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204

抑制剂 & 化合物

52

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T5817	PKC-theta inhibitor hcl PKC-theta inhibitor	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-theta inhibitor hcl 是一种选择性 PKC-θ 抑制剂 (IC50:12 nM)。
TP1955L	PKC β pseudosubstrate acetate PKC β pseudosubstrate醋酸盐,Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC β pseudosubstrate acetate (PKC β pseudosubstrate acetate (172308-76-8 Free base)) 是一种选择性的、细胞渗透的 PKC 抑制剂。
TP1956L	PKC ζ pseudosubstrate acetate PKC ζ pseudosubstrate acetate (799764-07-1 free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC ζ pseudosubstrate acetate 是蛋白激酶 C (PKC) ζ 的抑制剂；附着于细胞通透性触角足结构域载体肽。由 PKC ζ 假底物结构域的氨基酸 113-129 组成，通过二硫键连接到触角足结构域载体肽。 Antennapedia 肽在 4 或 37°C 时被完整细胞积极吸收，确保快速有效地吸收抑制肽。一旦进入细胞，二硫键在细胞质中被还原，导致抑制肽的释放。通过 PKC ζ 非依赖性途径诱导肥大细胞脱粒。
T8764	PKC-iota inhibitor 1	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-iota inhibitor 1 是一种蛋白激酶 C-iota(PKC-ι ℩)的抑制剂，IC50值为 0.34 μM。
T71993	PKC-9
	PKC-9 is a PKC-zeta inhibitor 9.
T5423	PKC-theta inhibitor	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-theta inhibitor 是一种PKC-θ抑制剂，IC50值为 12 nM。
T12494	PKC-IN-1	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-IN-1 是 ATP-竞争性可逆 PKC 抑制剂，对人 PKCβ 和 PKCα 的 Ki 值分别为 5.3 和 10.4 nM，对人 PKCα、PKCβI、PKCβII、PKCθ、PKCγ、PKC mu 和 PKCε 的IC50值分别为 2.3、8.1、7.6、25.6、57.5、314 和 808 nM。
T35826	PKC fragment (530-558)
	PKC fragment (530-558) 是蛋白激酶C (PKC) 的肽片段，是一种有效的 PKC 激活剂。Protein Kinase C (530-558) 可显著抑制破骨细胞骨吸收。
TP1053L	Protein Kinase C 19-31 acetate Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Protein Kinase C 19-31 acetate(121545-65-1 free base) 是一种蛋白激酶 C (PKC) 的肽抑制剂，源自 PKCa 的假底物调节结构域（残基 19-31），在 25 位用丝氨酸取代野生型丙氨酸作为蛋白激酶 C 底物肽，用于测试蛋白激酶 C 活性。
TP1955	PKC β pseudosubstrate
	Selective cell-permeable peptide inhibitor of protein kinase C (IC50 ~ 0.5 μM). Consists of amino acids 19 - 31 of PKC pseudosubstrate domain linked by a disulphide bridge to a cell permeabilisation Antennapedia domain vector peptide. The Antennapedia pep
TP1956	PKC ζ pseudosubstrate
	Inhibitor of protein kinase C (PKC) ζ; attached to cell permeabilisation Antennapedia domain vector peptide. Consists of amino acids 113 - 129 of PKC ζ pseudosubstrate domain linked by a disulphide bridge to the Antennapedia domain vector peptide. The Antennapedia peptide is actively taken up by intact cells, at 4 or 37°C, ensuring rapid and effective uptake of the inhibitor peptide. Once inside the cell, the disulphide bonds are subjected to reduction in the cytoplasm leading to release of the ...
T8376	PKCβ inhibitor 1 KUN79359	Apoptosis; PKC	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCβ inhibitor 1 (KUN79359) 是一种 ATP 竞争性和选择性PKCβ抑制剂，对人 PKCβ1 和 PKCβ2 的IC50分别为 21 和 5 nM。
T12496	PKC-theta inhibitor 1	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-theta inhibitor 1 is an inhibitor of PKCθ (Ki of 6 nM)
T61604	PKC-IN-4
	PKC-IN-4 (compound 7l) is a highly potent and orally active inhibitor of atypical protein kinase C (aPKC), exhibiting an IC 50 value of 0.52 μM. In vitro studies have demonstrated that PKC-IN-4 effectively suppresses NF-κB activity induced by TNF-α. Moreover, this compound effectively impedes the permeability of the retinal vasculature, induced by both VEGF and TNFα. [1]
T75885	PKC β pseudosubstrate TFA
	PKCβ pseudosubstrate TFA 是一种选择性的、细胞渗透的 PKC 抑制剂。
TP1053	Protein Kinase C (19-31) Protein Kinase C 19-31,PKC (19-31)
	Protein Kinase C (19-31), a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate pepti
T80509	PKC 20-28,myristoylated Myristoylated protein kinase C inhibitor 20-28	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC20-28,myristoylated（Myristoylated protein kinase C inhibitor 20-28）为具细胞渗透性之PKC抑制剂，可抑制AngII所诱导之IKca电流激活，用途涵盖癌症与心血管疾病研究。
T62945	Aurora A/PKC-IN-1
	Aurora A/PKC-IN-1 (Compound 2e) 是一种有效的 Aurora A (AurA) 和 PKC (α, β1, β2, θ) 双重抑制剂，作用于 AurA (IC50: 6.9 nM) 和 PKCα (IC50: 16.9 nM)。Aurora A/PKC-IN-1 对乳腺癌细胞表现出抗增殖和抗转移作用。
T81449	PKC-ε translocation inhibitor peptide	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKC-ε translocation inhibitor peptide，作为一种特定的PKC-ε易位抑制剂，能够特异性地调控FcγR介导的调理珠内化速率，而对FcαR运输不产生影响。
T35827L	PKCε Inhibitor Peptide acetate PKCε Inhibitor Peptide acetate(182683-50-7 Free base)	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	PKCε Inhibitor Peptide acetate 是一种特异性 PKCε 抑制剂，含有其特定受体活化 C 激酶 (RACK) 的位点。 PKCε Inhibitor Peptide acetate 抑制 PKCε 的转运，但不抑制 αPKC，βPKC 和 δPKC 的转运。
T17148	TPPB	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	TPPB 是可渗透细胞的苯并内酰胺衍生蛋白的激酶 C 激活剂，Ki 值为11.9 nM。
T3211	Midostaurin 米哚妥林,N-Benzoylstaurosporine,PKC412,CGP41231,CGP 41251,苯甲酰基十字孢碱	Others; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Others
	Midostaurin (PKC412) 是一种多靶点蛋白激酶抑制剂，有抗肿瘤活性，对 PKCα/β/γ、Syk、Flk-1、Akt、PKA、c-Kit、c-Fgr、c-Src、FLT3、PDFRβ和VEGFR1/2的IC50值范围为 22 到500 nM 之间。
T35407	Ζ-Stat	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	ζ-Stat 是非典型的、特异性的PKC-ζ抑制剂，IC50为 5 μM。ζ-Stat 能够减少黑色素瘤细胞系的增殖并诱导细胞凋亡，在体外显示除抗肿瘤活性。
T13314	VTX-27	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	VTX-27 是蛋白激酶 C θ (PKC θ) 的一种选择性抑制剂，对 PKC θ 和 PKC δ 的 Ki 值分别为 0.08 nM 和 16 nM。
TP1052	Protein Kinase C (19-31) (TFA)(121545-65-1,free) PKC (19-31) (TFA),Protein Kinase C (19-31) (TFA)
	Protein Kinase C (19-31) TFA, a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate p
T5600	Darovasertib LXS196	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Darovasertib (LXS196) 是一种有效的、选择性的和具有口服活性的蛋白激酶C(PKC) 抑制剂，有用于葡萄膜黑素瘤的研究潜力，对 PKCα、PKCθ 和 GSK3β 的 IC50值分别为 1.9、0.4 和 3.1 μM。
T7659	Bisindolylmaleimide IV	Others; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Others
	Bisindolylmaleimide IV 是一种蛋白激酶 C 细胞渗透抑制剂，其 IC50范围为 0.1-0.55 μM。它也抑制 PKA，IC50范围为3.1-11.8 μM。在细胞培养中，它有效抑制人巨细胞病毒(HCMV)复制，IC50为 0.2 μM。
T2441	TAS-301 TAS 301	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	TAS-301 是一种平滑肌迁移和增殖抑制剂，能够抑制 PDGF 诱导的 PKC 的活化，可抑制大鼠颈动脉球囊损伤后的内膜增厚。
T6515	Go6976 Gö 6976	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Go6976是蛋白激酶C (PKC)的小分子抑制剂。Go6976作为研究PKC 在各种生理和病理生理过程中的作用的工具，广泛应用于生物医学研究。
T6313	Go 6983 Goe 6983	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Go 6983 是一种PKC 抑制剂，能够作用于PKCα、PKCβ、PKCγ、PKCδ和PKCζ，IC50值分别为 7、7、6、10 和 60 nM。
T26019	R59949 R-59949,R 59949	Others; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Others
	R59949 是一种泛二酰甘油激酶(DGK)抑制剂，IC50为 300 nM。它通过提高内源性配体二酰甘油水平来激活蛋白激酶 C(PKC)。它强烈抑制 Ⅰ 型 DGKα 和 γ 的活性，中度减弱 Ⅱ 型 DGKθ 和 κ 的活性。
T6278	Sotrastaurin 索曲妥林,AEB071	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Sotrastaurin (AEB071) 是一种口服有效的泛 PKC 抑制剂，对 PKCθ、PKCβ、PKCα、PKCη、PKCδ 和 PKCε，Ki 分别为 0.22、0.64、0.95、1.8、2.1 和 3.2 nM。
T6280	Enzastaurin LY317615,恩扎妥林	Apoptosis; PKC; Autophagy	Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
	Enzastaurin (LY317615) 是一种PKCβ抑制剂，IC50值为 6 nM。它对 PKCβ 选择性是 PKCα，PKCγ 和 PKCε 的 6-20 倍。
T7604	Valrubicin Valstar,AD-32,戊柔比星	Antibiotic; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
	Valrubicin (AD-32) 是一种具有抗炎和抗肿瘤作用的化疗剂，能够抑制 TPA 和 PDBu 诱导的 PKC 活化，IC50值分别为 0.85 和 1.25 μM。
T7885	Afuresertib hydrochloride	ROCK; Akt; PKC	Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Stem Cells
	Afuresertib hydrochloride 是一个口服有效的，ATP 竞争性的选择性泛Akt 抑制剂，作用于Akt1、Akt2和Akt3，Ki 值分别为 0.08、2和 2.6 nM。
T14943	CGP60474	VEGFR; CDK; PKC	Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	CGP60474 是一种高效的抗内毒素药物，抑制细胞周期蛋白依赖激酶(CDK) ，抑制 CDK1/B、CDK2/E、CDK2/a、CDK4/D、CDK5/p25、CDK7/H 和 CDK9/T 的IC50分别为 26、3、4、216、10、200 和 13 nM。它是选择性和 ATP 竞争性PKC 抑制剂。
T11740	Delcasertib KAI-9803,BMS-875944	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Delcasertib (KAI-9803) 是一种有效且选择性的 δ-蛋白激酶 C (δPKC) 抑制剂，可改善急性心肌梗死动物模型的缺血再灌注损伤。
T14989	CMPD101	ROCK; GRK; PKC	Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; GPCR/G Protein; Stem Cells
	CMPD101 是膜透性的 GRK2/3高选择性小分子抑制剂，IC50分别为 18 nM 和 5.4 nM。它针对 GRK1、GRK5 ROCK-2 和 PKCα 的选择性较小，IC50值分别为 3.1 μM，2.3 μM，1.4 μM 和 8.1 μM，可研究心衰疾病。
T35827	Epsilon-V1-2 PKCε Inhibitor Peptide,Protein Kinase Cɛ Inhibitor Peptide,ɛV1-2
	Protein kinase C (PKC ) is a calcium-independent, phospholipid- and diacylglycerol-dependent serine/threonine kinase involved in diverse signaling pathways, including those involved in neuronal signaling, cytoskeletal function, and inflammation.[1] PKC inhibitor peptide is a synthetic peptide corresponding to an amino acid sequence found in the amino terminal C2 domain of most mammalian forms of PKC .[2] It selectively and reversibly inhibits the translocation of PKC to intracellular membrane...
T12148	N-Desmethyltamoxifen hydrochloride	Estrogen Receptor/ERR; Endogenous Metabolite; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Endocrinology/Hormones; Metabolism
	N-Desmethyltamoxifen hydrochloride 是 Tamoxifen 在人体内主要的三苯氧胺代谢物。它是蛋白激酶 C 抑制剂，也是人体 AML 细胞神经酰胺代谢的有效调节因子，可限制神经酰胺糖基化、水解和鞘氨醇磷酸化。
T7648	HA-100	Myosin; PKA; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	HA-100 是蛋白激酶和ROCK 抑制剂，抑制PKG，PKA，PKC 和MLC 激酶的IC50值分别为 4、8、12 和 240 μM。
T6588	Mitoxantrone 米托蒽醌,mitozantrone	Topoisomerase; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair
	Mitoxantrone (mitozantrone) 是一种拓扑异构酶 II 的抑制剂，也可抑制蛋白激酶C (PKC)，IC50值为8.5 μM。
T1911	Afuresertib GSK2110183C,GSK2110183	ROCK; Akt; PKC	Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Stem Cells
	Afuresertib (GSK2110183) 是一个选择性，ATP 竞争性，口服有效的泛 Akt 抑制剂，作用于 Akt1、Akt2和 Akt3，Ki 值分别为 0.08、2、2.6 nM。
T80071	PKCζ/ι pseudosubstrate inhibitor
	PKCζ/ι偽基質抑制劑對PKC酶家族表現廣譜抑制作用，並可能促成記憶功能障礙。
T76412	PKCδ Peptide Substrate
	PKCδPeptide Substrate 是一种δ-typePKC 的特异性底物，其序列与含有 Thr-431 的小鼠 eEF-1α 序列 422-443 相对应。
T83754	PKCδ Substrate TFA Protein Kinase Cδ Substrate
	PKCδ substrate是一种用于PKCδ的肽基底，常用于无细胞及细胞内测定中监测PKCδ活性。
T17019	TCS 21311 NIBR3049	GSK-3; JAK; PKC	Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; PI3K/Akt/mTOR signaling; Stem Cells
	TCS 21311 (NIBR3049) 是一种高选择性JAK3抑制剂，IC50为 8 nM，它的选择性是 JAK1、JAK2 和 TYK2 的100倍以上，还抑制PKCα、PKCθ和GSK3β，IC50值分别为 13、68 和 3 nM。
T14069	A-3 hydrochloride	CaMK; Casein Kinase; PKA; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Neuroscience; Stem Cells; Tyrosine Kinase/Adaptors
	A-3 hydrochloride 是一种细胞可渗透的、可逆的、ATP 竞争性非选择性拮抗剂。它抑制 PKA 、酪蛋白激酶 II 和肌球蛋白轻链激酶，Ki 值分别为4.3 µM、5.1 µM 和7.4 µM。它还抑制 PKC 和酪蛋白激酶 I 的活性，Ki 分别为 47 µM 和 80 µM。
T3689	Ruboxistaurin hydrochloride Ruboxistaurin,LY333531 HCl,LY 333531 hydrochloride,芦布妥林	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Ruboxistaurin hydrochloride (LY 333531 hydrochloride) 是蛋白激酶 C(PKC) 的同工酶选择性抑制剂，竞争性且可逆地抑制 PKCβI 和 PKCβII，IC50 值分别为 4.7 和 5.9 nM。
T6513	Bisindolylmaleimide I GF109203X,Go 6850,3-[1-[3-(二甲氨基)丙基]1H-吲哚-3-基]-4-(吲哚-3-基)1H-吡咯-2,5二酮	PDGFR; PKC	Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors
	Bisindolylmaleimide I (GF109203X) 是一种有效且高度选择性的蛋白激酶 C(PKC) 抑制剂，Ki 值为 14 nM。

化合物

PKC-theta inhibitor hcl

Cat.No: T5817

Synonym: PKC-theta inhibitor

Target: PKC

PKC β pseudosubstrate acetate

Cat.No: TP1955L

Synonym: PKC β pseudosubstrate醋酸盐,Protein kinase C beta pseudosubstrate,PKC beta pseudosubstrate,PKC β pseudosubstrate acetate (172308-76-8 Free base)

Target: PKC

PKC ζ pseudosubstrate acetate

Cat.No: TP1956L

Synonym: PKC ζ pseudosubstrate acetate (799764-07-1 free base)

Target: PKC

PKC-iota inhibitor 1

Cat.No: T8764

Target: PKC

Cat.No: T71993

PKC-theta inhibitor

Cat.No: T5423

Target: PKC

Cat.No: T12494

Target: PKC

PKC fragment (530-558)

Cat.No: T35826

Protein Kinase C 19-31 acetate

Cat.No: TP1053L

Synonym: Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate

Target: PKC

PKC β pseudosubstrate

Cat.No: TP1955

PKC ζ pseudosubstrate

Cat.No: TP1956

PKCβ inhibitor 1

Cat.No: T8376

Synonym: KUN79359

Target: Apoptosis, PKC

PKC-theta inhibitor 1

Cat.No: T12496

Target: PKC

Cat.No: T61604

PKC β pseudosubstrate TFA

Cat.No: T75885

Protein Kinase C (19-31)

Cat.No: TP1053

Synonym: Protein Kinase C 19-31,PKC (19-31)

PKC 20-28,myristoylated

Cat.No: T80509

Synonym: Myristoylated protein kinase C inhibitor 20-28

Target: PKC

Aurora A/PKC-IN-1

Cat.No: T62945

PKC-ε translocation inhibitor peptide

Cat.No: T81449

Target: PKC

PKCε Inhibitor Peptide acetate

Cat.No: T35827L

Synonym: PKCε Inhibitor Peptide acetate(182683-50-7 Free base)

Target: PKC

Cat.No: T17148

Target: PKC

Cat.No: T3211

Synonym: 米哚妥林,N-Benzoylstaurosporine,PKC412,CGP41231,CGP 41251,苯甲酰基十字孢碱

Target: Others, PKC

Cat.No: T35407

Target: PKC

Cat.No: T13314

Target: PKC

Protein Kinase C (19-31) (TFA)(121545-65-1,free)

Cat.No: TP1052

Synonym: PKC (19-31) (TFA),Protein Kinase C (19-31) (TFA)

Cat.No: T5600

Synonym: LXS196

Target: PKC

Bisindolylmaleimide IV

Cat.No: T7659

Target: Others, PKC

Cat.No: T2441

Synonym: TAS 301

Target: PKC

Cat.No: T6515

Synonym: Gö 6976

Target: PKC

Cat.No: T6313

Synonym: Goe 6983

Target: PKC

Cat.No: T26019

Synonym: R-59949,R 59949

Target: Others, PKC

Cat.No: T6278

Synonym: 索曲妥林,AEB071

Target: PKC

Cat.No: T6280

Synonym: LY317615,恩扎妥林

Target: Apoptosis, PKC, Autophagy

Cat.No: T7604

Synonym: Valstar,AD-32,戊柔比星

Target: Antibiotic, PKC

Afuresertib hydrochloride

Cat.No: T7885

Target: ROCK, Akt, PKC

Cat.No: T14943

Target: VEGFR, CDK, PKC

Cat.No: T11740

Synonym: KAI-9803,BMS-875944

Target: PKC

Cat.No: T14989

Target: ROCK, GRK, PKC

Cat.No: T35827

Synonym: PKCε Inhibitor Peptide,Protein Kinase Cɛ Inhibitor Peptide,ɛV1-2

N-Desmethyltamoxifen hydrochloride

Cat.No: T12148

Target: Estrogen Receptor/ERR, Endogenous Metabolite, PKC

Cat.No: T7648

Target: Myosin, PKA, PKC

Cat.No: T6588

Synonym: 米托蒽醌,mitozantrone

Target: Topoisomerase, PKC

Cat.No: T1911

Synonym: GSK2110183C,GSK2110183

Target: ROCK, Akt, PKC

PKCζ/ι pseudosubstrate inhibitor

Cat.No: T80071

PKCδ Peptide Substrate

Cat.No: T76412

PKCδ Substrate TFA

Cat.No: T83754

Synonym: Protein Kinase Cδ Substrate

Cat.No: T17019

Synonym: NIBR3049

Target: GSK-3, JAK, PKC

A-3 hydrochloride

Cat.No: T14069

Target: CaMK, Casein Kinase, PKA, PKC

Ruboxistaurin hydrochloride

Cat.No: T3689

Synonym: Ruboxistaurin,LY333531 HCl,LY 333531 hydrochloride,芦布妥林

Target: PKC

Bisindolylmaleimide I

Cat.No: T6513

Synonym: GF109203X,Go 6850,3-[1-[3-(二甲氨基)丙基]1H-吲哚-3-基]-4-(吲哚-3-基)1H-吡咯-2,5二酮

Target: PDGFR, PKC

Cat. No.	Product Name	Target	Signaling Pathways
TN1557	Decursinol angelate	ERK; VEGFR; PKC; JNK	Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Tyrosine Kinase/Adaptors
	Decursinol angelate 是从朝鲜当归根部分离得到的一种天然产物，是 PKC 激酶的激活剂，有细胞毒性，抗肿瘤和抗炎活性。
T5771	Hypocrellin A	Antibacterial; PKC; Parasite	Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
	Hypocrellin A 是一种天然的PKC 抑制剂，具有光诱导的抗肿瘤、抗真菌和抗病毒活性，还对 MHC 限制性抗原呈递发挥免疫调节作用。
T4S1335	Daphnoretin Dephnoretin,西瑞香素,Thymelol	Influenza Virus; Caspase; PKC	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
	Daphnoretin (Thymelol) 是从了哥王中提取得到的一种天然产物，具有抗癌和抗病毒活性。它通过在 G2/M 期连续阻断细胞并激活 caspase-3 通路导致 HOS 细胞死亡。
T6S0052	Chelerythrine Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine	Apoptosis; BCL; PKC; Autophagy	Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
	Chelerythrine (Broussonpapyrine) 是一种天然生物碱，为有效、选择性的 Ca2+/磷脂依赖性PKC 拮抗剂，IC50值为 0.7 μM。它具有抗肿瘤、抗糖尿病、抗炎的活性。它抑制BclXL-Bak BH3肽结合，IC50为 1.5 μM，并从 BclXL 取代了 Bax。它诱导细胞凋亡和自噬。
T5S2017	Ingenol (-)-Ingenol,巨大戟二萜醇,巨大戟醇	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Ingenol ((-)-Ingenol) 是一种PKC 激活剂，Ki 值为 30 μM，具有抗肿瘤活性。从 Ingenol 酯中配制新的衍生物可能是开发新的先导化合物以重新激活潜伏 HIV 的创新方法。Ingenol mebutate 是治疗光化性角化病的有效方法。
T3419	Chelerythrine chloride 白屈菜红碱,盐酸白屈菜红碱	Apoptosis; BCL; PKC; Autophagy	Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
	Chelerythrine chloride 是一种可渗透细胞的蛋白激酶 C 抑制剂，对磷酸盐受体具有竞争性，而对 ATP 是非竞争性的。它诱导细胞凋亡和自噬。
T22464	1,2-Dimyristoyl-sn-glycerol 1,2-DMG,1,2-二肉豆蔻酸甘油酯	Others; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Others
	1,2-Dimyristoyl-sn-glycerol (1,2-DMG) 是饱和二酰甘油的一种，可作为激活 PKC 的弱活性第二信使。
T4727	Taurolithocholic acid sodium salt 牛磺石胆酸钠,Sodium taurolithocholate	Others; Calcium Channel	Membrane transporter/Ion channel; Metabolism; Others
	Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂，可抑制放射性配体与毒蕈碱 M1 结合。
T11665	Ionomycin calcium SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)	Apoptosis; Calcium Channel; Antibacterial; Antibiotic; PKC	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
	Ionomycin calcium (SQ23377 calcium) 是选择性钙离子载体，也是一种由 Streptomyces conglobatus 产生的抗生素。它对二价阳离子具有高度特异性，还诱导蛋白激酶 C 激活。Ionomycin 促进细胞凋亡。
TN1136	Procyanidin A1 原花青素 A1,Proanthocyanidin A1,原花色素A1	LDL; Calcium Channel; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism
	Procyanidin A1 (Proanthocyanidin A1) 是一种原花青素二聚体，具有抗过敏作用，可抑制蛋白激酶 C 激活下游脱粒或 RBL-213 细胞内部储存的 Ca2+流入。
T3375	Verbascoside 毛蕊花苷,麦角甾苷,Kusaginin,Acteoside,TJC160	Apoptosis; PARP; Antibacterial; PKC; p53; HSV	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Microbiology/Virology
	Verbascoside (Kusaginin) 是从Lantana camara 中得到的糖苷类物质，是具有ATP 竞争性的PKC 抑制剂，IC50值为 25 µM，它还有抗炎，抗肿瘤，抗神经性疼痛等作用。
T3S1416	Decursin Decursinol angelate,前胡素,(+)-Decursin,紫花前胡素	Apoptosis; PKC	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling
	Decursin (Decursinol angelate) 是一种细胞毒性剂，是一种来自朝鲜当归根的有效蛋白激酶 C 激活剂。它通过 Hippo/YAP 信号通路抑制 HepG2 细胞的生长。它通过下调 CXCR7 表达来抑制胃癌中的肿瘤生长，迁移和侵袭。
T7792	Hispidin 6-[(1E)-2-(3,4-二羟基苯基)乙烯基]-4-羟基-2H-吡喃-2-酮	Endogenous Metabolite; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism
	Hispidin 是来自裂蹄木层孔菌的酚类天然产物，是一种 PKC 抑制剂，具有很强的抗氧化、抗癌、抗糖尿病和抗痴呆作用。
T5891	D-ERYTHRO-SPHINGOSINE trans-4-Sphingenine,erythro-C18-Sphingosine,Erythrosphingosine,鞘氨醇,D-鞘氨醇	Phosphatase; Endogenous Metabolite; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism
	D-erythro-Sphingosine (trans-4-Sphingenine) 是一种非常有效的p32激酶活化剂，EC50为 8 μM。它也是一种PP2A 激活剂，抑制蛋白激酶 C (PKC)。
TN1299	Desmethylglycitein 4',6,7-三羟基异黄酮,4',6,7-三羟异黄酮,6-羟基大豆苷元,6,7,4'-Trihydroxyisoflavone	PI3K; CDK; PKC	Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
	Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) 是大豆中苷元的代谢产物，具有抗氧化性和抗癌活性。它是蛋白激酶 C(PKC)α 的直接抑制剂，抑制正常人皮肤成纤维细胞中的太阳紫外线诱导的基质金属蛋白酶1。它在体内直接结合CDK1和CDK2，抑制 CDK1 和 CDK2 活性。
T9605	Sangivamycin BA-90912,桑霉素,NSC 65346	Nucleoside Antimetabolite/Analog; PKC	Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair
	Sangivamycin (NSC-65346) 是蛋白激酶 C (PKC) 的有效抑制剂 (Ki = 10 μM)。 Sangivamycin 对多种人类癌症细胞具有抗增殖活性。
T16791	Rottlerin Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525	CaMK; Apoptosis; Others; HIV Protease; PKA; PKC; Autophagy	Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Neuroscience; Others; Proteases/Proteasome; Tyrosine Kinase/Adaptors
	Rottlerin (NSC-56346) 是一种从Mallotus Philippinensis 中得到的天然产物，是 PKC 的特异性抑制剂，抑制HIV-1整合和狂犬病病毒感染。它通过活化 caspase 3 诱导细胞凋亡.
TQ0198	Phorbol 12-myristate 13-acetate 佛波醇12-十四酸酯13-乙酸酯,PMA	NF-κB; S1P Receptor; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; GPCR/G Protein; NF-κB
	Phorbol 12-myristate 13-acetate (PMA) 属于佛波酯类天然产物，是一种 PKC、SphK、NF-κB 的激活剂。Phorbol 12-myristate 13-acetate 可诱导 THP1 细胞分化。
T2A2481	Taurochenodeoxycholic Acid Chenodeoxycholyltaurine,TCDCA,Chenyltaurine,Taurochenodeoxycholate,12-Deoxycholyltaurine,牛磺鹅去氧胆酸	Apoptosis; TNF; Caspase; Endogenous Metabolite	Apoptosis; Metabolism; Proteases/Proteasome
	Taurochenodeoxycholic Acid (12-Deoxycholyltaurine) 是动物胆汁酸的主要生物活性物质之一，可诱导细胞凋亡，具有明显的抗炎和免疫调节作用。
TN2215	Taurochenodeoxycholic acid sodium 牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠	Apoptosis; Endogenous Metabolite	Apoptosis; Metabolism
	Taurochenodeoxycholic acid sodium (Sodium taurochenodeoxycholate) 是动物胆汁酸的主要生物活性物质之一。它可诱导细胞凋亡，具有抗炎和免疫调节作用。
T6S0923	Hypericin Hypericine,金丝桃素,Cyclosan	Apoptosis; Antiviral; Influenza Virus; Tyrosine Kinases; Antibacterial; PKC	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Tyrosine Kinase/Adaptors
	Hypericin (Cyclosan) 是贯叶连翘的提取物，有抗菌、抗病毒、抗肿瘤和抗抑郁作用。
T2851	Daphnetin 7,8-Dihydroxycoumarin,Daphnetol,瑞香素	EGFR; PKA; PKC; Parasite; Autophagy	Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
	Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物，有抗氧化、抗炎、抗疟疾和解热作用，可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。
T6680	Staurosporine Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素	Apoptosis; PKA; Antibacterial; Antibiotic; Src; PKC; Antifungal	Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
	Staurosporine (AM-2282) 是一种蛋白激酶抑制剂，对 PKC、PKA、c-Fgr、Phosphorylase kinase 和 TAOK2 均有抑制活性 (IC50=6/15/2/3/3000 nM)，具有 ATP 竞争性和非选择性。Staurosporine 也可以诱导凋亡。
TN1047	Ingenol mebutate Ingenol 3-Angelate,巨大戟醇甲基丁烯酸酯,PEP005	gp120/CD4; HIV Protease; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
	Ingenol mebutate (Ingenol 3-Angelate) 是 PKC 的有效激动剂，包括 PKC-α、PKC-β、PKC-γ、PKC-δ 和 PKC-ε，Kis 为 0.3、0.105、0.162、0.376 和 0.171 nM。 Ingenol mebutate 具有抗炎和抗肿瘤活性。
T4950	1,2-Dipalmitoyl-sn-glycerol 1,2-双棕榈酸甘油酯,(S)-1,2-Dipalmitin	Endogenous Metabolite; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism
	1,2-Dipalmitoyl-sn-glycerol ((S)-1,2-Dipalmitin) 是内源性代谢产物的一种。
TN4114	Gardenin A	ERK; LDL; MAPK; PKA; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Metabolism; Tyrosine Kinase/Adaptors
	Gardenin A 通过激活 MAPK/ERK、PKC 和 PKA 表现出神经营养作用。 Gardenin A 具有抗抑郁、抗惊厥和抗焦虑作用。
T2S0531	Pinoresinol dimethyl ether (+)-Eudesmin,松脂素二甲醚	Others; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Others
	Pinoresinol dimethyl ether 是一种非酚性呋喃木质素，从 Magnolia kobus 茎皮中分离得到，具有神经活性。它可刺激上游 MAPK、PKC 和 PKA 通路，诱导 PC12 细胞神经突起生长。
T3927	Phellopterin	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Phellopterin 是一种分离自P. trifoliata 中的天然产物。它能够调节 Akt 和 PKC 通路，抑制 TNF-alpha 诱导的 VCAM-1 表达，进而减少单核细胞与内皮细胞的粘附。
T5239	Cholesteryl sulfate sodium Cholesterol 3-Sulfate Sodium Salt,胆固醇硫酸酯钠盐,Sodium Cholesteryl Sulfate	Endogenous Metabolite; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism
	Cholesteryl sulfate sodium (Sodium Cholesteryl Sulfate) 是内源性代谢产物的一种。
T7285	Ionomycin	Calcium Channel	Membrane transporter/Ion channel; Metabolism
	Ionomycin 是一种钙离子载体和一种结合钙离子(Ca2+)的抗生素。它是由联合链霉菌(Streptomyces conglobatus)产生的。它在研究中用于提高细胞内钙水平(Ca2+)，并作为了解 Ca2+跨生物膜运输的研究工具。Ionomycin 可促进细胞凋亡，诱导蛋白激酶 C (PKC)活化。
T3863	Chikusetsusaponin IVa 竹节参皂苷IVa,Calenduloside F,竹节人参皂苷 IVA	AMPK	Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
	Chikusetsusaponin IVa (Calenduloside F) 是一种三萜皂苷中主要的活性成分，是一种蛋白激酶的激活剂，对血栓及一些代谢性疾病具有抵抗作用。
T3836	Eudesmin	MAPK; S6 Kinase	MAPK; PI3K/Akt/mTOR signaling
	Eudesmin 通过抑制S6K1信号通路来干扰成脂分化，具有抗肿瘤、抗炎和抗菌活性。
T3753	Sinapinic Acid Sinapic acid,芥子酸,Synapoic acid	Apoptosis; RAAS; Reactive Oxygen Species; HDAC	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
	Sinapinic Acid (Synapoic acid) 是从 Hydnophytum formicarumJack. 根中分离到的酚类，是HDAC 抑制剂，对ACE-I 的活性也有抑制作用。它有抗肿瘤活性，诱导肿瘤细胞凋亡，具有抗氧化、抗糖尿病的作用。
T6S1740	Nardosinone 苷松新酮,甘松新酮	Others	Others
	Nardosinone 是一个 dbcAMP 和 staurosporine 的神经生成作用增强剂，分离自Nardostachys chinensis 中。Nardosinone 可能成为一种有用的药理学工具，不仅可用于研究神经生长因子 (NGF) 的作用机理，而且可用于研究神经毒性物质的作用机理。
T5796	Plantainoside D Isoplantamajoside,车前草苷D	RAAS; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Endocrinology/Hormones
	Plantainoside D (Isoplantamajoside) 可以抑制 ACE ，IC50=2.17 mM。Plantainoside D 也是IKK-β抑制剂。
T13605	Cercosporin	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	Cercosporin is produced by a plant pathogen, Cercosporakikuchii, and the elsinochromes. Cercosporin is a potent photosensitizer with a short activation wavelength. Cercosporin contains the perylene quinone structural features necessary for PKC activity (I
T17198	UCN-02 7-epi-Hydroxystaurosporine	Others	Others
	UCN-02 is a selective protein kinase C inhibitor produced by Streptomyces strain N-12 (IC50s: 62 nM and 250 nM for PKC and protein kinase A (PKA), respectively).
T15638	K-252c	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	K-252c is a staurosporine analog isolated from Nocardiopsis sp. and is a cell-permeable PKC inhibitor (IC50: 2.45 μM). K-252c also inhibits β-lactamase, chymotrypsin, and malate dehydrogenase. K-252c causes apoptosis in human chronic myelogenous leukemia cancer cells.
T0610	Piceatannol 白皮杉醇,trans-Piceatannol,Astringenin	Apoptosis; Serine/threonin kinase; PKA; Syk; PKC; Autophagy	Angiogenesis; Apoptosis; Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; Metabolism; Tyrosine Kinase/Adaptors
	Piceatannol (Astringenin) 是一种Syk 抑制剂，可降低由 TNF 诱导的 iNOS 表达，可研究急性肺损伤。它是存在于各种水果和蔬菜中天然存在的多酚二苯乙烯，可诱导细胞自噬和凋亡，具有抗癌和抗炎特性。
T15636	K-252a Antibiotic K 252a,Antibiotic SF 2370,SF2370	Others	Others
	K-252a is a staurosporine analog isolated from Nocardiopsis sp. soil fungi. K-252a inhibits protein kinase (IC50: 470 nM, 140 nM, 270 nM, and 1.7 nM for PKC, PKA, Ca2+/calmodulin-dependent kinase type II, and phosphorylase kinase, respectively).
T75565	Vanicoside A
	Vanicoside A 是一种来自Polygonum pensylvanicum 的蛋白激酶 C (PKC)抑制剂。
T35895	Ingenol 3,20-dibenzoate
	Ingenol 3,20-dibenzoate is a powerful activator of protein kinase C (PKC) isoforms. It effectively induces the translocation of nPKC-delta, -epsilon, and -theta as well as PKC-mu from the cytosolic fraction to the particulate fraction. Through de novo synthesis of macromolecules, it triggers apoptosis with characteristic morphology. Moreover, Ingenol 3,20-dibenzoate enhances IFN-γ production and degranulation in NK cells, particularly when stimulated by NSCLC cells[1][2].
TN2844	(2R,3S)-Dihydrodehydroconiferyl alcohol	MAPK; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK
	(2R,3S)-Dihydrodehydroconiferyl alcohol can induce neurite outgrowth and enhance NGF-induced neurite outgrowth from PC12 cells by amplifying up-stream steps such as MAPK and PKC.
T15637	K-252b	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	K-252b is an indolocarbazole isolated from the actinomycete Nocardiopsis and is a PKC inhibitor. K-252b can be used to inhibit extracellular kinases of cells in culture because it can’t pass through the cell membrane freely.
TN2799	20-Deoxyingenol 3-angelate	PKC	Chromatin/Epigenetic; Cytoskeletal Signaling
	20-Deoxyingenol 3-angelate and ingenol 20-acetate 3-angelate are known as promoters of tumors of mouse skin. 20-Deoxyingenol 3-angelate can induce significant platelet aggregation accompanied by induction of phosphorylation of PKC substrates in platelets,
T68802	Vibsanin A
	Vibsanin A，作为一种蛋白激酶C (PKC) 激活剂，展现出对人类癌细胞系的抗增殖活性，同时也兼具HSP90抑制剂的功能。
T14831	Bryostatin 1	HIV Protease; PKC	Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
	Bryostatin 1 is a natural macrolide isolated from the bryozoan Bugula neritina and is a CNS)permeable PKC modulator. Bryostatin 1 binds to the isolated C1 domain of Munc13-1 and the full-length Munc13-1 protein (Kis: 8.07 nM and 0.45 nM).
TN3160	6-Deoxyisojacareubin	PKC; Antifection	Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
	6-Deoxyisojacareubin shows moderate inhibitory activity against the QGY-7703 cell line, with the IC50 value of 9.65 uM; it also possesses potency in the inhibition of protein kinase C (PKC).
TN3655	Cimiside E	ERK; TNF; ROS; Akt; PI3K; PKC; PPAR	Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Immunology/Inflammation; MAPK; Metabolism; PI3K/Akt/mTOR signaling
	Cimiside E has anti-inflammatory activity, it selectively inhibits TNF-α-induced expression of VCAM-1 at least by upregulation of PPAR-γ, and signals for ERK1/2, PI3K, and PKC are involved in this effect.Cimiside E may be an effective chemopreventive agen
TN4300	Isojacareubin	MAPK; PKC; Antifection	Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Microbiology/Virology
	Isojacareubin displays potent activity against H. pylori HP40 clinical isolate with MIC 23.9 uM, which is approximately two times greater than that of the standard drug amoxicillin. Isojacareubin is a potent inhibitor of protein kinase C (PKC), suppresses
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天然产物

Decursinol angelate

Cat.No: TN1557

Target: ERK, VEGFR, PKC, JNK

Cat.No: T5771

Target: Antibacterial, PKC, Parasite

Cat.No: T4S1335

Synonym: Dephnoretin,西瑞香素,Thymelol

Target: Influenza Virus, Caspase, PKC

Cat.No: T6S0052

Synonym: Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine

Target: Apoptosis, BCL, PKC, Autophagy

Cat.No: T5S2017

Synonym: (-)-Ingenol,巨大戟二萜醇,巨大戟醇

Target: PKC

Chelerythrine chloride

Cat.No: T3419

Synonym: 白屈菜红碱,盐酸白屈菜红碱

Target: Apoptosis, BCL, PKC, Autophagy

1,2-Dimyristoyl-sn-glycerol

Cat.No: T22464

Synonym: 1,2-DMG,1,2-二肉豆蔻酸甘油酯

Target: Others, PKC

Taurolithocholic acid sodium salt

Cat.No: T4727

Synonym: 牛磺石胆酸钠,Sodium taurolithocholate

Target: Others, Calcium Channel

Ionomycin calcium

Cat.No: T11665

Synonym: SQ23377 calcium,罗红霉素钙盐(链霉菌属载体)

Target: Apoptosis, Calcium Channel, Antibacterial, Antibiotic, PKC

Cat.No: TN1136

Synonym: 原花青素 A1,Proanthocyanidin A1,原花色素A1

Target: LDL, Calcium Channel, PKC

Cat.No: T3375

Synonym: 毛蕊花苷,麦角甾苷,Kusaginin,Acteoside,TJC160

Target: Apoptosis, PARP, Antibacterial, PKC, p53, HSV

Cat.No: T3S1416

Synonym: Decursinol angelate,前胡素,(+)-Decursin,紫花前胡素

Target: Apoptosis, PKC

Cat.No: T7792

Synonym: 6-[(1E)-2-(3,4-二羟基苯基)乙烯基]-4-羟基-2H-吡喃-2-酮

Target: Endogenous Metabolite, PKC

D-ERYTHRO-SPHINGOSINE

Cat.No: T5891

Synonym: trans-4-Sphingenine,erythro-C18-Sphingosine,Erythrosphingosine,鞘氨醇,D-鞘氨醇

Target: Phosphatase, Endogenous Metabolite, PKC

Desmethylglycitein

Cat.No: TN1299

Synonym: 4',6,7-三羟基异黄酮,4',6,7-三羟异黄酮,6-羟基大豆苷元,6,7,4'-Trihydroxyisoflavone

Target: PI3K, CDK, PKC

Cat.No: T9605

Synonym: BA-90912,桑霉素,NSC 65346

Target: Nucleoside Antimetabolite/Analog, PKC

Cat.No: T16791

Synonym: Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525

Target: CaMK, Apoptosis, Others, HIV Protease, PKA, PKC, Autophagy

Phorbol 12-myristate 13-acetate

Cat.No: TQ0198

Synonym: 佛波醇12-十四酸酯13-乙酸酯,PMA

Target: NF-κB, S1P Receptor, PKC

Taurochenodeoxycholic Acid

Cat.No: T2A2481

Synonym: Chenodeoxycholyltaurine,TCDCA,Chenyltaurine,Taurochenodeoxycholate,12-Deoxycholyltaurine,牛磺鹅去氧胆酸

Target: Apoptosis, TNF, Caspase, Endogenous Metabolite

Taurochenodeoxycholic acid sodium

Cat.No: TN2215

Synonym: 牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠

Target: Apoptosis, Endogenous Metabolite

Cat.No: T6S0923

Synonym: Hypericine,金丝桃素,Cyclosan

Target: Apoptosis, Antiviral, Influenza Virus, Tyrosine Kinases, Antibacterial, PKC

Cat.No: T2851

Synonym: 7,8-Dihydroxycoumarin,Daphnetol,瑞香素

Target: EGFR, PKA, PKC, Parasite, Autophagy

Cat.No: T6680

Synonym: Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素

Target: Apoptosis, PKA, Antibacterial, Antibiotic, Src, PKC, Antifungal

Ingenol mebutate

Cat.No: TN1047

Synonym: Ingenol 3-Angelate,巨大戟醇甲基丁烯酸酯,PEP005

Target: gp120/CD4, HIV Protease, PKC

1,2-Dipalmitoyl-sn-glycerol

Cat.No: T4950

Synonym: 1,2-双棕榈酸甘油酯,(S)-1,2-Dipalmitin

Target: Endogenous Metabolite, PKC

Cat.No: TN4114

Target: ERK, LDL, MAPK, PKA, PKC

Pinoresinol dimethyl ether

Cat.No: T2S0531

Synonym: (+)-Eudesmin,松脂素二甲醚

Target: Others, PKC

Cat.No: T3927

Target: GABA Receptor

Cholesteryl sulfate sodium

Cat.No: T5239

Synonym: Cholesterol 3-Sulfate Sodium Salt,胆固醇硫酸酯钠盐,Sodium Cholesteryl Sulfate

Target: Endogenous Metabolite, PKC

Cat.No: T7285

Target: Calcium Channel

Chikusetsusaponin IVa

Cat.No: T3863

Synonym: 竹节参皂苷IVa,Calenduloside F,竹节人参皂苷 IVA

Target: AMPK

Cat.No: T3836

Target: MAPK, S6 Kinase

Cat.No: T3753

Synonym: Sinapic acid,芥子酸,Synapoic acid

Target: Apoptosis, RAAS, Reactive Oxygen Species, HDAC

Cat.No: T6S1740

Synonym: 苷松新酮,甘松新酮

Target: Others

Plantainoside D

Cat.No: T5796

Synonym: Isoplantamajoside,车前草苷D

Target: RAAS, PKC

Cat.No: T13605

Target: PKC

Cat.No: T17198

Synonym: 7-epi-Hydroxystaurosporine

Target: Others

Cat.No: T15638

Target: PKC

Cat.No: T0610

Synonym: 白皮杉醇,trans-Piceatannol,Astringenin

Target: Apoptosis, Serine/threonin kinase, PKA, Syk, PKC, Autophagy

Cat.No: T15636

Synonym: Antibiotic K 252a,Antibiotic SF 2370,SF2370

Target: Others

Cat.No: T75565

Ingenol 3,20-dibenzoate

Cat.No: T35895

(2R,3S)-Dihydrodehydroconiferyl alcohol

Cat.No: TN2844

Target: MAPK, PKC

Cat.No: T15637

Target: PKC

20-Deoxyingenol 3-angelate

Cat.No: TN2799

Target: PKC

Cat.No: T68802

Cat.No: T14831

Target: HIV Protease, PKC

6-Deoxyisojacareubin

Cat.No: TN3160

Target: PKC, Antifection

Cat.No: TN3655

Target: ERK, TNF, ROS, Akt, PI3K, PKC, PPAR

Cat.No: TN4300

Target: MAPK, PKC, Antifection

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