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Androgen Receptor antagonist kit

Catalog No. CL0126

Androgen Receptor antagonist kit 包含雄激素受体拮抗剂,雄激素受体属于核受体超家族中的类固醇受体,与雄激素结合后,激活第二信使信号通路,调控靶基因的转录和翻译,从而影响生殖、骨骼肌、心血管、神经、免疫、造血系统的发育和稳态维持等方面。TargetMol 为您提供43种精选雄激素受体拮抗剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

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Androgen Receptor antagonist kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,500 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
T0272Nilutamide63612-50-0317.2210mMAndrogen Receptor
T0380Bicalutamide90357-06-5430.3710mMAndrogen Receptor; Autophagy
T0489Flutamide13311-84-7276.2110mMAndrogen Receptor
T1167Cyproterone acetate427-51-0416.9410mMAndrogen Receptor
T1541Drospirenone67392-87-4366.4910mMAndrogen Receptor; COX; Estrogen/progestogen Receptor; Glucocorticoid Receptor; progesterone receptor
T1596Chlormadinone acetate302-22-7404.9310mMAndrogen Receptor; progesterone receptor
T2236RU 58841154992-24-2369.3410mMAndrogen Receptor
T2339Apalutamide956104-40-8477.4310mMAndrogen Receptor; GABA Receptor
T2895Lupeol545-47-1426.7310mMAkt; Androgen Receptor; Apoptosis
T29913,3'-Diindolylmethane1968-05-4246.3110mMAndrogen Receptor; Autophagy
T3357Clascoterone19608-29-8402.5210mMAndrogen Receptor
T3393Triptophenolide74285-86-2312.410mMAndrogen Receptor
T6002Enzalutamide915087-33-1464.4410mMAndrogen Receptor; Autophagy
T6400AZD35141240299-33-5519.5610mMAndrogen Receptor
T6509Galeterone851983-85-2388.5510mMAndrogen Receptor; P450
T6829EPI-001227947-06-0394.8910mMAndrogen Receptor; Apoptosis; PPAR
T6889MI-1361628316-74-4470.5110mMAndrogen Receptor; Apoptosis; Epigenetic Reader Domain
T6915Darolutamide1297538-32-9398.8510mMAndrogen Receptor
T7440p,p'-DDE72-55-931810mMAndrogen Receptor; Drug Metabolite
T76902-hydroxy Flutamide52806-53-8292.2110mMAndrogen Receptor
T8592CTK8A3536926228-58-2276.3510mMAndrogen Receptor
T13273UT-342168525-92-4356.2710mMAndrogen Receptor
TQ0209Ailanthone981-15-7376.410mMAndrogen Receptor
TQ0214Dimethylcurcumin52328-98-0396.4310mMAndrogen Receptor
T19450N-desmethyl Enzalutamide1242137-16-1450.4110mMAndrogen Receptor
TCS1372Atraric acid4707-47-5196.210mMAndrogen Receptor; phosphatase
T8933JNJ-63576253 free base2110426-27-0502.5110mMAndrogen Receptor
T22263Bavdegalutamide2222112-77-6812.2910mMAndrogen Receptor
T12323ORM-153411297537-33-7396.8310mMAndrogen Receptor
T140082,2,5,7,8-Pentamethyl-6-Chromanol950-99-2220.3110mMAndrogen Receptor
T13272UT-1552031161-35-8405.3510mMAndrogen Receptor
T15445Proxalutamide1398046-21-3517.510mMAndrogen Receptor; SARS-CoV
T9246JNJ-635762532110428-64-1538.9710mMAndrogen Receptor
T10359AR antagonist 11818885-54-9278.7810mMAndrogen Receptor; Ligand for E3 Ligase; Ligands for Target Protein for PROTAC
T12146N-Desmethyl-Apalutamide1332391-11-3463.4110mMAndrogen Receptor; P450
T9179CLP-3094312749-73-8304.810mMAndrogen Receptor
T14116ACP-105899821-23-9290.7910mMAndrogen Receptor
T12928SK331928724-23-5500.3110mMAndrogen Receptor
T29111VPC-13566218464-59-6258.3210mMAndrogen Receptor
T20625Prochloraz67747-09-5376.6710mMAhR; Androgen Receptor; Antifungal; Estrogen Receptor/ERR
T24943VPC-1422819983-28-9246.3310mMAndrogen Receptor
T39695ARD-21282222111-87-5820.3810mMAndrogen Receptor
T21740RD162915087-27-3476.4510mMAndrogen Receptor

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产品应用

  • 信号通路研究
  • 预实验探索

包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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