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156

抑制剂 & 化合物

52

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Cat. No. Product Name Target Signaling Pathways
T8740 COH-SR4

COH-SR4 (Mitochondria uncoupler SR4)

Others; AMPK Chromatin/Epigenetic; Others; PI3K/Akt/mTOR signaling
COH-SR4 (COH-SR4 (Mitochondria uncoupler SR4)) 是线粒体氧化磷酸化的解偶联剂,可调节 amp 依赖性激酶 (ampk)-雷帕霉素 (mtor) 信号的哺乳动物靶点,并抑制 hepg2 肝癌细胞的增殖。它对白血病、黑色素瘤、乳腺癌和肺癌显示出强大的抗增殖活性。它是一种AMPK 活化剂,通过激活 AMPK 来抑制脂肪细胞分化,可用于肥胖及代谢紊乱相关的研究。
T81631 NV-354

Mitochondria modulator-1

Mitochondria modulator-1为线粒体调节剂,可促进ATP生成。该化合物展现出优良的口服生物利用度、血脑屏障透过性及稳定的血浆稳定性,展现出其研究线粒体疾病的潜力。
T72291 Mitochondria degrader-1

Mitochondria degrader-1 (实施例 5) 是一种通过自噬机制诱导受损线粒体降解的有效线粒体降解剂。适用于神经退行性疾病、癌症、炎症性疾病、年龄相关性疾病、代谢性疾病、线粒体疾病及唐氏病的研究。
T9423 Alkyne tyramide

Others Others
Alkyne tyramide 是抗坏血酸过氧化物酶 2 探针。它有助于鉴定 APEX 标记位点,明确线粒体蛋白的膜拓扑的分配。它显著提高了完整酵母细胞的 APEX 标记效率,比 APEX2 底物生物素苯酚具有更大的细胞壁渗透性。
T40130 Nur77 modulator 1

Nur77 modulator 1

Others Others
Nur77 modulator 1 可与Nur77结合,KD 为 3.58 μM。它上调 Nur77 表达,介导Nur77亚细胞定位,诱导Nur77 依赖的内质网应激和自噬,可导致细胞凋亡,Nur77 modulator 1显示出抗肝癌生物活性。
T3268 Mildronate

Kvaterin,米屈肼,Meldonium,Quaterin

Hydroxylase Metabolism
Mildronate (Meldonium) 是心血管保护药,能够竞争性的抑制 BBOX1和 OCTN2。作用于人重组 BBOX 的(IC50:34-62 μM)、人 OCTN2 (EC50:21 μM)。它 n 能够诱导长链脂肪酸代谢从线粒体向过氧化物酶体的重定向。
T5827 BI-6C9

Apoptosis; Others; Mitochondrial Metabolism Apoptosis; Metabolism; Others
BI-6C9 是一种高特异性的 BH3 相互作用结构域抑制剂,可阻止线粒体外膜电位和线粒体分裂,并保护细胞免受线粒体凋亡诱导因子释放和不依赖 caspase 的细胞死亡。
T9211 Mito-LND

Mito-Loidamine

OXPHOS; Reactive Oxygen Species; Mitochondrial Metabolism; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Mito-LND (Mito-Loidamine) 是一种有口服活性和靶向线粒体的氧化磷酸化抑制剂。它抑制线粒体生物能,刺激活性氧的形成,并诱导肺癌细胞自噬细胞死亡。
T1885 Siramesine hydrochloride

Lu 28-179 hydrochloride,西拉美新盐酸盐

Ferroptosis; Sigma receptor; lysosomal autophagy Apoptosis; Autophagy; GPCR/G Protein
Siramesine hydrochloride (Lu 28-179 hydrochloride) 是一种选择性 sigma-2 受体激动剂,可引发 Y 细胞的细胞死亡并在体内表现出有效的抗癌活性。Siramesine 对 sigma-2 受体具有亚纳摩尔亲和力,并且对 sigma-2 受体的选择性是 sigma-1 受体的 140 倍。
T6451 Clodronic acid disodium salt

Loron,Clodronate Disodium,氯屈膦酸二钠,Lodronate

Others Others
Clodronic acid disodium salt (Lodronate) 是一种口服具有活力的破骨细胞骨吸收 (osteoclastic bone resorption) 的抑制剂,是一代双磷酸盐。它可用于高骨转换状态、Paget’s 病和溶骨性骨转移中。
T0866 Propafenone

Rythmol,普罗帕酮,Propafenonum

Potassium Channel; MRP; Sodium Channel Immunology/Inflammation; Membrane transporter/Ion channel
Propafenone (Propafenonum) 是钠通道阻滞剂,它对 β 受体具有高亲和力 (IC50=32 nM)。它能够阻断瞬时外向钾电流 (Ito) (IC50: 4.9 nM) 和持续延迟整流器K+电流 (Isus) (IC50: 8.6 nM) ,具有抗心律失常的作用。它能够诱导线粒体功能障碍及诱导细胞凋亡,从而抑制食管癌增殖。
T6583 MG-101

ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I

Cysteine Protease; Proteasome Proteases/Proteasome; Ubiquitination
MG-101 (Calpain inhibitor I) 是一种有效的半胱氨酸蛋白酶抑制剂,能够抑制钙蛋白酶I (Ki:190 pM),钙蛋白酶II (Ki:220 pM),组织蛋白酶B (Ki:150 pM)和组织蛋白酶L (Ki:500 pM)。
T4620 Siramesine

西拉美新,Lu 28-179

Sigma receptor GPCR/G Protein
Siramesine (Lu 28-179) 是sigma-2受体激动剂,通过线粒体的不稳定溶酶体触发细胞死亡,有强大的抗癌活性。它对 sigma-2 受体具有亚纳摩尔亲和力,IC50为 0.12 nM。它对 sigma-2 受体的选择性是 sigma-1 受体的 140倍,IC50为 17 nM。
T9232 Mitochondrial fusion promoter M1

Mitochondrial Metabolism Metabolism
Mitochondrial fusion promoter M1 是一种线粒体动态调节剂,能够保持线粒体功能并促进细胞呼吸,减轻心肌缺血/再灌注大鼠的心脏损伤和大脑损伤。
T37657 Mitochondrial respiration-IN-1 hydrobromide

Mitochondrial respiration-IN-1 hydrobromide (compound 49) is a potent mitochondrial inhibitor (IC50=8.8 mg/mL). Mitochondrial respiration-IN-1 hydrobromide significantly reduces mitochondrial respiration in platelets[1].
T72138 Mitochondrial respiration-IN-2

Mitochondrial respiration-IN-2 是Virginiamycin M1 的氟衍生物。Mitochondrial respiration-IN-2 可以抑制胶质母细胞瘤干细胞的线粒体翻译。
T72137 Mitochondrial respiration-IN-3

Mitochondrial respiration-IN-3 是 Dalfopristin 的氟衍生物。Mitochondrial respiration-IN-3 具有细胞膜渗透性。Mitochondrial respiration-IN-3 可以抑制胶质母细胞瘤干细胞的线粒体翻译 (mitochondrial translation)。Mitochondrial respiration-IN-3 可用于癌症的研究
T19072 TMRE

四甲基若丹明乙酯酸铵,Tetramethylrhodamine ethyl ester perchlorate

Others Others
TMRE (Tetramethylrhodamine ethyl ester perchlorate) 是线粒体特异性染料 (λex=550 nm,λem=575 nm)。
T26982 Cerebrocrast

IOS 11212,IOS-11212,IOS11212

Others Others
Cerebrocrast (IOS-11212) 是具有抗炎和降血糖活性,促进大鼠肝脏线粒体中 H+ 和 Cl- 的共转运,阻断人血小板活化,可用于研究糖尿病。
T4168 Visomitin

SKQ1

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Visomitin (SKQ1) 是一种靶向线粒体的抗氧化剂,表现出高效的线粒体穿透能力和有效的抗氧化能力。
T77344 icFSP1

Apoptosis Apoptosis
icFSP1是一种线粒体相关凋亡诱导因子调节剂,具有抗肿瘤活性,可用于研究和治疗肿瘤疾病。
T77553 MHI-148

IR-808

MHI-148 是一种具有肿瘤靶向性的近红外七甲氨酸菁染料,可用于检测、诊断和研究癌症。MHI-148 可被肿瘤细胞的溶酶体和线粒体吸收并积累,但在正常细胞的溶酶体和线粒体不吸收。
T19428 Mito-TEMPO

Reactive Oxygen Species; Mitochondrial Metabolism Immunology/Inflammation; Metabolism; NF-κB
Mito-TEMPO 是一种线粒体靶向超氧化物歧化酶的模拟物。Mito-TEMPO 可以清除超氧化物和烷基自由基,防止线粒体的氧化、坏死和凋亡。
T14941 CGP37157

7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one

Na+/Ca2+ Exchanger Membrane transporter/Ion channel
CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) 是一种 Na+/Ca2+ 交换抑制剂,抑制 Na+ 诱导的豚鼠心脏线粒体中 Ca2+ 的释放,IC50 为 0.8 μM。
T4441 UK-5099

UK 5099,PF-1005023,UK5099

Others; Mitochondrial Metabolism Metabolism; Others
UK-5099 (PF-1005023) 是一种有效的线粒体丙酮酸转运蛋白(MPC) 抑制剂, 抑制丙酮酸依赖性 O2消耗的 IC50值为50 nM。
T8366 Mitochonic acid 5

MA-5

Mitochondrial Metabolism Metabolism
Mitochonic acid 5 (MA-5) 能够调节线粒体 ATP 合成,可与线粒体结合,并改善肾小管和心肌细胞损伤。
T5114 Pyridaben

Calcium Channel; Parasite Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Pyridaben 是一种METI 杀螨剂,可抑制复合物 I 处的线粒体电子转运。它对多种螨虫具有活性,通过滤纸接触给药,在 25 mg/mL、100 mg/mL 和 200 mg/mL 的剂量下,分别诱导 100% 的C. malaccensis,D. farina 和T. putrescentia 死亡率。
T9807 CPDS

Others Others
CPDS 是一种非渗透性硫醇剂,可影响多种线粒体功能。在大鼠肝线粒体中,它仅抑制 Pi/OH- 载体。它和丙二酸正丁酯都是完全抑制 Pi 进入所必需的。
T75342 MitoSOX Red

Reactive Oxygen Species; Mitochondrial Metabolism; Autophagy Autophagy; Immunology/Inflammation; Metabolism; NF-κB
MitoSOX Red 是一种具有特异性和细胞膜渗透性且靶向活细胞线粒体的新型荧光探针。MitoSOX Red 进入线粒体后会被超氧化物氧化,而不会被其他 ROS 或 RNS 生成系统氧化。MitoSOX Red 随后与线粒体内核酸结合,产生强红色荧光。MitoSOX Red 可以作为荧光指示剂,特异性检测超氧化物。超氧化物歧化酶 (Superoxide dismutase,SOD) 能够预防 MitoSOX Red 氧化。
T33412 MitoPQ

MitoParaquat

Glucokinase; transporter Metabolism
MitoPQ (MitoParaquat) 是一个线粒体靶向的小分子化合物。MitoPQ 选择性加强线粒体超氧化物和过氧化氢的含量,抑制胰岛素刺激的葡萄糖摄取和葡萄糖转运蛋白 4 (GLUT4) 向脂肪细胞和肌管中质膜的易位。MitoPQ 可用于研究线粒体氧化应激与调节的 GLUT4 转运。
T9558 KL-11743

transporter Metabolism
KL-11743 是葡萄糖竞争性 I 类葡萄糖转运蛋白抑制剂,口服有活性,能够抑制GLUT1 (IC50:115 nM) 、GLUT2 (IC50:137 nM) 、GLUT3 (IC50:90 nM) 及GLUT4 (IC50:68 nM) 。它能够特异性阻断葡萄糖代谢,也可与电子传递抑制剂协同作用诱导细胞死亡。
T7460 α-Cyano-4-hydroxycinnamic acid

α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基

Monocarboxylate transporter Membrane transporter/Ion channel
α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) 是非竞争性单羧酸盐转运蛋白 (MCTs) 抑制剂,可抑制线粒体丙酮酸转运蛋白,Ki 值为 6.3 μM。它可作为基质辅助激光解吸电离-飞行时间质谱 (MALDI-TOF) 分析的基质,可以促进肽离子化。
T37563 C22 Ceramide (d18:1/22:0)

Cer(d18:1/22:0),C22 Ceramide,Ceramide (d18:1/22:0)

C22 Ceramide (d18:1/22:0) (C22 Ceramide) 是一种从海绵Haliclona koremella 中分离出含有山嵛酸的长链神经酰胺,是一种内源性生物活性鞘脂。C22 Ceramide (d18:1/22:0) 可特异性抑制MCSR,降低离体大鼠肝线粒体和脂质体中 C16-神经酰胺通道的形成。
TP1095 Elamipretide

MTP-131,RX-31,SS-31

Others Others
Elamipretide (MTP-131) 是一种线粒体靶向抗氧化四肽 (D-Arg-dimethylTyr-Lys-Phe-NH2),可以减少有毒活性氧的产生并稳定心磷脂,具有血脑屏障渗透性。Elamipretide 是罕见病巴氏综合征的潜在治疗剂。
T2170 SKF-96365 hydrochloride

1-[2-(4-甲氧基)-2-[3-(4-甲氧基苯基)丙氧基]乙基]咪唑,SKF96365

Apoptosis; Potassium Channel; Calcium Channel; TRP/TRPV Channel; Autophagy Apoptosis; Autophagy; Membrane transporter/Ion channel; Metabolism
SKF-96365 hydrochloride (SKF96365) 是store-operated Ca2+entry 抑制剂,也是TRP channel 阻滞剂。它显著抑制豚鼠离体心脏 hERG、hKCNQ1/hKCNE1、hKir2.1 和 hKv4.3 电流,延长QTc 间期。它通过诱导结直肠癌细胞的细胞周期阻滞和凋亡起抗肿瘤作用。
T35689 MTP 131 acetate

Others Others
MTP 131 acetate 是一种小的线粒体靶向四肽。
T70270 SMTIN-P01

SMTIN-P01 is a mitochondria-targeted Hsp90 inhibitor. It is made from the isopropyl amine of the Hsp90 inhibitor PU-H71 being replaced with the mitochondria-targeting moiety triphenylphosphonium.
T22370 Mitoquinol mesylate

Others Others
Mitoquinol, a ubiquinone derivative, specifically accumulates in mitochondria due to the covalent attachment of the cation triphenylphosphonium. Mitoquinol is an antioxidant, protecting mitochondria from oxidative damage and preventing lipid peroxidation-
T28047 Mitoquinone-cyclodextrin

MitoQ10,Mitoubiquinone mesylate,MitoQ-10,MitoQ,Mito Q10,Mitoquinone mesylate-cyclodextrin

Mitoquinone-cyclodextrin is a 1:1 molar ratio complex of Mitoquinone mesylate with cyclodextrin. Mitoquinone mesylate is a mitochondria-targeted antioxidant designed to accumulate within mitochondria in vivo in order to protect against oxidative damage. M
T34892 TM608

TM-608,TM 608

TM608 is a potent selective c-Met inhibitor that targets mitochondria and kills erlotinib-resistant lung cancer cells, rapidly accumulates in mitochondria, and inhibits MET activation in high MET expression, erlotinib-resistant HCC827B cells (total cell l
T36240 AP219

AP39 is a compound used to increase the levels of hydrogen sulfide (H2S) within mitochondria. It consists of a mitochondria-targeting motif (triphenylphosphonium) coupled to an H2S-donating moiety (dithiolethione) by an aliphatic linker. AP219 is a control compound for AP39, containing the triphenylphosphonium scaffold but lacking the H2S-releasing portion.
T33404 MitoBADY

Mito-BADY,Mito BADY

Mitobady is a sensitive and specific Raman probe, which can be used for living cell imaging of mitochondria.
T12048 Mito-apocynin (C2)

Others Others
Mito-apocynin (C2) is an orally active mitochondria-targeted triphenylphosphonium (TPP)-based compound, has antineuroinflammatory effects.
T26242 SW IV-52

SW-IV-52,SW IV52,SW IV 52,SWIV52

SW IV-52 is an XIAP-inhibitor that acts as a second mitochondria-derived activator of caspases (SMAC) mimetic.
T35965 MitoTEMPOL

MitoTEMPOL is a mitochondria-targeting superoxide dismutase mimetic that reduces mitochondrial O2- to H2O2. Like the related compound MitoTEMPO , MitoTEMPOL combines an antioxidant moiety (here, TEMPOL, also known as 4-hydroxy-TEMPO) with the lipophilic cation triphenylphosphonium, which allows it to pass through lipid bilayers and accumulate in mitochondria. MitoTEMPOL has been used to elucidate the role of mitochondria-derived superoxide in mitochondrial, cellular, and whole animal signaling.
T22982 MitoPY1

Others Others
a fluorescent probe for imaging hydrogen peroxide (H2O2) in mitochondria of living cells
T40959 T0467

T0467

T0467 is a chemical compound that activates the translocation of parkin to the mitochondria in a PINK1-dependent manner in vitro. However, T0467 does not induce the accumulation of PINK1 in the mitochondria of dopaminergic neurons. As a result, T0467 shows promise as a potential compound for activating the PINK1-Parkin signaling pathway and can be utilized in research related to Parkinson's disease and related disorders.
T71866 Cochlioquinone B

Cochlioquinone B is a phytotoxin that inhibits NADH oxidase and NADH-2,3-dimethoxy-5-pentyl-1,4-benzoquinone reductase from heart mitochondria.
T35962 MitoPBN

MitoPBN is a mitochondria-targeted antioxidant. It accumulates in the mitochondria following the generation of a mitochondrial membrane potential by succinate, an effect that is blocked by addition of the mitochondrial membrane potential uncoupler FCCP . MitoPBN inhibits superoxide activation of mitochondrial uncoupling protein 1 (UCP1), UCP2, and UCP3 when used at a concentration of 250 nM in vitro but does not react with superoxide. It traps hydroxyl (IC50 = ~77 μM) and carbon-centered radical...
T11356 Gamitrinib TPP hexafluorophosphate

HSP Cytoskeletal Signaling; Metabolism
Gamitrinib TPP hexafluorophosphate is a potent HSP90 inhibitor that specifically targets the mitochondria, demonstrating notable anti-cancer activity. It functions by inhibiting the mitochondrial matrix, making it an effective compound in cancer treatment.

化合物

COH-SR4
Cat.No: T8740
Synonym: COH-SR4 (Mitochondria uncoupler SR4)
Target: Others, AMPK
NV-354
Cat.No: T81631
Synonym: Mitochondria modulator-1
Target:
Mitochondria degrader-1
Cat.No: T72291
Synonym:
Target:
Alkyne tyramide
Cat.No: T9423
Synonym:
Target: Others
Nur77 modulator 1
Cat.No: T40130
Synonym: Nur77 modulator 1
Target: Others
Mildronate
Cat.No: T3268
Synonym: Kvaterin,米屈肼,Meldonium,Quaterin
Target: Hydroxylase
BI-6C9
Cat.No: T5827
Synonym:
Target: Apoptosis, Others, Mitochondrial Metabolism
Mito-LND
Cat.No: T9211
Synonym: Mito-Loidamine
Target: OXPHOS, Reactive Oxygen Species, Mitochondrial Metabolism, Autophagy
Siramesine hydrochloride
Cat.No: T1885
Synonym: Lu 28-179 hydrochloride,西拉美新盐酸盐
Target: Ferroptosis, Sigma receptor, lysosomal autophagy
Clodronic acid disodium salt
Cat.No: T6451
Synonym: Loron,Clodronate Disodium,氯屈膦酸二钠,Lodronate
Target: Others
Propafenone
Cat.No: T0866
Synonym: Rythmol,普罗帕酮,Propafenonum
Target: Potassium Channel, MRP, Sodium Channel
MG-101
Cat.No: T6583
Synonym: ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I
Target: Cysteine Protease, Proteasome
Siramesine
Cat.No: T4620
Synonym: 西拉美新,Lu 28-179
Target: Sigma receptor
Mitochondrial fusion promoter M1
Cat.No: T9232
Synonym:
Target: Mitochondrial Metabolism
Mitochondrial respiration-IN-1 hydrobromide
Cat.No: T37657
Synonym:
Target:
Mitochondrial respiration-IN-2
Cat.No: T72138
Synonym:
Target:
Mitochondrial respiration-IN-3
Cat.No: T72137
Synonym:
Target:
TMRE
Cat.No: T19072
Synonym: 四甲基若丹明乙酯酸铵,Tetramethylrhodamine ethyl ester perchlorate
Target: Others
Cerebrocrast
Cat.No: T26982
Synonym: IOS 11212,IOS-11212,IOS11212
Target: Others
Visomitin
Cat.No: T4168
Synonym: SKQ1
Target: Reactive Oxygen Species
icFSP1
Cat.No: T77344
Synonym:
Target: Apoptosis
MHI-148
Cat.No: T77553
Synonym: IR-808
Target:
Mito-TEMPO
Cat.No: T19428
Synonym:
Target: Reactive Oxygen Species, Mitochondrial Metabolism
CGP37157
Cat.No: T14941
Synonym: 7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one
Target: Na+/Ca2+ Exchanger
UK-5099
Cat.No: T4441
Synonym: UK 5099,PF-1005023,UK5099
Target: Others, Mitochondrial Metabolism
Mitochonic acid 5
Cat.No: T8366
Synonym: MA-5
Target: Mitochondrial Metabolism
Pyridaben
Cat.No: T5114
Synonym:
Target: Calcium Channel, Parasite
CPDS
Cat.No: T9807
Synonym:
Target: Others
MitoSOX Red
Cat.No: T75342
Synonym:
Target: Reactive Oxygen Species, Mitochondrial Metabolism, Autophagy
MitoPQ
Cat.No: T33412
Synonym: MitoParaquat
Target: Glucokinase, transporter
KL-11743
Cat.No: T9558
Synonym:
Target: transporter
α-Cyano-4-hydroxycinnamic acid
Cat.No: T7460
Synonym: α-Cyano-4-hydroxycinnamic acid(α-CHCA),2-氰基-4-羟基
Target: Monocarboxylate transporter
C22 Ceramide (d18:1/22:0)
Cat.No: T37563
Synonym: Cer(d18:1/22:0),C22 Ceramide,Ceramide (d18:1/22:0)
Target:
Elamipretide
Cat.No: TP1095
Synonym: MTP-131,RX-31,SS-31
Target: Others
SKF-96365 hydrochloride
Cat.No: T2170
Synonym: 1-[2-(4-甲氧基)-2-[3-(4-甲氧基苯基)丙氧基]乙基]咪唑,SKF96365
Target: Apoptosis, Potassium Channel, Calcium Channel, TRP/TRPV Channel, Autophagy
MTP 131 acetate
Cat.No: T35689
Synonym:
Target: Others
SMTIN-P01
Cat.No: T70270
Synonym:
Target:
Mitoquinol mesylate
Cat.No: T22370
Synonym:
Target: Others
Mitoquinone-cyclodextrin
Cat.No: T28047
Synonym: MitoQ10,Mitoubiquinone mesylate,MitoQ-10,MitoQ,Mito Q10,Mitoquinone mesylate-cyclodextrin
Target:
TM608
Cat.No: T34892
Synonym: TM-608,TM 608
Target:
AP219
Cat.No: T36240
Synonym:
Target:
MitoBADY
Cat.No: T33404
Synonym: Mito-BADY,Mito BADY
Target:
Mito-apocynin (C2)
Cat.No: T12048
Synonym:
Target: Others
SW IV-52
Cat.No: T26242
Synonym: SW-IV-52,SW IV52,SW IV 52,SWIV52
Target:
MitoTEMPOL
Cat.No: T35965
Synonym:
Target:
MitoPY1
Cat.No: T22982
Synonym:
Target: Others
T0467
Cat.No: T40959
Synonym: T0467
Target:
Cochlioquinone B
Cat.No: T71866
Synonym:
Target:
MitoPBN
Cat.No: T35962
Synonym:
Target:
Gamitrinib TPP hexafluorophosphate
Cat.No: T11356
Synonym:
Target: HSP
Cat. No. Product Name Target Signaling Pathways
T7922 Kresoxim-Methyl

Others; Mitochondrial Metabolism; Antifungal Metabolism; Microbiology/Virology; Others
Kresoxim-methyl 是一种嗜球果伞素类杀菌剂,可抑制复合体 III 的呼吸,抑制苹果园分离株 V. inaequalis 的分生孢子萌发。
T0846 L-Carnitine

L(-)-Carnitine,Levocarnitine,左旋肉碱

Endogenous Metabolite; Fatty Acid Synthase Metabolism
L-Carnitine (L(-)-Carnitine) 是一种人内源性分子,在人体内以蛋氨酸和赖氨酸为底物进行生物合成,并参与脂肪酸代谢。L-Carnitine 将长链脂肪酰辅酶A 转运到线粒体。L-Carnitine 能够改善许多先天性代谢错误的代谢失衡。
T10148 4-Hydroxynonenal

4-羟基壬烯醛,4-HNE

Dehydrogenase; Endogenous Metabolite Metabolism
4-Hydroxynonenal (4-HNE) 是一种 α,β 不饱和羟基烯醛,可作为氧化/亚硝化应激生物标志物。它是ALDH2的底物和抑制剂。它可以调节许多信号传导过程,主要是通过与蛋白质,核酸和膜脂质中具有亲核官能团的共价加合物形成的。它通过线粒体在癌症中起重要作用。
TN7108 Urolithin C

Apoptosis; Calcium Channel; Reactive Oxygen Species; IGF-1R; Endogenous Metabolite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; NF-κB; Tyrosine Kinase/Adaptors
Urolithin C 属于多酚类,是鞣花酸的肠道微生物代谢产物,具有胰岛素分泌的葡萄糖依赖性激活活性。Urolithin C 是 L 型 Ca2+通道开放剂,可增强 Ca2+的流入。它通过线粒体介导的途径诱导细胞凋亡,并刺激活性氧的形成。
TL0006 Cichoric Acid

菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。
T2203 D-Carnitine hydrochloride

(S)-Carnitine Hydrochloride,L-Carnitine hydrochloride

Others; Endogenous Metabolite Metabolism; Others
D-Carnitine hydrochloride ((S)-Carnitine Hydrochloride) 已被用于研究麦角硫因素转运蛋白 SLC22A4 和肉毒碱转运蛋白 SLC22A5,也被用于使棕榈酸进入线粒体。
T1205 Chloramphenicol

Chlornitromycin,Levomycetin,Chloromycetin,氯霉素

ribosome; HIF/HIF Prolyl-Hydroxylase; Antibacterial; Antibiotic Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Chloramphenicol (Chloromycetin) 是一种广谱抗生素,有效抑制细菌蛋白质生物合成。它主要作用于细菌 70S 核糖体的 50S 亚基,对肽基转移酶有活性,抑制肽键的形成。
T3604 Sodium dichloroacetate

Sodium Dichloroacetate,DCA,BCA,bichloroacetic acid,二氯乙酸钠,Sodium dichloroacetate (DCA),二氯醋酸酯

Apoptosis; Dehydrogenase; Reactive Oxygen Species; PDK Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Sodium dichloroacetate (BCA) 是癌细胞线粒体中的一种代谢调节剂,具有抗癌活性。它抑制丙酮酸脱氢酶激酶,从而导致肿瘤微环境中的乳酸减少。它增加活性氧的产生并促进癌细胞凋亡,还可作为NKCC 抑制剂。
TN6714 Geranylgeraniol

FT-0626663,Tetraprenol,CJ24095,CJ 24095,FT0626663,香叶基香叶醇,CJ-24095

Apoptosis Apoptosis
Geranylgeraniol (FT0626663) 是一种类异戊二烯,存在于水果、蔬菜和谷物中,包括大米。 Geranylgeraniol (FT0626663) 抑制生长并诱导各种肿瘤细胞的凋亡。 Geranylgeraniol (FT0626663) 保护单核细胞免受他汀类药物诱导的细胞毒性并抑制分枝杆菌的生长。
TN3594 Cardanol (C15:1)

Apoptosis; Others Apoptosis; Others
Cardanol (C15:1) 存在于腰果壳液中,可诱导人黑色素瘤细胞线粒体相关的细胞凋亡。
T1068 Dithranol

1,8,9-trihydroxyanthracene,cignoline,蒽林,Anthralin

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Dithranol (cignoline) 是蒽醌衍生物,可破坏线粒体功能和结构,用于治疗皮肤病。
T33817 Orellanine

2-(1,3-dihydroxy-4-oxopyridin-2-yl)-1,3-dihydroxypyridin-4-one

Others Others
Orellanine 是一种从蘑菇 Cortinarius orellanus 中提取的肾毒性化合物。 Orellanine 强烈抑制 Madin-Darby 犬肾细胞和大鼠肝线粒体中大分子(蛋白质、RNA 和 DNA)的合成。
TN1274 4-Allylcatechol

2-羟基胡椒酚,4-Allylpyrocatechol,Hydroxychavicol

Others Others
4-Allylcatechol (Hydroxychavicol) 是合成黄樟素的一种中间体。
T6323 Oligomycin A

MCH 32,寡霉素A

ATPase; Antibiotic; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Oligomycin A (MCH 32) 是从链霉菌属中得到的一种线粒体F0F1-ATPase 抑制剂,抑制氧化磷酸化和线粒体偶联膜上发生的所有 ATP 依赖性过程。
T4S0800 Demethyleneberberine

P450; NOS; NF-κB; HIF; AMPK Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Demethyleneberberine 是从黄连中提取的一种天然产物,是线粒体靶向抗氧化剂。它也可作为AMPK 激活剂,用于非酒精性脂肪性肝病的研究。它通过抑制NF-κB 通路和调节 Th 细胞的平衡来减轻小鼠结肠炎并抑制炎症反应。
T27012 Chrysotoxine

Phenol, 4-[2-(3,4-dimethoxyphenyl)ethyl]-2,6-dimethoxy-,4-[2-(3,4-Dimethoxyphenyl)ethyl]-2,6-dimethoxyphenol,鼓槌石斛素

NF-κB NF-κB
Chrysotoxine (Phenol, 4-[2-(3,4-dimethoxyphenyl)ethyl]-2,6-dimethoxy-) 通过 NF-κB 调节和线粒体保护抑制 SH-SY5Y 细胞中 6-羟基多巴胺诱导的细胞凋亡。
T2731 Usnic Acid

Usniacin,松萝酸,地衣酸

Antibacterial; Autophagy Autophagy; Microbiology/Virology
Usnic Acid (Usniacin) 是地衣次生代谢产物,具有独特的二苯并呋喃骨架。它是一种抗菌剂、抗肿瘤剂和酶抑制剂。
T5715 (E)-Flavokawain A

(E)-1-(2-羟基-4,6-二甲氧基苯基)-3-(4-甲氧基苯基)-2-丙烯-1-酮,FLAVOKAVAIN A(P),卡瓦胡椒素A

Apoptosis; P450 Apoptosis; Metabolism
(E)-Flavokawain A 是一种来自卡瓦提取物的新型查尔酮,通过参与 Bax 蛋白依赖性和线粒体依赖性凋亡途径诱导膀胱癌细胞凋亡,并抑制小鼠肿瘤生长,具有抗癌作用。
T5055 For-Met-OH

fMet,N-甲酰甲硫氨酸,N-Formyl-L-methionine

Others; Endogenous Metabolite Metabolism; Others
For-Met-OH (N-Formyl-L-methionine) 是内源性代谢产物的一种。
T5S0285 Cistanoside A

肉苁蓉苷 A,肉苁蓉苷A

Others Others
Cistanoside A 是一种肉苁蓉中的苯丙素类化合物,能够抑制 NO 的聚集,但不影响诱导型一氧化氮合酶 iNOS 的 mRNA 和蛋白水平及其活性。它具有抗炎作用。
T2970 Rotenone

Rotenon,鱼藤酮,Paraderil,Barbasco,Rotocide,Dactinol

Apoptosis; Dehydrogenase; Mitochondrial Metabolism; p53; Autophagy Apoptosis; Autophagy; Metabolism
Rotenone (Rotocide) 属于天然产物,是一种植物杀虫剂。Rotenone 是一种线粒体电子传递复合物 I 抑制剂,可以促进线粒体产生活性氧,并诱导细胞凋亡。
T7050 alpha-Tocopherolquinone

托可醌,Metarene

Antioxidant oxidation-reduction
alpha-Tocopherolquinone (Metarene) 会下调线粒体的呼吸活动。在还原为生育酚氢醌后,它还显示出抗氧化活性。在大鼠缺氧期间,已发现它的水平升高。
T10662L Calcimycin

Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187

Apoptosis; Antibacterial; Antibiotic; Autophagy; Antifungal Apoptosis; Autophagy; Microbiology/Virology
Calcimycin (A-23187) 是抗生素和二价阳离子离子载体。它抑制革兰氏阳性细菌和一些真菌生长,也抑制 ATP 酶的活性并解耦哺乳动物细胞的氧化磷酸化。它通过增加细胞内钙浓度诱导 Ca2+依赖性细胞死亡。
T4S1335 Daphnoretin

Dephnoretin,西瑞香素,Thymelol

Influenza Virus; Caspase; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
Daphnoretin (Thymelol) 是从了哥王中提取得到的一种天然产物,具有抗癌和抗病毒活性。它通过在 G2/M 期连续阻断细胞并激活 caspase-3 通路导致 HOS 细胞死亡。
TN1911 Marein

马里苷,马里甙

transporter; Akt; HDAC; AMPK Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling
Marein 能通过CaMKK/AMPK/GLUT1促进葡萄糖摄取,IRS/Akt/GSK-3β增加糖原合成,并通过Akt/FoxO1减少糖异生,从而改善 HepG2 细胞中高葡萄糖诱导的胰岛素抵抗。它对甲基乙二醛诱导的 PC12 细胞损伤具有神经保护作用,还有抗氧化、降压、降血脂和抗糖尿病作用。
T3921 Punicalagin

安石榴甙,安石榴苷

SARS-CoV; HBV Microbiology/Virology
Punicalagin 是一种在石榴中发现的主要鞣花单宁,是可逆且非竞争性的3CLpro 抑制剂,有抗氧化、抗炎和抗癌作用。它有潜力研究 COVID-19 。
T4809 Pyrimidine

嘧啶,Metadiazine

Others; Endogenous Metabolite Metabolism; Others
Pyrimidine (Metadiazine) 是内源性代谢产物的一种。
T3926 Echinatin

刺甘草查尔酮,Retrochalcone

Free radical scavengers oxidation-reduction
Echinatin (Retrochalcone) 是分离自中草药甘草中,具有保肝和抗炎活性。在大鼠中,它可以被快速吸收和消除,并广泛分布,绝对生物利用度约为 6.81%。
T4838 (S)-Malic acid

L-(-)-Malic acid,(S)-(-)-HYDROXYSUCCINIC ACID,(S)-2-Hydroxysuccinic acid,L-苹果酸

Others; Endogenous Metabolite Metabolism; Others
(S)-Malic acid ((S)-2-Hydroxysuccinic acid) 是天然存在的二羧酸,是水果酸甜味的来源,常用作食品添加剂。
T4900 (±)-Methyl Jasmonate

(±)-茉莉酸甲酯,甲基茉莉酮酸酯,(±)-Jasmonic Acid methyl ester,Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate

Others; Endogenous Metabolite Metabolism; Others
Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate ((±)-Jasmonic Acid methyl ester) 是内源性代谢产物的一种。
T5S0045 Isofraxidin

6,8-Dimethoxyumbelliferone,异秦皮啶,Phytodolor,异嗪皮啶

MMP; ERK; p38 MAPK; TLR; COX Immunology/Inflammation; MAPK; Neuroscience; Proteases/Proteasome
Isofraxidin (Phytodolor) 是来自刺五加的香豆素成分,抑制MMP-7表达和人肝癌细胞侵袭。它作用于肝癌细胞,抑制ERK1/2磷酸化。它减弱iNOS 和COX-2表达,还抑制TLR4/髓样分化蛋白 2 复合物的形成。
T5287 N-Acetyl-L-aspartic acid

AC-ASP-OH,N-Acetylaspartic acid,N-乙酰-L-天门冬氨酸

Others; Endogenous Metabolite Metabolism; Others
N-Acetyl-L-aspartic acid (AC-ASP-OH) 是天冬氨酸的衍生物, 是由氨基酸天冬氨酸和乙酰辅酶 A 在神经元中合成的。
T4837 Itaconic acid

methylene-butanedioicaci,衣康酸

Others; Endogenous Metabolite Metabolism; Others
Itaconic acid (methylene-butanedioicaci) 是聚合物,化学物质和燃料的合成前体。Itaconic acid 可由真菌合成。它也是巨噬细胞特异性代谢产物。它介导巨噬细胞代谢和腹膜肿瘤之间的串扰。
TN5171 Tricetin

Apoptosis; Others; Nrf2 Apoptosis; Immunology/Inflammation; Others
Tricetin 是一种从石榴中分离出的类黄酮。Tricetin 是 Keap1-Nrf2 蛋白相互作用(PPI)的强效竞争性抑制剂,通过激活 Nrf2/HO-1 信号通路和阻止线粒体依赖性细胞凋亡通路,保护帕金森病患免受 6-OHDA 诱导的神经毒性的影响。Tricetin 通过 Akt/GSK-1β途径抑制鼻咽癌的迁移和指示性蛋白酶早老素-1(PS-1)表达。Tricetin 抑制由Egr-1介导的氧化LDL 诱导的内皮炎症,保护大鼠软骨细胞免受IL-1β诱导的炎症和细胞凋亡。
T4880 L-Dihydroorotic acid

Others; Endogenous Metabolite Metabolism; Others
L-Dihydroorotic acid 是一种能够通过二氢乳清酶,能够逆水解产生的无环 L-脲基琥珀酸。
T37714 Fuscin

Fuscin is a quinonoid fungal metabolite originally isolated from O. fuscum that has diverse biological activities. It inhibits binding of the ADP/ATP translocase inhibitor atractyloside to rat liver mitochondria in an ADP-dependent manner when used at a concentration of 50 μM in a radioligand binding assay. Fuscin (20 μM) reduces the glutathione content of rat liver mitochondria to 28% of controls and inhibits NADH oxidation in sonicated pigeon heart mitochondria preparations in a concentration-...
T38054 Avenaciolide

Avenaciolide is a water-insoluble fungal metabolite originally isolated from A. avenaceus. It inhibits glutamate transport in isolated rat liver mitochondria (Ki = 8 μM).
TN1572 Desacetylcinobufotalin

Others Others
Desacetylcinobufotalin has significant antitumor activity through induction apoptosis via mitochondria pathway, it also shows potent cytotoxic activities against HL-60 cell lines.
TN2039 Panaxydol

cAMP; p38 MAPK; JNK GPCR/G Protein; MAPK
Panaxydol has anti-cancer activity, can inhibit the growth and apoptosis of cancer cells, the signaling mechanisms involve a [Ca(2+)](i) increase, JNK and p38 MAPK activation, cAMP, MAP kinase and ROS generation through NADPH oxidase and mitochondria.
TN2191 Scutebarbatine A

BCL; Caspase Apoptosis; Proteases/Proteasome
Scutebarbatine A shows significant antitumor effects on A549 cells in vivo and in vitro via mitochondria-mediated apoptosis by up-regulating expressions of caspase-3 and 9, and down-regulating Bcl-2. Scutebarbatine A and barbatine A show a significant ability to protect cells against H2O2 with ED50 values of 5.0 and 16.8 μM, respectively.
T83281 6-(1-Hydroxyethyl)-5,6-dihydrochelerythrine

6-(1-Hydroxyethyl)-5,6-dihydrochelerythrine 显著影响细胞器特性,涉及早期内体、线粒体及自噬体(源自帕金森病患者的嗅觉细胞)。
TN5201 Uncarinic acid E

BCL; MEK; Caspase; PI3K; Antifection; p53 Apoptosis; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Uncarinic acid E has anti-cancer activity, it induces apoptosis in HepG2 cells via accumulation of p53, alters the Bax/Bcl-2 ratio, and activates caspases, resulting in cytochrome c release from the mitochondria. A mixture of uncarinic acid E and 27-O-p-(
T20123 L-Carnitine hydrochloride

L-Carnitine chloride,LC 80,Levocarnitine chloride,(R)-Carnitine hydrochloride,LC-80,LC80

Carnitine is a quaternary amine that occurs naturally in most mammalian tissue. Carnitine is present in relatively high concentrations in skeletal muscle and heart where it is involved in regulating energy metabolism. It has also been used to allow the en
T75630 Ganoderic acid Mf

Ganoderic acid Mf为具有抗肿瘤活性的三萜类化合物,能导致细胞周期在G1期停滞,并在正常细胞与癌细胞中显示高度选择性,通过线粒体介导途径促进细胞凋亡(apoptosis)。
T75629 Ganoderic acid Mk

Ganoderic acid Mk (GA-Mk)为来源于灵芝菌丝的三萜酸类化合物,能有效抑制细胞增殖,并通过线粒体途径诱导HeLa细胞的细胞凋亡(apoptosis),在宫颈癌研究中具有应用价值。
T4415 Katacine

Others Others
Katacine 抑制氧气消耗,并抑制电子通过线粒体呼吸链从氧化底物转移到分子氧的速度。 Katacine 是来自蓼科蓼科蓼属的 A 型原花青素聚合物在不同聚合阶段的混合物。 Katacine 是一种抗缺氧药。
TN6394 Alisol B acetate

Alisol B acetate can induce Bax nuclear translocation and apoptosis in human hormone-resistant prostate cancer PC-3 cells, the Bax activation and translocation from the cytosol to nucleus might be a crucial response to the apoptotic effect. Alisol B aceta
TMA1008 Ganoderic acid S

Others Others
A novel combination of triterpenoids includes at least ganoderic acid S (GAS), ganoderic acid T (GAT), ganoderic acid Me (GAMe), ganoderic acid R (GAR), and ganodermic acid S (GMAS), the composition is suitable for the treatment or prophylaxis of colon ca
TN3525 Boehmenan

ERK; Phosphatase; EGFR; PARP; MEK; Wnt/beta-catenin; Akt; Caspase; STAT; p53 Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; JAK/STAT signaling; MAPK; Metabolism; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
(±)-Boehmenan shows potent protein-tyrosine phosphatase 1B (PTP1B) inhibitory activity in vitro with the IC(50) values of 43.5 uM, it inhibits PTP1B activity in a competitive manner. Boehmenan exhibits the potent cytotoxic effects against many cancer cell
T79971 Asparanin A

Apoptosis Apoptosis
Asparanin A 是一种具有抗癌活性的凋亡 (apoptosis) 诱导剂。它能够通过线粒体和 PI3K/AKT 信号通路使细胞周期在 G0/G1 期停滞,并有效抑制癌细胞生长。此外,Asparanin A 在小鼠Ishikawa子宫内膜癌异种移植模型中显示出显著的体内抑制肿瘤生长效力。
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天然产物

Kresoxim-Methyl
Cat.No: T7922
Synonym:
Target: Others, Mitochondrial Metabolism, Antifungal
L-Carnitine
Cat.No: T0846
Synonym: L(-)-Carnitine,Levocarnitine,左旋肉碱
Target: Endogenous Metabolite, Fatty Acid Synthase
4-Hydroxynonenal
Cat.No: T10148
Synonym: 4-羟基壬烯醛,4-HNE
Target: Dehydrogenase, Endogenous Metabolite
Urolithin C
Cat.No: TN7108
Synonym:
Target: Apoptosis, Calcium Channel, Reactive Oxygen Species, IGF-1R, Endogenous Metabolite
Cichoric Acid
Cat.No: TL0006
Synonym: 菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid
Target: Reactive Oxygen Species, HIV Protease
D-Carnitine hydrochloride
Cat.No: T2203
Synonym: (S)-Carnitine Hydrochloride,L-Carnitine hydrochloride
Target: Others, Endogenous Metabolite
Chloramphenicol
Cat.No: T1205
Synonym: Chlornitromycin,Levomycetin,Chloromycetin,氯霉素
Target: ribosome, HIF/HIF Prolyl-Hydroxylase, Antibacterial, Antibiotic
Sodium dichloroacetate
Cat.No: T3604
Synonym: Sodium Dichloroacetate,DCA,BCA,bichloroacetic acid,二氯乙酸钠,Sodium dichloroacetate (DCA),二氯醋酸酯
Target: Apoptosis, Dehydrogenase, Reactive Oxygen Species, PDK
Geranylgeraniol
Cat.No: TN6714
Synonym: FT-0626663,Tetraprenol,CJ24095,CJ 24095,FT0626663,香叶基香叶醇,CJ-24095
Target: Apoptosis
Cardanol (C15:1)
Cat.No: TN3594
Synonym:
Target: Apoptosis, Others
Dithranol
Cat.No: T1068
Synonym: 1,8,9-trihydroxyanthracene,cignoline,蒽林,Anthralin
Target: Others, DNA/RNA Synthesis
Orellanine
Cat.No: T33817
Synonym: 2-(1,3-dihydroxy-4-oxopyridin-2-yl)-1,3-dihydroxypyridin-4-one
Target: Others
4-Allylcatechol
Cat.No: TN1274
Synonym: 2-羟基胡椒酚,4-Allylpyrocatechol,Hydroxychavicol
Target: Others
Oligomycin A
Cat.No: T6323
Synonym: MCH 32,寡霉素A
Target: ATPase, Antibiotic, Antifungal
Demethyleneberberine
Cat.No: T4S0800
Synonym:
Target: P450, NOS, NF-κB, HIF, AMPK
Chrysotoxine
Cat.No: T27012
Synonym: Phenol, 4-[2-(3,4-dimethoxyphenyl)ethyl]-2,6-dimethoxy-,4-[2-(3,4-Dimethoxyphenyl)ethyl]-2,6-dimethoxyphenol,鼓槌石斛素
Target: NF-κB
Usnic Acid
Cat.No: T2731
Synonym: Usniacin,松萝酸,地衣酸
Target: Antibacterial, Autophagy
(E)-Flavokawain A
Cat.No: T5715
Synonym: (E)-1-(2-羟基-4,6-二甲氧基苯基)-3-(4-甲氧基苯基)-2-丙烯-1-酮,FLAVOKAVAIN A(P),卡瓦胡椒素A
Target: Apoptosis, P450
For-Met-OH
Cat.No: T5055
Synonym: fMet,N-甲酰甲硫氨酸,N-Formyl-L-methionine
Target: Others, Endogenous Metabolite
Cistanoside A
Cat.No: T5S0285
Synonym: 肉苁蓉苷 A,肉苁蓉苷A
Target: Others
Rotenone
Cat.No: T2970
Synonym: Rotenon,鱼藤酮,Paraderil,Barbasco,Rotocide,Dactinol
Target: Apoptosis, Dehydrogenase, Mitochondrial Metabolism, p53, Autophagy
alpha-Tocopherolquinone
Cat.No: T7050
Synonym: 托可醌,Metarene
Target: Antioxidant
Calcimycin
Cat.No: T10662L
Synonym: Antibiotic A-23187,离子载体(钙镁盐混合物),A-23187
Target: Apoptosis, Antibacterial, Antibiotic, Autophagy, Antifungal
Daphnoretin
Cat.No: T4S1335
Synonym: Dephnoretin,西瑞香素,Thymelol
Target: Influenza Virus, Caspase, PKC
Marein
Cat.No: TN1911
Synonym: 马里苷,马里甙
Target: transporter, Akt, HDAC, AMPK
Punicalagin
Cat.No: T3921
Synonym: 安石榴甙,安石榴苷
Target: SARS-CoV, HBV
Pyrimidine
Cat.No: T4809
Synonym: 嘧啶,Metadiazine
Target: Others, Endogenous Metabolite
Echinatin
Cat.No: T3926
Synonym: 刺甘草查尔酮,Retrochalcone
Target: Free radical scavengers
(S)-Malic acid
Cat.No: T4838
Synonym: L-(-)-Malic acid,(S)-(-)-HYDROXYSUCCINIC ACID,(S)-2-Hydroxysuccinic acid,L-苹果酸
Target: Others, Endogenous Metabolite
(±)-Methyl Jasmonate
Cat.No: T4900
Synonym: (±)-茉莉酸甲酯,甲基茉莉酮酸酯,(±)-Jasmonic Acid methyl ester,Methyl 2-(3-oxo-2-(pent-2-en-1-yl)cyclopentyl)acetate
Target: Others, Endogenous Metabolite
Isofraxidin
Cat.No: T5S0045
Synonym: 6,8-Dimethoxyumbelliferone,异秦皮啶,Phytodolor,异嗪皮啶
Target: MMP, ERK, p38 MAPK, TLR, COX
N-Acetyl-L-aspartic acid
Cat.No: T5287
Synonym: AC-ASP-OH,N-Acetylaspartic acid,N-乙酰-L-天门冬氨酸
Target: Others, Endogenous Metabolite
Itaconic acid
Cat.No: T4837
Synonym: methylene-butanedioicaci,衣康酸
Target: Others, Endogenous Metabolite
Tricetin
Cat.No: TN5171
Synonym:
Target: Apoptosis, Others, Nrf2
L-Dihydroorotic acid
Cat.No: T4880
Synonym:
Target: Others, Endogenous Metabolite
Fuscin
Cat.No: T37714
Synonym:
Target:
Avenaciolide
Cat.No: T38054
Synonym:
Target:
Desacetylcinobufotalin
Cat.No: TN1572
Synonym:
Target: Others
Panaxydol
Cat.No: TN2039
Synonym:
Target: cAMP, p38 MAPK, JNK
Scutebarbatine A
Cat.No: TN2191
Synonym:
Target: BCL, Caspase
6-(1-Hydroxyethyl)-5,6-dihydrochelerythrine
Cat.No: T83281
Synonym:
Target:
Uncarinic acid E
Cat.No: TN5201
Synonym:
Target: BCL, MEK, Caspase, PI3K, Antifection, p53
L-Carnitine hydrochloride
Cat.No: T20123
Synonym: L-Carnitine chloride,LC 80,Levocarnitine chloride,(R)-Carnitine hydrochloride,LC-80,LC80
Target:
Ganoderic acid Mf
Cat.No: T75630
Synonym:
Target:
Ganoderic acid Mk
Cat.No: T75629
Synonym:
Target:
Katacine
Cat.No: T4415
Synonym:
Target: Others
Alisol B acetate
Cat.No: TN6394
Synonym:
Target:
Ganoderic acid S
Cat.No: TMA1008
Synonym:
Target: Others
Boehmenan
Cat.No: TN3525
Synonym:
Target: ERK, Phosphatase, EGFR, PARP, MEK, Wnt/beta-catenin, Akt, Caspase, STAT, p53
Asparanin A
Cat.No: T79971
Synonym:
Target: Apoptosis
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