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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T21806 HNHA

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
HNHA 是组蛋白去乙酰化酶抑制剂。它通过 p21诱导将细胞周期阻滞在 G1/S 期,抑制肿瘤生长及肿瘤新生血管形成。HNHA 可能是一种有效的抗乳腺癌药物。
T9244 σ1 Receptor antagonist-1

Sigma receptor GPCR/G Protein
σ1 Receptor antagonist-1 是高选择性的 sigma 1受体拮抗剂,pKi 为10.28。它抑制细胞生长,在 G0/G1 期阻滞细胞周期并诱导 MCF-7/ADR 细胞凋亡。
T6588 Mitoxantrone

米托蒽醌,mitozantrone

Topoisomerase; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair
Mitoxantrone (mitozantrone) 是一种拓扑异构酶 II 的抑制剂,也可抑制蛋白激酶C (PKC),IC50值为8.5 μM。
T15249 Estrogen receptor modulator 1

Estrogen Receptor/ERR Endocrinology/Hormones
Estrogen receptor modulator 1 是一种有效的、具有口服活性的、选择性雌激素受体(estrogen receptor)调节剂 (SERM),其 pIC50为 0.46。它能够诱导 Tamoxifen 耐药、激素非依赖性异种移植瘤的消退。
T2085 PQ401

IGF-1R Inhibitor II

Apoptosis; IGF-1R Apoptosis; Tyrosine Kinase/Adaptors
PQ401 (IGF-1R Inhibitor II) 是一种IGF-IR 抑制剂。在 MCF-7 细胞中,它抑制 IGF-I 刺激的 IGF-IR 自磷酸化,可有效抑制 IGF-I 刺激的 MCF-7 细胞生长。它诱导 caspase 介导的细胞凋亡,有用于乳腺癌和其他对 IGF-I 敏感的癌症的研究潜力。
T22288 (1E)-CFI-400437 dihydrochloride

CFI-400437 dihydrochloride

PLK Cell Cycle/Checkpoint
(1E)-CFI-400437 dihydrochloride (CFI-400437 dihydrochloride) 是一种选择性和有效的 polo 样激酶 4 (PLK4) 抑制剂,IC50为 0.6 nM。它还抑制 Aurora A、 Aurora B、 KDR 和 FLT-3,IC50分别为 0.37、0.21、0.48 和 0.18 μM,具有抗增殖活性。
T5882 3-Bromopyruvic acid

Hexokinase II Inhibitor II, 3-BP,3-溴丙酮酸,Bromopyruvic acid

Apoptosis; Hexokinase; Autophagy Apoptosis; Autophagy; Metabolism
3-Bromopyruvic acid (Hexokinase II Inhibitor II, 3-BP) 是己糖激酶 II 抑制剂,是针对肝癌细胞的一种抗肿瘤剂。
T0158 Mitoxantrone dihydrochloride

米托蒽醌二盐酸盐,盐酸米托蒽醌,Mitoxantrone 2HCl,Mitoxantrone hydrochloride,NSC-301739,mitozantrone dihydrochloride

Topoisomerase; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair
Mitoxantrone dihydrochloride (NSC-301739) 是一种拓扑异构酶 II 的抑制剂;也可抑制蛋白激酶C (PKC),IC50值为8.5 μM。
T6010 Idarubicin hydrochloride

盐酸伊达比星,Idamycin,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,4-Demethoxydaunorubicin hydrochloride,Idarubicin HCl,伊达比星盐酸盐,Zavedos

Topoisomerase; Antibacterial; Autophagy; Antifungal Autophagy; DNA Damage/DNA Repair; Microbiology/Virology
Idarubicin hydrochloride (Zavedos) 是一种蒽环类抗白血病药物,能抑制细菌和酵母菌生长,还抑制拓扑异构酶 II,干扰 DNA 复制和 RNA 转录。
T72470 Estrone O-sulfamate

Estrone 3-O-sulfamate

Others Others
Estrone O-sulfamate (Estrone 3-O-sulfamate) 是一种高效的的类固醇硫酸酯酶 (STS) 抑制剂。Estrone O-sulfamate 是一种胎盘微粒体抑制剂 (P.M.) ,IC50 值分别为 18 nM。Estrone O-sulfamate 在 MCF-7 细胞中对 STS 显示出抑制作用,IC50 值分别为 0.83 nM。Estrone O-sulfamate 可用于研究癌症。
T10325 ANI-7

Chk Cell Cycle/Checkpoint
ANI-7是芳香烃受体(AhR)途径的激活剂。ANI-7抑制多种癌症细胞的生长,并有效且选择性地抑制MCF-7乳腺癌症细胞的生长(GI50:0.56μM)。
T9541 CTB

Cholera Toxin B subunit

Epigenetic Reader Domain Chromatin/Epigenetic
CTB (Cholera Toxin B subunit) 是一种 p300 组蛋白乙酰转移酶的激活剂,可诱导 MCF-7 细胞凋亡。
T64348 Antiproliferative agent-16

Antiproliferative agent-16

Others Others
Antiproliferative agent-16 (Antiproliferative agent-16)是一种具有抗癌活性的吲哚酰肼-腙化合物。 Antiproliferative agent-16 对乳腺癌细胞表现出特异性 (对 MCF-7 细胞的 IC50 为 6.94 μM)。
T36488 LYG-202

LYG202,LYG 202

Apoptosis; ROS Apoptosis; Immunology/Inflammation
LYG-202是一种具有哌嗪替代的新型类黄酮,在体内和体外都具有抗肿瘤作用。LYG-202 诱导 MCF-7、MDA-MB-231 和 MDA-MB-435 细胞凋亡, 增加了细胞内 ROS 的产生。
T36970 STD1T

DUB Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Ubiquitination
STD1T 是一种具有选择性和有效性的脱泛素酶 USP2a 抑制剂,具有潜在的抗癌活性,可降低 HCT116 结肠和 MCF-7 乳腺癌细胞中的细胞周期蛋白 D1 蛋白水平。
T40233 (Iso)-MS4322

(Iso)-YS43-22,MS4322 (isomer),YS43-22 (isomer)

Histone Methyltransferase Chromatin/Epigenetic
(Iso)-MS4322 ((Iso)-YS43-22) 是一种具有选择性和强效性的蛋白质精氨酸甲基转移酶 5 (PRMT5) 降解剂,具有潜在的抗癌活性,有效地降低 MCF-7 细胞中的 PRMT5 蛋白水平,可抑制多种癌细胞的生长。
T28589 Ro 41-5253

Ro-41-5253,Ro 415253

Apoptosis; Retinoid Receptor Apoptosis; Metabolism
Ro 41-5253 是一种具有口服活性的 RARα 拮抗剂,是过氧化物酶体增殖物激活受体 (PPAR)-γ 的配体和部分激动剂,具有抗肿瘤活性,抑制 MCF-7 和 ZR-75.1 雌激素受体阳性乳腺癌细胞的增殖并诱导细胞凋亡。
T83627 Pim-1 kinase inhibitor 8

Pim; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling
Pim-1 kinase inhibitor 8 是一种高效的 Pim-1 kinase 抑制剂,具有抗癌活性,可有效抑制细胞迁移。Pim-1 kinase inhibitor 8 对 MCF-7 和 HepG2 细胞有细胞毒性,是研究乳腺癌的候选化合物。
T77575 P-gb-IN-1

P-gp Membrane transporter/Ion channel; Neuroscience
P-gb-IN-1 是一种有效的 P-糖蛋白 (P-gp) 抑制剂,通过抑制 P-gp 外流展现出逆转活性。P-gb-IN-1 通过与残基 Asn 721 和 Met 986 形成氢键相互作用从而显示出对 P-gp 的抑制作用。P-gb-IN-1 在 MCF-7/ADR 细胞中显示出低毒性。
T7057 Methylstat

Histone Demethylase; Others Chromatin/Epigenetic; Others
Methylstat 是一种含有 Jumonji C 结构域的组蛋白去甲基化酶 (JMJD) 抑制剂的甲酯前药,具有良好的细胞渗透性。在体外试验中,methylstat 的游离酸可抑制 JMJD2A、JMJD2C、JMJD2E、PHF8 和 JMJD3,IC50 值分别约为 4.3、3.4、5.9、10 和 43 µM。 Methylstat 抑制 JMJD2C 敏感的食管癌细胞系 KYSE150 的生长,GI50 为 5.1 µM,而 methylstat 的游离酸在高达 100 µM 时不抑制细胞生长。 Methylstat 以浓度依赖性方式在多个位点诱导组蛋白高甲基化(KYSE150 细胞中 H3K4me3 和 H3K9me3 的 EC50 = 10.3 和 8.6 µM,MCF-7 细胞中的 EC50 分别为 6.7 和 6.3 µM)。
T1960 YL-109

AhR; Aryl Hydrocarbon Receptor Immunology/Inflammation; Metabolism
YL-109是一种抗肿瘤剂,可以通过芳烃受体 AhR 信号传导诱导 Hsp70 相互作用蛋白 (CHIP) 表达,具有抑制乳腺癌细胞生长和侵袭性的能力。
T2283 PX-12

2-[(1-甲基丙基)二硫代]-1H-咪唑,IV-2,PX12

Thioredoxin Metabolism
PX-12 (PX12) 是一种可逆的硫氧还蛋白-1(Trx-1)抑制剂,能够抑制 MCF-7 细胞(IC50:1.9 μM)和HT-29 细胞(IC50:2.9 μM)的生长。
T18981 DMA

Others Others
DMA 是一种荧光试剂 (λex=340 nm, λem=478 nm)。
T68147 T-900607

Microtubule Associated Cytoskeletal Signaling
T-900607是一种新型微管蛋白活性剂,通过独特的作用机制破坏微管聚合。t-900607具有心脏毒性。
T36696 DMBA

7,12-Dimethylbenz[a]anthracene (DMBA) is a polycyclic aromatic hydrocarbon (PAH) that has been found in tobacco smoke and diesel exhaust and has carcinogenic activity.1,2It undergoes metabolic activation by numerous enzymes, including the cytochrome P450 (CYP450) isoform CYP1B1, as well as microsomal epoxide hydrolase (mEH), producing a variety of reactive metabolites that form DNA adductsin vivo, and it has been commonly used to induce tumor formation in various rodent models.2,3,1DMBA increase...
T61899 VEGFR2-IN-1

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
VEGFR2-IN-1 是一种具有选择性和高效性的 VEGFR2 抑制剂,具有抗肿瘤活性,可抑制细胞的增殖和迁移,可用于研究乳腺癌。
T4464 Irosustat

667-Coumate,BN83495,STX64

Others Others
Irosustat (667-Coumate) 是类固醇硫酸酯酶抑制剂(IC50:8 nM),具有抗乳腺癌作用。
T72076 H2-Gamendazole

HSP Cytoskeletal Signaling; Metabolism
H2-Gamendazole 是一种抑制精子发生和癌症治疗的新型化合物,可作为热休克蛋白和/或延伸因子1 α的抑制剂,是 Hsp90调节剂。
T73582 EB1

MNK MAPK
EB1 是一种具有有效性和选择性的 MNK 激酶抑制剂,对 MNK1和 MNK2 具有抑制作用 IC50 分别为 0.69 μM 和 9.4 μM。EB1 抑制癌细胞的生长,促进细胞凋亡,抑制 eIF4E 磷酸化。
T10133 3'-Azido-3'-deoxy-5-methylcytidine

Antiviral; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
3'-Azido-3'-deoxy-5-methylcytidine 抑制 HIV-1 逆转录酶 (EC50 = 0.06 μM),是异嗜性鼠白血病相关逆转录病毒 (XMRV, CC50 = 43.5 μM) 的有效抑制剂。
T13685 ERD-308

Others Others
ERD-308 induces >95% of ER degradation at concentrations as low as 5 nM in both cell lines (DC50 (concentration causing 50% of protein degradation) of 0.17 nM and 0.43 nM in MCF-7 and T47D ER+ cells, respectively).ERD-308 is a highly potent PROTAC degrade
T13292 VDR agonist 1

Others Others
VDR agonist 1 (compound 28) 是一种非甾体类维生素 D 受体 (VDR)的激动剂, 在MCF-7 细胞中测得其IC50值为 690 nM。VDR agonist 1 通过上调 p21 和 p27 的表达来抑制细胞周期,通过增加 BAX 的表达来促进细胞凋亡,降低 Bcl-2 的表达,具有治疗乳腺癌的潜力。
T16357 DA-3003-1

NSC 663284

Phosphatase Metabolism
DA-3003-1 (DA-3003-1) 是一种可渗透进细胞膜且具有有效性和选择性的 Cdc25 dual specificity phosphatase 抑制剂,具有抗肿瘤活性,对 Cdc25B2、Cdc25A、Cdc25B2 和 Cdc25C具有抑制作用。
T27078 CPUY201112

CPUY 201112,CPUY-201112

CPUY201112, a novel inhibitor of heat shock protein Hsp90, induces p53-mediated apoptosis in MCF-7 cells.
T62905 GLS-1-IN-1

GLS-1-IN-1 (compound 1d) 是一种 GLS-1 抑制剂,能够抑制 Hep G2、MCF 7MCF 10A 细胞。
T63676 Bcl-2-IN-6

Bcl-2-IN-6 是 Bcl-2 (b 细胞淋巴瘤-2) 的有效抑制剂,可下调 Bcl-2 的表达,并提高 p53、Bax、caspase-7 mRNA 的表达。Bcl-2-IN-7 能够诱导乳腺癌 MCF-7 细胞周期阻滞和凋亡。Bcl-2-IN-7 能够作用于 MCF-7 细胞 (IC50: 20.91 μM)、LoVo 细胞 (IC50: 22.30 μM)、HepG2 细胞 (IC50: 42.29 μM) 和 A549 细胞 (IC50: 48.00 μM) 均显示出良好的抗肿瘤效果。
T31936 GLL398

GLL 398,GLL-398

GLL398 is an oral selective estrogen receptor down-regulating agent that strongly binds to ERα (IC50 =1.14 nM) and effectively degrades ERα in MCF-7 breast cancer cells (IC50 = 0.21 μM).
T79109 Estrogen receptor modulator 8

Estrogen Receptor/ERR Endocrinology/Hormones
Estrogen receptor modulator8 (compound 4) 为一口服活性化合物,作用为抑制雌激素受体/ERR α(IC50=0.437 nM,MCF-7 细胞)。此化合物能有效抑制MCF-7细胞的增殖,其IC50值仅为0.1 nM。
T60555 Antiproliferative agent-3

Antiproliferative agent-3 (comp 4) 对 MCF-7 癌细胞表现出良好的活性,IC50值为 0.19 nM。
T82715 Cisplatin-resistant cells-IN-1

Cisplatin-resistant cells-IN-1(化合物8)对顽固的铂类药物抗性细胞具有较高的细胞毒性。在低纳摩尔浓度范围内(IC50:0.14–1.79 μM in A549/A549-R, K562/K562-R, and MCF-7/MCF-7TamR cells),该化合物能有效降低代谢活性。
T63521 Bcl-2-IN-7

Bcl-2-IN-7 是 Bcl-2(b 细胞淋巴瘤 -2) 的有效抑制剂,能够下调 Bcl-2 的表达,提高 p53、Bax、caspase-7 mRNA 的表达,能够诱导乳腺癌 MCF-7 细胞周期阻滞和凋亡。Bcl-2-IN-7MCF-7 细胞 (IC50: 20.17 μM)、LoVo 细胞 (IC50: 22.64 μM)、HepG2 细胞 (IC50:45.57 μM) 和 A549 细胞 (IC50: 51.50 μM)均表现出良好的抗肿瘤活性。
T63455 PI3K/Akt/mTOR-IN-3

PI3K/Akt/mTOR-IN-3 是 PI3K/Akt/mTOR 的有效抑制剂。PI3K/Akt/mTOR-IN-3 能够抑制 MCF-7 细胞 (IC50: 0.77 μM)、HeLa 细胞 (IC50: 1.23 μM) 和 HepG2 细胞(IC50: 4.57 μM)。PI3K/Akt/mTOR-IN-3 在 4 μM 浓度下可抑制 MCF-7 和 HeLa 细胞的迁移。PI3K/Akt/mTOR-IN-3 能够将细胞周期阻滞在 S 期,并诱导细胞凋亡 (apoptosis)。
T39203 Raloxifene 6-Monomethyl Ether

Compound 7, or Raloxifene 6-Monomethyl Ether, is a derivative of Raloxifene that effectively inhibits estrogen receptor α. It also displays the inhibitory effects on MCF-7 cells, with an IC50 of 250 nM and a pIC50 of 6.6.
T79727 EGFR/CDK2-IN-2

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
EGFR/CDK2-IN-2(compound 6a)是一种针对EGFR和CDK-2的双重抑制剂,具有19.6 nM和87.9 nM的IC50s。该化合物能在MCF-7细胞内诱导凋亡,并在S期引发细胞周期停滞。此外,EGFR/CDK2-IN-2展现出IC50为0.39 μM的显著抗癌活性,对MCF-7细胞具有强效的细胞毒性。
T22159 TCS HDAC6 20b

TCS HDAC6 20b 是一种HDAC6选择性抑制剂,可阻断雌激素受体 α 阳性乳腺癌 MCF-7 细胞的生长。
T83017 Antiproliferative agent-40

抗增殖剂-40(化合物9)对HT1080和MCF-7细胞系展示了明显的抑制效果,其IC50值分别为52 μM和8.2 μM。
T83874 S-72

S-72是一种微管聚合抑制剂,以1, 3, 10 µM的浓度在无细胞测定中抑制微管聚合,并在MCF-7和耐紫杉醇的MCF-7/T乳腺癌细胞中降低细胞活性(IC50分别为15.64和26.32 nM)。50 nM浓度的S-72能抑制MCF-7MCF-7/T细胞的迁移和侵袭,并减少划痕实验中的伤口闭合百分比。100 nM的S-72在MCF-7/T细胞中诱导G2/M期的细胞周期阻滞以及凋亡,并在同一浓度下抑制这些细胞中干扰素基因激活剂(STING)的激活。以每天15 mg/kg的剂量,S-72抑制了耐紫杉醇的MCF-7/T和MX-1/T小鼠异种移植模型中的肿瘤生长。
T72523 Antitumor agent-46

Antitumor agent-46 是一种抗肿瘤剂。Antitumor agent-46 对 MCF-7 细胞具有明显更高的抗增殖活性,IC50值为 2.08 µM。
T80537 Ac-AAVALLPAVLLALLAP-LEHD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-LEHD-CHO 是半胱天冬酶4、5和9的抑制剂,能够对Neocarzinostatin处理的MCF-7细胞展现保护效果。
T79729 EGFR/CDK2-IN-4

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
EGFR/CDK2-IN-4(化合物4c)是一种EGFR与CDK-2的双重抑制剂,其IC50值分别为89.6 nM和165.4 nM。该化合物在MCF-7细胞中能诱导(apoptosis)凋亡,并导致细胞周期在S期停滞。EGFR/CDK2-IN-4显示出显著的抗癌细胞毒性,对MCF-7细胞的IC50为2.74 μM。

化合物

HNHA
Cat.No: T21806
Synonym:
Target: HDAC
σ1 Receptor antagonist-1
Cat.No: T9244
Synonym:
Target: Sigma receptor
Mitoxantrone
Cat.No: T6588
Synonym: 米托蒽醌,mitozantrone
Target: Topoisomerase, PKC
Estrogen receptor modulator 1
Cat.No: T15249
Synonym:
Target: Estrogen Receptor/ERR
PQ401
Cat.No: T2085
Synonym: IGF-1R Inhibitor II
Target: Apoptosis, IGF-1R
(1E)-CFI-400437 dihydrochloride
Cat.No: T22288
Synonym: CFI-400437 dihydrochloride
Target: PLK
3-Bromopyruvic acid
Cat.No: T5882
Synonym: Hexokinase II Inhibitor II, 3-BP,3-溴丙酮酸,Bromopyruvic acid
Target: Apoptosis, Hexokinase, Autophagy
Mitoxantrone dihydrochloride
Cat.No: T0158
Synonym: 米托蒽醌二盐酸盐,盐酸米托蒽醌,Mitoxantrone 2HCl,Mitoxantrone hydrochloride,NSC-301739,mitozantrone dihydrochloride
Target: Topoisomerase, PKC
Idarubicin hydrochloride
Cat.No: T6010
Synonym: 盐酸伊达比星,Idamycin,4-demethoxydaunorubicin (NSC256439, 4-DMDR) HCl,4-Demethoxydaunorubicin hydrochloride,Idarubicin HCl,伊达比星盐酸盐,Zavedos
Target: Topoisomerase, Antibacterial, Autophagy, Antifungal
Estrone O-sulfamate
Cat.No: T72470
Synonym: Estrone 3-O-sulfamate
Target: Others
ANI-7
Cat.No: T10325
Synonym:
Target: Chk
CTB
Cat.No: T9541
Synonym: Cholera Toxin B subunit
Target: Epigenetic Reader Domain
Antiproliferative agent-16
Cat.No: T64348
Synonym: Antiproliferative agent-16
Target: Others
LYG-202
Cat.No: T36488
Synonym: LYG202,LYG 202
Target: Apoptosis, ROS
STD1T
Cat.No: T36970
Synonym:
Target: DUB
(Iso)-MS4322
Cat.No: T40233
Synonym: (Iso)-YS43-22,MS4322 (isomer),YS43-22 (isomer)
Target: Histone Methyltransferase
Ro 41-5253
Cat.No: T28589
Synonym: Ro-41-5253,Ro 415253
Target: Apoptosis, Retinoid Receptor
Pim-1 kinase inhibitor 8
Cat.No: T83627
Synonym:
Target: Pim, PKC
P-gb-IN-1
Cat.No: T77575
Synonym:
Target: P-gp
Methylstat
Cat.No: T7057
Synonym:
Target: Histone Demethylase, Others
YL-109
Cat.No: T1960
Synonym:
Target: AhR, Aryl Hydrocarbon Receptor
PX-12
Cat.No: T2283
Synonym: 2-[(1-甲基丙基)二硫代]-1H-咪唑,IV-2,PX12
Target: Thioredoxin
DMA
Cat.No: T18981
Synonym:
Target: Others
T-900607
Cat.No: T68147
Synonym:
Target: Microtubule Associated
DMBA
Cat.No: T36696
Synonym:
Target:
VEGFR2-IN-1
Cat.No: T61899
Synonym:
Target: VEGFR
Irosustat
Cat.No: T4464
Synonym: 667-Coumate,BN83495,STX64
Target: Others
H2-Gamendazole
Cat.No: T72076
Synonym:
Target: HSP
EB1
Cat.No: T73582
Synonym:
Target: MNK
3'-Azido-3'-deoxy-5-methylcytidine
Cat.No: T10133
Synonym:
Target: Antiviral, HIV Protease
ERD-308
Cat.No: T13685
Synonym:
Target: Others
VDR agonist 1
Cat.No: T13292
Synonym:
Target: Others
DA-3003-1
Cat.No: T16357
Synonym: NSC 663284
Target: Phosphatase
CPUY201112
Cat.No: T27078
Synonym: CPUY 201112,CPUY-201112
Target:
GLS-1-IN-1
Cat.No: T62905
Synonym:
Target:
Bcl-2-IN-6
Cat.No: T63676
Synonym:
Target:
GLL398
Cat.No: T31936
Synonym: GLL 398,GLL-398
Target:
Estrogen receptor modulator 8
Cat.No: T79109
Synonym:
Target: Estrogen Receptor/ERR
Antiproliferative agent-3
Cat.No: T60555
Synonym:
Target:
Cisplatin-resistant cells-IN-1
Cat.No: T82715
Synonym:
Target:
Bcl-2-IN-7
Cat.No: T63521
Synonym:
Target:
PI3K/Akt/mTOR-IN-3
Cat.No: T63455
Synonym:
Target:
Raloxifene 6-Monomethyl Ether
Cat.No: T39203
Synonym:
Target:
EGFR/CDK2-IN-2
Cat.No: T79727
Synonym:
Target: EGFR
TCS HDAC6 20b
Cat.No: T22159
Synonym:
Target:
Antiproliferative agent-40
Cat.No: T83017
Synonym:
Target:
S-72
Cat.No: T83874
Synonym:
Target:
Antitumor agent-46
Cat.No: T72523
Synonym:
Target:
Ac-AAVALLPAVLLALLAP-LEHD-CHO
Cat.No: T80537
Synonym:
Target: Caspase
EGFR/CDK2-IN-4
Cat.No: T79729
Synonym:
Target: EGFR
Cat. No. Product Name Target Signaling Pathways
TN1768 Iriflophenone

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Iriflophenone 是从 Aquilaria sinensis 中分离得到,能诱导 MCF-7 和 T-47D 人乳腺癌细胞增殖。
T5724 Neogambogic acid

neo-gambogic acid,新藤黄酸

Apoptosis; Others; Antibacterial Apoptosis; Microbiology/Virology; Others
Neogambogic acid 是藤黄的有效成分,可诱导细胞凋亡并具有抗癌作用。它有效抑制耐甲氧西林的金黄色葡萄球菌。
T2882 Genistin

染料木甙,Genistoside,Genistein glucoside,Genistein 7-glucoside,Genistine,Genistein 7-O-β-D-glucopyranoside,染料木苷

Apoptosis; Estrogen Receptor/ERR; Others Apoptosis; Endocrinology/Hormones; Others
Genistin (Genistoside) 是一种植物雌激素家族的异黄酮,是一种抗脂肪生成剂。它通过调节ERalpha 信号通路抑制乳腺癌细胞生长和促进凋亡细胞死亡。
T7786 Tryptanthrin

DNA gyrase DNA Damage/DNA Repair
Tryptanthrin 是一种口服具有活性的细胞内Leukotriene (LT) biosynthesis 抑制剂。 它能够降低大鼠胸膜炎模型中的 LTB4 水平,并抑制人全血中Leukotriene 的形成 (IC50= 10 µM)。
T19768 γ-Tocotrienol

gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol,γ-生育三烯酚

Others Others
γ-Tocotrienol (Plastochromanol) 是一种维生素 E 的活性形式。
TN7041 (-)-Epipodophyllotoxin

Apoptosis Apoptosis
(-)-Epipodophyllotoxin 是一种从八角莲中分离的癌细胞抗增殖剂,在 HeLa 细胞和 MCF-7 细胞中的GI50值分别为 0.36 和 0.24 μM。它可在体外抑制有丝分裂纺锤体组装。
T12581 Puerarin-4'-O-β-D-glucopyranoside

Puerarin4'-O-glucoside,葛根素-4'-Β-D-葡萄糖苷

Others Others
Puerarin-4'-O-β-D-glucopyranoside (Puerarin4'-O-glucoside) 是一种从葛根 (PLR) 中提取的异黄酮。它具有雌激素活性和抗 MCF-7 人乳腺癌细胞增殖作用。
T83321 4-Demethyldeoxypodophyllotoxin

Chk Cell Cycle/Checkpoint
4-Demethyldeoxypodophyllotoxin 是一种来自 Podophyllum peltatum 根部的芳基四氢萘木酚素类化合物,具有抗癌活性,可调节 MCF-7乳腺癌细胞中的Chk-2信号通路。
TMA2270 Alisol F 24-acetate

P-gp Membrane transporter/Ion channel; Neuroscience
Alisol F 24-acetate 是一种从 Alisma plantago-aquatica Linn [1] 中分离出来的天然产物。 Alisol F 24 Acetate 通过抑制 P-糖蛋白介导的药物流出来增强 MCF-7/DOX 细胞的化学敏感性和凋亡。
T4S0544 Furanodienone

呋喃二烯酮,莪术呋喃二烯酮

Apoptosis; HER Angiogenesis; Apoptosis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Furanodienone 是来源于姜黄根茎的一种主要生物活性成分,可诱导细胞凋亡。
T4519 Alisol A

Alisol-A,泽泻醇 A

Autophagy Autophagy
Alisol A (Alisol-A) 是泽泻中的一种三萜类天然产物,可能是一种自噬诱导剂,具有抗癌活性。
T3411 Curdione

莪术二酮,(+)-Curdione

P450 Metabolism
Curdione ((+)-Curdione) 是一种具有高生物活性的倍半萜类物质,从莪术中分离获得,具有抑制血小板聚集、抵抗血栓形成的作用。
TJS0387 Desoxyrhaponticin

去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin

Apoptosis; Fatty Acid Synthase Apoptosis; Metabolism
Desoxyrhaponticin (Deoxyrhaponticin) 是来自西藏营养食品唐古特大黄中的一种二苯乙烯苷。它是脂肪酸合成酶抑制剂,抑制细胞内 FAS 活性,下调人乳腺癌 MCF-7细胞中 FAS 的表达。它是控制糖尿病餐后高血糖的潜在药物。
T3S1416 Decursin

Decursinol angelate,前胡素,(+)-Decursin,紫花前胡素

Apoptosis; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling
Decursin (Decursinol angelate) 是一种细胞毒性剂,是一种来自朝鲜当归根的有效蛋白激酶 C 激活剂。它通过 Hippo/YAP 信号通路抑制 HepG2 细胞的生长。它通过下调 CXCR7 表达来抑制胃癌中的肿瘤生长,迁移和侵袭。
T5S2358 Dehydrocorydaline

Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline (13-Methylpalmatine) 是一种生物碱。它调节Bax,Bcl-2蛋白表达,激活caspase-7,caspase-8,并使PARP 失活。它能增强p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T3S2344 β,β-Dimethylacrylshikonin

β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin

ERK; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; MAPK; Metabolism
β,β-Dimethylacrylshikonin (Dimethylacrylshikonin) 是一种萘醌衍生物,从 Arnebia nobilis 中提取得到。它利用 PI3K 通路诱导 eNOS、VEGF 和 HIF-1α 的表达,促进血管生成,具有抗肿瘤活性。
T6S1315 Oroxylin A

千层纸素A,6-Methoxybaicalein,Baicalein 6-methyl ether

Virus Protease; HIF/HIF Prolyl-Hydroxylase; Autophagy Autophagy; Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Oroxylin A (Baicalein 6-methyl ether) 是一种有活性的黄酮,具有较强的抗癌作用。
T3729 Ethyl gallate

Nipagallin A,Phyllemblin,gallic acid ethyl ester,没食子酸乙酯

MMP; NF-κB; Akt; Antibacterial Cytoskeletal Signaling; Microbiology/Virology; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Ethyl gallate (gallic acid ethyl ester) 是一种非类黄酮酚过氧化氢清除剂。
T2S1865 Octyl gallate

Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯

Antioxidant; Influenza Virus; Reactive Oxygen Species; Antibacterial; Antifungal; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) 具有抗菌、抗氧化作用,有选择性和敏感性的荧光特性,广泛用作食品添加剂。它对 HSV-1,水泡性口炎病毒和脊髓灰质炎病毒有显著的抗病毒作用。
T17155 Trabectedin

Ecteinascidin 743,曲贝替定,ET-743

Apoptosis; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB
Trabectedin (Ecteinascidin 743) 是一种四氢异喹啉生物碱,有抗肿瘤的活性, 通过与 DNA 的小沟结合,阻断应激诱导的蛋白质的转录,诱导 DNA 骨架裂解和癌细胞凋亡,并增加 MCF-7 和 MDA-MB-453 细胞中 ROS 的生成。Trabectedin 在软组织肉瘤和卵巢癌中具有的研究价值。
TN5538 6-Methoxykaempferol

Others Others
6-Methoxykaempferol 是一种存在于 brazilian propolis 中的黄酮。6-Methoxykaempferol 对癌细胞具有抗增殖活性,对离体大鼠脑突触体的神经保护作用,可降低的谷胱甘肽水平。6-Methoxykaempferol 表现出一定的脂肪酶活性,可用于恶病质的治疗。
T8724 6-Methoxydihydrosanguinarine

Others Others
6-Methoxydihydrosanguinarine 是一种从M. cordata 果实中分离出的生物碱,它对 MCF-7 细胞系(IC50:0.61 μM)和 SF-268 细胞系(IC50:0.54 μM)具有强的细胞毒性。
T2902 Costunolide

Costus lactone,NSC 106404,Costunolid,(+)-Costunolide,木香烃内酯

Apoptosis; Endogenous Metabolite; Telomerase Apoptosis; DNA Damage/DNA Repair; Metabolism
Costunolide (Costus lactone) 是一种天然的倍半萜内酯,具有抗氧化、抗炎、抗过敏、骨重塑、神经保护、促进毛发生长、抗癌和抗糖尿病的特性,可诱导乳腺癌细胞周期阻滞和凋亡。
T1174 Topotecan hydrochloride

SKF 104864A,SKFS 104864A,NSC609699,Nogitecan HCl,NSC 609669,盐酸拓扑替康,Topotecan HCl

Apoptosis; Topoisomerase; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair
Topotecan hydrochloride (NSC609699) 是一种具有抗癌活性的拓扑异构酶I 抑制剂。
TN2249 (+)-Syringaresinol

Sirtuin; Antifection Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology
(+)-Syringaresinol shows antioxidant potential, it exhibits cytoprotective activity in cultured MCF-7 cells stressed by H2O2.
T40940 7,3′,5′-Trihydroxyflavanone

7,3′,5′-Trihydroxyflavanone, a flavanoid derivative, promotes apoptotic cell death in MCF-7 cells by augmenting Bax expression. Additionally, this compound demonstrates antioxidant properties.
T83301 5,7-Dimethoxy-2,3-phenanthrenediol

5,7-Dimethoxy-2,3-phenanthrenediol 表现出雌激素活性,能够促进MCF-7细胞的增殖,并增强ERβ在MCF-7细胞系中的表达。
TN1578 Dihydroconiferyl alcohol

Others Others
Dihydroconiferyl alcohol exhibits cytoprotective activity in cultured MCF-7 cells stressed by H2O2.
T83089 Anticancer agent 149

Anticanceragent 149 (compound 3) 是一种从薯蓣 (DM) 根茎中分离出的抗癌剂,其对MCF-7 细胞呈现选择性细胞毒活性,特有IC50值为31.41 μM。
T75484 Clionamine B

Clionamine B, 一种海绵 Cliona celata 分离出来的刺激自噬的氨基类固醇,强烈刺激人乳腺癌 MCF-7 细胞的自噬。
T81529 Peganumine A

Peganumine A,一种天然产物,源自Peganum harmala,具备对HL-60、MCF-7、PC-3、HepG2细胞线显示出细胞毒性作用,其IC50值依次为5.8、38.5、40.2、55.4 µM[1]< /sup>。
TN4903 Regiolone

Caspase Apoptosis; Proteases/Proteasome
Regiolone demonstrates phytotoxicity. Regiolone also has anti-proliferative and apoptotic activities, it can induce apoptosis in MCF-7 cells through the caspase-3 independent pathway.
T69368 GKK1032B

GKK1032B is a fungal metabolite that has antiproliferative and antibacterial activities. GKK1032B inhibits the growth of HeLa S3 cervical and MCF-7 breast cancer cells and Vero cells. It also inhibits the growth of B. subtilis and M. tuberculosis.
TN3429 Aphagranin A

Others Others
Aphagranin A exhibits strong antiproliferative activity against the growth of six lines of human cancer cells (MCF-7, A549, HepG2, Bel-7402, SGC-7901, and BGC-823.
T75490 27-O-(tert-Butyldimethylsilyl)withaferin A

27-O-(tert-Butyldimethylsilyl)withaferin A (compound 9a) 为一种天然茄内酯类化合物,具备诱导细胞凋亡 (apoptosis) 的能力。该化合物对人类癌细胞系HeLa、A-549、MCF-7以及正常Vero细胞展现出抗增殖活性。
TN2288 Uralenol

乌拉尔醇

Others; Estrogen/progestogen Receptor; Tyrosinase Endocrinology/Hormones; Others; Proteases/Proteasome
Uralenol significantly shows the inhibitory activities against the PTP1B enzyme; it also shows inhibitory activities on mushroom tyrosinase using l-tyrosine as substrate( IC50 =49.5 μM). Uralenol shows potent anti-proliferation effects on ER-positive breast cancer MCF-7 cells in vitro.
T73403 Aviculin

Aviculin 是一种木聚糖苷,是一种有效的抗癌剂 (anticanceragent)。Aviculin 可降低 MCF-7 细胞代谢活性到 50% 以下,IC50为 75.47 μM。Aviculin 通过内在凋亡途径诱导乳腺癌细胞凋亡 (apoptosis)。Aviculin 增加了 caspase-9、caspase-7和 PARP 的表达。Aviculin 使 Bax/Bcl-2 的比值升高。
TN3049 4-Methoxycinnamyl alcohol

Others Others
4-Methoxycinnamyl alcohol 对MCF-7、HeLa 和DU145癌症细胞系显示出毒性,IC50值分别为14.24、7.82和22.10μg/mL。4-methoxycinnamyl alcohol 是从Foeniculum vulgare 中分离出来的。4-Methoxycinnamyl alcohol 没有显示出凋亡作用,却在10μg/mL DNA 碎片研究显示48小时后发生了坏死。
TN3084 5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone

Estrogen Receptor/ERR; Others Endocrinology/Hormones; Others
5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone 具有抗癌活性,体外对 ER 阳性乳腺癌MCF-7细胞表现出较强的抗增殖作用,对MCF-7细胞的IC50值为4.41 uM。5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone 能显著下调雌激素受体-α (ER-α)的表达浓度,并能抑制人乳腺癌细胞系BCAP-37异种移植模型体内的肿瘤生长。
TN5657 Goniotriol

Goniotriol shows antimycobacterial activity against Mycobacterium tuberculosis (MIC =100 microg/mL). It exhibits antiplasmodial activity against Plasmodium falciparum (IC50=2.6 microg/mL). Goniotriol shows cytotoxicity against cancer cells, KB, BC1, NCI-H
TN5647 Confluentin

Confluentin has antimicrobial activity against the gram-positive bacteria.Confluentin significantly inhibits compound 48/80-induced histamine release from rat peritoneal mast cells. Confluentin also shows weak cytotoxicity against four human tumor cell li
T1166 Ellipticine

玫瑰树碱,NSC 71795,Elliptisine

Topoisomerase DNA Damage/DNA Repair
Ellipticine (Elliptisine) 是一种有效的抗肿瘤剂,抑制 DNA 拓扑异构酶 II 活性,对白血病、神经母细胞瘤和胶质母细胞瘤有部分活性。
TN2767 2'-Hydroxygenistein

鲁冰花

Antifection Microbiology/Virology
2'-Hydroxygenistein has antifungal activity, dimerization of it causes a remarkable increase of antifungal activity. It shows significant concentration-dependent inhibitory effects on the release of beta-glucuronidase and lysozyme from rat neutrophils in response to formyl-Met-Leu-Phe/cytochalasin B. 2'-Hydroxygenistein of genistein can enhance its antioxidant activity and cell cytotoxicity in MCF-7 human breast cancer cells.
TN4552 Methyl p-hydroxyphenyllactate

Others Others
Methyl para-hydroxyphenyllactate(MeHPLA) can suppress the cellular proliferation of estrogen-sensitive MCF-7 breast cancer cells in vitro and to suppress the growth of rat uteri in vivo, high affinity of MeHPLA for the type II estrogen binding site (EBS)
TN5930 Ocotillone

Ocotillone has potent antibacterial activity against Gram-negative bacteria, P. aeruginosa and S. typhimurium, that are without hemolytic activity, whereas it has weak antimicrobial activity against Gram-positive bacteria and fungi. Ocotillone shows only
T3P2855 Chamigrenal

EGFR; NOS; PAFR; COX; Prostaglandin Receptor Angiogenesis; GPCR/G Protein; Immunology/Inflammation; JAK/STAT signaling; Neuroscience; Tyrosine Kinase/Adaptors
β-Chamigrenal has anti-inflammatory activity, it has inhibitory effects on lipopolysaccharide-induced nitric oxide and prostaglandin E2 production in RAW 264.7 macrophages. Chamigrenal shows platelet-activating factor antagonistic activity and the IC(50)
T83597 (+)-Menthyl acetate

(+)-Menthyl acetate是一种从Cunila angustifolia Benth精油中分离得到的化学化合物。它对MCF-7细胞株具有较高的选择性,其半抑制浓度(IC50)为34.0 μg/mL,而对SK-Mel-28细胞株的选择性较低,IC50为279.9 μg/mL,并且对A549细胞没有致死作用。
TN3870 Iriflophenone 2-O-Rhamnoside

Dimethylmatairesinol

Others Others
Dimethylmatairesinol can reduce the amount of Immunoglobulin E (IgE) secreted by human myeloma U266 cells, it has potential as an anti-allergic agent. Dimethylmatairesinol also exhibits significant cytotoxicity against three human tumor cells(A-549 lung c
T37452 Stephacidin B

Stephacidin B is a fungal metabolite that has been found inA. ochraceus.1Dimeric stephacidin B is rapidly converted to a monomer, avrainvillamide ,in vitro.2Stephacidin B is cytotoxic to a variety of cancer cells, including testosterone-independent PC3 and -sensitive LNCaP prostate cancer cells (IC50s = 0.37 and 0.06 μM, respectively) and estradiol-independent SK-BR-3 and -sensitive MCF-7 breast cancer cells (IC50s = 0.32 and 0.27 μM, respectively).1It induces apoptosis in HepG2 and Huh7 hepatoc...
T35754 Aszonapyrone A

Aszonapyrone A is a meroditerpene fungal metabolite that has been found in Neosartorya and has diverse biological activities.1,2,3 It inhibits the growth of MCF-7, NCI H460, and A375-C5 cancer cells (GI50s = 13.6, 11.6, and 10.2 μM, respectively).1 Aszonapyrone A is active against multidrug-resistant isolates of S. aureus, E. faecalis, and E. faecium (MICs = 8, 16, and 16 μg/ml, respectively) and inhibits S. aureus biofilm formation.2 It is also active against P. falciparum in vitro (IC50 = 1.34...
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天然产物

Iriflophenone
Cat.No: TN1768
Synonym:
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Neogambogic acid
Cat.No: T5724
Synonym: neo-gambogic acid,新藤黄酸
Target: Apoptosis, Others, Antibacterial
Genistin
Cat.No: T2882
Synonym: 染料木甙,Genistoside,Genistein glucoside,Genistein 7-glucoside,Genistine,Genistein 7-O-β-D-glucopyranoside,染料木苷
Target: Apoptosis, Estrogen Receptor/ERR, Others
Tryptanthrin
Cat.No: T7786
Synonym:
Target: DNA gyrase
γ-Tocotrienol
Cat.No: T19768
Synonym: gamma Tocotrienol,gammaTocotrienol,gamma-Tocotrienol,D-gamma-Tocotrienol,Plastochromanol,γ-生育三烯酚
Target: Others
(-)-Epipodophyllotoxin
Cat.No: TN7041
Synonym:
Target: Apoptosis
Puerarin-4'-O-β-D-glucopyranoside
Cat.No: T12581
Synonym: Puerarin4'-O-glucoside,葛根素-4'-Β-D-葡萄糖苷
Target: Others
4-Demethyldeoxypodophyllotoxin
Cat.No: T83321
Synonym:
Target: Chk
Alisol F 24-acetate
Cat.No: TMA2270
Synonym:
Target: P-gp
Furanodienone
Cat.No: T4S0544
Synonym: 呋喃二烯酮,莪术呋喃二烯酮
Target: Apoptosis, HER
Alisol A
Cat.No: T4519
Synonym: Alisol-A,泽泻醇 A
Target: Autophagy
Curdione
Cat.No: T3411
Synonym: 莪术二酮,(+)-Curdione
Target: P450
Desoxyrhaponticin
Cat.No: TJS0387
Synonym: 去氧土大黄苷,Deoxyrhapontin,脱氧土大黄苷,Deoxyrhaponticin
Target: Apoptosis, Fatty Acid Synthase
Decursin
Cat.No: T3S1416
Synonym: Decursinol angelate,前胡素,(+)-Decursin,紫花前胡素
Target: Apoptosis, PKC
Dehydrocorydaline
Cat.No: T5S2358
Synonym: Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
β,β-Dimethylacrylshikonin
Cat.No: T3S2344
Synonym: β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin
Target: ERK, HIF/HIF Prolyl-Hydroxylase
Oroxylin A
Cat.No: T6S1315
Synonym: 千层纸素A,6-Methoxybaicalein,Baicalein 6-methyl ether
Target: Virus Protease, HIF/HIF Prolyl-Hydroxylase, Autophagy
Ethyl gallate
Cat.No: T3729
Synonym: Nipagallin A,Phyllemblin,gallic acid ethyl ester,没食子酸乙酯
Target: MMP, NF-κB, Akt, Antibacterial
Octyl gallate
Cat.No: T2S1865
Synonym: Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯
Target: Antioxidant, Influenza Virus, Reactive Oxygen Species, Antibacterial, Antifungal, HSV
Trabectedin
Cat.No: T17155
Synonym: Ecteinascidin 743,曲贝替定,ET-743
Target: Apoptosis, Reactive Oxygen Species
6-Methoxykaempferol
Cat.No: TN5538
Synonym:
Target: Others
6-Methoxydihydrosanguinarine
Cat.No: T8724
Synonym:
Target: Others
Costunolide
Cat.No: T2902
Synonym: Costus lactone,NSC 106404,Costunolid,(+)-Costunolide,木香烃内酯
Target: Apoptosis, Endogenous Metabolite, Telomerase
Topotecan hydrochloride
Cat.No: T1174
Synonym: SKF 104864A,SKFS 104864A,NSC609699,Nogitecan HCl,NSC 609669,盐酸拓扑替康,Topotecan HCl
Target: Apoptosis, Topoisomerase, Autophagy
(+)-Syringaresinol
Cat.No: TN2249
Synonym:
Target: Sirtuin, Antifection
7,3′,5′-Trihydroxyflavanone
Cat.No: T40940
Synonym:
Target:
5,7-Dimethoxy-2,3-phenanthrenediol
Cat.No: T83301
Synonym:
Target:
Dihydroconiferyl alcohol
Cat.No: TN1578
Synonym:
Target: Others
Anticancer agent 149
Cat.No: T83089
Synonym:
Target:
Clionamine B
Cat.No: T75484
Synonym:
Target:
Peganumine A
Cat.No: T81529
Synonym:
Target:
Regiolone
Cat.No: TN4903
Synonym:
Target: Caspase
GKK1032B
Cat.No: T69368
Synonym:
Target:
Aphagranin A
Cat.No: TN3429
Synonym:
Target: Others
27-O-(tert-Butyldimethylsilyl)withaferin A
Cat.No: T75490
Synonym:
Target:
Uralenol
Cat.No: TN2288
Synonym: 乌拉尔醇
Target: Others, Estrogen/progestogen Receptor, Tyrosinase
Aviculin
Cat.No: T73403
Synonym:
Target:
4-Methoxycinnamyl alcohol
Cat.No: TN3049
Synonym:
Target: Others
5,7,3',4'-Tetrahydroxy-3-methoxy-8,5'-diprenylflavone
Cat.No: TN3084
Synonym:
Target: Estrogen Receptor/ERR, Others
Goniotriol
Cat.No: TN5657
Synonym:
Target:
Confluentin
Cat.No: TN5647
Synonym:
Target:
Ellipticine
Cat.No: T1166
Synonym: 玫瑰树碱,NSC 71795,Elliptisine
Target: Topoisomerase
2'-Hydroxygenistein
Cat.No: TN2767
Synonym: 鲁冰花
Target: Antifection
Methyl p-hydroxyphenyllactate
Cat.No: TN4552
Synonym:
Target: Others
Ocotillone
Cat.No: TN5930
Synonym:
Target:
Chamigrenal
Cat.No: T3P2855
Synonym:
Target: EGFR, NOS, PAFR, COX, Prostaglandin Receptor
(+)-Menthyl acetate
Cat.No: T83597
Synonym:
Target:
Iriflophenone 2-O-Rhamnoside
Cat.No: TN3870
Synonym: Dimethylmatairesinol
Target: Others
Stephacidin B
Cat.No: T37452
Synonym:
Target:
Aszonapyrone A
Cat.No: T35754
Synonym:
Target:
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