首页 工具
登录
购物车

搜索结果

Search Results for " gastric "

302

抑制剂 & 化合物

60

天然产物

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
TP1309 Gastric mucin

Antibacterial; Antibiotic Microbiology/Virology
Gastric mucin 是一种能保护胃肠道免受酸、蛋白酶、致病微生物和机械创伤影响的糖蛋白。
T78543 Acetyl Gastric Inhibitory Peptide (human) TFA

Human N-acetyl GIP TFA

AcetylGastric Inhibitory Peptide(human) TFA 是一种葡萄糖依赖性胰岛素释放多肽的改性脂肪酸衍生物,具有增强的抗高血糖和促胰岛素作用。它主要用于糖尿病、胰岛素抵抗和肥胖的科研领域。
T76309 Gastric Inhibitory Peptide, porcine

Gastric Inhibitory Peptide, porcine 为葡萄糖依赖性胰岛素促进多肽,包含42个氨基酸构成的肠道激素,对脂肪及葡萄糖代谢产生影响。
T37589 GIP (3-42), human

Gastric Inhibitory Polypeptide (3-42) (human)

IGF-1R Tyrosine Kinase/Adaptors
GIP (3-42), human (Gastric Inhibitory Polypeptide (3-42) (human)) 是一种多肽,可充当葡萄糖依赖性促胰岛素多肽 (GIP) 受体拮抗剂,在体内调节胰岛素分泌和 GIP 的代谢作用,可用于研究2型糖尿病。
T76310 Acetyl Gastric Inhibitory Peptide (human)

AcetylGastric Inhibitory Peptide(human),一种脂肪酸衍生的葡萄糖依赖性胰岛素多肽类似物,具备改善抗高血糖和胰岛素敏感性的特性。适用于糖尿病、胰岛素抵抗及肥胖研究。
T76308 Gastric Inhibitory Polypeptide (1-30), porcine

Gastric Inhibitory Polypeptide (1-30), porcine 缺乏天然胃抑制多肽 (GIP) C 端 12 个氨基酸残基,能够增强胰岛素和生长抑素的释放而发挥生物活性。
T17030 Tegoprazan

ATPase; Proton pump Membrane transporter/Ion channel
Tegoprazan 是一种口服有效的、高选择性胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,能够控制胃酸分泌和运动,在体外检测的对猪、犬、人的 H+/K+-ATP 酶的 IC50为0.29-0.52 μM。
T76307 [Tyr0] Gastric Inhibitory Peptide (23-42), human

[Tyr0]Gastric Inhibitory Peptide(23-42), human,属于葡萄糖依赖性促胰岛素多肽(GIP)类,具有抑制胃酸分泌并促进胰岛素释放的功能。它在糖尿病和肥胖症的研究中有应用价值。
T83694 Gastric Inhibitory Peptide (1-42) (porcine) TFA

GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42)

胃抑制肽(GIP) (1-42)是一种内源性的42氨基酸肽类肠促素激素,能诱导胰岛素分泌。该激素在肠道神经内分泌K细胞和颌下腺中表达,并在餐后释放到循环中。GIP (1-42)抑制由组胺、五肽和胰岛素引起的胃酸和胃蛋白酶分泌,增加葡萄糖诱导的胰岛素释放,并在大鼠中刺激胃排空。
T83710 Gastric Inhibitory Peptide (22-51) (human) TFA

GIP (22-51),Glucose-dependent Insulinotropic Peptide (22-51)

胃抑制肽(GIP) (22-51) 是一种具有30个氨基酸的前动脉硬化肽,对应于GIP前体蛋白proGIP的第22至51个氨基酸残基,已在人类血浆中发现。在1 µM的浓度下使用,该肽能引起在巨峰细胞分化的THP-1细胞和分离的人类主动脉内皮细胞中IκB-α的降解和NF-κB的核转移。在体内,GIP (22-51) 增加了ApoE-/-小鼠的动脉粥样硬化病变面积和斑块形成。
T82332 Gastric Inhibitory Polypeptide (6-30) amide (human)

Gastric Inhibitory Polypeptide (6-30) amide (human) 为一种肠促胰岛素激素,主要应用于糖尿病研究领域。
T4579 Pentagastrin

五肽胃泌素,ICI-50123

Others; cholecystokinin GPCR/G Protein; Others
Pentagastrin (ICI-50123) 是一种选择性的胆囊收缩素 B(CCKB) 受体激动剂,IC50=11 nM。它能够增强胃粘膜对酸的防御机制,并保护胃粘膜免受损伤。
T38612 Linaprazan glurate

Others Others
Linaprazan glurate 抑制外源性或内源性刺激的胃酸分泌。 Linaprazan glurate 可用于胃肠道炎症性疾病和消化性溃疡疾病的研究。
T83696 Gastric Inhibitory Peptide 1 (3-42) (human) TFA

Glucose-dependent Insulinotropic Polypeptide 3-42,GIP-1 (3-42)

胃抑制肽1(GIP-1) (3-42)是肠促胰岛素激素GIP的一个肽段,同时也是GIP受体的拮抗剂。它通过血清二肽基肽酶4(DDP-4)从GIP中形成。GIP-1 (3-42) (100 nM)在减少BRIN-BD11胰腺细胞的胰岛素分泌方面起作用。在以25 nmol/kg剂量给药的ob/ob糖尿病小鼠模型中,它能增加血浆葡萄糖水平并降低血浆胰岛素水平。
T22724 Dimaprit dihydrochloride

NOS; NO Synthase; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Dimaprit dihydrochloride 是组胺H2受体的一种选择性激动剂,可刺激胃酸的分泌。它还抑制nNOS,IC50值为 49 μM。
T4981 Anisotropine Methylbromide

Prostaglandin Receptor; AChR GPCR/G Protein; Immunology/Inflammation; Neuroscience
Anisotropine Methylbromide 是一种抗胆碱能药物,已用于缓解胃肠道痉挛和抑制胃酸分泌。
T15500 HPi1

Others; Antibacterial Microbiology/Virology; Others
HPi1 是一种有口服活性的,针对幽门螺杆菌的选择性抗菌剂,IC50为 0.24 μM,MIC 为 0.08-0.16 μg/mL。
T6710 Troxipide

曲昔派特,曲昔匹特,Aplace

Others Others
Troxipide (Aplace) 是非分泌型胃保护剂,是口服具有活力的胃炎和胃溃疡的防御因子的增强剂,具有抗溃疡、抗炎和粘液分泌作用。
T1787 Levobupivacaine

Sodium Channel Membrane transporter/Ion channel
Levobupivacaine 是一种氨基酰胺类局麻药,属于n-alkylsubstituted pipecoloxylidide 家族。它是bupivacaine 的 S-对映异构体。
T9929 Ramucirumab

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
Ramucirumab 是一种人 VEGFR-2 拮抗剂,具有抗实体瘤活性。它是人源化单克隆抗体,能够与 VEGFR-2 结合,阻碍 VEGFR 配体 VEGF-A,VEGF-C 和 VEGF-D 结合。
T2319 Acotiamide monohydrochloride trihydrate

Acotiamide hydrochloride,YM-443 HCl,盐酸阿考替胺,Z-338 HCl

AChE Neuroscience
Acotiamide monohydrochloride trihydrate (Z-338 HCl) 是一种首创的、具有口服活性的胃肠动力药。它通过促毒蕈碱受体拮抗作用和乙酰胆碱酯酶(AChE)抑制作用增强肠神经元释放的乙酰胆碱,从而增强胃排空和胃部适应性,有潜力用于功能性消化不良的研究。
T2676 PF-04217903

c-Met/HGFR Tyrosine Kinase/Adaptors
PF04217903 是一种高效的、 ATP 竞争性的c-Met 激酶抑制剂(Ki=4.8 nM),相对于 208 个激酶,PF04217903 显示出 1000 倍以上的选择性。它抗血管生成作用。
T8599 Betazole dihydrochloride

盐酸倍他唑,Betazole hydrochloride

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Betazole dihydrochloride (Betazole hydrochloride) 是吡唑类组胺,是一种口服活性 H2受体激动剂,能诱导胃酸分泌,导致胆总管压力立即显著升高。它作为一种诊断剂,用于研究胃酸分泌能力。
T22368 Metyrosine

甲酪氨酸,α-Methyltyrosine

COX Immunology/Inflammation; Neuroscience
Metyrosine (α-Methyltyrosine) 是一种选择性酪氨酸羟化酶抑制剂,可显著抑制高 COX-2 活性和有效控制血压,具有抗炎和抗溃疡作用。
T1756L Ilaprazole

IY81149,艾普拉唑,IY 81149,IY-81149

Proton pump; TOPK MAPK; Membrane transporter/Ion channel
Ilaprazole (IY-81149) 是一种具有口服活性质子泵抑制剂,以剂量依赖性方式不可逆地抑制H+/K+-ATPase,在兔壁细胞制剂中的IC50为 6 μM。它也是一种有效的T 细胞起源蛋白激酶(TOPK)抑制剂,用于胃溃疡的研究。
T6700 Tenatoprazole

泰妥拉唑,TU-199

Proton pump Membrane transporter/Ion channel
Tenatoprazole (TU-199) 是一种口服有效的,基于咪唑吡啶的质子泵抑制剂。它抑制猪胃H+/K+-ATP 酶活性,IC50为6.2 μM。它阻断泛素与 ESCRT-1 因子 Tsg101 的相互作用,抑制几种包膜病毒的产生,包括 EBV。
T0865 Ranitidine Hydrochloride

AH19065,盐酸雷尼替丁

P450; Antibacterial; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Ranitidine Hydrochloride (AH19065) 是一种具有口服活性的组胺 H2 受体选择性拮抗剂,IC50为 3.3 μM。它还是一种CYP2C19和CYP2C9的弱抑制剂,可抑制胃液分泌。
T6540 Ibuprofen Lysine

布洛芬赖氨酸盐,Neoprofen

COX Immunology/Inflammation; Neuroscience
Ibuprofen Lysine (Neoprofen) 是一种非甾体抗炎药。
T1052 Proglumide

二丙谷酰胺

cholecystokinin GPCR/G Protein
Proglumide (Binoside) 是一种非肽的、口服具有活性的胆囊收缩素(CCK)-A/B 受体拮抗剂。它能够选择性阻断 CCK 在中枢神经系统中的作用。它能够抑制胃分泌,具有保护胃十二指肠粘膜的能力,并表现出抗癫痫和抗氧化活性。
T0081 Lafutidine

拉呋替丁,FRG-8813

5-HT Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Lafutidine (FRG-8813) 是一种组胺受体 H2RA 拮抗剂,可抑制胃酸分泌,具有胃粘膜保护作用,可用于研究胃食管反流疾病。
T3610 Ranitidine

雷尼替丁,HSDB 3925,Ranitidin

P450; Antibacterial; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Ranitidine (HSDB 3925) 是一种选择性的,具有口服活性的组胺 H2 受体拮抗剂,IC50为 3.3 μM。它还一种是CYP2C19和CYP2C9的弱抑制剂,可抑制胃液分泌。
T1562 Rebamipide

Proamipide,OPC12759,瑞巴派特

Free radical scavengers; COX; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience; oxidation-reduction
Rebamipide (OPC12759) 是一种粘膜保护剂,可诱导COX-2表达,增加PGE2水平,并以 COX-2 依赖性方式增强胃粘膜防御。
T1756 Ilaprazole sodium

IY-81149 sodium,艾普拉唑钠

Proton pump; TOPK MAPK; Membrane transporter/Ion channel
Ilaprazole sodium (IY-81149 sodium) 是一种具有口服活性质子泵抑制剂,以剂量依赖性方式不可逆地抑制 H+/K+-ATPase,在兔壁细胞制剂中的 IC50为 6 μM。它也是一种有效的 T 细胞起源蛋白激酶(TOPK)抑制剂,用于胃溃疡的研究。
T0157 Roxatidine Acetate hydrochloride

HOE 760,盐酸罗沙替丁醋酸酯,Roxatidine Acetate HCl

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Roxatidine Acetate hydrochloride (HOE 760) 是一种特异性和竞争性的组胺 H2 受体拮抗剂,能抑制胃酸分泌,可用于胃溃疡和十二指肠溃疡的研究。
T11139 (E/Z)-BCI

NSC 150117

Apoptosis; Phosphatase Apoptosis; Metabolism
(E/Z)-BCI (NSC-150117) 是一种DUSP6抑制剂,可通过激活 Nrf2 信号和抑制 NF-κB 通路,减弱 LPS 诱导的巨噬细胞炎症和 ROS 生成,具有抗炎活性。
T11826 LCH-7749944

GNF-PF-2356

Apoptosis; PAK Apoptosis; Cytoskeletal Signaling
LCH-7749944 (GNF-PF-2356) 是一种 PAK4抑制剂,IC50为 14.93 μM。它通过下调 PAK4/c-Src/EGFR/cyclin D1 途径有效抑制人胃癌细胞的增殖,并诱导凋亡。
T2325 Neratinib

HKI-272,来那替尼

EGFR; HER Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Neratinib (HKI-272) 是一种口服的、不可逆的酪氨酸激酶抑制剂,对 HER2 和 EGFR 的 IC50值分别为 59 和 92 nM。
T0686 Orlistat

Ro-18-0647,奥利司他,Tetrahydrolipstatin

Apoptosis; Others; Fatty Acid Synthase Apoptosis; Metabolism; Others
Orlistat (Tetrahydrolipstatin) 是一种不可逆的胰腺和胃脂肪酶抑制剂,也是一种脂肪酸合成酶抑制剂,可研究肥胖症,具有抗动脉粥样硬化作用。
T1394 Ibuprofen

Brufen,(±)-Ibuprofe,布洛芬,Motrin,Advil

COX Immunology/Inflammation; Neuroscience
Ibuprofen (Advil) 是一种丙酸衍生物和非甾体抗炎药 (NSAID),具有抗炎、镇痛和解热作用。它是COX-1和COX-2的抑制剂,IC50值分别为 13 和 370 μM,导致前列腺素和血栓素前体的形成减少。
T14975 CJ-42794

CJ-042794

Others Others
CJ-42794 (CJ-042794)是前列腺素受体 EP4的选择性拮抗剂, 抑制[3H]-PGE2与 EP4受体结合的平均 pKi 为8.5, 对 EP4选择性比 EP1, EP2和 EP3高200多倍。
T1552 Itopride hydrochloride

盐酸伊托必利,HSR803,盐酸依托必利,Ganaton

Dopamine Receptor; AChE GPCR/G Protein; Neuroscience
Itopride hydrochloride (Ganaton) 是一种促胃动力的 Benzamide 衍生物,是一种乙酰胆碱酯酶 (AChE) 和多巴胺受体 D2 (D2DR) 抑制剂。
T0674 Lansoprazole

兰索拉唑,A-65006,AG-1749

Proton pump; Phospholipase; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Lansoprazole (A-65006) 是一种可抑制胃酸生成的质子泵抑制剂。它是中性鞘磷脂酶的外泌体抑制剂。
T0498 Salsalate

Disalicylic acid,Salicylsalicylic acid,Sasapyrine,NSC-49171,双水杨酸酯

Reactive Oxygen Species; COX Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Salsalate (Sasapyrine) 是一种有效的抗风湿药物,是一种非乙酰化水杨酸盐,可以绕过胃的吸收,也可以避免环氧合酶的抑制。它具有抗炎活性,降低血糖水平、胰岛素抵抗和细胞因子表达,可用于研究 2 型糖尿病。
T8388 Vonoprazan

TAK-438 (free base),沃诺拉赞

Proton pump Membrane transporter/Ion channel
Vonoprazan (TAK-438 (free base)) 是一种质子泵抑制剂,是口服活性钾竞争性酸阻断剂,有抗分泌作用。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50值为 19 nM。它可用于研究胃酸相关疾病。
T8505 SC-236

4-(5-(4-氯苯基)-3-(三氟甲基)-1H-,Sc 236

Apoptosis; COX; PPAR Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience
SC-236 (Sc 236) 是一种具有口服活性的COX-2特异性抑制剂和PPARγ激动剂。它可通过 c-Jun 氨基端抑制激活蛋白-1活性,在小鼠模型中通过抑制 ERK 的磷酸化发挥抗炎作用。
T19763 Cetraxate hydrochloride

DV-1006,DV 1006,Cetraxate HCl,盐酸西曲酸酯,DV1006

Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism
Cetraxate hydrochloride (DV10062) 是一种有效的顶体蛋白酶 (acrosomal proteinase acrosin) 抑制剂,Ki 和 IC50分别为 0.94 μM 和 3.3 μM。它是一种口服有活性的抗溃疡试剂 (anti-ulcer),具有粘膜保护作用,可用于研究胃溃疡。
T21254 Vonoprazan Fumarate

TAK-438,TAK 438,Vonoprazan Fumurate,TAK438,富马酸沃诺拉赞

Proton pump Membrane transporter/Ion channel
Vonoprazan Fumarate (TAK438) 是质子泵的有效抑制剂,是口服有效的高效钾竞争性酸阻断剂,具有抗分泌活性。在 pH 为 6.5 时,它抑制猪胃微粒体中的 H+,K+-ATPase 酶活性,IC50为 19 nM。它被开发用于研究酸相关疾病,如消化性溃疡和胃食管反流病。
T37588 GIP (1-30) amide, porcine

This GIP fragment has potent insulinotropic activity in the isolated, perfused rat pancreas but greatly reduced somatostatinotropic activity in the isolated perfused rat stomach. The site responsible for insulinotropic activity apparently lies between residues 19 and 30 of GIP.
T6566 Levobupivacaine hydrochloride

Levobupivacaine HCl,(S)-(-)-Bupivacaine HCl,盐酸左布比卡因,(S)-(-)-Bupivacaine monohydrochloride

Sodium Channel Membrane transporter/Ion channel
Levobupivacaine hydrochloride ((S)-(-)-Bupivacaine monohydrochloride) 是有效的钠通道阻滞剂。
T7615 Xenopsin

爪蟾肽,Xenopsin(2TFA)

Others Others
Xenopsin (Xenopsin(2TFA)) 是一种神经降压素样八肽,来自于非洲爪蟾皮肤,能够抑制胃泌素刺激的胃酸分泌。

化合物

Gastric mucin
Cat.No: TP1309
Synonym:
Target: Antibacterial, Antibiotic
Acetyl Gastric Inhibitory Peptide (human) TFA
Cat.No: T78543
Synonym: Human N-acetyl GIP TFA
Target:
Gastric Inhibitory Peptide, porcine
Cat.No: T76309
Synonym:
Target:
GIP (3-42), human
Cat.No: T37589
Synonym: Gastric Inhibitory Polypeptide (3-42) (human)
Target: IGF-1R
Acetyl Gastric Inhibitory Peptide (human)
Cat.No: T76310
Synonym:
Target:
Gastric Inhibitory Polypeptide (1-30), porcine
Cat.No: T76308
Synonym:
Target:
Tegoprazan
Cat.No: T17030
Synonym:
Target: ATPase, Proton pump
[Tyr0] Gastric Inhibitory Peptide (23-42), human
Cat.No: T76307
Synonym:
Target:
Gastric Inhibitory Peptide (1-42) (porcine) TFA
Cat.No: T83694
Synonym: GIP (1-42),Glucose-dependent Insulinotropic Polypeptide (1-42)
Target:
Gastric Inhibitory Peptide (22-51) (human) TFA
Cat.No: T83710
Synonym: GIP (22-51),Glucose-dependent Insulinotropic Peptide (22-51)
Target:
Gastric Inhibitory Polypeptide (6-30) amide (human)
Cat.No: T82332
Synonym:
Target:
Pentagastrin
Cat.No: T4579
Synonym: 五肽胃泌素,ICI-50123
Target: Others, cholecystokinin
Linaprazan glurate
Cat.No: T38612
Synonym:
Target: Others
Gastric Inhibitory Peptide 1 (3-42) (human) TFA
Cat.No: T83696
Synonym: Glucose-dependent Insulinotropic Polypeptide 3-42,GIP-1 (3-42)
Target:
Dimaprit dihydrochloride
Cat.No: T22724
Synonym:
Target: NOS, NO Synthase, Histamine Receptor
Anisotropine Methylbromide
Cat.No: T4981
Synonym:
Target: Prostaglandin Receptor, AChR
HPi1
Cat.No: T15500
Synonym:
Target: Others, Antibacterial
Troxipide
Cat.No: T6710
Synonym: 曲昔派特,曲昔匹特,Aplace
Target: Others
Levobupivacaine
Cat.No: T1787
Synonym:
Target: Sodium Channel
Ramucirumab
Cat.No: T9929
Synonym:
Target: VEGFR
Acotiamide monohydrochloride trihydrate
Cat.No: T2319
Synonym: Acotiamide hydrochloride,YM-443 HCl,盐酸阿考替胺,Z-338 HCl
Target: AChE
PF-04217903
Cat.No: T2676
Synonym:
Target: c-Met/HGFR
Betazole dihydrochloride
Cat.No: T8599
Synonym: 盐酸倍他唑,Betazole hydrochloride
Target: Histamine Receptor
Metyrosine
Cat.No: T22368
Synonym: 甲酪氨酸,α-Methyltyrosine
Target: COX
Ilaprazole
Cat.No: T1756L
Synonym: IY81149,艾普拉唑,IY 81149,IY-81149
Target: Proton pump, TOPK
Tenatoprazole
Cat.No: T6700
Synonym: 泰妥拉唑,TU-199
Target: Proton pump
Ranitidine Hydrochloride
Cat.No: T0865
Synonym: AH19065,盐酸雷尼替丁
Target: P450, Antibacterial, Histamine Receptor
Ibuprofen Lysine
Cat.No: T6540
Synonym: 布洛芬赖氨酸盐,Neoprofen
Target: COX
Proglumide
Cat.No: T1052
Synonym: 二丙谷酰胺
Target: cholecystokinin
Lafutidine
Cat.No: T0081
Synonym: 拉呋替丁,FRG-8813
Target: 5-HT Receptor, Histamine Receptor
Ranitidine
Cat.No: T3610
Synonym: 雷尼替丁,HSDB 3925,Ranitidin
Target: P450, Antibacterial, Histamine Receptor
Rebamipide
Cat.No: T1562
Synonym: Proamipide,OPC12759,瑞巴派特
Target: Free radical scavengers, COX, Prostaglandin Receptor
Ilaprazole sodium
Cat.No: T1756
Synonym: IY-81149 sodium,艾普拉唑钠
Target: Proton pump, TOPK
Roxatidine Acetate hydrochloride
Cat.No: T0157
Synonym: HOE 760,盐酸罗沙替丁醋酸酯,Roxatidine Acetate HCl
Target: Histamine Receptor
(E/Z)-BCI
Cat.No: T11139
Synonym: NSC 150117
Target: Apoptosis, Phosphatase
LCH-7749944
Cat.No: T11826
Synonym: GNF-PF-2356
Target: Apoptosis, PAK
Neratinib
Cat.No: T2325
Synonym: HKI-272,来那替尼
Target: EGFR, HER
Orlistat
Cat.No: T0686
Synonym: Ro-18-0647,奥利司他,Tetrahydrolipstatin
Target: Apoptosis, Others, Fatty Acid Synthase
Ibuprofen
Cat.No: T1394
Synonym: Brufen,(±)-Ibuprofe,布洛芬,Motrin,Advil
Target: COX
CJ-42794
Cat.No: T14975
Synonym: CJ-042794
Target: Others
Itopride hydrochloride
Cat.No: T1552
Synonym: 盐酸伊托必利,HSR803,盐酸依托必利,Ganaton
Target: Dopamine Receptor, AChE
Lansoprazole
Cat.No: T0674
Synonym: 兰索拉唑,A-65006,AG-1749
Target: Proton pump, Phospholipase, Antibacterial
Salsalate
Cat.No: T0498
Synonym: Disalicylic acid,Salicylsalicylic acid,Sasapyrine,NSC-49171,双水杨酸酯
Target: Reactive Oxygen Species, COX
Vonoprazan
Cat.No: T8388
Synonym: TAK-438 (free base),沃诺拉赞
Target: Proton pump
SC-236
Cat.No: T8505
Synonym: 4-(5-(4-氯苯基)-3-(三氟甲基)-1H-,Sc 236
Target: Apoptosis, COX, PPAR
Cetraxate hydrochloride
Cat.No: T19763
Synonym: DV-1006,DV 1006,Cetraxate HCl,盐酸西曲酸酯,DV1006
Target: Serine/threonin kinase
Vonoprazan Fumarate
Cat.No: T21254
Synonym: TAK-438,TAK 438,Vonoprazan Fumurate,TAK438,富马酸沃诺拉赞
Target: Proton pump
GIP (1-30) amide, porcine
Cat.No: T37588
Synonym:
Target:
Levobupivacaine hydrochloride
Cat.No: T6566
Synonym: Levobupivacaine HCl,(S)-(-)-Bupivacaine HCl,盐酸左布比卡因,(S)-(-)-Bupivacaine monohydrochloride
Target: Sodium Channel
Xenopsin
Cat.No: T7615
Synonym: 爪蟾肽,Xenopsin(2TFA)
Target: Others
Cat. No. Product Name Target Signaling Pathways
T5043 Lentinan

Others Others
Lentinan 是一种 β-葡聚糖,从香菇中提取获得。它在日本已被批准用作胃癌的生物反应调节剂。
T3862 Irigenin

NF-κB; Integrin Cytoskeletal Signaling; NF-κB
Irigenin 可通过特异性和选择性地阻断 Extra Domain A 域的 C-C 环上α9β1和α4β1整合素结合位点,介导其抗转移作用。可通过增强胃癌细胞中促凋亡分子的表达来敏化 TRAIL 诱导的凋亡,具有抗癌作用。
T4034 Solamargine

Solamargin,δ-Solanigrine,澳洲茄边碱

Apoptosis; p38 MAPK; P-gp; STAT Apoptosis; JAK/STAT signaling; MAPK; Membrane transporter/Ion channel; Neuroscience; Stem Cells
Solamargine (δ-Solanigrine) 是一种来源于茄属植物的类固醇 Solasodine 的衍生物,诱导非选择性细胞毒性和 P-gp 抑制作用。它通过下调 MMP-2 和 MMP-9 的表达和活性来显著抑制 HepG2 细胞的迁移和侵袭,在多种癌症中均表现出抗癌活性。
T5S2360 Corydaline

Corydalin,紫堇碱,延胡索甲素,(+)-Corydaline

P450; Virus Protease; Opioid Receptor; AChE Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Corydaline (Corydalin) 是从 Corydalis yanhusuo 提取的一种异喹啉生物碱,是一种新型促动力植物药的主要活性成分之一。它促进胃排空和小肠转运,促进胃的调节,具有抗乙酰胆碱酯酶、抗过敏和镇痛活性。
T3S0509 Gaultherin

COX Immunology/Inflammation; Neuroscience
Gaultherin 是一种分离自 Gaultheria yunnanensis 中的天然水杨酸酯衍生物。它是一种非甾体类抗炎药,具有止痛和抗炎作用,与 Aspirin 相比没有胃溃疡作用。
TN2078 Pinocembrin chalcone

2',4',6'-Trihydroxychalcone,Pinocembrinchalcone

Calcium Channel; Tyrosinase; Antibacterial; Antifection Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Proteases/Proteasome
Pinocembrin chalcone 是一种具有抗诱变作用的酪氨酸酶抑制剂。 Pinocembrin 查尔酮可用于预防胃溃疡的研究。
T4S1881 Aconine

乌头原碱,Jesaconine

Others; NF-κB NF-κB; Others
Aconine (Jesaconine) 是一种退热药,有胃麻醉作用,能够抑制核因子 κB 受体活化剂配体诱导的 NF-κB 激活。
TN6577 Bletilloside A

3-Methoxyshancigusin I

Others Others
Bletilloside A(3-Methoxyshancigusin I) 是从条纹苜蓿的块茎中分离出一种新型葡萄糖苷,具有抗胃溃疡活性。
TC0039 Vasicinone

Others Others
Vasicinone 是一种喹唑啉类生物碱,分离自凡士林植物中。它是具有研究帕金森病和其他氧化应激相关神经退行性疾病的潜力。
T0743 DL-Carnitine

Carnitina,Carnitine,卡尼丁

Others Others
DL-Carnitine (Carnitina) 是肝脏和横纹肌的成分。在治疗上它用于刺激胰腺和胃的分泌并治疗高脂蛋白血症。
T2203 D-Carnitine hydrochloride

(S)-Carnitine Hydrochloride,L-Carnitine hydrochloride

Others; Endogenous Metabolite Metabolism; Others
D-Carnitine hydrochloride ((S)-Carnitine Hydrochloride) 已被用于研究麦角硫因素转运蛋白 SLC22A4 和肉毒碱转运蛋白 SLC22A5,也被用于使棕榈酸进入线粒体。
T2S1975 Ponicidin

冬凌草乙素,Rubescensine B

Apoptosis; JAK; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
Ponicidin (Rubescensine B) 是来源于冬凌草的一种二萜,具有免疫调节、抗炎、抗病毒和抗癌作用。它可诱导胃癌细胞凋亡,降低 JAK2 和 STAT3 的磷酸化水平。
T21651 Lansoprazole sodium

兰索拉唑钠,Lansoprazole (sodium), AG-1749 sodium

Proton pump; Phospholipase; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Lansoprazole sodium (Lansoprazole (sodium)) 是一种质子泵抑制剂,是中性鞘磷脂酶的外泌体抑制剂,能抑制胃酸生成。
T5S1389 Escin IB

七叶皂苷B,七叶皂苷 IB

5-HT Receptor; NO Synthase GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escin IB 是一种皂苷,分离自马栗子种子的皮和胚乳中,能够抑制 pancreatic lipase 的活性。
T20604L Litorin acetate(55749-97-8 Free base)

Bombesin Receptor GPCR/G Protein
Litorin acetate 是一种两栖类铃蟾肽衍生物,是一种铃蟾肽受体激动剂。它刺激平滑肌收缩,刺激胃泌素、胃酸和胰腺分泌,抑制体内营养。
TN1560 Dehydroeffusol

去氢厄弗酚,5-Ethenyl-1-Methylphenanthrene-2,7-Diol,Dehydro Effusol

MMP; ERK; GPR; Others Endocrinology/Hormones; GPCR/G Protein; MAPK; Others; Proteases/Proteasome
Dehydroeffusol (Dehydro Effusol) 通过选择性诱导肿瘤抑制性内质网应激和中度细胞凋亡来抑制胃癌细胞生长和致瘤性,具有抗癌、抗焦虑和镇静作用。
TN1103 Diphyllin

山荷叶素,二叶草素

ATPase; Proton pump; Influenza Virus; HIV Protease Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Diphyllin 是一种从Justicia procumbens 中分离的芳基萘木脂素,是HIV-1的有效抑制剂,IC50 为 0.38 μM。它是V-ATPase 抑制剂,IC50值为 17 nM,可抑制人破骨细胞中的溶酶体酸化。它抑制NO 产生,IC50值为 50 μM ,具有抗癌和抗炎活性。
T0965 Histamine

Ergamine,组胺

5-HT Receptor; Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine (Ergamine) 是通过组胺的酶促脱羧衍生的胺。它是一种强大的胃分泌兴奋剂、支气管平滑肌的收缩剂、血管扩张剂以及中枢作用的神经递质。
T6S2038 Ziyuglycoside II

Apoptosis; Antioxidant; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Ziyuglycoside II 是从地榆中提取的一种三萜皂苷,可诱导活性氧 产生和凋亡,具有抗炎和抗癌作用。
T37152 3-Methyl-2-cyclopenten-1-one

Endogenous Metabolite Metabolism
3-Methyl-2-cyclopenten-1-one 可作为食品添加剂,在 2-5 ppm 下可改善肉类和肉制品的风味。添加3-Methyl-2-cyclopenten-1-one 在对雄性Wistar 大鼠口服给药时显示出胃细胞保护活性。
T6S1302 Carnosol

Nrf2; Endogenous Metabolite; S6 Kinase Immunology/Inflammation; MAPK; Metabolism; PI3K/Akt/mTOR signaling
Carnosol 是 Nrf2激活剂,增加 Nrf2 的水平以及能促进血红素氧合酶 1(HMOX1) 表达。它是核糖体 S6激酶(RSK2)抑制剂,可用于胃癌相关研究,IC50值约为 5.5 μM。
T6534 Histamine dihydrochloride

组胺二盐酸盐,peremin,Ceplene,Histamine 2HCl

Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine dihydrochloride (Ceplene) 是 Histamine 的二盐酸形式。Histamine 是一种有机氮化合物,是一种强效的胃分泌兴奋剂,支气管平滑肌收缩剂,血管舒张剂,也是一种中枢作用的神经递质。
T3727 Methyl syringate

Syringic Acid Methyl Ester,丁香酸甲酯

TRP/TRPV Channel Membrane transporter/Ion channel
Methyl syringate (Syringic Acid Methyl Ester) 是水仙花蜜的化学标记物,是有效的细菌和真菌漆酶酚介质。它也是TRPA1激动剂。
T3S2312 Poncirin

枸橘苷,Isosakuranetin-7-neohesperidoside

Apoptosis; Others Apoptosis; Others
Poncirin (Isosakuranetin-7-neohesperidoside) 是从三叶草中分离出来的一种天然产物,具有抗炎活性。 它防止脂肪生成,增强间充质干细胞中的成骨细胞分化,增加骨矿物质密度,改善小梁微结构,可能反映 GIO 小鼠的骨形成增加和骨吸收减少。
T2A2532 L-Histidine

Glyoxaline-5-alanine,L-(-)-Histidine,L-组氨酸,histidine,组氨酸,L-Hisidine

Mitochondrial Metabolism; Endogenous Metabolite Metabolism
L-Histidine (L-(-)-Histidine) 是人类生长和组织修复所需的一种半必需氨基酸(儿童应从食物中获得)。 L-Histidine 是线粒体谷氨酰胺转运的抑制剂。
T40615 N,N'-Dimethylthiourea

N,N-二甲基硫脲,DMTU

Antioxidant oxidation-reduction
N,N'-Dimethylthiourea (DMTU) 是一种分离自黑蒜的化合物。N,N'-Dimethylthiourea 具有口服活性的羟基自由基 (•OH) 的清除剂,通过活化的中性粒细胞在体外阻止 •OH 的产生。N,N'-Dimethylthiourea 通过发挥 •OH 清除和抗炎作用,防止水浸限制应激诱导的大鼠胃粘膜损伤。
T4S0867 Pogostone

DHELWANGIN,广藿香酮

Apoptosis; Antibacterial; Autophagy Apoptosis; Autophagy; Microbiology/Virology
Pogostone (DHELWANGIN) 是从薄荷中分离出,对革兰氏阴性菌、革兰氏阳性菌、大肠埃希菌等具有强效抗菌、抗真菌活性。它诱导细胞凋亡和自噬。
T0962 L-Hyoscyamine

Daturine,Hyoscyamine,L-莨菪碱,L-天仙子胺

AChR Neuroscience
L-Hyoscyamine (Daturine) 是从山莨菪中提取的一种托烷生物碱,是竞争性的毒蕈碱受体拮抗剂。它是 Atropine 的左旋异构体。
TN2601 12-O-Methylcarnosic acid

Reductase Endocrinology/Hormones; Metabolism
12-O-Methylcarnosic acid 是分离自小叶丹参的丙酮提取物的一种二萜肉桂酸,可抑制 5α-还原酶 (5α-reductase) 活性,IC50为 61.7 μM。它抑制 LNCaP 细胞的增殖。它具有抗微生物活性、抗氧化和抗癌活性。
T4S1619 L-Hyoscyamine sulfate

Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate,硫酸天仙子胺水合物,L-莨菪碱硫酸盐

AChR Neuroscience
L-Hyoscyamine sulfate (Levsin Sulfate) 是来自山莨菪的一种托烷生物碱,是竞争性的毒蕈碱受体拮抗剂。它是 Atropine 的左旋异构体。
T3S2344 β,β-Dimethylacrylshikonin

β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin

ERK; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; MAPK; Metabolism
β,β-Dimethylacrylshikonin (Dimethylacrylshikonin) 是一种萘醌衍生物,从 Arnebia nobilis 中提取得到。它利用 PI3K 通路诱导 eNOS、VEGF 和 HIF-1α 的表达,促进血管生成,具有抗肿瘤活性。
T3779 Crocin II

Crocin 2,西红花苷II,Crocetin gentiobiosylglucosyl ester,藏红花,Tricrocin,Crocin B

Caspase; COX; NO Synthase Apoptosis; Immunology/Inflammation; Neuroscience; Proteases/Proteasome
Crocin II (Crocetin gentiobiosylglucosyl ester) 是从栀子果实中分离出来的一种天然产物,具有抗氧化、抗癌和抗抑郁活性。它抑制 iNOS 和 COX-2的蛋白质和 m-RNA 的表达,还抑制NO 产生,IC50值为 31.1 μM。
T6S1684 8-Gingerol

Antioxidant; Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology; oxidation-reduction
8-Gingerol 分离自姜的根状茎,是口服有效的 TRPV1激活剂,EC50值为5.0 µM。8-Gingerol 抑制 COX-2,还能抑制体外 H. pylori 的生长。
T4S0797 Berberine

小檗碱,Berberin,Umbellatine,黄连素

Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic; Autophagy Autophagy; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Berberine (Umbellatine) 是从中草药黄连中分离出来的一种生物碱抗生素。它诱导活性氧生成并抑制 DNA 拓扑异构酶,具有抗肿瘤特性。
TN4932 Sageone

PARP; Akt; Caspase; Antifection Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Sageone represents a promising anticancer agent against gastric cancer that warrants further study, it synergizes with cisplatin cytotoxicity in SNU-1 human gastric cancer cells.Sageone also shows antiviral activity.
T20604 Litorin

Litorin, an amphibian bombesin peptide derivative, is found to suppress the nutriment, to stimulate the contraction of smooth muscle, to stimulate gastrin, gastric acid, and pancreatic secretion.
TN4465 Luvangetin

COX; Prostaglandin Receptor; Antifection GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Luvangetin may have anti-inflammatory activity, it can inhibit NO and PGE2 production in LPS-stimulated BV2 cells. Luvangetin shows significant protection against pylorus-ligated and aspirin-induced gastric ulcers in rats and cold restraint stress-induced
TN3605 Casegravol

Others Others
Casegravol shows antiproliferative activity against human gastric adenocarcinoma (MK-1), human uterus carcinoma (HeLa), and murine melanoma (B16F10) cells.
TN3740 Cyclocommunol

PAFR GPCR/G Protein
Cyclocommunol exhibits cytotoxicity against hepatocellular carcinoma (SMMC-7721) and gastric carcinoma (BGC-823 and SGC-7901) cell lines. It also shows strong inhibition of arachidonic acid (AA)- and collagen-induced platelet aggregation.
TN3852 Dihydrolicoisoflavone

Antifection Microbiology/Virology
Dihydrolicoisoflavone A possesses weaker anti-H. pylori activity, it may be useful chemopreventive agents for peptic ulcer or gastric cancer in H. pylori-infected individuals.
TN1810 Jatropholone B

Others Others
Jatropholone B shows antiproliferative activity against cancer cell lines. It also has gastroprotective activity in preventing the gastric lesions in mice.
TN1302 6,8-Diprenylorobol

6,8-二异戊烯基香豌豆苷元

Others; HIV Protease; Antifection Microbiology/Virology; Others; Proteases/Proteasome
6,8-Diprenylorobol possesses weaker anti-H. pylori activity, it may be a useful chemopreventive agent for peptic ulcer or gastric cancer in H. pylori-infected individuals.
TN4489 Manassantin A

ERK; cAMP; TNF; NF-κB; MAPK; COX; HIF; Prostaglandin Receptor; JNK; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; GPCR/G Protein; Immunology/Inflammation; JAK/STAT signaling; MAPK; Neuroscience; NF-κB; Stem Cells
Manassantin A is a high potent HIF-1 inhibitor, it protects the gastric mucosa from ethanol-induced acute gastric injury, and suggest that these protective effects might be associated with COX/PGE2 stimulation, inhibition of iNOS production and NF-κB act
TN3495 Benzyl ferulate

TNF; Antifection Apoptosis; Microbiology/Virology
Benzyl ferulate has antimicrobial activity. It also shows good anti-proliferative against three gastro-intestinal cancer cell lines(HCT-116 colon carcinoma, KYSE-30 oesophageal squamous cancer, and NCI-N87 gastric carcinoma).
TN3726 Cudraflavone B

IκB/IKK; MAO; ROS; Akt; COX; PI3K; Nrf2; Autophagy Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling
Cudraflavone B has anti-proliferative activity, mouse brain monoamine oxidase (MAO) inhibitory effects, apoptotic actions in human gastric carcinoma cells and mouse melanoma cells, and hepatoprotective activity. It may be a lead for the development of a potential candidate for human oral squamous cell carcinoma cells.
T83258 7(18)-Dehydroschisandro A

7(18)-Dehydroschisandro A (化合物2) 是从Schizandra chinensis Baill分离得到的木脂素,对激性胃溃疡显示出抑制效果。
TN6010 Picrasidine S

Picrasidine S shows the potent cytotoxicity against human HeLa cervical, gastric MKN-28, and mouse melanoma B-16 cancer cells, it also shows the potent antibacterial activity against two strains of pathogenic bacteria methicillin-resistant Staphylococcus
T83257 7(8)-Dehydroschisandrol A

7(8)-Dehydroschisandrol A (Compound 4a)为从Schizandra chinensis Baill分离的木脂素,对激性胃溃疡表现出较弱抑制效果。
T80702 α-Thevetin B

α-Thevetin B(Compound 24), 一种从Thevetia peruviana分离得到的心脏苷,用于肺癌、胃癌和胰腺癌的研究。
TN1913 Marmin

Calcium Channel; Antifection; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
Marmin have anti-ulcer effects, which are ascribed primarily to the maintenance of the mucosal barrier integrity and inhibition of gastric motor activity and secondarily due to the prevention of the effects of endogenous acetylcholine and histamine.
------------------------ 更多 ------------------------

天然产物

Lentinan
Cat.No: T5043
Synonym:
Target: Others
Irigenin
Cat.No: T3862
Synonym:
Target: NF-κB, Integrin
Solamargine
Cat.No: T4034
Synonym: Solamargin,δ-Solanigrine,澳洲茄边碱
Target: Apoptosis, p38 MAPK, P-gp, STAT
Corydaline
Cat.No: T5S2360
Synonym: Corydalin,紫堇碱,延胡索甲素,(+)-Corydaline
Target: P450, Virus Protease, Opioid Receptor, AChE
Gaultherin
Cat.No: T3S0509
Synonym:
Target: COX
Pinocembrin chalcone
Cat.No: TN2078
Synonym: 2',4',6'-Trihydroxychalcone,Pinocembrinchalcone
Target: Calcium Channel, Tyrosinase, Antibacterial, Antifection
Aconine
Cat.No: T4S1881
Synonym: 乌头原碱,Jesaconine
Target: Others, NF-κB
Bletilloside A
Cat.No: TN6577
Synonym: 3-Methoxyshancigusin I
Target: Others
Vasicinone
Cat.No: TC0039
Synonym:
Target: Others
DL-Carnitine
Cat.No: T0743
Synonym: Carnitina,Carnitine,卡尼丁
Target: Others
D-Carnitine hydrochloride
Cat.No: T2203
Synonym: (S)-Carnitine Hydrochloride,L-Carnitine hydrochloride
Target: Others, Endogenous Metabolite
Ponicidin
Cat.No: T2S1975
Synonym: 冬凌草乙素,Rubescensine B
Target: Apoptosis, JAK, STAT
Lansoprazole sodium
Cat.No: T21651
Synonym: 兰索拉唑钠,Lansoprazole (sodium), AG-1749 sodium
Target: Proton pump, Phospholipase, Antibacterial
Escin IB
Cat.No: T5S1389
Synonym: 七叶皂苷B,七叶皂苷 IB
Target: 5-HT Receptor, NO Synthase
Litorin acetate(55749-97-8 Free base)
Cat.No: T20604L
Synonym:
Target: Bombesin Receptor
Dehydroeffusol
Cat.No: TN1560
Synonym: 去氢厄弗酚,5-Ethenyl-1-Methylphenanthrene-2,7-Diol,Dehydro Effusol
Target: MMP, ERK, GPR, Others
Diphyllin
Cat.No: TN1103
Synonym: 山荷叶素,二叶草素
Target: ATPase, Proton pump, Influenza Virus, HIV Protease
Histamine
Cat.No: T0965
Synonym: Ergamine,组胺
Target: 5-HT Receptor, Endogenous Metabolite, Histamine Receptor
Ziyuglycoside II
Cat.No: T6S2038
Synonym:
Target: Apoptosis, Antioxidant, Reactive Oxygen Species
3-Methyl-2-cyclopenten-1-one
Cat.No: T37152
Synonym:
Target: Endogenous Metabolite
Carnosol
Cat.No: T6S1302
Synonym:
Target: Nrf2, Endogenous Metabolite, S6 Kinase
Histamine dihydrochloride
Cat.No: T6534
Synonym: 组胺二盐酸盐,peremin,Ceplene,Histamine 2HCl
Target: Endogenous Metabolite, Histamine Receptor
Methyl syringate
Cat.No: T3727
Synonym: Syringic Acid Methyl Ester,丁香酸甲酯
Target: TRP/TRPV Channel
Poncirin
Cat.No: T3S2312
Synonym: 枸橘苷,Isosakuranetin-7-neohesperidoside
Target: Apoptosis, Others
L-Histidine
Cat.No: T2A2532
Synonym: Glyoxaline-5-alanine,L-(-)-Histidine,L-组氨酸,histidine,组氨酸,L-Hisidine
Target: Mitochondrial Metabolism, Endogenous Metabolite
N,N'-Dimethylthiourea
Cat.No: T40615
Synonym: N,N-二甲基硫脲,DMTU
Target: Antioxidant
Pogostone
Cat.No: T4S0867
Synonym: DHELWANGIN,广藿香酮
Target: Apoptosis, Antibacterial, Autophagy
L-Hyoscyamine
Cat.No: T0962
Synonym: Daturine,Hyoscyamine,L-莨菪碱,L-天仙子胺
Target: AChR
12-O-Methylcarnosic acid
Cat.No: TN2601
Synonym:
Target: Reductase
L-Hyoscyamine sulfate
Cat.No: T4S1619
Synonym: Hyoscyamine sulfate hydrate,Levsin Sulfate,Hyoscyamine Sulphate,硫酸天仙子胺水合物,L-莨菪碱硫酸盐
Target: AChR
β,β-Dimethylacrylshikonin
Cat.No: T3S2344
Synonym: β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin
Target: ERK, HIF/HIF Prolyl-Hydroxylase
Crocin II
Cat.No: T3779
Synonym: Crocin 2,西红花苷II,Crocetin gentiobiosylglucosyl ester,藏红花,Tricrocin,Crocin B
Target: Caspase, COX, NO Synthase
8-Gingerol
Cat.No: T6S1684
Synonym:
Target: Antioxidant, Antibacterial, TRP/TRPV Channel
Berberine
Cat.No: T4S0797
Synonym: 小檗碱,Berberin,Umbellatine,黄连素
Target: Reactive Oxygen Species, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic, Autophagy
Sageone
Cat.No: TN4932
Synonym:
Target: PARP, Akt, Caspase, Antifection
Litorin
Cat.No: T20604
Synonym:
Target:
Luvangetin
Cat.No: TN4465
Synonym:
Target: COX, Prostaglandin Receptor, Antifection
Casegravol
Cat.No: TN3605
Synonym:
Target: Others
Cyclocommunol
Cat.No: TN3740
Synonym:
Target: PAFR
Dihydrolicoisoflavone
Cat.No: TN3852
Synonym:
Target: Antifection
Jatropholone B
Cat.No: TN1810
Synonym:
Target: Others
6,8-Diprenylorobol
Cat.No: TN1302
Synonym: 6,8-二异戊烯基香豌豆苷元
Target: Others, HIV Protease, Antifection
Manassantin A
Cat.No: TN4489
Synonym:
Target: ERK, cAMP, TNF, NF-κB, MAPK, COX, HIF, Prostaglandin Receptor, JNK, STAT
Benzyl ferulate
Cat.No: TN3495
Synonym:
Target: TNF, Antifection
Cudraflavone B
Cat.No: TN3726
Synonym:
Target: IκB/IKK, MAO, ROS, Akt, COX, PI3K, Nrf2, Autophagy
7(18)-Dehydroschisandro A
Cat.No: T83258
Synonym:
Target:
Picrasidine S
Cat.No: TN6010
Synonym:
Target:
7(8)-Dehydroschisandrol A
Cat.No: T83257
Synonym:
Target:
α-Thevetin B
Cat.No: T80702
Synonym:
Target:
Marmin
Cat.No: TN1913
Synonym:
Target: Calcium Channel, Antifection, Histamine Receptor
--------- 更多 ---------
共302条,每页50条 1 2 3 4 5 6 7
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼