium Cholesteryl Sulfate
Target: Endogenous Metabolite, PKC
POPE
Cat.No: TF0083
Synonym:
Target:
Taurodeoxycholate sodium salt
Cat.No: TN2349
Synonym: Sodium taurodeoxylate,牛磺脱氧胆酸钠
Target: Endogenous Metabolite
Cymen-ar-ol
Cat.No: TN7022
Synonym:
Target: Antibacterial
Nortrachelogenin
Cat.No: TN4675
Synonym: (-)-Wikstromol,(-)-Nortrachelogenin
Target: Apoptosis, Antifungal
2,6-Diaminoheptanedioic acid
Cat.No: T4889
Synonym:
Target: Others, Endogenous Metabolite
Araloside X
Cat.No: T3S0289
Synonym:
Target: Calcium Channel
Alkaline Phosphatase
Cat.No: T35951
Synonym:
Target: Others
Glycerophospholipids, cephalins
Cat.No: T38141
Synonym: Phosphatidylethanolamines (egg)
Target:
Lecithin
Cat.No: T3237
Synonym: Phospholutein,卵磷脂,L-α-磷脂酰胆碱,L-α-Phosphatidylcholine,Phosphatidylcholines
Target: Others, Endogenous Metabolite
Genistein 8-c-glucoside
Cat.No: T13701
Synonym: G8CG
Target: Mitochondrial Metabolism
Phosphoenolpyruvic acid tricyclohexylammoniu​m salt
Cat.No: T12451
Synonym: PEP 3 CHA,phosphoenolpyruvic-acid-tricyclohexylammonium-salt,phosphoenolpyruvic-acid-tricyclohexylammoniu-m-salt,磷酸烯醇丙酮酸三(环已胺)盐
Target: Others
Tioconazole
Cat.No: T0146
Synonym: UK-20349,Vagistat,噻康唑
Target: Antibiotic, Antifection, Antifungal
Oligomycin A
Cat.No: T6323
Synonym: MCH 32,寡霉素A
Target: ATPase, Antibiotic, Antifungal
Methyl protodioscin
Cat.No: T3771
Synonym: 山药,Smilax saponin B,NSC-698790
Target: Apoptosis
Robinetin
Cat.No: TN2158
Synonym: 3,3',4',5',7-Pentahydroxyflavone,洋槐黄素
Target: Anti-infection, HIV Protease, Antibacterial
L-Aspartic aicd sodium
Cat.No: T19554
Synonym: L-Aspartic acid sodium,Sodium L-aspartate
Target: Others, Sodium Channel, Endogenous Metabolite
Atractyloside potassium salt
Cat.No: T3S0156
Synonym: Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐
Target: Others
Cepharanthine
Cat.No: T0131
Synonym: NSC-623442,千金藤碱,千金藤素
Target: Apoptosis, TNF, HIV Protease, Autophagy
DSPS
Cat.No: T21437
Synonym: Phosphatidylserine(36:0),磷脂酰丝氨酸,Dioctadecanoylphosphatidylserine,Distearoyl phosphatidylserine
Target: Others
Lipopolysaccharides, Escherichiacoli (11C)
Cat.No: T41078
Synonym: LPS E. coli O55:B5,Lipopolysaccharide, E. coli O111:B4
Target: Others
Higenamine hydrochloride
Cat.No: T3232
Synonym: Higenamine HCl,Demethylcoclaurine hydrochloride,盐酸去甲乌头碱,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride
Target: Adrenergic Receptor
Trimyristin
Cat.No: T4852
Synonym: Trimyristoylglycerol,Tritetradecanoin,三肉豆蔻酸甘油酯,Glyceryl trimyristate,甘油三肉豆蔻酸酯,1,2,3-Tritetradecanoylglycerol
Target: Phosphatase, Endogenous Metabolite, AChE
(+)-Magnoflorine
Cat.No: T3S1319
Synonym: Escholin,Magnoflorine,Thalictrin,Escholine,木兰花碱
Target: Others, Antifungal
Terbinafine
Cat.No: T6702
Synonym: Terbinex,特比萘芬,SF 86-327,Lamisil,TDT 067
Target: Antibacterial, Antibiotic, Antifungal
Lipopolysaccharides
Cat.No: T11855
Synonym: 脂多糖,LPS
Target: Others
Leupeptin Hemisulfate
Cat.No: T6564
Synonym: 亮肽素
Target: Serine Protease, Cysteine Protease
1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine
Cat.No: T5238
Synonym: 1,2-Dipalmitoyl-sn-glycero-3-PE,L-磷脂酰乙醇胺,1,2-Dipalmitoyl-sn-glycerol-3-Phosphoethanolamine,1,2-DPPE
Target: Others, Endogenous Metabolite
(-)-Epicatechin gallate
Cat.No: T2732
Synonym: 表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG
Target: Virus Protease, COX, Autophagy
Ethyl cinnamate
Cat.No: TN1624
Synonym:
Target: Calcium Channel, ROS, NO Synthase
Roemerine
Cat.No: TN2160
Synonym: (-)-Roemerine
Target: Antibiotic
Glycol chitosan
Cat.No: T13708
Synonym: 羟乙基脱乙酰壳多糖,乙二醇壳聚糖
Target: Antibacterial
Hederacolchiside A1
Cat.No: T2P2806
Synonym: 黑海常春藤苷A1,革叶常春藤皂苷 A1,Raddeanoside R13
Target: Apoptosis, ERK, MEK, Akt, PI3K, Parasite, mTOR
Deslanoside
Cat.No: T8183
Synonym: 洋地黄,去乙酰西地兰,Desacetyllanatoside C,Deacetyllanatoside C
Target: ATPase, Drug Metabolite
Bacoside A
Cat.No: T3426
Synonym:
Target: MMP, Others, TNF, Dopamine Receptor, NOS, ROS
Cortisone acetate
Cat.No: T0034
Synonym: 醋酸可的松,Cortisone 21-acetate,NSC 49420
Target: Glucocorticoid Receptor, Endogenous Metabolite
Cholesteryl linoleate
Cat.No: T5214
Synonym: CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯
Target: Others, Endogenous Metabolite
1-Docosanol
Cat.No: T0884
Synonym: Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol
Target: Antifection, HSV
Hyaluronic acid sodium
Cat.No: T5004
Synonym: 透明质酸钠,Sodium Hyaluronate
Target: Others
Calycosin-7-O-β-D-glucoside
Cat.No: T3388
Synonym: 毛蕊异黄酮苷,calycosin-7-O-beta-D-glucopyranoside,Calycosin-7-O-beta-D-glucoside
Target: MMP, Reactive Oxygen Species
Demethyleneberberine
Cat.No: T4S0800
Synonym:
Target: P450, NOS, NF-κB, HIF, AMPK
Lariciresinol
Cat.No: TN1853
Synonym: (+)-落叶松树脂醇
Target: VEGFR, Antifection
Dehydrocorydaline nitrate
Cat.No: T2S2362
Synonym: 去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱
Target: BCL, Others, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Neferine
Cat.No: T5S1097
Synonym: (R)-1,2-Dimethoxyaporphine,(-)-Neferine,甲基莲心碱
Target: Apoptosis, NF-κB, Autophagy
Echinatin
Cat.No: T3926
Synonym: 刺甘草查尔酮,Retrochalcone
Target: Free radical scavengers
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