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Cat. No. Product Name Target Signaling Pathways
TP2030 Gastrin I, human

Gastrin I (human)

cholecystokinin GPCR/G Protein
Gastrin I, human (Gastrin I (human)) 是胃中产生的内源性肽,通过 CCK2 受体增加大鼠的胃蛋白酶原和酸分泌。
TP1240 Adrenocorticotropic Hormone (ACTH) (18-39), human TFA

CLIP (human) (TFA)

Others Others
Adrenocorticotropic Hormone (ACTH) (18-39), human TFA (CLIP human TFA) 是一种似皮质促素中叶肽,由垂体中叶的促黑素细胞产生。
TP1143L Fibrinopeptide A, human acetate

Fibrinopeptide A, human acetate(25422-31-5 free base),Human fibrinopeptide A acetate

Others Others
Fibrinopeptide A, human acetate (Human fibrinopeptide A acetate)(25422-31-5 free base) 是一种 16 个残基的短多肽,由凝血酶从纤维蛋白原上切割下来。纤维蛋白肽 A (FPA) 由纤维蛋白原蛋白的 N 末端 Aα 区域在被凝血酶切割后产生。
TP1174 Endothelin-2 (49-69), human

Human endothelin-2,Endothelin-2, human,Endothelin-2 (human, canine),人内皮素2

Others Others
Endothelin-2 (49-69), human (Human endothelin-2) 是一种由 21 个氨基酸组成的血管活性肽。它可与 G 蛋白连接的跨膜受体,ET-RA 和ET-RB 结合。
T7489 MART-1 (26-35) (human)

MART-1 (26-35) human

Others Others
MART-1 (26-35) (human) (MART-1 (26-35) human) 是一种 MART-1 蛋白 26 到 35 氨基酸片段。
TP1187 C-Type Natriuretic Peptide (CNP) (1-22), human

CNP (1-22), human

RAAS Endocrinology/Hormones
C-Type Natriuretic Peptide (CNP) (1-22), human 是一种利钠肽受体 B (NPR-B) 激动剂,是一种 CNP 的 1-22 片段。它对生理激动剂组胺和 5-HT 刺激或直接由 Forskolin 刺激的 cAMP 合成具有抑制作用。其中CNP 是一种有效的、内皮衍生的松弛剂和生长抑制因子。
TP2018L GIP (human) acetate

GIP (human) acetate(100040-31-1 Free base)

IGF-1R Tyrosine Kinase/Adaptors
GIP (human) acetate 是葡萄糖依赖性胰岛素分泌的刺激剂和胃酸分泌的弱抑制剂。 GIP (human) acetate 在脂质代谢和肥胖的发展中起着至关重要的作用。
T8221 Insulin (human)

INSULIN,甘精胰岛素,胰岛素,Insulin(human)

IGF-1R Tyrosine Kinase/Adaptors
Insulin (human) 是一种多肽激素,可以促进糖原的合成,调节血液中的葡萄糖水平。Insulin (human) 具有降血糖活性,临床上用于治疗糖尿病患者的高血糖。
TP1082L Neuropeptide AF (human) acetate

Neuropeptide AF (93-110), human Acetate,Neuropeptide AF (human) acetate (192387-38-5 Free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) 属于抗阿片类神经肽,是 Neuropeptide AF (human) 衍生物,可调节脂肪细胞代谢。
TP1923L1 ELA-14(human) acetate

ELA-14(human) acetate (1886973-05-2 free base)

Apelin receptor; Arrestin GPCR/G Protein
ELA-14(human) acetate 是 ELA 的一个片段,它与 APJ 结合,激活 Gαi1 和 β-arrestin-2 信号通路,并类似于其亲本内源性肽诱导受体内化。
T7577 Angiotensin III, human, mouse

血管紧张素III,Angiotensin III, human, mouse(3TFA)

RAAS Endocrinology/Hormones
Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA)) 是一种七肽,是血管紧张素 2 型受体 (AT2R) 激动剂,能够作用于 AT2R (IC50:0.648 nM)及 AT1R (IC50:21.1nM)。
T19584L TNF-α (31-45), human acetate

TNF-α (31-45), human acetate(144796-71-4 free base)

Others Others
TNF-α (31-45), human acetate(144796-71-4 free base) 是一种肿瘤坏死因子-α 的肽。
TP1900L1 Hemopressin (human, mouse) acetate

Hemopressin (human, mouse) acetate(1314035-51-2 free base)

Cannabinoid Receptor GPCR/G Protein
Hemopressin (human, mouse) acetate(1314035-51-2 free base) 是一种衍生自血红蛋白 α1 链的九肽,是从大鼠脑匀浆中分离出来的。 Hemopressin 是 CB1 大麻素受体的口服活性、选择性和反向激动剂。 Hemopressin 在炎性疼痛模型中发挥镇痛作用。
T8231 Adrenocorticotropic Hormone (ACTH) (1-39), human

ACTH (1-39), human,丝拉克肽

Others Others
Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) 是黑皮质素受体激动剂。
T40412L BAD (103-127) (human) acetate

BAD (103-127) (human) acetate (331762-68-6 Free base)

Others Others
BAD (103-127) (human) acetate 是一种来自于 BAD 的 BH3结构域的25-mer Bad 多肽,可拮抗 Bcl-xl 的作用。
TP1257L Adrenomedullin (AM) (22-52), human acetate

Adrenomedullin (AM) (22-52), human acetate(159899-65-7 Free base)

CGRP Receptor GPCR/G Protein; Neuroscience
Adrenomedullin (AM) (22-52), human acetate 是猫后肢血管床中 CGRP 受体和肾上腺髓质素受体的拮抗剂。
TP1295 Angiotensin I (human, mouse, rat)

Angiotensin 1 Human,血管紧张素 1 (人)

Others Others
Angiotensin I (human, mouse, rat) 是血管紧张素Ⅱ的前体物质,在血管紧张素转化酶 (ACE) 的参与下裂解成血管紧张素Ⅱ。
TP2092L Apelin-17 (human, bovine) acetate

Apelin-17 (human, bovine) acetate(217082-57-0 free base)

HIV Protease Microbiology/Virology; Proteases/Proteasome
Apelin-17 (human, bovine) acetate(217082-57-0 free base) 是一种内源性 apelin 受体激动剂。有效抑制毛喉素刺激的 cAMP 积累 (pIC50 = 9.94)。
TP1219 Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate

ANP (1-28), human, porcineANP(1-28)

Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate 是颗粒鸟苷酸环化酶的刺激剂,已被发现通过增加环鸟苷单磷酸的合成来保护分离的心肌细胞免受复氧诱导的高收缩。Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate 也有助于在反复运动期间刺激脂解,并在运动期间控制脂解。
TP1880L1 PAMP-12 (human, porcine) acetate

PAMP-12 (human, porcine) acetate(196305-05-2 free base)

Others Others
PAMP-12 (human, porcine) acetate (PAMP-12 (human, porcine) acetate (196305-05-2 free base)) 是 ir-PAMP 的主要成分,由 AM 前体加工而成,PAMP-20 也是如此,并且可能参与心血管控制。
TP1144L Corticotropin-releasing factor (human) acetate

Corticotropin-releasing factor (human) acetate (86784-80-7 Free base)

CRFR GPCR/G Protein
Corticotropin-releasing factor (human) acetate 刺激垂体前叶合成和分泌促肾上腺皮质激素。
T19309L1 Endothelin 1 (swine, human) acetate

Endothelin 1 (swine, human) acetate(117399-94-7 free base)

Endothelin Receptor GPCR/G Protein
Endothelin 1 (swine, human) acetate(117399-94-7 free base) 是一种合成肽,其序列为人和猪内皮素 1。它是一种有效的内源性血管收缩剂,通过两种类型的受体 ETA 和 ETB 起作用。
TP1627L Prepro VIP (111-122), human acetate

Prepro VIP (111-122), human acetate(123025-94-5 free base)

Others Others
Prepro VIP (111-122), human acetate(123025-94-5 free base) 是一种前血管活性肠多肽 (VIP) 衍生肽,对应于残基 111-122。
TP1737L Urotensin II (114-124), human acetate

Urotensin II (114-124), human acetate(251293-28-4 free base)

GPR Endocrinology/Hormones; GPCR/G Protein
Urotensin II (114-124), human acetate(251293-28-4 free base) 是一种 11 个氨基酸残基肽,是一种有效的血管收缩剂和孤儿受体 GPR14 的激动剂。
TP1244L1 Adrenocorticotropic Hormone (ACTH) (1-10), human acetate

Adrenocorticotropic Hormone (ACTH) (1-10), human acetate(2791-05-1 Free base)

Others Others
Adrenocorticotropic Hormone (ACTH) (1-10), human acetate 是促肾上腺皮质激素的一个片段。 Adrenocorticotropic Hormone (ACTH) (1-10), human acetate 仅在 100 和 1000 nM 时具有较弱的 α-MSH 效力。
T21608L β-Interleukin I (163-171), human Acetate

β-Interleukin I (163-171), human Acetate(106021-96-9 Free base)

Others Others
β-Interleukin I (163-171), human Acetate 是一种参与调节免疫反应、炎症反应和造血的肽。
TP1732L Galanin (1-30), human acetate

醋酸甘丙肽,Galanin (1-30), human acetate(119418-04-1 Free base)

Others Others
Galanin (1-30), human acetate (Galanin ) 是一种 30 个氨基酸的神经肽。 它是 GalR1 和 GalR2 受体的激动剂,Kis 均为 1 nM。
TP1618L PACAP-38 (31-38), human, mouse, rat acetate

PACAP-38 (31-38), human, mouse, rat acetate(138764-85-9 Free base)

PACAP GPCR/G Protein
PACAP-38 (31-38), human, mouse, rat acetate 是 PAC1 受体的激活剂。PACAP-38 (31-38), human, mouse, rat acetate 对交感神经元 NPY 和儿茶酚胺的产生具有强效、有效和持续的刺激作用,可用于神经营养和神经保护研究。
TP1007L β-Amyloid (1-42), acetate (human)

β-Amyloid (1-42), human acetate (107761-42-2 Free base)

β-Amyloid (1-42), acetate (human) 是由 42 个氨基酸组成的肽,是 β-Amyloid 的一部分,常用于阿尔茨海默病造模。
TP1628L Activated Protein C (390-404), human acetate

Activated Protein C (390-404), human acetate(146340-20-7 Free base)

APC Cell Cycle/Checkpoint
Activated Protein C (390-404), human acetate (Activated Protein C ) 抑制 APC 抗凝活性。
TP2499 Human IgE Pentapeptide HEPP acetate

Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base)

Human IgE Pentapeptide HEPP acetate 是一种五肽,在几种不同体系中均不能产生 IgE 抑制作用,可用于治疗结膜炎。
TP2056L Acetyl-Calpastatin (184-210)(human) acetate

Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )

Cysteine Protease Proteases/Proteasome
Acetyl-Calpastatin (184-210)(human) acetate 是一种有效,选择性和可逆的钙蛋白酶 (calpain) 抑制剂,对 μ-钙蛋白酶和组织蛋白酶 L 的 Ki 值分别为 0.2 nM 和 6 μM。
T38193L β-Endorphin (1-27) (human) acetate

β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
β-Endorphin (1-27) (human) acetate 存在于大脑垂体和下丘脑中,具有镇痛活性。 β-Endorphin (1-27) (human) acetate 是一种阿片受体激动剂,对 μ-阿片受体和 δ-阿片受体具有较好的亲和力。
TP1996 MCH(human, mouse, rat)

MCH (human, mouse, rat),黑色素聚集激酶素(MCH)( 大鼠)

GPR; Melanin-concentrating Hormone Receptor (MCHR) Endocrinology/Hormones; GPCR/G Protein
MCH(human, mouse, rat) 是MCH-R 肽激动剂,对 CHO 细胞系中 MCH-2R 高度敏感,激活 MCH-1R 和 MCH-2R 的IC50 值分别为 0.3 和 1.5 nM,EC50值对分别为 3.9 和 0.1 nM。
T39392L C-Type Natriuretic Peptide (CNP) (1-22), human acetate

C-Type Natriuretic Peptide (CNP) (1-22), human acetate(1966153-17-2 Free base)

Others Others
C-Type Natriuretic Peptide (CNP) (1-22), human acetate 是一种利钠肽受体 B (NPR-B) 的激动剂,一种内皮衍生的松弛剂和生长抑制因子。 C-Type Natriuretic Peptide (CNP) (1-22), human acetate 抑制由组胺和 5-HT 或直接由毛喉素刺激的 cAMP 合成。
T38470 Obestatin(human)

Obestatin (human) is a 23-amino acid amidated peptide that interacts with GPR39 to regulate appetite and gastrointestinal motility. Its properties also make it suitable for weight loss. Nonetheless, Obestatin (human) is unable to permeate the cell membrane.
T21649L GnRH Associated Peptide (GAP) (1-13), human Acetate

GnRH Associated Peptide (GAP) (1-13), human Acetate (100111-07-7 Free base)

Others Others
GnRH Associated Peptide (GAP) (1-13), human Acetate 被发现是催乳素分泌的有效抑制剂并刺激促性腺激素的释放。用对应于 GAP 序列的肽进行主动免疫导致催乳素分泌大大增加。
TP2044L α-CGRP (human) acetate

人类降钙素基因相关肽 1,α-CGRP (human) acetate (90954-53-3 free base)

Others Others
α-CGRP (human) acetate 是一种由 37 个氨基酸组成的调节性神经肽。它是一种有效的血管扩张剂,具有正性肌力作用和变时性作用。
TP1651L Proinsulin C-peptide human acetate

醋酸胰岛素原C-肽(55-89),人,Proinsulin C-peptide human acetate (33017-11-7 Free base)

Others Others
Proinsulin C-peptide human acetate (Proinsulin C-peptide human acetate (33017-11-7 Free base)) 是一种由31个氨基酸残基组成的多肽,它连接胰岛素原的 A 链和 B 链以确保正确折叠,具有生物活性并调节细胞功能。
TP1070L PACAP (1-27), human, ovine, rat acetate

PACAP 1-27 acetate,PACAP (1-27), human, ovine, rat acetate(127317-03-7 free base)

PACAP GPCR/G Protein
PACAP (1-27), human, ovine, rat acetate (PACAP 1-27 acetate)(127317-03-7 free base) 是一种新的神经肽,最初从牛下丘脑中分离出来,也存在于人和大鼠中。
TP1359L Amyloid β Peptide (42-1)(human) acetate

Amyloid β Peptide (42-1)(human) acetate(317366-82-8 free base)

Beta Amyloid Neuroscience
Amyloid β Peptide (42-1)(human) acetate 是淀粉样蛋白 β 肽 (1-42) 的无活性形式。Amyloid β Peptide (42-1)(human) acetate 是由 42 个氨基酸组成的肽,其在阿尔茨海默病的发病机制中起关键作用。
TP1004L Beta-MSH (1-22) (human) acetate

Beta-MSH (1-22) (human) acetate (17908-57-5 Free base),醋酸Β-促黑激素(人)

Melanocortin Receptor GPCR/G Protein; Neuroscience
Beta-MSH (1-22) (human) acetate (Beta-MSH (1-22) (human) acetate (17908-57-5 Free base)) 是一种 22 肽,是一种内源性黑皮质素 4 受体 (MC4-R) 激动剂。
TP1705 Gastrin I (1-14), human

Others Others
Gastrin I (1-14), human 是人胃泌素 I 肽的 1-14 片段。其中Gastrin I 是内源性胃肠肽激素。Gastrin 是胃酸分泌的主要激素调节剂。
T21484 BNP (1-32), human

Others Others
BNP (1-32), human 是一种脑利钠肽。
TP2030L1 Gastrin I (human) acetate

Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐

cholecystokinin GPCR/G Protein
Gastrin I (human) acetate (Gastrin-17 acetate) 是在胃中产生的内源性肽,通过胆囊收缩素 2 (CCK2) 受体增加胃酸分泌。
TP1842L Angiotensinogen (1-14), human acetate

Endogenous Metabolite Metabolism
Angiotensinogen (1-14), human acetate 是血管紧张素原的片段,它是肾素-血管紧张素系统的被动底物。
TP1863L Glucagon (19-29), human acetate

Glucagon Receptor GPCR/G Protein
Glucagon (19-29), human acetate 是一种从胰高血糖素加工而来的 COOH 末端片段,是一种有效的胰岛素分泌抑制剂。
TP1949L PEN (human) aceate

GPCR19 GPCR/G Protein
PEN (human) aceate 是丰富的下丘脑神经肽之一,源自 ProSAAS 前蛋白,是 GPR83 的内源性配体。
TP1116L Kinetensin acetate(103131-69-7 free base)

Kinetensin (human) acetate

Neurotensin Receptor GPCR/G Protein
Kinetensin acetate(103131-69-7 free base) 是从经胃蛋白酶处理的人血浆中分离出来的。它是一种神经降压素样肽。
TP1188L Cortistatin 14, human, rat acetate

Somatostatin GPCR/G Protein
Cortistatin 14, human, rat acetate 是一种与 somatostatin-14 结构相似的神经肽,具有抗惊厥、神经保护作用和显着的抗炎特性。 Cortistatin 14, human, rat acetate 通过与生长抑素受体结合并发挥其功能。

化合物

Gastrin I, human
Cat.No: TP2030
Synonym: Gastrin I (human)
Target: cholecystokinin
Adrenocorticotropic Hormone (ACTH) (18-39), human TFA
Cat.No: TP1240
Synonym: CLIP (human) (TFA)
Target: Others
Fibrinopeptide A, human acetate
Cat.No: TP1143L
Synonym: Fibrinopeptide A, human acetate(25422-31-5 free base),Human fibrinopeptide A acetate
Target: Others
Endothelin-2 (49-69), human
Cat.No: TP1174
Synonym: Human endothelin-2,Endothelin-2, human,Endothelin-2 (human, canine),人内皮素2
Target: Others
MART-1 (26-35) (human)
Cat.No: T7489
Synonym: MART-1 (26-35) human
Target: Others
C-Type Natriuretic Peptide (CNP) (1-22), human
Cat.No: TP1187
Synonym: CNP (1-22), human
Target: RAAS
GIP (human) acetate
Cat.No: TP2018L
Synonym: GIP (human) acetate(100040-31-1 Free base)
Target: IGF-1R
Insulin (human)
Cat.No: T8221
Synonym: INSULIN,甘精胰岛素,胰岛素,Insulin(human)
Target: IGF-1R
Neuropeptide AF (human) acetate
Cat.No: TP1082L
Synonym: Neuropeptide AF (93-110), human Acetate,Neuropeptide AF (human) acetate (192387-38-5 Free base)
Target: Opioid Receptor
ELA-14(human) acetate
Cat.No: TP1923L1
Synonym: ELA-14(human) acetate (1886973-05-2 free base)
Target: Apelin receptor, Arrestin
Angiotensin III, human, mouse
Cat.No: T7577
Synonym: 血管紧张素III,Angiotensin III, human, mouse(3TFA)
Target: RAAS
TNF-α (31-45), human acetate
Cat.No: T19584L
Synonym: TNF-α (31-45), human acetate(144796-71-4 free base)
Target: Others
Hemopressin (human, mouse) acetate
Cat.No: TP1900L1
Synonym: Hemopressin (human, mouse) acetate(1314035-51-2 free base)
Target: Cannabinoid Receptor
Adrenocorticotropic Hormone (ACTH) (1-39), human
Cat.No: T8231
Synonym: ACTH (1-39), human,丝拉克肽
Target: Others
BAD (103-127) (human) acetate
Cat.No: T40412L
Synonym: BAD (103-127) (human) acetate (331762-68-6 Free base)
Target: Others
Adrenomedullin (AM) (22-52), human acetate
Cat.No: TP1257L
Synonym: Adrenomedullin (AM) (22-52), human acetate(159899-65-7 Free base)
Target: CGRP Receptor
Angiotensin I (human, mouse, rat)
Cat.No: TP1295
Synonym: Angiotensin 1 Human,血管紧张素 1 (人)
Target: Others
Apelin-17 (human, bovine) acetate
Cat.No: TP2092L
Synonym: Apelin-17 (human, bovine) acetate(217082-57-0 free base)
Target: HIV Protease
Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
Cat.No: TP1219
Synonym: ANP (1-28), human, porcineANP(1-28)
Target:
PAMP-12 (human, porcine) acetate
Cat.No: TP1880L1
Synonym: PAMP-12 (human, porcine) acetate(196305-05-2 free base)
Target: Others
Corticotropin-releasing factor (human) acetate
Cat.No: TP1144L
Synonym: Corticotropin-releasing factor (human) acetate (86784-80-7 Free base)
Target: CRFR
Endothelin 1 (swine, human) acetate
Cat.No: T19309L1
Synonym: Endothelin 1 (swine, human) acetate(117399-94-7 free base)
Target: Endothelin Receptor
Prepro VIP (111-122), human acetate
Cat.No: TP1627L
Synonym: Prepro VIP (111-122), human acetate(123025-94-5 free base)
Target: Others
Urotensin II (114-124), human acetate
Cat.No: TP1737L
Synonym: Urotensin II (114-124), human acetate(251293-28-4 free base)
Target: GPR
Adrenocorticotropic Hormone (ACTH) (1-10), human acetate
Cat.No: TP1244L1
Synonym: Adrenocorticotropic Hormone (ACTH) (1-10), human acetate(2791-05-1 Free base)
Target: Others
β-Interleukin I (163-171), human Acetate
Cat.No: T21608L
Synonym: β-Interleukin I (163-171), human Acetate(106021-96-9 Free base)
Target: Others
Galanin (1-30), human acetate
Cat.No: TP1732L
Synonym: 醋酸甘丙肽,Galanin (1-30), human acetate(119418-04-1 Free base)
Target: Others
PACAP-38 (31-38), human, mouse, rat acetate
Cat.No: TP1618L
Synonym: PACAP-38 (31-38), human, mouse, rat acetate(138764-85-9 Free base)
Target: PACAP
β-Amyloid (1-42), acetate (human)
Cat.No: TP1007L
Synonym: β-Amyloid (1-42), human acetate (107761-42-2 Free base)
Target:
Activated Protein C (390-404), human acetate
Cat.No: TP1628L
Synonym: Activated Protein C (390-404), human acetate(146340-20-7 Free base)
Target: APC
Human IgE Pentapeptide HEPP acetate
Cat.No: TP2499
Synonym: Human IgE Pentapeptide HEPP acetate (62087-72-3 Free base)
Target:
Acetyl-Calpastatin (184-210)(human) acetate
Cat.No: TP2056L
Synonym: Acetyl-Calpastatin (184-210) (human) acetate(123714-50-1 Free base )
Target: Cysteine Protease
β-Endorphin (1-27) (human) acetate
Cat.No: T38193L
Synonym: β-Endorphin (1-27) (human) acetate(76622-84-9 Free base)
Target: Opioid Receptor
MCH(human, mouse, rat)
Cat.No: TP1996
Synonym: MCH (human, mouse, rat),黑色素聚集激酶素(MCH)( 大鼠)
Target: GPR, Melanin-concentrating Hormone Receptor (MCHR)
C-Type Natriuretic Peptide (CNP) (1-22), human acetate
Cat.No: T39392L
Synonym: C-Type Natriuretic Peptide (CNP) (1-22), human acetate(1966153-17-2 Free base)
Target: Others
Obestatin(human)
Cat.No: T38470
Synonym:
Target:
GnRH Associated Peptide (GAP) (1-13), human Acetate
Cat.No: T21649L
Synonym: GnRH Associated Peptide (GAP) (1-13), human Acetate (100111-07-7 Free base)
Target: Others
α-CGRP (human) acetate
Cat.No: TP2044L
Synonym: 人类降钙素基因相关肽 1,α-CGRP (human) acetate (90954-53-3 free base)
Target: Others
Proinsulin C-peptide human acetate
Cat.No: TP1651L
Synonym: 醋酸胰岛素原C-肽(55-89),人,Proinsulin C-peptide human acetate (33017-11-7 Free base)
Target: Others
PACAP (1-27), human, ovine, rat acetate
Cat.No: TP1070L
Synonym: PACAP 1-27 acetate,PACAP (1-27), human, ovine, rat acetate(127317-03-7 free base)
Target: PACAP
Amyloid β Peptide (42-1)(human) acetate
Cat.No: TP1359L
Synonym: Amyloid β Peptide (42-1)(human) acetate(317366-82-8 free base)
Target: Beta Amyloid
Beta-MSH (1-22) (human) acetate
Cat.No: TP1004L
Synonym: Beta-MSH (1-22) (human) acetate (17908-57-5 Free base),醋酸Β-促黑激素(人)
Target: Melanocortin Receptor
Gastrin I (1-14), human
Cat.No: TP1705
Synonym:
Target: Others
BNP (1-32), human
Cat.No: T21484
Synonym:
Target: Others
Gastrin I (human) acetate
Cat.No: TP2030L1
Synonym: Gastrin I (human) acetate(10047-33-3 free base),Gastrin-17 acetate,Little gastrin I acetate,胃膜素醋酸盐
Target: cholecystokinin
Angiotensinogen (1-14), human acetate
Cat.No: TP1842L
Synonym:
Target: Endogenous Metabolite
Glucagon (19-29), human acetate
Cat.No: TP1863L
Synonym:
Target: Glucagon Receptor
PEN (human) aceate
Cat.No: TP1949L
Synonym:
Target: GPCR19
Kinetensin acetate(103131-69-7 free base)
Cat.No: TP1116L
Synonym: Kinetensin (human) acetate
Target: Neurotensin Receptor
Cortistatin 14, human, rat acetate
Cat.No: TP1188L
Synonym:
Target: Somatostatin
Cat. No. Product Name Target Signaling Pathways
TP2167 β-CGRP, human acetate

β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate

CGRP Receptor GPCR/G Protein; Neuroscience
β-CGRP, human acetate 是降钙素肽之一,通过受体活性修饰蛋白 (RAMP) 和降钙素受体样受体 (CRLR) 的复合物发挥作用(对于 CRLR/RAMP1 和 CRLR,IC50:1 nM 和 300 nM /RAMP2 在单元格中)。
T7040 Angiotensin II human

DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Angiotensin II human (Ang II) 是一种生物活性肽,一种血管收缩剂。Angiotensin II 可以与 AT1R 和 AT2R 相互作用,调节人类血压,刺激交感神经,增加醛固酮生物合成和肾脏活动。
T13433 β-Endorphin, human

Others Others
β-Endorphin, human, a prominent endogenous peptide, existing in the hypophysis cerebri and hypothalamus,and is an agonist of opioid receptor.
T41030 γ-Globulins from human blood

γ-Globulins, a protein fraction found in human blood, comprise a class of proteins with potent antibody activity that safeguards against bacterial and viral infections. These γ-globulins are specifically utilized in the treatment of common variable immunodeficiency.
T6377 Aloperine

Apoptosis; Virus Protease; HIV Protease; Antibiotic; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Aloperine 是一种在苦参类植物中的生物碱,其具有抗癌,抗炎、抗肿瘤和抗病毒特性,可用于研究过敏性接触性皮炎湿疹和其他皮肤炎症。
TN2283 Tripterifordin

HIV Protease Microbiology/Virology; Proteases/Proteasome
Tripterifordin 在 H9 淋巴细胞中显示出抗 HIV 复制活性,EC50值为 3100 nM。
T2S1040 Jolkinolide B

ERK; IL Receptor; BCL; p38 MAPK; TNF; NF-κB; Akt; Caspase; PI3K; JAK; JNK; STAT; mTOR Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; JAK/STAT signaling; MAPK; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Jolkinolide B 是一种从 Euphorbia fischeriana Steud 的根中分离出来的具有生物活性的二萜。 Jolkinolide B 诱导癌细胞凋亡。 Jolkinolide B 可用于预防和治疗骨溶解的研究。
T3020 Sclareol

Apoptosis; Others Apoptosis; Others
Sclareol 是一种从快乐鼠尾草中分离出来的拉丹型二萜,对多种人类 Y 细胞系具有生长抑制和细胞毒活性,诱导细胞凋亡。
T9503 PHYTOSPHINGOSINE

Apoptosis Apoptosis
Phytosphingosine 是具有抗癌作用的一种磷脂。在癌细胞中,它通过 caspase 8 的激活和 Bax 转位诱导细胞凋亡。
T10021 1-Methylxanthine

Endogenous Metabolite Metabolism
1-Methylxanthine 是咖啡因衍生物,是咖啡因和茶碱 (1,3-二甲基黄嘌呤,TP) 在人体尿代谢产物,能够提高肿瘤细胞的放射敏感性。
TQ0217 Gomisin G

戈米辛G,戈米辛 G

P450; HIV Protease Metabolism; Microbiology/Virology; Proteases/Proteasome
Gomisin G 是一种有抗HIV 活性的天然产物。
T11363 Ganoderic acid F

Others Others
Ganoderic acid F 是一种灵芝酸。它具有抗肿瘤和抗转移的活性,与抑制血管生成和涉及细胞增殖和细胞死亡,致癌作用,氧化应激,钙信号传导和内质网应激的蛋白质改变等机制相关。
TN4417 Larixyl acetate

Others Others
Larixyl acetate 是一种生物活性化学物质。
T0474 Erythromycin ethylsuccinate

EES,琥乙红霉素

ribosome; HIV Protease; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Erythromycin ethylsuccinate (EES) 是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗 HIV-1病毒活性。
T2942 Psoralen

Ficusin,Furocoumarin,补骨脂素,psoralene

Apoptosis; Influenza Virus; HIV Protease; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
Psoralen (Ficusin) 是从补骨脂种子中提取的一种香豆素。它具有如抗癌、抗氧化、抗抑郁、抗癌、抗菌、抗病毒等多种生物学特性。
Fr16741 Oxindole

2-吲哚酮,板蓝根,Indolin-2-one

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Oxindole (Indolin-2-one) 是一种芳族杂环砌块,其衍生物是激酶抑制剂研究中的主要成分。
TN2069 Picrocrocin

藏红花,苦番紅花素

Apoptosis Apoptosis
Picrocrocin 是一种从椰菜花中发现的类胡萝卜素,对 SKMEL-2 人恶性黑色素瘤细胞具有生长抑制作用,具有抗癌作用。
T10005L 1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium

Endogenous Metabolite Metabolism
1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium 是一种人内源性代谢物,是一种磷酸酯。
T5061 Lumichrome

7,8-Dimethylalloxazine,光色素

Others Others
Lumichrome (7,8-Dimethylalloxazine) 是人类体内的内源性化合物,由核黄素光降解产生。它利用 p53 依赖机制抑制人肺癌细胞生长并诱导凋亡。
T2865 Oleanolic Acid

Oleanic acid,Caryophyllin,齐墩果酸

HIV Protease; Endogenous Metabolite; Antibiotic; Autophagy Autophagy; Metabolism; Microbiology/Virology; Proteases/Proteasome
Oleanolic Acid (Caryophyllin) 是具有抗癌活性的一种天然产物。
T0966 Sennoside A

番泻苷A,NSC 112929,番泻苷 A

MAO; HIV Protease Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Sennoside A (NSC-112929) 是在番泻叶的叶子和豆荚中大量发现的蒽醌苷,抑制 HIV-1 复制。
T3822 Bellidifolin

Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Bellidifolin (Bellidifoline) 是从獐牙菜的茎中提取的一种呫吨酮,它能作为病毒蛋白 R 的抑制剂,具有保肝、降血糖、抗炎、抗氧化、抗肿瘤作用。
T6841 Fumagillin

NSC9168,烟曲霉素,Amebacilin

Others; HIV Protease; Antibiotic; Parasite Microbiology/Virology; Others; Proteases/Proteasome
Fumagillin (Amebacilin) 由烟曲霉菌中提取的一种抗菌药,有抗阿米巴活性。它通过抑制 HIV-1 viral protein R 活性来抑制 HIV‐1感染。
TN1103 Diphyllin

山荷叶素,二叶草素

ATPase; Proton pump; Influenza Virus; HIV Protease Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Diphyllin 是一种从Justicia procumbens 中分离的芳基萘木脂素,是HIV-1的有效抑制剂,IC50 为 0.38 μM。它是V-ATPase 抑制剂,IC50值为 17 nM,可抑制人破骨细胞中的溶酶体酸化。它抑制NO 产生,IC50值为 50 μM ,具有抗癌和抗炎活性。
T8689 Chloroquine

CQ,氯喹

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine 是一种 Toll 样受体抑制剂,可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性,广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。
T8116 Azulene

甘菊蓝,奥苷菊环,Bicyclo[5.3.0]Decapentaene

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Azulene (Bicyclo[5.3.0]Decapentaene) 是萘的异构体,具有高抗HIV 活性。它是从洋甘菊精油中分离出来的一种化学支架。
T5S1133 Ganoderic acid D

灵芝酸D,灵芝酸 D

Apoptosis; Sirtuin Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Ganoderic acid D 是高度氧化的四环三萜,是灵芝的主要活性成分,可诱导 HeLa 人宫颈癌细胞凋亡。它上调 SIRT3的蛋白质表达并通过 SIRT3 诱导脱乙酰化的亲环蛋白 D 。它抑制结肠癌细胞的能量重编程,包括结肠癌细胞中的葡萄糖摄取,乳酸、丙酮酸和乙酰辅酶的产生。
T2177 Kaempferol

Kempferol,山柰酚,山奈酚,Robigenin

Apoptosis; Estrogen Receptor/ERR; Mitophagy; Estrogen/progestogen Receptor; HIV Protease; Endogenous Metabolite; Parasite; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; Metabolism; Microbiology/Virology; Proteases/Proteasome
Kaempferol (Robigenin) 属于天然类黄酮,是一种 ERRα 和 ERRγ 的反向激动剂。Kaempferol 具有抗肿瘤、抗炎、抗氧化、抗菌和抗病毒等多种活性。
T0492 Dimethyl fumarate

富马酸二甲酯,DMF

Reactive Oxygen Species; HIV Protease; Nrf2; Endogenous Metabolite; Autophagy Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Dimethyl fumarate (DMF) 是具有口服活性且可透过血脑屏障的Nrf2激活剂,可诱导抗氧化剂基因表达上调。它是一种富马酸盐衍生物,可作抗炎和免疫调节剂,可研究多发性硬化症。
T2S0731 Trilobatin

三叶苷,三叶甙,P-Phlorizin

Amylase Metabolism
Trilobatin (P-Phlorizin) 是源自Lithocarpus polystachyusRehd 的甜味剂,是一种HIV-1抑制剂,靶向 Gp41 包膜蛋白,具有神经保护作用。它还是SGLT1/2抑制剂,可选择性诱导人肝母细胞瘤细胞增殖。
T0437 Inosine

INO 495,NSC 20262,肌苷

ROS; Endogenous Metabolite; Adenosine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Inosine (NSC-20262) 是由腺苷分解代谢产生的一种内源性嘌呤核苷,是腺苷受体A1R 和A2AR 的激动剂,具有抗炎免疫调节,抗伤害和神经保护作用。
TN2004 Obtusin

1,7-二羟基-2,3,8-三甲氧基-6-甲基蒽-9,10-二酮,决明素

MAO; Monoamine Oxidase Metabolism; Neuroscience
Obtusin 是来自决明子种子,是一种高度选择性和竞争性的人单胺氧化酶-A 抑制剂,IC50=11.12 μM,Ki=6.15 μM。它在神经退行性疾病,尤其是焦虑和抑郁中起预防作用。
T2789 Scutellarin

黄岑素,野黄芩苷,Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide

Akt; HIV Protease; STAT Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Scutellarin (Scutellarein-7-glucuronide) 是从黄芩中分离的黄酮,可抑制破骨细胞中 RANKL 介导的 MAPK 和 NF-κB 信号通路,并下调 HCC 细胞中的 STAT3/Girdin/Akt 信号通路。
T4962 Zingibroside R1

Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Zingibroside R1 (Ginsenoside Z-R1) 是分离自Panax japonicasC. A. Meyer 根部的一种三萜皂苷,有HIV-1、抗肿瘤和抗血管生成活性。它对 EAT 细胞的 2-脱氧-D-葡萄糖的摄取具有抑制作用,IC50值为91.3 μM。
T1284 Megestrol acetate

SC10363,醋酸甲地孕酮,BDH1298

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。
T1131 Ivermectin

MK-933,伊维菌素

Mitophagy; GluCls; P2X Receptor; SARS-CoV; HIV Protease; Antibiotic; Parasite; Autophagy; HSV Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ivermectin (MK-933) 是谷氨酸门控氯离子通道激活剂,具有抗寄生虫活性。它特异性抑制Impα/β1 介导的核导入,还抑制牛疱疹病毒 1 复制并抑制BoHV-1DNA 聚合酶的核输入。它具有很强的抗病毒活性。它也是P2X4和 α7nAChRs 的正异构效应物。
T2728 Limonin

Dictamnolactone,Limonoic acid 3,19:16,17 dilactone,柠檬苦素,Obaculactone,Citrolimonin

Apoptosis; HIV Protease; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome
Limonin (Citrolimonin) 是柑橘类水果中富含的一种三萜类天然产物,具有抗病毒和抗肿瘤活性。
T7991 2-Hydroxycinnamic acid

邻羟基肉桂酸(邻香豆酸),(E)-3-(2-羟基苯基)丙烯酸

Others; SARS-CoV; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
2-Hydroxycinnamic acid 是从肉桂的甲醇提取物中分离出的一种天然产物,具有光氧化活性。它对HIV/SARS-CoV S 假病毒的感染具有抑制作用,IC50为 0.3 mM。
TN2883 3',4'-Dimethoxyflavone

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。
T16791 Rottlerin

Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525

CaMK; Apoptosis; Others; HIV Protease; PKA; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Neuroscience; Others; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Rottlerin (NSC-56346) 是一种从Mallotus Philippinensis 中得到的天然产物, 是 PKC 的特异性抑制剂,抑制HIV-1整合和狂犬病病毒感染。它通过活化 caspase 3 诱导细胞凋亡.
T3122 Fangchinoline

Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline

Apoptosis; FAK; HIV Protease; Autophagy Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Fangchinoline (Tetrandrine B) 是从Stephaniatetrandra 中分离出来的,一种具有广泛生物学活性的天然产物。它是新型HIV-1抑制剂,通过损害 gp160 蛋白水解过程来抑制 HIV-1 复制。它靶向Focal adhesion kinase (FAK)并抑制肿瘤细胞中 FAK 介导的的信号传导途径。
T3730 Methyl gallate

NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯

Reactive Oxygen Species; HIV Protease; Reverse Transcriptase; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Methyl gallate (Gallincin) 是具有抗氧化,抗癌和抗炎活性的植物酚类。它也可抑制细菌活性。它还具有抗HIV-1和HIV-1酶的抑制活性。
T4P2931 Linoleic acid

9,12-octadecadienoic acid,亚油酸,α-亚油酸,acidelinoleique,9,12-Linoleic acid

Others; Endogenous Metabolite Metabolism; Others
Linoleic acid (9,12-octadecadienoic acid) 是一种多不饱和脂肪酸,存在于坚果、种子和植物性油中。它是膜磷脂的一部分,作为膜流动性的结构成分来维持表皮透皮水屏障。它通过氧化作用引起血红蛋白和红细胞损伤。
TN6796 2'-FUCOSYLLACTOSE

2'-Fucosyl-D-lactose,2'-岩藻糖基乳糖

Others Others
2'-FUCOSYLLACTOSE (2'-Fucosyl-D-lactose) 是一种含岩藻糖的寡糖。
T5782 Bevirimat

YK FH312,MPC-4326,PA-457,贝韦立马

HIV Protease Microbiology/Virology; Proteases/Proteasome
Bevirimat (PA-457) 是一种 HIV-1 成熟抑制剂,可在病毒体成熟过程中阻断 Gag 衣壳 (CA) 前体 CA-SPI 裂解为成熟的 CA 蛋白。
T2830 Betulinic acid

白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid

Apoptosis; Mitophagy; NF-κB; HIV Protease; Topoisomerase; Endogenous Metabolite; Aminopeptidase; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Betulinic acid (ALS-357) 是从白桦树皮中分离出来的一种五环三萜类天然产物,是真核细胞拓扑异构酶 I 的抑制剂,IC50值为 5 μM,具有抗逆转录病毒、抗疟疾、抗癌和抗炎特性。
T2775 Baicalin

黄芩苷,黄岑苷,Baicalein 7-O-β-D-glucuronide

NF-κB; HIV Protease; GABA Receptor; Autophagy Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome
Baicalin (Baicalein 7-O-β-D-glucuronide) 是一种从黄芩中分离出来的脯氨酰内肽酶抑制剂,具有抗氧化、抗肿瘤、抗 HIV 的特性。
T7203 Oglufanide

奥谷法奈,L-Glutamyl-L-tryptophan,H-Glu-Trp-OH

VEGFR; HCV Protease; Endogenous Metabolite Angiogenesis; Metabolism; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Oglufanide (H-Glu-Trp-OH) 是一种从小牛胸腺中分离出来的二肽免疫调节剂,可抑制血管内皮生长因子,可刺激细胞内细菌感染和对丙型肝炎病毒的免疫反应。
T6S2391 L-Chicoric Acid

(-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸,是一种选择性可逆的 HIV-1 整合酶抑制剂,IC50约为 100 nM。它还可抑制 HIV-1 复制。
T0070 Pentoxifylline

Oxpentifylline,PTX,己酮可可碱,BL-191

HIV Protease; PDE; Adenosine Receptor; Autophagy Autophagy; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Pentoxifylline (PTX) 是一种具有口服活性的磷酸二酯酶非选择性抑制剂,具有免疫调节、抗炎、抗纤溶、抗增殖和血液流变学改善作用。它可研究周围血管疾病、脑血管疾病和其他一些涉及局部微循环缺陷的疾病。
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天然产物

β-CGRP, human acetate
Cat.No: TP2167
Synonym: β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate
Target: CGRP Receptor
Angiotensin II human
Cat.No: T7040
Synonym: DRVYIHPF,Angiotensin II,Hypertensin II,血管紧张素Ⅱ,Ang II,血管紧张素II
Target: Apoptosis, RAAS
β-Endorphin, human
Cat.No: T13433
Synonym:
Target: Others
γ-Globulins from human blood
Cat.No: T41030
Synonym:
Target:
Aloperine
Cat.No: T6377
Synonym:
Target: Apoptosis, Virus Protease, HIV Protease, Antibiotic, Autophagy
Tripterifordin
Cat.No: TN2283
Synonym:
Target: HIV Protease
Jolkinolide B
Cat.No: T2S1040
Synonym:
Target: ERK, IL Receptor, BCL, p38 MAPK, TNF, NF-κB, Akt, Caspase, PI3K, JAK, JNK, STAT, mTOR
Sclareol
Cat.No: T3020
Synonym:
Target: Apoptosis, Others
PHYTOSPHINGOSINE
Cat.No: T9503
Synonym:
Target: Apoptosis
1-Methylxanthine
Cat.No: T10021
Synonym:
Target: Endogenous Metabolite
Gomisin G
Cat.No: TQ0217
Synonym: 戈米辛G,戈米辛 G
Target: P450, HIV Protease
Ganoderic acid F
Cat.No: T11363
Synonym:
Target: Others
Larixyl acetate
Cat.No: TN4417
Synonym:
Target: Others
Erythromycin ethylsuccinate
Cat.No: T0474
Synonym: EES,琥乙红霉素
Target: ribosome, HIV Protease, Antibacterial, Antibiotic, Autophagy
Psoralen
Cat.No: T2942
Synonym: Ficusin,Furocoumarin,补骨脂素,psoralene
Target: Apoptosis, Influenza Virus, HIV Protease, DNA/RNA Synthesis
Oxindole
Cat.No: Fr16741
Synonym: 2-吲哚酮,板蓝根,Indolin-2-one
Target: Others, HIV Protease
Picrocrocin
Cat.No: TN2069
Synonym: 藏红花,苦番紅花素
Target: Apoptosis
1,2-Dipalmitoyl-sn-glycerol 3-phosphate sodium
Cat.No: T10005L
Synonym:
Target: Endogenous Metabolite
Lumichrome
Cat.No: T5061
Synonym: 7,8-Dimethylalloxazine,光色素
Target: Others
Oleanolic Acid
Cat.No: T2865
Synonym: Oleanic acid,Caryophyllin,齐墩果酸
Target: HIV Protease, Endogenous Metabolite, Antibiotic, Autophagy
Sennoside A
Cat.No: T0966
Synonym: 番泻苷A,NSC 112929,番泻苷 A
Target: MAO, HIV Protease
Bellidifolin
Cat.No: T3822
Synonym: Bellidifoline,龙胆山酮酚,Bellidifolium,雏菊叶龙胆酮
Target: Others, HIV Protease
Fumagillin
Cat.No: T6841
Synonym: NSC9168,烟曲霉素,Amebacilin
Target: Others, HIV Protease, Antibiotic, Parasite
Diphyllin
Cat.No: TN1103
Synonym: 山荷叶素,二叶草素
Target: ATPase, Proton pump, Influenza Virus, HIV Protease
Chloroquine
Cat.No: T8689
Synonym: CQ,氯喹
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
Azulene
Cat.No: T8116
Synonym: 甘菊蓝,奥苷菊环,Bicyclo[5.3.0]Decapentaene
Target: Others, HIV Protease
Ganoderic acid D
Cat.No: T5S1133
Synonym: 灵芝酸D,灵芝酸 D
Target: Apoptosis, Sirtuin
Kaempferol
Cat.No: T2177
Synonym: Kempferol,山柰酚,山奈酚,Robigenin
Target: Apoptosis, Estrogen Receptor/ERR, Mitophagy, Estrogen/progestogen Receptor, HIV Protease, Endogenous Metabolite, Parasite, Autophagy
Dimethyl fumarate
Cat.No: T0492
Synonym: 富马酸二甲酯,DMF
Target: Reactive Oxygen Species, HIV Protease, Nrf2, Endogenous Metabolite, Autophagy
Trilobatin
Cat.No: T2S0731
Synonym: 三叶苷,三叶甙,P-Phlorizin
Target: Amylase
Inosine
Cat.No: T0437
Synonym: INO 495,NSC 20262,肌苷
Target: ROS, Endogenous Metabolite, Adenosine Receptor
Obtusin
Cat.No: TN2004
Synonym: 1,7-二羟基-2,3,8-三甲氧基-6-甲基蒽-9,10-二酮,决明素
Target: MAO, Monoamine Oxidase
Scutellarin
Cat.No: T2789
Synonym: 黄岑素,野黄芩苷,Breviscapin,Breviscapinun,Breviscapine,Scutellarein-7-glucuronide
Target: Akt, HIV Protease, STAT
Zingibroside R1
Cat.No: T4962
Synonym: Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1
Target: HIV Protease
Megestrol acetate
Cat.No: T1284
Synonym: SC10363,醋酸甲地孕酮,BDH1298
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, HIV Protease, Autophagy
Ivermectin
Cat.No: T1131
Synonym: MK-933,伊维菌素
Target: Mitophagy, GluCls, P2X Receptor, SARS-CoV, HIV Protease, Antibiotic, Parasite, Autophagy, HSV
Limonin
Cat.No: T2728
Synonym: Dictamnolactone,Limonoic acid 3,19:16,17 dilactone,柠檬苦素,Obaculactone,Citrolimonin
Target: Apoptosis, HIV Protease, Endogenous Metabolite
2-Hydroxycinnamic acid
Cat.No: T7991
Synonym: 邻羟基肉桂酸(邻香豆酸),(E)-3-(2-羟基苯基)丙烯酸
Target: Others, SARS-CoV, HIV Protease
3',4'-Dimethoxyflavone
Cat.No: TN2883
Synonym:
Target: Others, PARP
Rottlerin
Cat.No: T16791
Synonym: Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525
Target: CaMK, Apoptosis, Others, HIV Protease, PKA, PKC, Autophagy
Fangchinoline
Cat.No: T3122
Synonym: Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline
Target: Apoptosis, FAK, HIV Protease, Autophagy
Methyl gallate
Cat.No: T3730
Synonym: NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯
Target: Reactive Oxygen Species, HIV Protease, Reverse Transcriptase, Antibacterial
Linoleic acid
Cat.No: T4P2931
Synonym: 9,12-octadecadienoic acid,亚油酸,α-亚油酸,acidelinoleique,9,12-Linoleic acid
Target: Others, Endogenous Metabolite
2'-FUCOSYLLACTOSE
Cat.No: TN6796
Synonym: 2'-Fucosyl-D-lactose,2'-岩藻糖基乳糖
Target: Others
Bevirimat
Cat.No: T5782
Synonym: YK FH312,MPC-4326,PA-457,贝韦立马
Target: HIV Protease
Betulinic acid
Cat.No: T2830
Synonym: 白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid
Target: Apoptosis, Mitophagy, NF-κB, HIV Protease, Topoisomerase, Endogenous Metabolite, Aminopeptidase, Autophagy
Baicalin
Cat.No: T2775
Synonym: 黄芩苷,黄岑苷,Baicalein 7-O-β-D-glucuronide
Target: NF-κB, HIV Protease, GABA Receptor, Autophagy
Oglufanide
Cat.No: T7203
Synonym: 奥谷法奈,L-Glutamyl-L-tryptophan,H-Glu-Trp-OH
Target: VEGFR, HCV Protease, Endogenous Metabolite
L-Chicoric Acid
Cat.No: T6S2391
Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸
Target: Others, HIV Protease
Pentoxifylline
Cat.No: T0070
Synonym: Oxpentifylline,PTX,己酮可可碱,BL-191
Target: HIV Protease, PDE, Adenosine Receptor, Autophagy
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