313
20
5
14
41
Cat. No. | Product Name | ||
---|---|---|---|
L1510 | 核受体化合物库 | 531 compounds | |
531 个核受体作用化合物的独特集合,可用于高通量筛选和高内涵筛选; | |||
L2700 | 肾上腺素能受体化合物库 | 193 compounds | |
193 种特异靶向肾上腺素受体的生物活性小分子化合物的集合,是相关疾病药物筛选的有效工具; | |||
L3300 | 组胺&褪黑色素化合物库 | 153 compounds | |
153 种生物活性小分子化合物,用于高通量、高内涵筛选; | |||
L2800 | 5-羟色胺分子库 | 268 compounds | |
268 种生物活性小分子化合物,用于高通量、高内涵筛选; | |||
L2610 | 神经递质受体化合物库 | 1513 compounds | |
1513 种与神经递质受体相关的化合物,用于高通量、高内涵筛选; |
Cat. No. | Product Name | Form | Specificity Of Inhibition |
---|---|---|---|
CL0070 |
GABA Receptor inhibitor kit
GABA Receptor inhibitor kit |
||
CL0079 |
Adenosine Receptor inhibitor kit
Adenosine Receptor inhibitor kit |
||
CL0078 |
Glucocorticoid Receptor inhibitor/activator kit
Glucocorticoid Receptor inhibitor/activator kit |
||
CL0060 |
Estrogen Receptor inhibitor kit
Estrogen Receptor inhibitor kit |
||
CL0059 |
Dopamine Receptor inhibitor kit
Dopamine Receptor inhibitor kit |
||
CL0126 |
Androgen Receptor antagonist kit
Androgen Receptor antagonist kit |
||
CL0144 |
Endothelin Receptor antagonist kit
Endothelin Receptor antagonist kit |
||
CL0051 |
Adrenergic Receptor antagonist/agonist kit
Adrenergic Receptor antagonist/agonist kit |
||
CL0046 |
5-HT Receptor antagonist/agonist kit
5-HT Receptor antagonist/agonist kit |
||
CL0097 |
Prostaglandin Receptor antagonist/agonist kit
Prostaglandin Receptor antagonist/agonist kit |
||
CL0088 |
Angiotensin Receptor inhibitor kit
Angiotensin Receptor inhibitor kit |
||
CL0049 |
Histamine Receptor antagonist kit
Histamine Receptor antagonist kit |
||
CL0110 |
Progesterone Receptor agonist/antagonist/modulator kit
Progesterone Receptor agonist/antagonist/modulator kit |
||
CL0148 |
LPL Receptor antagonist/agonist kit
LPL Receptor antagonist/agonist kit |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11175 |
Elenbecestat
E2609 |
Beta-Secretase; BACE | Neuroscience |
Elenbecestat (E2609) 是一种高效、有口服活性的,能透过 CNS 的 BACE-1抑制剂,它有用于阿尔茨海默病 (AD) 的研究潜力。 | |||
T8848 |
GPR34 receptor antagonist 2
Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-,gpr34-receptor-antagonist-2 |
Others | Others |
GPR34 receptor antagonist 2 (Tyrosine, N-[(2E)-3-(4'-chloro[1,1'-biphenyl]-4-yl)-1-oxo-2-propen-1-yl]-O-(phenylmethyl)-) 是一种GPR34受体拮抗剂,可用于研究免疫疾病、炎性疾病。 | |||
T30191L |
Atecegatran TFA
Atecegatran TFA(917904-13-3 Free base),AR-H067637 TFA |
Others | Others |
Atecegatran TFA 常被当作一种抗凝血剂,可用来治疗心血管疾病。 | |||
T38836L |
Protease-Activated Receptor-1, PAR-1 Agonist acetate
|
Protease-activated Receptor | GPCR/G Protein |
Protease-Activated Receptor-1, PAR-1 Agonist acetate 是一种选择性蛋白酶激活受体 1 (PAR-1) 激动剂肽。 它对应于 PAR1 栓系配体,可以选择性地模拟凝血酶通过该受体的作用。 | |||
T1824 |
TGR5 Receptor Agonist
|
GPCR19 | GPCR/G Protein |
TGR5 Receptor Agonist 是一种TGR5(GPCR19)激动剂。 | |||
T78646 |
Estrogen receptor antagonist 8
|
Estrogen/progestogen Receptor | Endocrinology/Hormones |
Estrogen receptor antagonist 8 作为一种雌激素受体(ER)拮抗剂,具有抗子宫活性和潜在的抗肿瘤活性,可用于研究卵巢功能障碍。 | |||
T15785 |
LPA1 receptor antagonist 1
LPA1 R antagonist 1 |
LPA Receptor | GPCR/G Protein |
LPA1 receptor antagonist 1(LPA1 R antagonist 1) 是一种具有选择性和高效性的溶血磷脂酸 (LPA1) 受体拮抗剂( IC50 : 25 nM),可用于研究特发性肺纤维化。 | |||
T10058 |
A2B receptor antagonist 1
|
Adenosine Receptor | GPCR/G Protein; Neuroscience |
A2B receptor antagonist 1 是一个有效的 A2B 腺苷受体 (A2B adenosine receptor) 拮抗剂。 | |||
T21723L |
Epidermal Growth Factor Receptor Peptide Acetate
Epidermal Growth Factor Receptor Peptide Acetate(96249-43-3 Free base) |
Others | Others |
Epidermal Growth Factor Receptor Peptide Acetate (Epidermal Growth Factor Receptor Peptide Acetate (96249-43-3 Free base)) 存在于细胞表面,通过与其特异性配体的结合而被激活。EGFR 属于受体酪氨酸激酶(RTK) 的 ErbB 家族。 | |||
T9579L |
GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate (2401892-71-3 Free base) |
Glucagon Receptor | GPCR/G Protein |
GLP-1 receptor agonist 9 citrate 是 GLP-1 的激动剂。 | |||
T10307 |
AMPA receptor modulator-1
|
iGluR | Membrane transporter/Ion channel; Neuroscience |
AMPA receptor modulator-1可被谷氨酸激活,从而调节离子通道。 | |||
T11137 |
(E)-GABAB receptor antagonist 1
|
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
(E)-GABAB receptor antagonist 1 是 GABAB receptor antagonist 1 的反式结构。(E)-GABAB receptor antagonist 1 降低 GABA 诱导的 IP3 (三磷酸肌醇) 产生,IC50 为 37.9 μM。GABAB receptor antagonist 1是选择性的 GABAB (γ-氨基丁酸) 受体的负变构调节剂。 | |||
T14338 |
Atabecestat
JNJ-54861911 |
BACE | Neuroscience |
Atabecestat (JNJ-54861911) is a potent brain-penetrant and orally active β-site amyloid precursor protein cleaving enzyme 1 (BACE1) inhibitor, achieves robust and high CSF Aβ reduction and it is tolerated and displays a sustained pharmacokinetic (PK) and | |||
TP1422 |
Interleukin (IL)-6 Receptor
|
Others | Others |
Interleukin (IL)-6 Receptor 是一种肽,来源于白细胞介素6受体。 | |||
T12404 |
CCK-A receptor inhibitor 1
|
cholecystokinin | GPCR/G Protein |
CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50:340 nM)。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。 | |||
T11211 |
EP4 receptor antagonist 1
|
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
EP4 receptor antagonist 1 是一种有效的特异性前列腺素 EP4受体拮抗剂,对人和小鼠 EP4受体的 IC50分别为6.1 nM 和16.2 nM。 EP4 receptor antagonist 1 可用于癌症免疫治疗的研究。 | |||
T15249 |
Estrogen receptor modulator 1
|
Estrogen Receptor/ERR | Endocrinology/Hormones |
Estrogen receptor modulator 1 是一种有效的、具有口服活性的、选择性雌激素受体(estrogen receptor)调节剂 (SERM),其 pIC50为 0.46。它能够诱导 Tamoxifen 耐药、激素非依赖性异种移植瘤的消退。 | |||
T7011 |
Verubecestat
MK-8931,维罗司他 |
Beta-Secretase; BACE | Neuroscience |
Verubecestat (MK-8931) 是一种高亲和力的、具有口服活性的BACE1和BACE2抑制剂,Ki 分别为 2.2 nM 和 0.38 nM。它可以有效降低 Aβ40,并具有潜力用于阿尔茨海默氏病。 | |||
T19589 |
trans-2-Undecenoic acid
(E)-2-Undecenoic acid,反-2-十一烯酸,(E)-Undec-2-enoic acid |
Others | Others |
trans-2-Undecenoic acid ((E)-Undec-2-enoic acid) 是一种 α,β-不饱和羧酸,其特征在于酸二聚体,相应的二聚体通过羧基 C=O···H-O 的分子间氢键连接。 | |||
T3177 |
Orexin 2 Receptor Agonist
OX2R |
OX Receptor | GPCR/G Protein; Neuroscience |
Orexin 2 Receptor Agonist (OX2R) 是一种选择性有效的OX2R 激动剂, EC50为23 nM。 | |||
T11349 |
GABAA receptor agent 1
|
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
GABAA receptor agent 1 是GABAA 受体的高亲和力配体,有抗惊厥活性。 | |||
T12910 |
Sigma-1 receptor antagonist 1
|
Sigma receptor | GPCR/G Protein |
Sigma-1 receptor antagonist 1 是一种有效、特异性的 sigma-1 受体拮抗剂。 Sigma-1 receptor antagonist 1 具有抗神经性疼痛活性,可用于治疗神经性疼痛研究。 | |||
T7740 |
Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA(245443-52-1(free base)) |
Protease-activated Receptor | GPCR/G Protein |
Protease-Activated Receptor-4 diTFA 是蛋白酶激活受体 4 (PAR4) 激动剂。 | |||
T7674 |
Thrombin Receptor Activator for Peptide
|
Protease-activated Receptor | GPCR/G Protein |
Thrombin Receptor Activator for Peptide 也称为凝血因子 II 受体 (1-5) 或蛋白酶激活受体 1 (1-5),用于研究冠心病 (CHD)。 | |||
T11077 |
Dopamine D2 receptor antagonist-1
|
Others | Others |
Dopamine D2 receptor antagonist-1,一种对多巴胺D2受体(D2R)表现出亚毫摩尔级别亲和力的负变构调节剂(NAM)。 | |||
T37792 |
A2A receptor antagonist 1
CPI-444 analog,A2A receptor antagonist 1 |
Adenosine Receptor | GPCR/G Protein; Neuroscience |
A2A receptor antagonist 1 (CPI-444 analog)是腺苷 A2A 和 A1受体的拮抗剂,Ki 值分别为4和264 nM。 | |||
T5829 |
H4 Receptor antagonist 1
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
H4 Receptor antagonist 1 是选择性组胺 H4受体反向激动剂,其IC50值为19 nM。 | |||
T10499 |
H3 receptor-MO-1
|
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
H3 receptor-MO-1 是一种有效的组胺 H3 受体 (histamine H3 receptor) 调节剂,可用于研究神经分裂和认知障碍。 | |||
T13253 |
Umibecestat
CNP520 |
BACE | Neuroscience |
Umibecestat 是一种β-位点淀粉样前体蛋白裂解酶-1 (BACE-1) 抑制剂,对人 BACE-1 和小鼠 BACE-1 的 IC50 分别为 11 nM 和 10 nM,可用于阿尔茨海默病的研究。 | |||
T37908 |
Glucocorticoid receptor agonist-1
|
Glucocorticoid Receptor | Endocrinology/Hormones |
Glucocorticoid receptor agonist-1是一种强效糖皮质激素受体激动剂,其 IC50 值为 2.8 nM。 | |||
T2636 |
Decernotinib
VX-509,VRT-831509 |
Tyrosine Kinases; JAK | Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors |
Decernotinib (VRT-831509) 是一种可口服的JAK3抑制剂,对JAK3、JAK1、JAK2 和 TYK2 的Ki 值分别为 2.5、11、13 和 11 nM。 | |||
T4031 |
S1p receptor agonist 1
S1p-receptor-agonist-1 |
S1P Receptor; LPL Receptor | GPCR/G Protein |
S1p receptor agonist 1 (S1p-receptor-agonist-1) 是有口服活性的S1P 受体激动剂,具有诱导 S1P1 内化的活性,EC50为9.83 nM。它有潜力用于关节炎和实验性自身免疫性脑炎)的相关研究。 | |||
T12911 |
Sigma-1 receptor antagonist 2
|
Sigma receptor | GPCR/G Protein |
Sigma-1 receptor antagonist 2 是有效的sigma 1受体选择性拮抗剂,与 σ1 和 σ2 受体结合的Ki 分别为 3.88 和 1288 nM。 | |||
T22009 |
CB2 receptor agonist 2
ZINC72105556,4-Quinolone-3-Carboxamide Furan CB2 Agonist,CB2受体拮抗剂2 |
Cannabinoid Receptor | GPCR/G Protein |
CB2 receptor agonist 2 (ZINC72105556) 是有效和选择性的 CB2 受体激动剂。对 CB2 的 Ki 为 8.5 nM。CB2 receptor agonist 2 对 CB2 具有高亲和力和选择性。 | |||
T14127 |
Adenosine A1 receptor activator T62
|
Adenosine Receptor | GPCR/G Protein; Neuroscience |
Adenosine A1 receptor activator T62 是腺苷 A1 受体的变构增强剂,有镇痛作用。 | |||
T60087 |
cFMS Receptor Inhibitor IV
5-cyano-N-(2,5-di(piperidin-1-yl)phenyl)furan-2-carboxamide |
c-Fms | Tyrosine Kinase/Adaptors |
cFMS Receptor Inhibitor IV 是 c-Fms 酪氨酸激酶的抑制剂。 | |||
T67915 |
Succinate/succinate receptor antagonist 1
|
Others | Others |
Succinate/succinate receptor antagonist 1 是一种有效的琥珀酸受体拮抗剂。Succinate/succinate receptor antagonist 1 中断牙龈组织中的琥珀酸信号,抑制琥珀酸受体 1 (SucnRl Antagonist 1) 的激活,对琥珀酸受体 1的 IC50 值为 20 μΜ。Succinate/succinate receptor antagonist 1 可用于治疗牙周病。 | |||
T22216 |
10-Undecen-1-ol
|
Others | Others |
10-Undecen-1-ol 是由蓖麻油酸转化得到,是一种能够引入官能团的共聚单体。 | |||
T31095 |
Crinecerfont
SSR125543,SSR 125543,SSR-125543,SSR125543A,SSR 125543A,SSR-125543A |
CRFR | GPCR/G Protein |
Crinecerfont (SSR-125543) 是促肾上腺皮质激素释放因子 1 受体 (CRF1) 的特异性拮抗剂,可用于经典先天性肾上腺增生的研究。 | |||
T10250 |
ADRA1D receptor antagonist 1 HCl
ADRA1D receptor antagonist 1 HCl(1191908-24-3 free base) |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
ADRA1D receptor antagonist 1 HCl 是一种具有口服活性、高效性和选择性的 α1D 肾上腺素受体拮抗剂(Ki:1.6 nM),具有潜在的抗增殖活性。 | |||
T9157 |
GP130 receptor agonist-1
N-(4-Fluorophenyl)-4-phenyl-2-thiazolami |
Interleukin | Immunology/Inflammation |
GP130 receptor agonist-1 (N-(4-Fluorophenyl)-4-phenyl-2-thiazolami) 是一种有效的、口服有活性的、可透过血脑屏障的 GP130受体激动剂。它对 NMDA 诱导的神经毒性具有神经保护作用。 | |||
T7513 |
Protease-Activated Receptor-2, amide
蛋白酶活化的受体-2,酰胺,SLIGKV-NH2,H-丝氨酰亮氨酰异亮氨酰甘氨酰赖氨酰缬氨酰NH2 |
Protease-activated Receptor | GPCR/G Protein |
Protease-Activated Receptor-2, amide (SLIGKV-NH2) 是 PAR2 的激动剂,IC50为 10.4 M。 | |||
T9244 |
σ1 Receptor antagonist-1
|
Sigma receptor | GPCR/G Protein |
σ1 Receptor antagonist-1 是高选择性的 sigma 1受体拮抗剂,pKi 为10.28。它抑制细胞生长,在 G0/G1 期阻滞细胞周期并诱导 MCF-7/ADR 细胞凋亡。 | |||
T7332 |
(E)-2-Decenoic acid
trans-2-Decenoic acid,反式-2-癸烯酸 |
Others | Others |
(E)-2-Decenoic acid (trans-2-Decenoic acid) 是一种存在于蜂王浆中的脂肪酸。 | |||
T61813 |
AMPA receptor antagonist-3
|
iGluR | Membrane transporter/Ion channel; Neuroscience |
AMPA receptor antagonist-3 是一种AMPA 受体拮抗剂。 | |||
T12912 |
Sigma-1 receptor antagonist 3
|
Sigma receptor; HER | Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Sigma-1 receptor antagonist 3 是 Sigma-1受体选择性拮抗剂,Ki 为 1.14 nM。它抑制 hERG,IC50为 1.54μM。它在神经性疼痛方面有研究的价值。 | |||
T77508 |
A2B receptor antagonist 2 hydrochloride
|
||
A2B receptor antagonist 2 hydrochloride 是腺苷受体 A2B 的拮抗剂(rA1 的 Ki = 2.30 μM,rA2A 的 Ki = 6.8 μM,hA2B 的 3.44 μM) | |||
TP1704 |
Galanin Receptor Ligand M35 TFA
|
Neuropeptide Y Receptor | GPCR/G Protein; Neuroscience |
Galanin Receptor Ligand M35 TFA(142846-71-7 free base) 是一种高亲和力配体和甘丙肽受体拮抗剂 (Kd=0.1 nM)。 | |||
T61068 |
AMPA receptor antagonist-2
|
iGluR | Membrane transporter/Ion channel; Neuroscience |
AMPA receptor antagonist-2是一种AMPA 受体拮抗剂。 | |||
T21620 |
Adenosine receptor antagonist 4
|
Adenosine Receptor | GPCR/G Protein; Neuroscience |
Adenosine receptor antagonist 4 是一种腺苷受体拮抗剂。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8240 |
Cis-5-Dodecenoic Acid
|
Others | Others |
Cis-5-Dodecenoic Acid 是一种单不饱和脂肪酸,具有 C12 链作为主链,C5 位具有顺式双键。 | |||
T0306 |
10-Undecenoic acid
Undecylenic acid,Undecenoic acid,10-十一烯酸 |
Endogenous Metabolite; Antibiotic; Antifungal | Metabolism; Microbiology/Virology |
10-Undecenoic acid (Undecylenic acid) 是一种天然或合成的抑菌脂肪酸,具有抗真菌活性。 | |||
T0744 |
10-Undecenoic acid zinc salt
Zinc diundec-10-enoate,Zinc 10-undecenoate,Zinc undecylenate,十一烯酸锌 |
Antibiotic; Antifungal | Microbiology/Virology |
10-Undecenoic acid zinc salt (Zinc undecylenate) 是一种天然的或合成的抗真菌脂肪酸, 在乳膏中可局部用于治疗湿疹、真菌感染、癣和其他皮肤病。 锌具有收敛作用。 | |||
T8271 |
10Z-Nonadecenoic acid
|
Endogenous Metabolite | Metabolism |
10Z-Nonadecenoic acid 是一种长链脂肪酸,具有抗肿瘤特性。 | |||
T8241 |
cis-10-Heptadecenoic acid
|
Others | Others |
cis-10-Heptadecenoic acid 是反刍动物脂肪的次要成分。 | |||
TQ0251 |
(Z)-2-decenoic acid
(Z)-dec-2-enoic acid,(Z)-2-癸烯酸,cis-2-Decenoic acid,cis-dec-2-enoic acid |
Others | Others |
(Z)-2-decenoic acid (cis-dec-2-enoic acid) 是一种由铜绿假单胞菌产生的不饱和脂肪酸。它能够诱导一系列革兰氏阴性细菌(包括铜绿假单胞菌)和革兰氏阳性细菌形成的生物膜发生分散反应。它能够抑制生物膜发育。 | |||
TN6057 |
1-Methyl-2-[(Z)-6-undecenyl]-4(1H)-quinolone
(Z)-1-Methyl-2-(undec-6-enyl)quinolin-4(1H)-one |
||
(Z)-1-Methyl-2-(undec-6-enyl)quinolin-4(1H)-one shows strong inhibitory activity on leukotriene biosynthesis in human polymorphonuclear granulocytes, and it is very effective against mycobacteria. | |||
TN6899 |
1-Octadecene
|
||
1-Octadecene is a natural product. | |||
T75560 | 4(1H)-Quinolinone, 1-methyl-2-(5Z)-5-undecen-1-yl- | ||
4(1H)-Quinolinone, 1-methyl-2-(5Z)-5-undecen-1-yl- (化合物2) 是一种从蛇床子提取的喹诺酮类生物碱。该化合物对耐甲氧西林金黄色葡萄球菌(MRSA)表现出活性,其最小抑制浓度(MIC)值对ATCC 33591和ATCC 25923株分别为32 μg/mL和16 μM/mL。 | |||
T75507 | 1-Methyl-2-(8E)-8-tridecenyl-4(1H)-quinolinone | ||
1-Methyl-2-(8E)-8-tridecenyl-4(1H)-quinolinone 对幽门螺杆菌菌株 51 表现出有效的抗菌活性,MIC50 值和 MIC90 值分别为 22 µM 和 50 µM。该化合物展现了在研究胃及十二指肠溃疡方面的潜力。 | |||
TN6440 |
Pieceid-2''-O-gallate
|
||
Pieceid-2''-O-gallate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6440,CAS号为 105304-51-6。 | |||
T80018 |
cis-2-Dodecenoic acid
|
||
cis-2-Dodecenoic acid,最初在Burkholderia cenocepacia中被发现,能够干扰细菌的群体感应系统,从而抑制细菌生物膜的形成和毒力因子的产生。 | |||
TN6927 |
trans-2-Dodecenal
|
||
trans-2-Dodecenal is a natural product. | |||
TN7037 |
(Z)-9-nonadecene
9-Nonadecene |
Others | Others |
(Z)-9-nonadecene (9-Nonadecene) 首次在 T. melanocephalum 中被发现。它是下颌腺中的主要成分,而虹膜在尾腺中产生。 | |||
T83228 |
9-O-Methylstecepharine
|
||
9-O-Methylstecepharine(化合物 7)为Stephania cepharantha中检出的生物碱。 | |||
T78467 |
trans-10-Heptadecenoic acid
|
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trans-10-Heptadecenoic acid 是一种能在特定酶作用下参与生物合成与代谢过程的反式脂肪酸。在 2,4-二烯酰基-CoA 还原酶与 Delta3,Delta2-烯酰基-CoA 异构酶催化下,trans-10-Heptadecenoic acid 可合成聚羟基链烷酸酯。当缺乏 2,4-二烯酰基-CoA 还原酶时,该化合物则经由多功能酶 (MFE) 中的烯酰辅酶 A 水合酶 II 进行降解。此外,trans-10-Heptadecenoic acid 能通过还原酶依赖性与直接 MFE 依赖性途径引起细胞内的碳外流。 | |||
TN6843 |
1-Hexadecene
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1-Hexadecene is a natural product. | |||
TN6906 |
1-Pentadecene [Standard Material for GC]
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1-Pentadecene [Standard Material for GC] is a natural product. | |||
T34931 |
Trichodecenin II
Trichodecenin-II,4-Decenoyl-gly-gly-leu-aib-gly-leu-lol |
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Trichodecenin II is a peptaibol isolated from Trichoderma viride. | |||
T6627 |
Phosphoramidon Disodium
Phosphoramidon Disodium Salt,磷酰胺二钠 |
RAAS; Neprilysin; Others | Endocrinology/Hormones; Metabolism; Others |
Phosphoramidon Disodium (Phosphoramidon Disodium Salt) Salt 是一种金属蛋白酶 (metalloprotease) 抑制剂 。Phosphoramidon Disodium Salt 抑制内皮素转化酶 (ECE) ,中性肽内切酶 (NEP) 和血管紧张素转换酶 (ACE) 的IC50分别为 3.5 ,0.034 和 78 μM。 |
Cat. No. | Product Name | Species | Expression System |
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TMPY-01929 |
ECE1 Protein, Human, Recombinant (His)
RP3-329E20.1,endothelin converting enzyme 1,ECE |
Human | HEK293 Cells |
Endothelin-converting enzyme 1, also known as ECE-1, is a single-pass type II membrane protein which belongs to thepeptidase M13 family. ECE-1 converts big endothelin-1 to endothelin-1. ECE-1 is a membrane metalloprotease that generates endothelin from its direct precursor big endothelin. Four isoforms of ECE-1 are produced from a single gene through the use of alternate promoters. These isoforms share the same extracellular catalytic domain and contain unique cytosolic tails, which resul... | |||
TMPY-01891 |
ECE2 Protein, Human, Recombinant (His)
endothelin converting enzyme 2,UNQ403/PRO740,KIAA0604 |
Human | HEK293 Cells |
ECE2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 80.2 kDa and the accession number is P0DPD8. | |||
TMPY-00782 |
ECE2 Protein, Human, Recombinant (hFc)
endothelin converting enzyme 2,KIAA0604,UNQ403/PRO740 |
Human | HEK293 Cells |
ECE2 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 105 kDa and the accession number is P0DPD8. | |||
TMPY-01725 |
Leptin Receptor Protein, Human, Recombinant (His)
LEPRD,OB-R,OBR,LEP-R,CD295,leptin receptor |
Human | HEK293 Cells |
Leptin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 95 kDa and the accession number is P48357-1. | |||
TMPY-03739 |
Transferrin Receptor/TFRC Protein, Cynomolgus, Rhesus, Recombinant (His)
transferrin receptor |
Cynomolgus,Rhesus | HEK293 Cells |
Transferrin Receptor/TFRC Protein, Cynomolgus, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.5 kDa and the accession number is XP_005545315.1&NP_001244232.1. | |||
TMPY-02294 |
Transferrin Receptor/TFRC Protein, Mouse, Recombinant (His)
2610028K12Rik,p90,E430033M20Rik,AI426448,TFR,AU015758,Mtvr1,... |
Mouse | HEK293 Cells |
Transferrin Receptor/TFRC Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 78.3 kDa and the accession number is Q62351. | |||
TMPY-01873 |
Transferrin Receptor/TFRC Protein, Human, Recombinant (His)
TFR1,p90,CD71,TFR,transferrin receptor,T9,TRFR,TR |
Human | HEK293 Cells |
Transferrin Receptor/TFRC Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.4 kDa and the accession number is AAA61153.1. | |||
TMPY-05096 |
Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc)
CD71,T9,transferrin receptor,TFR1,p90,TRFR,TFR,TR |
Human | HEK293 Cells |
Transferrin Receptor/TFRC Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 103.6 kDa and the accession number is CAA25527.1. | |||
TMPY-01053 |
Prolactin Receptor Protein, Human, Recombinant (His)
hPRLrI,PRLR,MFAB,HPRL,prolactin receptor |
Human | HEK293 Cells |
Prolactin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26 kDa and the accession number is P16471-1. | |||
TMPY-01146 |
Insulin Receptor Protein, Human, Recombinant (long isoform, His)
HHF5,CD220,insulin receptor |
Human | HEK293 Cells |
Insulin Receptor Protein, Human, Recombinant (long isoform, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 107 kDa and the accession number is P06213-1. | |||
TMPH-03388 |
Transferrin Receptor/TFRC Protein, Rat, Recombinant (His & SUMO)
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Rat | E. coli |
Transferrin Receptor/TFRC Protein, Rat, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 35.9 kDa and the accession number is Q99376. | |||
TMPY-03860 |
Endothelin B Receptor Protein, Human, Recombinant (mFc)
ET-B,endothelin receptor type B,ETB,ETBR,ETRB,ET-BR... |
Human | HEK293 Cells |
Endothelin B Receptor Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 34.4 kDa and the accession number is P24530-1. | |||
TMPY-01566 |
Prolactin Receptor Protein, Mouse, Recombinant (His & hFc)
prolactin receptor,Prlr,Pr-3,Pr-1,Prlr-rs1,AI987712 |
Mouse | HEK293 Cells |
Prolactin Receptor Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 52.5 kDa and the accession number is Q08501-1. | |||
TMPY-02706 |
Vitamin D Receptor/VDR Protein, Human, Recombinant (His)
PPP1R163,vitamin D (1,25- dihydroxyvitamin D3) rece... |
Human | Baculovirus Insect Cells |
Vitamin D Receptor/VDR Protein, Human, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 50 kDa and the accession number is P11473. | |||
TMPY-01221 |
Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His & hFc)
NgR1,reticulon 4 receptor,NgR,Rtn4r,NOGOR |
Mouse | HEK293 Cells |
Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 73.8 kDa and the accession number is Q99PI8. | |||
TMPY-05025 |
Thrombin Receptor Protein, Human, Recombinant (His)
TR,PAR1,HTR,coagulation factor II (thrombin) recept... |
Human | HEK293 Cells |
Thrombin Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 10.2 kDa and the accession number is A0A024RAP7. | |||
TMPY-02984 |
Prolactin Receptor Protein, Mouse, Recombinant (His)
Pr-1,Pr-3,AI987712,prolactin receptor,Prlr,Prlr-rs1 |
Mouse | HEK293 Cells |
Prolactin Receptor Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26 kDa and the accession number is P07321. | |||
TMPY-03144 |
Nogo Receptor/RTN4R Protein, Human, Recombinant (His)
NGR,reticulon 4 receptor,NOGOR |
Human | HEK293 Cells |
Nogo Receptor/RTN4R Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 46.8 kDa and the accession number is Q9BZR6. | |||
TMPK-01200 |
Nogo Receptor/RTN4R Protein, Cynomolgus, Recombinant (His)
NGR,NOGOR,RTN4R,NgR1,Nogo receptor,Nogo-66 rece... |
Cynomolgus | HEK293 Cells |
NOGO Receptor 1 (RTN4R) regulates axonal growth, as well as axon regeneration after injury. The gene maps to the 22q11.2 schizophrenia susceptibility locus and is thus a strong functional and positional candidate gene.RTN4R may modulate the genetic risk or clinical expression of schizophrenia in a subset of patients and identify additional studies that will be necessary to clarify the role of RTN4R in psychiatric phenotypes. | |||
TMPY-00177 |
Ebola virus EBOV (subtype Bundibugyo, strain Uganda 2007) Glycoprotein/GP-RBD (Receptor Binding Domain) Protein (hFc)
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EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Bundibugyo, strain Uganda 2007) Glycoprotein/GP-RBD (Receptor Binding Domain) Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 57.6 kDa and the accession number is B8XCN0. | |||
TMPY-00178 |
Ebola virus EBOV (subtype Zaire, strain Mayinga 1976) Glycoprotein/GP-RBD (Receptor Binding Domain) Protein (hFc)
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EBOV | HEK293 Cells |
Ebola virus EBOV (subtype Zaire, strain Mayinga 1976) Glycoprotein/GP-RBD (Receptor Binding Domain) Protein (hFc) is expressed in HEK293 mammalian cells with Fc tag. The predicted molecular weight is 57.6 kDa and the accession number is Q05320. | |||
TMPY-02987 |
Vitamin D Receptor/VDR Protein, Mouse, Recombinant (His)
vitamin D (1,25- dihydroxyvitamin D3) receptor,Nr1i... |
Mouse | Baculovirus Insect Cells |
Vitamin D Receptor/VDR Protein, Mouse, Recombinant (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 49.28 kDa and the accession number is P48281. | |||
TMPY-01149 |
Insulin Receptor Protein, Human, Recombinant (short isoform, His)
Insulin Receptor,HHF5,CD220 |
Human | HEK293 Cells |
Insulin Receptor Protein, Human, Recombinant (short isoform, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 106 kDa and the accession number is P06213-2. | |||
TMPY-04395 |
Insulin Receptor Protein, Human, Recombinant (His & GST)
HHF5,insulin receptor,CD220 |
Human | Baculovirus Insect Cells |
Insulin Receptor Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 72.3 kDa and the accession number is P06213-1. | |||
TMPH-00932 |
Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO)
Nuclear receptor subfamily 3 group C member 4,AR,NR... |
Human | E. coli |
Androgen receptor Protein, Human, Recombinant (His & Myc & SUMO) is expressed in E. coli. | |||
TMPH-02390 |
Odorant receptor Protein, Larimichthys crocea, Recombinant (His)
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Larimichthys crocea | E. coli |
Odorant receptor Protein, Larimichthys crocea, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 37.0 kDa and the accession number is F2XEX3. | |||
TMPJ-00378 |
Transferrin Receptor/TFRC Protein, Human, Recombinant (aa 101-760, His)
p90,TfR,T9,Trfr,Transferrin receptor protein 1,TR |
Human | HEK293 Cells |
Transferrin receptor protein 1 (TFRC) belongs to the peptidase M28 family that is synthesized as a 172 amino acid (aa). TFRC regulated by cellular iron levels through binding of the iron regulatory proteins, IRP1 and IRP2, to iron-responsive elements in the 3'-UTR. It binds one transferrin or HFE molecule per subunit and binds the HLA class II histocompatibility antigen, DR1. It Interacts with SH3BP3 and STEAP3, facilitates TFRC endocytosis in erythroid precursor cells. Cellular uptake of iron o... | |||
TMPY-00874 |
Leptin Receptor Protein, Human, Recombinant (His & hFc)
LEP-R,OBR,CD295,OB-R,LEPRD,leptin receptor |
Human | HEK293 Cells |
Leptin Receptor Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 121.4 kDa and the accession number is P48357-1. | |||
TMPY-01056 |
Nogo Receptor/RTN4R Protein, Human, Recombinant (His & hFc)
NOGOR,reticulon 4 receptor,NGR |
Human | HEK293 Cells |
Nogo Receptor/RTN4R Protein, Human, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 73 kDa and the accession number is Q9BZR6. | |||
TMPY-01163 |
Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His)
Rtn4r,NgR,NgR1,reticulon 4 receptor,NOGOR |
Mouse | HEK293 Cells |
Nogo Receptor/RTN4R Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 47 kDa and the accession number is Q99PI8. | |||
TMPY-00317 |
Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc)
CTR,calcitonin receptor,CRT,CTR1,CT-R |
Human | HEK293 Cells |
Calcitonin receptor Protein, Human, Recombinant (aa 25-154, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 43.9 kDa and the accession number is P30988-1. | |||
TMPH-02023 |
Renin receptor Protein, Human, Recombinant (His)
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Human | E. coli |
Renin receptor Protein, Human, Recombinant (His) is expressed in E. coli. | |||
TMPY-04787 |
West Nile Virus (WNV) (lineage 2, strain Nea Santa-Greece-2010) E/Envelope Protein (His)
WNV-E Protein |
WNV | P. pastoris (Yeast) |
West Nile Virus (WNV) (lineage 2, strain Nea Santa-Greece-2010) E/Envelope Protein (His) is expressed in yeast with His tag. The predicted molecular weight is 12.9 kDa and the accession number is AED99787.1. | |||
TMPY-05617 |
Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated
TRFR,p90,TR,TFR,CD71,TFR1,T9,transferrin receptor |
Human | HEK293 Cells |
Transferrin Receptor/TFRC Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 77.4 kDa and the accession number is P02786. | |||
TMPH-02641 |
ECEL1 Protein, Mouse, Recombinant (His & Myc)
Ecel1,Endothelin-converting enzyme-like 1,Dine,Xce,... |
Mouse | E. coli |
May contribute to the degradation of peptide hormones and be involved in the inactivation of neuronal peptides. | |||
TMPY-00181 |
Endothelin B Receptor Protein, Human, Recombinant (His)
ETBR,ET-B,ET-BR,ETB,HSCR2,endothelin receptor type ... |
Human | HEK293 Cells |
Endothelin B Receptor Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 9.5 kDa and the accession number is P24530-1. | |||
TMPY-00085 |
Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc)
CTR,CTR1,CT-R,calcitonin receptor,CRT |
Human | HEK293 Cells |
Calcitonin receptor Protein, Human, Recombinant (aa 1-153, hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 42.1 kDa and the accession number is P30988-2. | |||
TMPY-02434 |
Prolactin Receptor Protein, Rat, Recombinant (His)
prolactin receptor,RATPRLR,MGC105486 |
Rat | HEK293 Cells |
Prolactin Receptor Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 26 kDa and the accession number is P05710-1. | |||
TMPY-05283 |
Insulin Receptor Protein, Human, Recombinant (long isoform, His), Biotinylated
CD220,Insulin Receptor,HHF5 |
Human | HEK293 Cells |
Insulin Receptor Protein, Human, Recombinant (long isoform, His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 107 kDa and the accession number is P06213-1. | |||
TMPY-06661 |
Transferrin Receptor/TFRC Protein, Rat, Recombinant (His)
transferrin receptor |
Rat | HEK293 Cells |
Transferrin Receptor/TFRC Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 78.59 kDa and the accession number is Q99376. | |||
TMPY-02648 |
PACAP receptor/ADCYAP1R1 Protein, Human, Recombinant (hFc)
adenylate cyclase activating polypeptide 1 (pituitary) r... |
Human | HEK293 Cells |
Pituitary adenylate cyclase activating polypeptide (PACAP, Adcyap1) activation of PAC1 receptors ( Adcyap1r1) significantly increases excitability of guinea pig cardiac neurons. This modulation of excitability is mediated in part by plasma membrane G protein-dependent activation of adenylyl cyclase and downstream signaling cascades. Studies point to the potential role of the (pituitary) adenylate cyclase activating polypeptide receptor 1 (ADCYAP1R1) gene, which has been implicated in stress resp... |