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895

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T0850 Primaquine diphosphate

Primaquine phosphate,磷酸伯氨喹,Primaquine bisphosphate,磷酸伯安喹

Antibiotic; Parasite Microbiology/Virology
Primaquine diphosphate 是一种合成的 8-氨基喹啉衍生物,具有抗疟特性。它是一种能破坏间日疟原虫和卵形疟原虫肝脏晚期和潜在组织形态的化合物。
T0462 Cilostazol

西洛他唑,OPC 21,OPC 13013

PDE; Autophagy Autophagy; Metabolism
Cilostazol (OPC 21) 是一种选择性的心血管系统中磷酸二酯酶 3 亚型PDE 3A 的抑制剂,IC50值为 0.2 μM。
T0425 Pefloxacin Mesylate

Pefloxacinium mesylate,甲磺酸培氟沙星

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate (Pefloxacinium mesylate) 是一种抗菌化合物,可抑制DNA 旋转酶阻断DNA 复制。
T7212 Delavirdine mesylate

U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate)

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Delavirdine mesylate (BHAP-U 90152(mesylate)) 是一种口服活性非核苷逆转录酶抑制剂。它抑制 HIV-1 病毒复制,可以用于艾滋病的相关研究。它选择性地抑制 HIV-1 逆转录酶,其选择性超过 DNA 聚合酶 α 和 DNA 聚合酶 δ 。
T3335 Darunavir Ethanolate

地瑞那韦乙醇盐,UIC 94017,Darunavir Ethanolate,TMC114,达芦那韦乙醇

HIV Protease Microbiology/Virology; Proteases/Proteasome
Darunavir Ethanolate (UIC 94017) 是一种HIV 蛋白酶抑制剂,可以用于 HIV/AIDS 的相关研究。对野生型 HIV-1 蛋白酶的Ki 值为1 nM。
T2589 Dolasetron Mesylate hydrate

Dalasetron Mesylate Hydrate,多拉司琼甲磺酸盐一水合物

5-HT Receptor GPCR/G Protein; Neuroscience
Dolasetron Mesylate hydrate (Dalasetron Mesylate Hydrate) 是一种选择性血清素受体拮抗剂,可竞争性阻断血清素对 5HT3 受体的作用,从而抑制化疗和放疗引起的恶心和呕吐。
T0225 Pizotifen Malate

Pizotyline (malate),BC-105 (malate),BC-105,苯噻啶苹果酸盐

5-HT Receptor GPCR/G Protein; Neuroscience
Pizotifen Malate (BC-105 malate) 是5-HT2受体的拮抗剂,对5-HT1C 有高亲和力。
T2226 Pergolide mesylate

甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Pergolide mesylate salt(LY127809) 是一种有效的,具有口服活性的多巴胺 D1和 D2受体激动剂,是一种 Ergoline 衍生物,可用于帕金森氏病和高泌乳素血症的研究。
T8541 Lenvatinib mesylate

仑伐替尼甲酸盐,E7080 (mesylate),乐伐替尼

VEGFR; FGFR; c-RET; PDGFR; c-Kit Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Lenvatinib mesylate (E7080 (mesylate)) 是一种口服具有活力的,多靶点酪氨酸激酶抑制剂,能够抑制血管内皮生长因子受体(VEGFR1-3),成纤维细胞生长因子受体(FGFR1-4),干细胞因子受体(KIT),血小板衍生生长因子受体(PDGFR),转染期间重排(RET),具有效抗癌作用。
T77705 Diethyl 2,4-dimethylpyrrole-3,5-dicarboxylate

Diethyl 3,5-dimethyl-1H-pyrrole-2,4-dicarboxylate

Others Others
Diethyl 2,4-dimethylpyrrole-3,5-dicarboxylate 是一种生化试剂,可用于研究生化反应。
T0535 Memantine Related Compound B

美金刚杂质B,3,5-Dimethyl-1-adamantanol

Others Others
Memantine Related Compound B (3,5-Dimethyl-1-adamantanol) 是Memantine 的杂质。
T7593 Levomefolate calcium

左旋甲状腺素钙,L-5-甲基四氢叶酸钙

Antifolate Cell Cycle/Checkpoint
Levomefolate calcium 是一种人工形式的叶酸。它是叶酸的一种辅酶形式,是膳食补充剂中生物利用度更高的替代品。
T11558 Hexyl gallate

没食子酸己酯,Gallic acid hexyl ester,Hexyl 3,4,5-trihydroxybenzoate

Antibacterial Microbiology/Virology
Hexyl gallate (Gallic acid hexyl ester) 是没食子酸的烷基酯衍生物,对恶性疟原虫具有很强的抗疟活性,IC50为 0.11 mM。它具有抗菌活性,通过抑制 RhlR 抑制鼠李糖脂和绿脓杆菌素的产生。
T6963 Reboxetine mesylate

瑞波西汀甲磺酸盐,FCE20124 mesylate,Edronax,PNU155950E mesylate,PNU 155950E,甲磺酸瑞波西汀

Adrenergic Receptor; Norepinephrine GPCR/G Protein; Neuroscience
Reboxetine mesylate (FCE20124 mesylate) 是一种高效、选择性的,特异性的去甲肾上腺素再摄取抑制剂(NARI),能够抑制去甲肾上腺素再摄取(Ki=8 nM),可用于抑郁症的研究。
T0794 Mepenzolate Bromide

Colibantil,Cantil,溴美喷酯,Cantilaque

AChR Neuroscience
Mepenzolate Bromide (Colibantil) 是一种可口服的毒蕈碱受体拮抗剂,对hM2R 和hM3R 的Ki 分别为 0.68 和 2.6 nM。它是GPR109A 抑制剂,可用于抑制与肠易激综合征相关的胃肠道过度运动。
T7386 Bretylium tosylate

溴苄乙胺,托西溴苄铵

Others Others
Bretylium tosylate 是交感神经和肾上腺素神经的阻断剂,是血管收缩的神经递质突触前释放的抑制剂。
TP1945L1 Pep2m, myristoylated acetate

Pep2m, myristoylated acetate(1423381-07-0 free base)

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Pep2m, myristoylated acetate(1423381-07-0 free base) 是一种细胞可渗透的肉豆蔻酰化形式的 pep2m。 GluA2(AMPA 受体)亚基的 C 末端与 N-乙基马来酰亚胺敏感融合蛋白 (NSF)(一种调节 AMPA 受体功能的蛋白质)之间相互作用的肽抑制剂。降低 CA1 神经元中的突触后电流、培养的海马神经元中 AMPA 介导的电流和 AMPA 受体表面表达。
TP2137L pp60 c-src (521-533) (phosphorylated) acetate

Others Others
pp60 c-src (521-533) (phosphorylated) acetate 是粘着斑形成和细胞扩散的调节剂。它还调节细胞运动,是由促运动透明质酸受体 RHAMM 触发的信号通路中的关键成分。
T10432L AZD-8529 mesylate

GluR Neuroscience
AZD-8529 mesylate 是高度选择性的可口服mGluR2正向调节剂,EC50值为 285 nM。它在 20-25 M 时,对 mGluR1、3、4、5、6、7 和 8 亚型没有显示正变构调节剂反应。
T23453 Tetrindole mesylate

MAO Metabolism; Neuroscience
Tetrindole mesylate 是一种 MAO-A 抑制剂。
T1492 Gemifloxacin mesylate

LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate

DNA gyrase; Topoisomerase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
Gemifloxacin mesylate (Gemifloxacin mesylate) 是一种喹诺酮类口服广谱抗菌剂,可研究轻中度肺炎和慢性支气管炎的急性细菌性发作。
T0547 FlutaMide Related CoMpound B

Others Others
FlutaMide Related CoMpound B 用作医药中间体。
T40122 L-Histidine benzyl ester bistosylate

Others Others
L-Histidine benzyl ester bistosylate may serve as an activator for HutP, an RNA-binding protein.
T3086 Mesoridazine Besylate

Mesoridazine benzenesulfonate,Serentil,苯磺酸美索达嗪

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Mesoridazine Besylate (Serentil) 是一种哌啶类精神安定药,属于称为吩噻嗪类的药物,用于治疗精神分裂症。它是硫利达嗪的代谢物。
T22313 Dolasetron Mesylate

多拉司琼甲磺酸盐,甲磺酸多拉司琼,Anzemet hydrate,MDL-73147EF

Others; 5-HT Receptor GPCR/G Protein; Neuroscience; Others
Dolasetron Mesylate (MDL-73147EF) 是 5-HT3 受体的拮抗剂,可用于治疗化疗后呕吐和恶心的研究。
T9154 Sodium taurodeoxycholate hydrate

牛磺去氧胆酸钠,Taurodeoxycholic acid sodium salt monohydrate

Others Others
Sodium taurodeoxycholate hydrate (Taurodeoxycholic acid sodium salt monohydrate) 已用于一项研究,以评估亚胶束浓度的胆汁盐对脂质双层膜的影响。
TQ0041 Ningetinib Tosylate

VEGFR; c-Met/HGFR; TAM Receptor Angiogenesis; Tyrosine Kinase/Adaptors
Ningetinib Tosylate 是口服具有活力的、小分子酪氨酸激酶抑制剂,能够抑制 c-Met (IC50:6.7 nM),VEGFR2 (IC50:1.9 nM) 和 Axl (IC50<1.0 nM)。
T7026L Kukoamine B mesylate

Antioxidant oxidation-reduction
Kukoamine B mesylate 是从地骨皮中提取得到的新型阳离子生物碱,具有抗氧化活性,抑制 Kupffer 和 RAW 264。7 细胞中的 LPS 内化,可用于研究急性炎症和糖尿病。
T5988 Dimethyl biphenyl-4,4'-dicarboxylate

Biphenyl dimethyl dicarboxylate,联苯二甲酸二甲酯

Others Others
Dimethyl biphenyl-4,4'-dicarboxylate (Biphenyl dimethyl dicarboxylate) 是一种保肝剂,提取自五味子中,能够诱导 IFN 相关的信号转导。
T2429 Olverembatinib dimesylate

GZD824 Dimesylate,HQP1351

Bcr-Abl Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
Olverembatinib dimesylate (GZD824 Dimesylate) 是一种高效的、口服具有活性的pan-Bcr-Abl 抑制剂,具有抗肿瘤活性。它能广泛而有效地抑制突变型 Bcr-Abl。它对天然的 Bcr-Abl 和 Bcr-AblT315I 作用的IC50值分别为 0.34 nM 和 0.68 nM。
T9497 Niraparib tosylate monohyrate

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
Niraparib tosylate monohyrate 也称为 MK-4827,是一种聚 (ADP-核糖) 聚合酶 (PARP) 抑制剂,具有潜在的抗肿瘤活性。 MK4827 抑制 PARP 活性,增强 DNA 链断裂的积累,促进基因组不稳定性和细胞凋亡。 PARP 蛋白家族通过碱基切除修复 (BER) 途径检测和修复单链 DNA 断裂。
T50107 ethyl 2-[3,5-bis(trifluoromethyl)phenyl]-3-oxo-2,3-dihydro-1H-pyrazole-4-carboxylate

Others Others
ethyl 2-[3,5-bis(trifluoromethyl)phenyl]-3-oxo-2,3-dihydro-1H-pyrazole-4-carboxylate 是一种合成化合物,属于姜黄素家族。它通过抑制NF-κB 信号通路参与免疫反应和炎症的调节,通过激活Nrf2信号通路参与抗氧化反应的调节,通过抑制Akt 信号通路参与细胞存活和增殖的调节。
T4978 Sarpogrelate hydrochloride

盐酸沙格雷酯,MCI-9042

5-HT Receptor GPCR/G Protein; Neuroscience
Sarpogrelate hydrochloride (MCI-9042) 是一种选择性5-HT2R 拮抗剂,可用于研究与血栓形成有关的血管疾病,对 5-HT2A、5-HT2B 和 5-HT2C 受体的pKi 值分别为 8.52、6.57 和 7.43。
T0117 Suplatast (Tosilate)

IPD 1151T,甲磺司特,Suplatast tosilate,Suplatast Tosylate

IL Receptor; Interleukin Immunology/Inflammation
Suplatast Tosilate (IPD 1151T) 是一种口服有活性的 Th2 细胞因子抑制剂,能够阻碍 Th2 细胞产生 IL-4 和 IL-5 ,并对 IgE 的合成具有抑制作用。它是一种抗过敏剂,它具有抗纤维化、抗哮喘及抗炎特性。
T39437 Cevidoplenib dimesylate

Syk Angiogenesis; Tyrosine Kinase/Adaptors
Cevidoplenib dimesylate 是一种脾酪氨酸激酶 (Syk) 抑制剂,具有抗炎和免疫调节特性。
T13639 Deferasirox (Fe3+ chelate)

Apoptosis Apoptosis
Deferasirox (Fe3+ chelate) 是一种可口服的铁螯合剂,具有潜在的抗癌活性,抑制 MCL-1 的抗凋亡活性,可用于研究铁超负荷。
T0372 Gabexate mesylate

甲磺酸加贝酯,FOY

Factor Xa; Serine Protease; Proteasome Metabolism; Proteases/Proteasome; Ubiquitination
Gabexate mesylate (FOY) 是一种非抗原的类胰蛋白酶丝氨酸蛋白酶抑制剂。
T6275 Obatoclax Mesylate

Obatoclax,GX15-070,奥巴克拉甲磺酸盐

BCL; Parasite; Autophagy Apoptosis; Autophagy; Microbiology/Virology
Obatoclax Mesylate (GX15-070) 是泛 BCL-2家族蛋白抑制剂,对 BCL-2 的 Ki 值为 220 nM。它是 BH3 模拟物,具有抗癌和广谱抗寄生虫活性。它诱导自噬依赖性细胞死亡,并靶向细胞周期蛋白 D1 进行蛋白酶体降解。
T1459 Cisatracurium besylate

顺苯磺酸阿曲库铵,顺苯磺阿曲库铵,51W89

Adrenergic Receptor; AChR; Autophagy Autophagy; GPCR/G Protein; Neuroscience
Cisatracurium besylate (51W89) 是一种用于静脉内给药的非去极化骨骼肌松弛剂。
T0504 Cyclandelate

安脉生,BS 572,环扁桃酯,3,5,5-Trimethylcyclohexyl mandelate

Acyltransferase Metabolism
Cyclandelate (BS 572) 是直接作用的平滑肌松弛剂,用于扩张血管。
T41194 FFN 102 mesylate

Others Others
FFN 102 mesylate 是pH 响应型荧光假神经递质(FFN),作为选择性多巴胺转运蛋白(DAT)和VMAT2底物。FFN 102 mesylate 与38个中枢神经系统受体(包括多巴胺和血清素受体)无明显结合。它的Ex-max在pH 值5时为340 nm,在pH 值7.5时为370 nm,在pH 值为5和7.5时,Em-max为435 nm。
T2531 Eprosartan Mesylate

SKF-108566J,甲磺酸依普罗沙坦

RAAS Endocrinology/Hormones
Eprosartan Mesylate (SKF-108566J) 是一种具有选择性、竞争性血管紧张素 II 受体拮抗剂,是具有口服活性的非肽。它结合血管紧张素 II 受体,在大鼠和人类肾上腺皮质膜中的IC50值分别为 9.2 nM 和 3.9 nM,可用作降压剂。
T6651 Safinamide mesylate

PNU-151774E,FCE28073,PNU-151774E,NW-1015,EMD 1195686 mesylate,沙芬酰胺甲磺酸盐

MAO; Monoamine Oxidase Metabolism; Neuroscience
Safinamide mesylate (EMD 1195686 mesylate) 是选择性的、有效的、可逆的单胺氧化酶 B 的抑制剂,对 MAO-A 选择性较低。它能够阻断钠通道和调节谷氨酸释放。它具有神经保护作用,可用于研究帕金森病、缺血脑卒中等疾病。
T0425L Pefloxacin Mesylate Dihydrate

Pefloxacinium mesylate dihydrate,1589 RB,甲磺酸培氟沙星二水合物

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate Dihydrate (1589 RB) 是一种抗菌素,能通过抑制DNA 旋转酶阻断细菌DNA 复制。
T0113 Mebhydrolin napadisylate

Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,美海屈林萘二磺酸盐,Omeril,Diazoline

5-HT Receptor; AChR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mebhydrolin napadisylate (Incidal) 是一种抗组胺药,用于缓解组胺释放引起的过敏症状,如鼻过敏和过敏性皮肤病。
T20168 Aurothiomalate sodium

金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate

Others; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Others
Aurothiomalate sodium (Miochrysin) 是一种选择性的致癌 PKCι信号传导抑制剂,可抑制肿瘤细胞增殖。它是一种硫氧还蛋白还原酶 (TrxR) 抑制剂,也是一种抗风湿剂。
T6962 Rasagiline Mesylate

TVP1012,甲磺酸雷沙吉兰,AGN1135,Azilect

Apoptosis; MAO; Autophagy; Monoamine Oxidase Apoptosis; Autophagy; Metabolism; Neuroscience
Rasagiline Mesylate (AGN1135) 是一种高效的,不可逆的选择性线粒体单胺氧化酶 (MAO) 抑制剂,抑制大鼠脑 MAO B 和 MAO A 的IC50分别为 4.43 nM 和 412 nM。
T13174 TMPyP4 tosylate

TMP 1363

DNA/RNA Synthesis; Telomerase Cell Cycle/Checkpoint; DNA Damage/DNA Repair
TMPyP4 tosylate (TMP 1363) 是四链体 (G-quadruplex) 的特异性配体,抑制四链体和 IGF-1 之间的相互作用。它也是端粒酶抑制剂,在骨肉瘤细胞系中显示抗肿瘤作用。
T77351 tert-Butyl5-bromo-1H-indole-1-carboxylate

N-Boc-5-bromoindole

Tert-Butyl5-bromo-1H-indole-1-carboxylate (N-Boc-5-bromoindole) 是一种具有治疗疼痛,炎症和其他病症潜力的吲哚衍生物。
T3608 Carbasalate calcium

Rheomin,Omegin,Alcacyl,Iromin,卡巴匹林钙,Solupsan,Carbasalate Calcium

Platelet aggregation Others
Carbasalate calcium (Rheomin) 是抗炎和解热剂,可用于研究疼痛的缓解。

化合物

Primaquine diphosphate
Cat.No: T0850
Synonym: Primaquine phosphate,磷酸伯氨喹,Primaquine bisphosphate,磷酸伯安喹
Target: Antibiotic, Parasite
Cilostazol
Cat.No: T0462
Synonym: 西洛他唑,OPC 21,OPC 13013
Target: PDE, Autophagy
Pefloxacin Mesylate
Cat.No: T0425
Synonym: Pefloxacinium mesylate,甲磺酸培氟沙星
Target: Topoisomerase, Antibacterial, Antibiotic
Delavirdine mesylate
Cat.No: T7212
Synonym: U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate)
Target: HIV Protease, Reverse Transcriptase
Darunavir Ethanolate
Cat.No: T3335
Synonym: 地瑞那韦乙醇盐,UIC 94017,Darunavir Ethanolate,TMC114,达芦那韦乙醇
Target: HIV Protease
Dolasetron Mesylate hydrate
Cat.No: T2589
Synonym: Dalasetron Mesylate Hydrate,多拉司琼甲磺酸盐一水合物
Target: 5-HT Receptor
Pizotifen Malate
Cat.No: T0225
Synonym: Pizotyline (malate),BC-105 (malate),BC-105,苯噻啶苹果酸盐
Target: 5-HT Receptor
Pergolide mesylate
Cat.No: T2226
Synonym: 甲磺酸培高利特,Pergolide mesylate salt,LY127809,Pergolide methanesulfonate
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Lenvatinib mesylate
Cat.No: T8541
Synonym: 仑伐替尼甲酸盐,E7080 (mesylate),乐伐替尼
Target: VEGFR, FGFR, c-RET, PDGFR, c-Kit
Diethyl 2,4-dimethylpyrrole-3,5-dicarboxylate
Cat.No: T77705
Synonym: Diethyl 3,5-dimethyl-1H-pyrrole-2,4-dicarboxylate
Target: Others
Memantine Related Compound B
Cat.No: T0535
Synonym: 美金刚杂质B,3,5-Dimethyl-1-adamantanol
Target: Others
Levomefolate calcium
Cat.No: T7593
Synonym: 左旋甲状腺素钙,L-5-甲基四氢叶酸钙
Target: Antifolate
Hexyl gallate
Cat.No: T11558
Synonym: 没食子酸己酯,Gallic acid hexyl ester,Hexyl 3,4,5-trihydroxybenzoate
Target: Antibacterial
Reboxetine mesylate
Cat.No: T6963
Synonym: 瑞波西汀甲磺酸盐,FCE20124 mesylate,Edronax,PNU155950E mesylate,PNU 155950E,甲磺酸瑞波西汀
Target: Adrenergic Receptor, Norepinephrine
Mepenzolate Bromide
Cat.No: T0794
Synonym: Colibantil,Cantil,溴美喷酯,Cantilaque
Target: AChR
Bretylium tosylate
Cat.No: T7386
Synonym: 溴苄乙胺,托西溴苄铵
Target: Others
Pep2m, myristoylated acetate
Cat.No: TP1945L1
Synonym: Pep2m, myristoylated acetate(1423381-07-0 free base)
Target: PKC
pp60 c-src (521-533) (phosphorylated) acetate
Cat.No: TP2137L
Synonym:
Target: Others
AZD-8529 mesylate
Cat.No: T10432L
Synonym:
Target: GluR
Tetrindole mesylate
Cat.No: T23453
Synonym:
Target: MAO
Gemifloxacin mesylate
Cat.No: T1492
Synonym: LB-20304a,甲磺酸吉米沙星,SB-265805S,Gemifloxacin mesylate
Target: DNA gyrase, Topoisomerase, Antibacterial
FlutaMide Related CoMpound B
Cat.No: T0547
Synonym:
Target: Others
L-Histidine benzyl ester bistosylate
Cat.No: T40122
Synonym:
Target: Others
Mesoridazine Besylate
Cat.No: T3086
Synonym: Mesoridazine benzenesulfonate,Serentil,苯磺酸美索达嗪
Target: Dopamine Receptor, 5-HT Receptor
Dolasetron Mesylate
Cat.No: T22313
Synonym: 多拉司琼甲磺酸盐,甲磺酸多拉司琼,Anzemet hydrate,MDL-73147EF
Target: Others, 5-HT Receptor
Sodium taurodeoxycholate hydrate
Cat.No: T9154
Synonym: 牛磺去氧胆酸钠,Taurodeoxycholic acid sodium salt monohydrate
Target: Others
Ningetinib Tosylate
Cat.No: TQ0041
Synonym:
Target: VEGFR, c-Met/HGFR, TAM Receptor
Kukoamine B mesylate
Cat.No: T7026L
Synonym:
Target: Antioxidant
Dimethyl biphenyl-4,4'-dicarboxylate
Cat.No: T5988
Synonym: Biphenyl dimethyl dicarboxylate,联苯二甲酸二甲酯
Target: Others
Olverembatinib dimesylate
Cat.No: T2429
Synonym: GZD824 Dimesylate,HQP1351
Target: Bcr-Abl
Niraparib tosylate monohyrate
Cat.No: T9497
Synonym:
Target: PARP
ethyl 2-[3,5-bis(trifluoromethyl)phenyl]-3-oxo-2,3-dihydro-1H-pyrazole-4-carboxylate
Cat.No: T50107
Synonym:
Target: Others
Sarpogrelate hydrochloride
Cat.No: T4978
Synonym: 盐酸沙格雷酯,MCI-9042
Target: 5-HT Receptor
Suplatast (Tosilate)
Cat.No: T0117
Synonym: IPD 1151T,甲磺司特,Suplatast tosilate,Suplatast Tosylate
Target: IL Receptor, Interleukin
Cevidoplenib dimesylate
Cat.No: T39437
Synonym:
Target: Syk
Deferasirox (Fe3+ chelate)
Cat.No: T13639
Synonym:
Target: Apoptosis
Gabexate mesylate
Cat.No: T0372
Synonym: 甲磺酸加贝酯,FOY
Target: Factor Xa, Serine Protease, Proteasome
Obatoclax Mesylate
Cat.No: T6275
Synonym: Obatoclax,GX15-070,奥巴克拉甲磺酸盐
Target: BCL, Parasite, Autophagy
Cisatracurium besylate
Cat.No: T1459
Synonym: 顺苯磺酸阿曲库铵,顺苯磺阿曲库铵,51W89
Target: Adrenergic Receptor, AChR, Autophagy
Cyclandelate
Cat.No: T0504
Synonym: 安脉生,BS 572,环扁桃酯,3,5,5-Trimethylcyclohexyl mandelate
Target: Acyltransferase
FFN 102 mesylate
Cat.No: T41194
Synonym:
Target: Others
Eprosartan Mesylate
Cat.No: T2531
Synonym: SKF-108566J,甲磺酸依普罗沙坦
Target: RAAS
Safinamide mesylate
Cat.No: T6651
Synonym: PNU-151774E,FCE28073,PNU-151774E,NW-1015,EMD 1195686 mesylate,沙芬酰胺甲磺酸盐
Target: MAO, Monoamine Oxidase
Pefloxacin Mesylate Dihydrate
Cat.No: T0425L
Synonym: Pefloxacinium mesylate dihydrate,1589 RB,甲磺酸培氟沙星二水合物
Target: Topoisomerase, Antibacterial, Antibiotic
Mebhydrolin napadisylate
Cat.No: T0113
Synonym: Incidal,Diazolin,Mebhydroline 1,5-naphthalenedisulfonate salt,美海屈林萘二磺酸盐,Omeril,Diazoline
Target: 5-HT Receptor, AChR, Histamine Receptor
Aurothiomalate sodium
Cat.No: T20168
Synonym: 金硫丁二钠,Myocrisin,Myocrisine,Miochrysin,Sodium aurothiomalate,Myochrysine,gold sodium thiomalate
Target: Others, PKC
Rasagiline Mesylate
Cat.No: T6962
Synonym: TVP1012,甲磺酸雷沙吉兰,AGN1135,Azilect
Target: Apoptosis, MAO, Autophagy, Monoamine Oxidase
TMPyP4 tosylate
Cat.No: T13174
Synonym: TMP 1363
Target: DNA/RNA Synthesis, Telomerase
tert-Butyl5-bromo-1H-indole-1-carboxylate
Cat.No: T77351
Synonym: N-Boc-5-bromoindole
Target:
Carbasalate calcium
Cat.No: T3608
Synonym: Rheomin,Omegin,Alcacyl,Iromin,卡巴匹林钙,Solupsan,Carbasalate Calcium
Target: Platelet aggregation
Cat. No. Product Name Target Signaling Pathways
TN7174 methyl 5-bromo-1H-pyrrole-2-carboxylate

甲基 5-溴-1H-吡咯-2-甲酸酯,ZINC13379818

Others Others
methyl 5-bromo-1H-pyrrole-2-carboxylate 是一种海洋来源的天然产物,存在于Lissodendoryx sp.。
TMS0418 Dihydroergotoxine mesylate

甲磺酸二氢麦角碱,Ergoloid mesylates,甲磺酸双氢麦角毒碱

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Dihydroergotoxine mesylate (Ergoloid mesylates) 是系列生物碱盐混合物,对GABAA 受体高结合活性。它主要用于改善与衰老相关的精神退化的症状和身体症状。
TN2349 Taurodeoxycholate sodium salt

Sodium taurodeoxylate,牛磺脱氧胆酸钠

Endogenous Metabolite Metabolism
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
T5112 DI-N-OCTYL PHTHALATE

Others Others
DI-N-OCTYL PHTHALATE 用作增塑剂和添加剂。用于毒理学研究以及通过邻苯二甲酸盐从食品接触材料 (FCM) 迁移到食品中而发生的食品污染风险评估研究。
T8319 Butyl isobutyl phthalate

ButylIsobutylPhthalate,邻苯二甲酸-1-丁酯-2-异丁酯

Glucosidase Metabolism
Butyl isobutyl phthalate (ButylIsobutylPhthalate) 是一种非竞争性 α-葡萄糖苷酶抑制剂,IC50=38 μM,可以从海带的根状茎中分离得到。它具有降血糖作用,可用于糖尿病相关的研究。
T3730 Methyl gallate

NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯

Reactive Oxygen Species; HIV Protease; Reverse Transcriptase; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Methyl gallate (Gallincin) 是具有抗氧化,抗癌和抗炎活性的植物酚类。它也可抑制细菌活性。它还具有抗HIV-1和HIV-1酶的抑制活性。
T3682 (-)-Catechin gallate

(-)-Catechin 3-O-gallate,儿茶素没食子酸酯,几茶素没食子酸酯,(-)-Catechin 3-gallate

Others; COX Immunology/Inflammation; Neuroscience; Others
(-)-Catechin gallate ((-)-Catechin 3-O-gallate) 是绿茶儿茶素中的微量组分,可抑制COX-1和COX-2活性。它抑制人 Beta-secretase,对氯喹敏感的恶性疟原虫 NF54 和耐氯喹的恶性疟原虫 K1 具有抗疟原虫活性。
T6293 Mycophenolate Mofetil

TM-MMF,吗替麦考酚酯,RS 61443

Apoptosis; Dehydrogenase; Drug Metabolite Apoptosis; Metabolism
Mycophenolate Mofetil (TM-MMF) 是 Mycophenolic acid 的吗啉乙酯前药。它通过抑制肌苷一磷酸脱氢酶抑制从头嘌呤合成,显示出选择性淋巴细胞抗增殖作用。
T15245 Erythromycin estolate

Phtalic anhydride,ilosone

Antibacterial Microbiology/Virology
Erythromycin estolate 是红霉素的衍生物,属于大环内酯类抗生素,常用于研究多种细菌感染。酯酸红霉素对胆汁酸转运有抑制作用,可引起肝损伤,主要是胆汁淤积性肝炎。
TN1608 (-)-Epigallocatechin-3-(3''-O-methyl) gallate

(-)-EGCG-3''-O-ME

Antioxidant; Antibacterial Microbiology/Virology; oxidation-reduction
(-)-Epigallocatechin-3-(3''-O-methyl) gallate ((-)-EGCG-3''-O-ME) 是从茶叶中分离出的一种天然产物,具有很强的抗氧化、细胞毒性和抗菌活性,可增强蚀刻漂洗粘合剂与牙本质的粘合稳定性。
T22366 Methyl cyclohexanecarboxylate

Hexahydrobenzoic acid methyl ester,环己甲酸甲酯,Methyl hexahydrobenzoate

Others; Endogenous Metabolite Metabolism; Others
Methyl cyclohexanecarboxylate (Methyl hexahydrobenzoate) 是一种内源性代谢物,用作化学合成的原料。环己烷羧酸甲酯是一种具有浆果味、酯味和水果味的调味成分。
TN2330 Phenethyl ferulate

Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯

Lipoxygenase; COX Immunology/Inflammation; Metabolism; Neuroscience
Phenethyl ferulate (Caffeic Acid 3-Methyl Phenethyl Ester) 对化学诱导的结肠癌具有化学预防特性,可增强偶氮甲烷诱导的结肠肿瘤的细胞凋亡。 它抑制环氧合酶(COX) 和 5-脂氧合酶 (5-LOX) ,IC50 值分别为 4.35 和 5.75 μM。
T4394 Methyl Isoferulate

Others Others
Methyl Isoferulate 从毛竹叶中分离纯化。
TN1925 Methyl anthranilate

Others; Antibacterial Microbiology/Virology; Others
Methyl anthranilate 是一种植物香料提取物,在食品加工业中广泛用于制备食用香精和食品添加剂。它是一种群体感应抑制剂和抗温和气单胞菌的生物膜剂。
TQ0316 Ingenol-5,20-acetonide-3-O-angelate

Ingenol 5,20-acetonide 3-angelate,Ingenol 3-angelate 5,20-acetonide,巨大戟醇-5,20-缩丙酮-3-当归酸酯

Others Others
Ingenol-5,20-acetonide-3-O-angelate (Ingenol 5,20-acetonide 3-angelate) 是一种天然产物。
TN6710 Methyl acetylsalicylate

ACETYLSALICYLIC ACID METHYL ESTER,乙酰水杨酸甲酯

Others Others
Methyl acetylsalicylate (ACETYLSALICYLIC ACID METHYL ESTER) 是一种从豌豆中分离出来的天然产物。抑制胶原蛋白诱导的人富含血小板的血浆聚集。
T5429 Theaflavin 3,3'-digallate

茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG

Virus Protease; Antioxidant; HIV Protease; HSV Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。
T6752 S-Adenosyl-L-methionine disulfate tosylate

S-腺苷蛋氨酸对甲苯磺酸硫酸盐,Ademetionine disulfate tosylate

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
S-Adenosyl-L-methionine disulfate tosylate (Ademetionine disulfate tosylate) 是一种主要生物甲基供体,在所有哺乳动物细胞中合成,但在肝脏中含量较高。
T20648 Dodecyl gallate

没食子酸月桂酯,NSC-133463,Nipagallin LA,Lauryl gallate,Progallin LA,NSC 133463,NSC133463

Others Others
Dodecyl gallate (Progallin LA) 是一种抗氧化剂,普遍用作食品制造及制药和化妆品行业中。它还对动物病毒,如非洲猪瘟病毒(ASFV)具有作用活性。
T2818 Methyl Vanillate

Reactive Oxygen Species; Wnt/beta-catenin; Endogenous Metabolite Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells
Methyl vanillate 是一种枳椇属植物中的提取物,是Wnt/β-catenin 信号通路活化剂,是一种香草酸的甲酯。它具有抗氧化作用。
T5119 Dicyclo hexyl Phthalate

Others Others
Dicyclo hexyl Phthalate 是一种固体增塑剂。
T0281 Meclocycline sulfosalicylate salt

磺基水杨酸甲氯环素,Meclutin,Mecloderm,甲环素磺基水杨酸盐,Meclan Cream

Antibacterial; Antibiotic Microbiology/Virology
Meclocycline sulfosalicylate salt (Mecloderm) 是一种具有广谱抗菌活性的四环素抗生素,可预防皮肤细菌感染。
T3729 Ethyl gallate

Nipagallin A,Phyllemblin,gallic acid ethyl ester,没食子酸乙酯

MMP; NF-κB; Akt; Antibacterial Cytoskeletal Signaling; Microbiology/Virology; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Ethyl gallate (gallic acid ethyl ester) 是一种非类黄酮酚过氧化氢清除剂。
T2929 Ethyl Vanillate

香兰酸乙酯,Ethylprotal,香草酸乙酯,Bourbonal

Antioxidant; Antifungal Microbiology/Virology; oxidation-reduction
Ethyl Vanillate (Bourbonal) 是一种杀菌剂,抑制17β-HSD2,其IC50为 1.3 µM。它是一种香草醛类似物,是一种调味剂,具有很强的抗氧化活性。
TN7138 Methyl 5-hydroxy-1H-indole-3-carboxylate

ZINC40836050,5-羟基-1H-吲哚-3-甲酸甲酯,5-hydroxy-1H-indole-3-carboxylic acid methyl ester,Methyl5-hydroxy-1H-indole-3-carboxylate

Others Others
Methyl 5-hydroxy-1H-indole-3-carboxylate (5-hydroxy-1H-indole-3-carboxylic acid methyl ester) 是一种海洋来源的天然产物,存在于Hyrtios erectus。
T5868 Methyl indole-3-carboxylate

吲哚-3-甲酸甲酯,Methyl 3-indolecarboxylate,3-吲哚甲酸甲酯

Others; Antibacterial Microbiology/Virology; Others
Methyl indole-3-carboxylate (Methyl 3-indolecarboxylate) 是一种从Sorangium cellulosumSoce895 菌株中分离出来的天然产物。它对革兰氏阳性诺卡氏菌的MIC 值为 33.3 μg/mL。
T4S0553 Theaflavin-3'-Gallate

茶黄素-3-没食子酸酯,Theaflavin 2B,THEAFLAVIN 3'-O-GALLATE,茶黄素-3'-没食子酸酯

Others Others
Theaflavin-3'-Gallate (Theaflavin 2B) 是红茶茶黄素单体,是红茶生物学上重要的活性成分,对健康有益。它以时间和浓度依赖性方式与还原型谷胱甘肽直接反应。它充当促氧化剂并在癌细胞中诱导氧化应激。
TQ0099 20-O-Acetylingenol-3-angelate

巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1

Others Others
20-O-Acetylingenol-3-angelate (Euphorbia factor Pe1) 是一种天然化合物,存在于植物英加的叶子和茎中。它具有多种生物活性,包括抑制肿瘤生长、抗炎、抗真菌和抗氧化作用。
T3S1866 Propyl gallate

没食子酸丙酯;3,4,5-三羟基苯甲酸丙酯、倍酸丙酯、五倍子酸丙酯,Tenox PG,没食子酸丙酯,n-Propyl gallate,Gallic acid propyl esterZ

Antioxidant oxidation-reduction
Propyl gallate (Gallic acid propyl esterZ) 是常见的食品抗氧化剂。它能阻碍乙二醛、丙烯醛、甲基乙二醛的生成。
TWA2417 Sodium taurocholate

牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium

Others Others
Sodium taurocholate (Taurocholate Sodium) hydrate 具有显著的生物学效应,例如通过上调 VEGF-A 的表达抑制肝动脉结扎所致的胆道损伤。对免疫系统具有一定的调节作用。
TN2030 P-Hydroxyphenethyl trans-ferulate

反式-阿魏酸对羟基苯乙酯

5-HT Receptor GPCR/G Protein; Neuroscience
p-Hydroxyphenethyl trans-ferulate 具有抗高血糖 (酵母α-葡萄糖苷酶,IC5019.24 ± 1.73 µmol L-1),抗氧化,抗炎活性,也具有抗癌特性和血清素能特性。
T4S0554 Theaflavine-3,3'-digallate

TFBG,theaflavin digallate,3,3’-二没食子酸酯茶黄素

Others Others
Theaflavine-3,3'-digallate (theaflavin digallate) 和乳酸一起可以减少单纯疱疹病毒的传播。
T0335 Sodium salicylate

水杨酸钠,Salicylic acid sodium salt,2-Hydroxybenzoic acid sodium salt

Apoptosis; NF-κB; COX; S6 Kinase; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; MAPK; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling
Sodium salicylate (2-Hydroxybenzoic acid sodium salt) 是一种S6K 的抑制剂,可抑制COX-2活性。它还是一种NF-κB 抑制剂,可降低炎症基因的表达,促进老化肌肉的修复。
T4589 9'''-Methyl salvianolate B

9’’’-丹酚酸B单甲酯,9'''-丹酚酸B单甲酯,9'''-MethyllithosperMate B

Others Others
9'''-MethyllithosperMate B 是一种从 Cynoglossum columnaeTen 中获得的一种天然提取物。
T1276 Danofloxacin mesylate

甲磺酸达氟沙星,CP 76136-27

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Danofloxacin mesylate (CP 76136-27) 是一种兽医用氟喹诺酮类抗菌素。
T0606 Monobutyl Phthalate

邻苯二甲酸单丁酯,Mono-n-butyl phthalate,Butyl hydrogen phthalate

Others Others
Monobutyl Phthalate (Butyl hydrogen phthalateButyl hydrogen phthalate) 是邻苯二甲酸二丁酯的主要代谢物,是一种胚胎毒物,具有抗雄激素作用。
T20250 Phenyl salicylate

NSC-33406,NSC 33406,水杨酸苯酯,NSC33406

Others Others
Phenyl salicylate (NSC-33406) 是一种化学物质。由水杨酸与苯酚加热合成。
T3051 Theaflavin-3-gallate

茶黄素-3-没食子酸酯,茶黄素 3-没食子酸酯,茶黄素 -3-没食子酸,Theaflavine-3-Gallate

Others Others
Theaflavin-3-gallate (Theaflavine-3-Gallate) 是红茶茶黄素单体,是红茶生物学上重要的活性成分,对健康有益。它以时间和浓度依赖性方式与还原型谷胱甘肽直接反应。它充当促氧化剂并在癌细胞中诱导氧化应激。
T4961 9''-Methyl salvianolate B

9'-Methyl lithospermate B,9’-丹酚酸B单甲酯,9''-丹酚酸B单甲酯

Others Others
9'-Methyl lithospermate B 是一种酚类化合物,提取自 RadixSalvia miltiorrhizae。
T2S1865 Octyl gallate

Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯

Antioxidant; Influenza Virus; Reactive Oxygen Species; Antibacterial; Antifungal; HSV Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Octyl gallate (Octyl 3,4,5-trihydroxybenzoate) 具有抗菌、抗氧化作用,有选择性和敏感性的荧光特性,广泛用作食品添加剂。它对 HSV-1,水泡性口炎病毒和脊髓灰质炎病毒有显著的抗病毒作用。
T2821 Ethyl ferulate

Ethyl 4'-hydroxy-3'-methoxycinnamate,Ethyl 3-(4-hydroxy-3-methoxyphenyl)acrylate,阿魏酸乙酯,Ferulic acid ethyl ester,乙基阿魏酸

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Ethyl ferulate (Ethyl 4'-hydroxy-3'-methoxycinnamate) 是一种从大茴香分离得到的阿魏酸的天然亲酯衍生物,能够诱导血红素氧合酶 1 ,保护大鼠神经元免受氧化应激。它能够保护神经元,使其受 β 淀粉样肽(1-42)导致的全身性的氧化应激和神经毒性。
TN1557 Decursinol angelate

ERK; VEGFR; PKC; JNK Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Tyrosine Kinase/Adaptors
Decursinol angelate 是从朝鲜当归根部分离得到的一种天然产物,是 PKC 激酶的激活剂,有细胞毒性,抗肿瘤和抗炎活性。
T1687L Doxycycline (hyclate)

Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate

MMP; ribosome; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。
TN1625 Ethyl salicylate

Others Others
Ethyl salicylate 是一种天然产物。
T3S0012 coniferyl ferulate

P-gp; GST Membrane transporter/Ion channel; Neuroscience; oxidation-reduction
Coniferyl ferulate 是从川芎中提取的一种天然产物,是强效的谷胱甘肽 S-转移酶抑制剂,强抑制人胎盘型谷胱甘肽 S-转移酶,IC50为 0.3 μM。它还可逆转多药耐药性并下调 P-糖蛋白。
TN1162 Dibutyl phthalate

邻苯二甲酸二丁酯,1,2-Benzenedicarboxylic acid

Antifection Microbiology/Virology
1,2-Benzenedicarboxylic acid is one kind of allelochemical shows stronger allelopathic effect on itself than on wheat and pigeonpea.
T2732 (-)-Epicatechin gallate

表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG

Virus Protease; COX; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience
(-)-Epicatechin gallate ((-)-Epicatechin 3-O-gallate) 抑制环加氧酶-1 的IC50值为 7.5 μM。
T0516 Dehydrocholate sodium

去氢胆酸钠,Sodium dehydrocholate

Endogenous Metabolite; Lipid Metabolism
Dehydrocholate sodium 是胆液排泄增多剂,能够提高胆汁输出,清除提高的胆汁酸负载。
T2988 (-)-Epigallocatechin Gallate

Epigallocatechol Gallate,(-)-表没食子儿茶素没食子酸酯,EGCG

Ferroptosis; Reactive Oxygen Species; HIV Protease; Mitochondrial Metabolism; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
(-)-Epigallocatechin Gallate (EGCG) 是茶类黄酮,具有强大的抗氧化,抗炎和抗癌作用。它可抑制EGFR 信号传导,有抗癌作用。它是谷氨酸脱氢酶 1/2 抑制剂。它通过激活细胞色素c 氧化酶来诱导氧化磷酸化。
T0399 Methyl salicylate

Gaultheria oil,Methyl 2-hydroxybenzoate,2-Carbomethoxyphenol,Betula oil,水杨酸甲酯,Natural wintergreen oil,Wintergreen oil

COX; TRP/TRPV Channel Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience
Methyl salicylate (Gaultheria oil) 是从番泻叶中提取的一种天然三萜皂苷,是一种局部缓解疼痛和抗炎作用的药物。 它还用作食品和烟草制品中的农药、变性剂、香料成分和调味剂。
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天然产物

methyl 5-bromo-1H-pyrrole-2-carboxylate
Cat.No: TN7174
Synonym: 甲基 5-溴-1H-吡咯-2-甲酸酯,ZINC13379818
Target: Others
Dihydroergotoxine mesylate
Cat.No: TMS0418
Synonym: 甲磺酸二氢麦角碱,Ergoloid mesylates,甲磺酸双氢麦角毒碱
Target: GABA Receptor
Taurodeoxycholate sodium salt
Cat.No: TN2349
Synonym: Sodium taurodeoxylate,牛磺脱氧胆酸钠
Target: Endogenous Metabolite
DI-N-OCTYL PHTHALATE
Cat.No: T5112
Synonym:
Target: Others
Butyl isobutyl phthalate
Cat.No: T8319
Synonym: ButylIsobutylPhthalate,邻苯二甲酸-1-丁酯-2-异丁酯
Target: Glucosidase
Methyl gallate
Cat.No: T3730
Synonym: NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯
Target: Reactive Oxygen Species, HIV Protease, Reverse Transcriptase, Antibacterial
(-)-Catechin gallate
Cat.No: T3682
Synonym: (-)-Catechin 3-O-gallate,儿茶素没食子酸酯,几茶素没食子酸酯,(-)-Catechin 3-gallate
Target: Others, COX
Mycophenolate Mofetil
Cat.No: T6293
Synonym: TM-MMF,吗替麦考酚酯,RS 61443
Target: Apoptosis, Dehydrogenase, Drug Metabolite
Erythromycin estolate
Cat.No: T15245
Synonym: Phtalic anhydride,ilosone
Target: Antibacterial
(-)-Epigallocatechin-3-(3''-O-methyl) gallate
Cat.No: TN1608
Synonym: (-)-EGCG-3''-O-ME
Target: Antioxidant, Antibacterial
Methyl cyclohexanecarboxylate
Cat.No: T22366
Synonym: Hexahydrobenzoic acid methyl ester,环己甲酸甲酯,Methyl hexahydrobenzoate
Target: Others, Endogenous Metabolite
Phenethyl ferulate
Cat.No: TN2330
Synonym: Caffeic Acid 3-Methyl Phenethyl Ester,阿魏酸苯乙酯,阿魏酸苯乙醇酯
Target: Lipoxygenase, COX
Methyl Isoferulate
Cat.No: T4394
Synonym:
Target: Others
Methyl anthranilate
Cat.No: TN1925
Synonym:
Target: Others, Antibacterial
Ingenol-5,20-acetonide-3-O-angelate
Cat.No: TQ0316
Synonym: Ingenol 5,20-acetonide 3-angelate,Ingenol 3-angelate 5,20-acetonide,巨大戟醇-5,20-缩丙酮-3-当归酸酯
Target: Others
Methyl acetylsalicylate
Cat.No: TN6710
Synonym: ACETYLSALICYLIC ACID METHYL ESTER,乙酰水杨酸甲酯
Target: Others
Theaflavin 3,3'-digallate
Cat.No: T5429
Synonym: 茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG
Target: Virus Protease, Antioxidant, HIV Protease, HSV
S-Adenosyl-L-methionine disulfate tosylate
Cat.No: T6752
Synonym: S-腺苷蛋氨酸对甲苯磺酸硫酸盐,Ademetionine disulfate tosylate
Target: DNA/RNA Synthesis
Dodecyl gallate
Cat.No: T20648
Synonym: 没食子酸月桂酯,NSC-133463,Nipagallin LA,Lauryl gallate,Progallin LA,NSC 133463,NSC133463
Target: Others
Methyl Vanillate
Cat.No: T2818
Synonym:
Target: Reactive Oxygen Species, Wnt/beta-catenin, Endogenous Metabolite
Dicyclo hexyl Phthalate
Cat.No: T5119
Synonym:
Target: Others
Meclocycline sulfosalicylate salt
Cat.No: T0281
Synonym: 磺基水杨酸甲氯环素,Meclutin,Mecloderm,甲环素磺基水杨酸盐,Meclan Cream
Target: Antibacterial, Antibiotic
Ethyl gallate
Cat.No: T3729
Synonym: Nipagallin A,Phyllemblin,gallic acid ethyl ester,没食子酸乙酯
Target: MMP, NF-κB, Akt, Antibacterial
Ethyl Vanillate
Cat.No: T2929
Synonym: 香兰酸乙酯,Ethylprotal,香草酸乙酯,Bourbonal
Target: Antioxidant, Antifungal
Methyl 5-hydroxy-1H-indole-3-carboxylate
Cat.No: TN7138
Synonym: ZINC40836050,5-羟基-1H-吲哚-3-甲酸甲酯,5-hydroxy-1H-indole-3-carboxylic acid methyl ester,Methyl5-hydroxy-1H-indole-3-carboxylate
Target: Others
Methyl indole-3-carboxylate
Cat.No: T5868
Synonym: 吲哚-3-甲酸甲酯,Methyl 3-indolecarboxylate,3-吲哚甲酸甲酯
Target: Others, Antibacterial
Theaflavin-3'-Gallate
Cat.No: T4S0553
Synonym: 茶黄素-3-没食子酸酯,Theaflavin 2B,THEAFLAVIN 3'-O-GALLATE,茶黄素-3'-没食子酸酯
Target: Others
20-O-Acetylingenol-3-angelate
Cat.No: TQ0099
Synonym: 巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1
Target: Others
Propyl gallate
Cat.No: T3S1866
Synonym: 没食子酸丙酯;3,4,5-三羟基苯甲酸丙酯、倍酸丙酯、五倍子酸丙酯,Tenox PG,没食子酸丙酯,n-Propyl gallate,Gallic acid propyl esterZ
Target: Antioxidant
Sodium taurocholate
Cat.No: TWA2417
Synonym: 牛黄胆酸钠(牛胆酸钠,牛胆酸钠盐,牛磺膽酸鈉,牛磺胆酸钠,牛磺胆酸钠盐,牛胆酸钠水合物,水合牛磺胆酸钠,牛胆酸钠(混合物),牛黄胆酸钠(水合),牛磺胆酸钠(标准品)),Taurocholate Sodium
Target: Others
P-Hydroxyphenethyl trans-ferulate
Cat.No: TN2030
Synonym: 反式-阿魏酸对羟基苯乙酯
Target: 5-HT Receptor
Theaflavine-3,3'-digallate
Cat.No: T4S0554
Synonym: TFBG,theaflavin digallate,3,3’-二没食子酸酯茶黄素
Target: Others
Sodium salicylate
Cat.No: T0335
Synonym: 水杨酸钠,Salicylic acid sodium salt,2-Hydroxybenzoic acid sodium salt
Target: Apoptosis, NF-κB, COX, S6 Kinase, Autophagy
9'''-Methyl salvianolate B
Cat.No: T4589
Synonym: 9’’’-丹酚酸B单甲酯,9'''-丹酚酸B单甲酯,9'''-MethyllithosperMate B
Target: Others
Danofloxacin mesylate
Cat.No: T1276
Synonym: 甲磺酸达氟沙星,CP 76136-27
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Monobutyl Phthalate
Cat.No: T0606
Synonym: 邻苯二甲酸单丁酯,Mono-n-butyl phthalate,Butyl hydrogen phthalate
Target: Others
Phenyl salicylate
Cat.No: T20250
Synonym: NSC-33406,NSC 33406,水杨酸苯酯,NSC33406
Target: Others
Theaflavin-3-gallate
Cat.No: T3051
Synonym: 茶黄素-3-没食子酸酯,茶黄素 3-没食子酸酯,茶黄素 -3-没食子酸,Theaflavine-3-Gallate
Target: Others
9''-Methyl salvianolate B
Cat.No: T4961
Synonym: 9'-Methyl lithospermate B,9’-丹酚酸B单甲酯,9''-丹酚酸B单甲酯
Target: Others
Octyl gallate
Cat.No: T2S1865
Synonym: Gallic acid octyl ester,n-Octylgallate,Octyl 3,4,5-trihydroxybenzoate,Progallin O,Stabilizer GA-8,没食子酸辛酯
Target: Antioxidant, Influenza Virus, Reactive Oxygen Species, Antibacterial, Antifungal, HSV
Ethyl ferulate
Cat.No: T2821
Synonym: Ethyl 4'-hydroxy-3'-methoxycinnamate,Ethyl 3-(4-hydroxy-3-methoxyphenyl)acrylate,阿魏酸乙酯,Ferulic acid ethyl ester,乙基阿魏酸
Target: Reactive Oxygen Species
Decursinol angelate
Cat.No: TN1557
Synonym:
Target: ERK, VEGFR, PKC, JNK
Doxycycline (hyclate)
Cat.No: T1687L
Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate
Target: MMP, ribosome, Antibacterial, Antibiotic
Ethyl salicylate
Cat.No: TN1625
Synonym:
Target: Others
coniferyl ferulate
Cat.No: T3S0012
Synonym:
Target: P-gp, GST
Dibutyl phthalate
Cat.No: TN1162
Synonym: 邻苯二甲酸二丁酯,1,2-Benzenedicarboxylic acid
Target: Antifection
(-)-Epicatechin gallate
Cat.No: T2732
Synonym: 表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG
Target: Virus Protease, COX, Autophagy
Dehydrocholate sodium
Cat.No: T0516
Synonym: 去氢胆酸钠,Sodium dehydrocholate
Target: Endogenous Metabolite, Lipid
(-)-Epigallocatechin Gallate
Cat.No: T2988
Synonym: Epigallocatechol Gallate,(-)-表没食子儿茶素没食子酸酯,EGCG
Target: Ferroptosis, Reactive Oxygen Species, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite, Autophagy
Methyl salicylate
Cat.No: T0399
Synonym: Gaultheria oil,Methyl 2-hydroxybenzoate,2-Carbomethoxyphenol,Betula oil,水杨酸甲酯,Natural wintergreen oil,Wintergreen oil
Target: COX, TRP/TRPV Channel
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