LPL Receptor antagonist/agonist kit 包含脂蛋白脂肪酶LPL 拮抗剂/激动剂,LPL 是脂肪细胞、心肌细胞、骨骼肌细胞、乳腺细胞以及巨噬细胞等实质细胞合成和分泌的一种糖蛋白,催化脂蛋白中TG 水解,以供组织氧化供能和贮存,参与VLDL 和HDL 之间的载脂蛋白和磷脂的转换。另外,LPL 还具有增加CM 残粒结合到LPL 受体上的能力,促进CM 残粒摄取。TargetMol 为您提供22种精选LPL 拮抗剂/激动剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T2171 | SEW​2871 | 256414-75-2 | 440.36 | 10mM | LPL Receptor; S1P Receptor |
T2539 | Fingolimod hydrochloride | 162359-56-0 | 343.93 | 10mM | LPL Receptor; PAK; S1P Receptor; TRP/TRPV Channel |
T3258 | Ponesimod | 854107-55-4 | 460.97 | 10mM | LPL Receptor; S1P Receptor |
T3961 | CYM-5541 | 945128-26-7 | 316.44 | 10mM | LPL Receptor; S1P Receptor |
T4031 | S1p receptor agonist 1 | 1514888-56-2 | 409.45 | 10mM | LPL Receptor; S1P Receptor |
T6403 | Siponimod | 1230487-00-9 | 516.6 | 10mM | LPL Receptor; S1P Receptor |
T6923 | Ozanimod | 1306760-87-1 | 404.46 | 10mM | LPL Receptor; S1P Receptor |
T7360 | GSK2018682 | 1034688-30-6 | 440.88 | 10mM | LPL Receptor; S1P Receptor |
T7832 | Ibrolipim | 133208-93-2 | 451.25 | 10mM | LPL Receptor |
T7939 | Fingolimod | 162359-55-9 | 307.47 | 10mM | LPL Receptor; PAK; S1P Receptor |
T10305 | Amiselimod hydrochloride | 942398-84-7 | 413.9 | 10mM | LPL Receptor; S1P Receptor |
T17183 | TY-52156 | 934369-14-9 | 364.27 | 10mM | LPL Receptor; S1P Receptor |
T15629 | JTE-013 | 383150-41-2 | 408.29 | 10mM | Apoptosis; LPL Receptor; S1P Receptor |
T8840 | PF-543 hydrochloride | 1706522-79-3 | 502.1 | 10mM | Apoptosis; Autophagy; LPL Receptor; S1P Receptor |
T15032 | CYM50308 | 1345858-76-5 | 405.46 | 10mM | LPL Receptor; S1P Receptor |
T22703 | CYM-5520 | 1449747-00-5 | 345.4 | 10mM | LPL Receptor; S1P Receptor |
TQ0227 | Etrasimod | 1206123-37-6 | 457.48 | 10mM | LPL Receptor; S1P Receptor |
T9199 | GLPG2938 | 2130996-00-6 | 503.4 | 10mM | LPL Receptor; S1P Receptor |
T9464 | CYM50358 | 1314212-39-9 | 389.27 | 10mM | LPL Receptor |
T28169 | NIBR-0213 | 1233332-14-3 | 464.98 | 10mM | LPL Receptor |
T12086 | Mocravimod hydrochloride | 509088-69-1 | 480.45 | 10mM | LPL Receptor |
T12821 | S1PR1 modulator 1 | 2328109-05-1 | 408.51 | 10mM | LPL Receptor |