93
83
12
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T76774 |
Ponsegromab
PF 06946860 |
TGF-beta/Smad | Stem Cells |
Ponsegromab (PF 06946860) 是一种具有选择性和有效性的人源化抗 GDF15 抗体抑制剂。 Ponsegromab 具有抗恶病质活性,通过与 GDF15 结合来阻止其与 GFRAL 结合,从而中断 GDF15/GFRAL 介导的信号传导。 Ponsegromab 具有潜在的抗癌活性,可用于治疗患有癌症厌食-恶病质综合征的癌症患者。 | |||
T3467 |
Miransertib
ARQ-092,AKT inhibitor 2 |
Akt; Parasite | Cytoskeletal Signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling |
Miransertib (ARQ-092) 是一种具有口服活性的,选择性和变构性Akt 抑制剂。它有效抑制利什曼原虫,还是 AKT1-E17K 突变蛋白抑制剂,可研究PI3K/AKT 驱动的肿瘤和 Proteus 综合征。 | |||
T68141 |
Seganserin
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Seganserin 是一种非选择性5-羟色胺2-HT 受体拮抗剂,可逆转了氟西汀和喹帕嗪对黄体酮诱导的食欲亢进,抑郁和痛觉的抑制作用,逆转氟西汀和喹帕嗪诱导的抗抑郁和镇痛作用。 | |||
T1066 |
Ketanserin
R41468,凯他色林,Ketanserin tartrate,酮色林,Ketanserinum |
Potassium Channel; 5-HT Receptor; Autophagy | Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Ketanserin (Ketanserinum) 是一种喹唑啉衍生物和 5-羟色胺受体亚型 2 拮抗剂,具有潜在的抗高血压和抗血小板活性。它也浓度依赖性抑制 hERG 电流,IC50为 0.11 μM。 | |||
T7350 |
Nelotanserin
1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲,APD125 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Nelotanserin (APD125) 是5-HT2A 强完全逆向激动剂,5-HT2C 中等强度的部分反向激动剂和5-HT2B 的弱反向激动剂,IC50s 值分别为 1.7、79 和 791 nM。 | |||
T6946 |
Pimavanserin tartrate
ACP-103,ACP-103 tartrate,Nuplazid,Pimavanserin,匹莫范色林 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Pimavanserin tartrate (Nuplazid) 是一种有效的5-HT 2A 受体反向激动剂,pIC50和 pKi 值分别为8.73和9.3,用于治疗与帕金森病相关的精神病。 | |||
T6247 |
Onvansertib
NMS-P937,NMS-1286937 |
Apoptosis; PLK | Apoptosis; Cell Cycle/Checkpoint |
Onvansertib (NMS-1286937) 是一种可口服的高选择性PLK1抑制剂,IC50值为 2 nM。 | |||
T16759 |
Ritanserin
利坦丝林,R 55667 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Ritanserin (R 55667) 是一种长效、高效、相对选择性、可口服的5-HT2受体拮抗剂,IC50值为 0.9 nM。 | |||
T1478 |
Ondansetron hydrochloride dihydrate
盐酸昂丹司琼,SN 307,NSC 665799,GR 38032,Ondansetron hydrochloride |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Ondansetron hydrochloride dihydrate (GR 38032) 是5- HT3受体拮抗剂,可治疗化疗后的恶心和呕吐,有抗焦虑和抗精神病作用。 | |||
T5389 |
Volinanserin
M 100907,MDL100907,氟利色林 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Volinanserin (MDL100907) 是选择性的5-HT2受体拮抗剂,Ki 值为 0.36 nM,可用于精神疾病的研究。它对 5-HT2 受体的选择性比 5-HT1c、α-1 肾上腺素能受体和 σ 受体高 300 倍。 | |||
T22964 |
Glemanserin
MDL11939 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Glemanserin (MDL11939) 是一种特异性 5-HT2A 拮抗剂,对兔、人和大鼠 5-HT2A 的 Ki 值为 0.54 nM、2.5 nM 和 2.89 nM。 | |||
T37979 |
N-Desmethyl Pimavanserin
AC-279 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
N-Desmethyl Pimavanserin (AC-279) 是 Pimavanserin (一种 5-HT2A 受体反向激动剂)的活性代谢物,可用于治疗失眠等睡眠障碍。 | |||
T8451 |
Tropanserin
MDL 72422 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tropanserin (MDL 72422) 是一种 5-羟色胺受体拮抗剂,抑制5-HT3受体活性。Tropanserin 具有抗焦虑活性,可用于治疗抑郁症和认知障碍。 | |||
T62083 |
Camonsertib
ATR inhibitor 4,RP-3500 |
ATM/ATR | DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling |
Camonsertib (RP-3500) 是一种选择性的、口服具有活力的 ATR 激酶抑制剂 (ATRi),在生化试验中的 IC50: 1.00 nM,表现出有效的抗肿瘤作用。RP-3500 对 ATR 的选择性是 mTOR 的 30 倍 (IC50: 120 nM),是 ATM、DNA-PK 和 PI3Kα 激酶的 2,000 倍以上。 | |||
T23445 |
Anxiolytic/nonsedative agent-1
TCS 1205 |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Anxiolytic/nonsedative agent-1 (TCS 1205) 是一种有效的选择性 GABAA 激动剂。Anxiolytic/nonsedative agent-1 对牛脑膜中的 BzR 显示出明显的亲和力,对 α1β2γ2、α2β2γ2、α5β3γ2 的 Kis 分别为 14、121、239 nM。Anxiolytic/nonsedative agent-1 在体外表现出 α2 选择性功效,在体内表现出抗焦虑选择性作用。 | |||
T14968 |
Cinanserin hydrochloride
SQ 10643 |
Influenza Virus; 5-HT Receptor | GPCR/G Protein; Microbiology/Virology; Neuroscience |
Cinanserin hydrochloride (SQ 10643) 是一种高亲和力拮抗剂,对 5-HT2 受体的Ki 值为 41 nM。它也是严重急性呼吸综合征冠状病毒的 3C 样蛋白酶抑制剂。 | |||
T1517 |
Benserazide hydrochloride
Benserazide HCl,盐酸苄丝肼,Serazide,Ro 4-4602 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Benserazide hydrochloride (Ro 4-4602) 是一种芳香族 L-氨基酸脱羧酶(AADC)的抑制剂,常用于帕金森病。 | |||
T23631 |
Adatanserin
WY-50324,WY 50324,WAY SEB 324,WY50324 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Adatanserin (WY 50324) 是一种混合型 5-HT1A 受体部分激动剂,也是一种 5-HT2A 和 5-HT2C 受体拮抗剂,具有潜在的神经保护活性,可用于研究焦虑和抑郁症。 | |||
T67914 |
Insecticidal agent 364
|
mTOR; Autophagy | Autophagy; PI3K/Akt/mTOR signaling |
Insecticidal agent 364是一种雷帕霉素激酶靶蛋白的选择性小分子抑制剂。Insecticidal agent 364具有抗肿瘤活性,通过抑制mTOR, Insecticidal agent 364旨在破坏参与癌细胞生长和存活的信号通路,从而潜在地抑制肿瘤生长。 | |||
T3350 |
Selonsertib
GS-4997 |
Apoptosis; ASK; MAPK | Apoptosis; MAPK |
Selonsertib (GS-4997) 是一种选择性的,具有生物口服可利用的凋亡信号调节激酶1 抑制剂,pIC50为 8.3。它具有潜在的抗炎、抗肿瘤和抗纤维化活性。 | |||
T21428 |
Mianserin
Lantanon,Lumin,Norval,Lerivon,Depnon |
Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Mianserin 是H1受体反向激动剂,是四环抗抑郁药(TeCA)治疗家族中的一种精神活性化合物,具有抗抑郁、抗焦虑、止吐、促氧、催眠和抗组胺作用,可作为去甲肾上腺素和特定的血清素联合用药能治疗抑郁症。 | |||
T1180 |
Blonanserin
布南色林,AD-5423 |
Dopamine Receptor; Sigma receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Blonanserin (AD-5423) 是一种有效的5-HT2A 和多巴胺 D2 受体拮抗剂,Ki 为 0.812 和 0.142 nM,是一种非典型的抗精神病试剂。 | |||
T2076 |
Pimavanserin
ACP-103,匹莫范色林 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Pimavanserin (ACP-103) 是特异性的 5-HT2A 受体反向激动剂,在基于细胞的功能测定中,平均 pIC50值为8.7。它是非典型抗精神病药,用于治疗帕金森病患者的幻觉和精神病。 | |||
T15270 |
Fananserin
RP 62203,法南色林 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Fananserin 是一种有效的、特异性的、口服活性的 5-HT2 拮抗剂(大鼠 5-HT2A 的 Ki = 0.37 nM)。 Fananserin 是人 D4 受体的拮抗剂 (Ki = 2.93 nM)。 | |||
T6615 |
Ondansetron
GR-C507/75,GR 38032,昂丹司琼,GR 38032F,SN 307,恩丹西酮 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Ondansetron (GR 38032) 是一种血清素 5-HT3 受体拮抗剂,主要用作止吐剂。 | |||
T27020 |
Cilansetron
KC-9946,KC9946,DU-123265,DU123265 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Cilansetron 是一种具有有效性和选择性的 5-HT3 受体拮抗剂,可用于结肠炎引发的相关疾病。 | |||
T6616 |
Ondansetron hydrochloride
SN 307,盐酸昂丹司琼,帕罗西汀杂质A,Ondansetron HCl,Emeset,GR 38032 HCl,NSC 665799,Zofran |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Ondansetron hydrochloride (Zofran) 是5-HT3受体的拮抗剂,可用作化疗后止吐剂。 | |||
T4297 |
Flibanserin
BIMT-17BS,氟立班丝氨,Girosa,BIMT-17 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Flibanserin (Girosa) 一种具有口服活性的 5-HT1A 受体激动剂和 5-HT2A 受体拮抗剂,Ki 值分别为 1 和 49 nM。它与多巴胺 D4 受体结合,Ki 值在 4 到 24 nM 之间。它是一种血清素能抗抑郁药,用于治疗性欲减退症。 | |||
T9833 |
Opiranserin hydrochloride
|
P2X Receptor; GlyT; 5-HT Receptor | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Opiranserin hydrochloride 是甘氨酸转运蛋白 2 型 (GlyT2) 和 5-羟色胺受体 2A (5HT2A) 的双重拮抗剂,IC50 分别为 0.86 和 1.3 μM。它显示对 rP2X3 的拮抗活性 (IC50=0.87 μM)。它正在开发为用于治疗术后疼痛的注射剂。 | |||
T1066L |
Ketanserin tartrate
KJK 945 tartrate,KJK-945 tartrate,KJK945 tartrate |
5-HT Receptor; Serotonin Transporter; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Ketanserin tartrate (KJK-945 tartrate) 是 5-HT2A 受体和α1-肾上腺素能受体拮抗剂,具有抗高血压活性,抑制血清素诱导的血管收缩和血小板活化,可用于研究系统性硬化症。 | |||
T29645 |
Adatanserin hydrochloride
WY50324 hydrochloride |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Adatanserin hydrochloride (WY50324 hydrochloride) 是一种新型 5-HT(1A)/5-HT(2) 受体配体,具有潜在的神经保护作用,抑制内源性氨基酸缺血性外排,可用于研究抑郁症和焦虑症。 | |||
T22243 |
Anserine
L-鹅肌肽,L-Anserine |
Endogenous Metabolite | Metabolism |
Anserine (L-Anserine) 是 Carnosine 的甲基化形式,是口服具有活性的天然二肽,存在于脊椎动物的骨骼肌。它不会被血清肌肽酶裂解,能够作为生化缓冲液,螯合剂,抗糖化剂和抗氧化剂。它能够改善阿尔茨海默氏病模型小鼠的记忆功能。 | |||
T12477 |
Uzansertib phosphate
INCB053914 phosphate |
Pim | Chromatin/Epigenetic; JAK/STAT signaling |
Uzansertib phosphate (INCB053914 phosphate) 是一种可口服的 ATP 竞争性泛-PIM 激酶抑制剂,对多种血液肿瘤细胞系具有广泛的抗增殖活性,对 PIM1、PIM2 和 PIM3 的 IC50分别为 0.24 、30 和 0.12 nM。 | |||
T11217 |
Eplivanserin
依利色林,SR-46349 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Eplivanserin (SR-46349) 是一种有效和特异性的 5-HT2A 受体拮抗剂,Kd 值为 1.14 nM,在大鼠皮质膜中 IC50 值为 5.8 nM。 | |||
T27020L |
isomer-Cilansetron
|
Others | Others |
isomer-Cilansetron 是 Cilansetron 的异构体。 | |||
T29913 |
Altanserin
R-53200,R53200,R 53200 |
||
Altanserin can binds to the 5-HT2A receptor. Labeled with the isotope fluorine-18 it is used as a radioligand in positron emission tomography (PET) studies of the brain. | |||
T12446 |
Phenserine
(-)-Eseroline phenylcarbamate,(-)-Phenserine |
AChR | Neuroscience |
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE. | |||
T39090 |
Uzansertib
INCB053914 |
||
Uzansertib (INCB053914) is a potent ATP-competitive pan-PIM kinase inhibitor. It exhibits exceptional inhibitory activity against PIM1, PIM2, and PIM3 with IC50 values of 0.24 nM, 30 nM, and 0.12 nM, respectively. Furthermore, Uzansertib demonstrates significant anti-proliferative effects against an assorted range of hematologic tumor cell lines. | |||
T39126 |
Zunsemetinib
CDD-450,ATI-450 |
||
Zunsemetinib (CDD-450) is a potent and specific inhibitor of the p38α-MK2 pathway, exerting its effects through oral administration. It has proven activity against immuno-inflammatory diseases, making it a valuable tool for research in this area. | |||
T26768 |
Benanserin HCl
Benanserin Hydrochloride,BAS,Benanserin,Benzyl antiserotonin |
||
Benanserin HCl is a serotonin antagonist. It causes psychotropic effects in humans. | |||
T34918 |
Trelanserin
SL650472,SL-650472,SL 650472 |
||
Trelanserin (SL-650472) is an antagonist of the serotonin receptor. | |||
T1517L |
Benserazide
Ro-44602,Ro44602,Ro 44602,Serazide |
||
Benserazide is an inhibitor of dopa decarboxylase. It is often given with levodopa in the treatment of Parkinson's to prevent the conversion of levodopa to dopamine in the periphery, thereby increasing the amount that reaches the central nervous system an | |||
T9901A-011 |
Lunsekimig
SAR443765 |
||
Lunsekimig (SAR443765) 是一种 IL-13/TSLP 双抗,将靶向 IL-13 和靶向 TSLP 的重链可变区 (VHH) 连接在一起的纳米抗体,可用于哮喘研究。 | |||
T16399 |
Opiranserin
|
P2X Receptor; GlyT; 5-HT Receptor | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Opiranserin 是一种非阿片类和非 NSAID 镇痛候选药物,是 2 型甘氨酸转运蛋白 (GlyT2) 和 5-羟色胺受体 2A (5HT2A) 的双重拮抗剂,IC50分别为 0.86 和 1.3 μM。它可用于术后疼痛的研究,对 rP2X3 有拮抗作用,IC50为0.87 μM。 | |||
T82064 |
Insecticidal agent 6
|
Parasite | Microbiology/Virology |
Insecticidal agent 6(化合物 Im)是昆虫兰尼碱受体(RyRs)的抑制剂,该化合物对 S. frugiperda RyRs 具有强效的抑制作用,其 EC50 值为0.6308 µM。该化合物在鳞翅目害虫中展现出卓越的杀虫效果,适用于病虫害研究。 | |||
T25568 |
Ketanserinol
Reduced ketanserin |
||
Ketanserinol is the metabolite of ketanserin. Ketanserin is a hypotensive drug with 5-HT2 receptor antagonism, used to reverse pulmonary hypertension caused by protamine. | |||
T83106 |
Anselamimab
|
||
Anselamimab (CAEL-101) 为一种靶向血清淀粉样蛋白 A1 (SAA1) 的人源 IgG1-κ 抗淀粉样蛋白原纤维抗体。 | |||
T30936 |
Cilansetron Hydrochloride
KC-9946,KC9946,KC 9946 |
||
Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance. | |||
T70439 |
Galdansetron hydrochloride
|
||
Galdansetron hydrochloride is a serotonin antagonist and anti-emetic. | |||
T71292 |
Rivipansel sodium
|
||
Rivipansel sodium is a glycomimetic drug candidate that acts as a pan-selectin antagonist and reverses acute vascular occlusions in sickle cell mice. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN2245 |
Sunset Yellow FCF
Food Yellow 3,Orange Yellow S,Sunset yellow,CI 15985 |
Androgen Receptor | Endocrinology/Hormones |
Sunset Yellow FCF (Sunset yellow) 是一种橙色偶氮染料,吸光度具有pH 依赖性。Sunset Yellow FCF 可在食品,化妆品和药品中使用,在许多食品中用作着色剂食品添加剂,它们可能具有细胞毒性和遗传毒性,因此在使用这些材料作为食品添加剂时必须小心。 | |||
T3829 |
Ginsenoside F3
人参皂苷F3 |
Others; IFNAR; Interleukin | Immunology/Inflammation; Others |
Ginsenoside F3 是一种皂苷,提取自Panax ginseng 叶片。它能够调节1 型 (IL-2, IFN-γ) 及 2 型细胞因子(IL-4 and IL-10) 的产生和表达,有免疫增强的作用。 | |||
T11398 |
Ginsenoside Ra3
人参皂苷 RA3,人参皂苷RA3 |
Others | Others |
Ginsenoside Ra3 是分离自人参中,具有抗癌作用。 | |||
T3918 |
Ginsenoside Rb3
人参皂苷 Rb3,Gypenoside IV,人参皂苷Rb3 |
NF-κB; COX; NO Synthase | Immunology/Inflammation; Neuroscience; NF-κB |
Ginsenoside Rb3 (Gypenoside IV) 是从三七中提取的一种天然产物。它在 293T 细胞系中抑制 TNFα 诱导的NF-κB 转录活性,IC50为 8.2 μM。它还抑制COX-2和iNOSmRNA 的诱导。 | |||
T2822 |
Ginsenoside Rb1
Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III |
ATPase; Mitophagy; IRAK; NF-κB; Autophagy; HSV | Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB |
Ginsenoside Rb1 (Gypenoside Ⅲ) 是中药人参的成分,可能具有抑制或阻止肿瘤生长的特性。 | |||
T2873 |
Ginsenoside Rg2
Chikusetsusaponin I,Panaxoside Rg2,人参皂苷Rg2,Prosapogenin C2,(20S)Ginsenoside Rg2,人参皂苷 Rg2 |
Beta Amyloid; GSK-3; NF-κB | Neuroscience; NF-κB; PI3K/Akt/mTOR signaling; Stem Cells |
Ginsenoside Rg2 (Chikusetsusaponin I) 是一种人参的主要活性成分。它能够降低Aβ1-42积聚,抑制脂多糖介导的VCAM-1和ICAM-1表达的增加。 | |||
T3830 |
20(R)-Ginsenoside Rg2
20R-Ginsenoside Rg2,20R-人参皂苷Rg2,20(R)-人参皂苷 Rg2 |
IL Receptor | Immunology/Inflammation |
20(R)-Ginsenoside Rg2 (20R-Ginsenoside Rg2) 是一种人参皂苷。它能够抑制肺癌 NCI-H1650 细胞,具有抗癌作用。 | |||
T6S1485 |
Ginsenoside Rh4
人参皂苷Rh4 |
Others | Others |
Ginsenoside Rh4 可以安全地用作佐剂,具有低溶血作用或无溶血作用。它具有细胞毒活性,其苷元对癌细胞系具有杀伤作用。 | |||
T2959 |
Ginsenoside Rh2
20(S)-Rh2,20S-Ginsenoside Rh2,人参皂苷Rh2,20(S)-Ginsenoside Rh2,人参皂苷 Rh2 |
Apoptosis; EGFR; Caspase; Endogenous Metabolite | Angiogenesis; Apoptosis; JAK/STAT signaling; Metabolism; Proteases/Proteasome; Tyrosine Kinase/Adaptors |
Ginsenoside Rh2 (20(S)-Ginsenoside Rh2) 诱导caspase-8和caspase-9活化。它以多途径方式诱导癌细胞凋亡。 | |||
T4S1519 |
Pseudoginsenoside RT5
拟人参皂苷RT5 |
Others | Others |
Pseudoginsenoside RT5 分离于 Panax quinquefolium 中。它通过促进神经生长和提高认知能力,具有抗癫痫、抗抑郁活性,还具有抗菌、抗肿瘤、抗疟疾等活性。 | |||
T6S1487 |
Ginsenoside Rg5
人参皂苷Rg5,人参皂甙 Rg5 |
NF-κB; COX; IGF-1R | Immunology/Inflammation; Neuroscience; NF-κB; Tyrosine Kinase/Adaptors |
Ginsenoside Rg5 是红参的主要成分,可阻断IGF-1与其受体的结合,IC50约为90 nM。它还通过抑制NF-κB p65的 DNA 结合活性来抑制COX-2的 mRNA 表达。它可促进血管生成和改善高血压,具有抗炎和治疗阿尔茨海默病的潜力。 | |||
T3919 |
Ginsenoside Rb2
Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2 |
GPR; Others; Influenza Virus; Endogenous Metabolite | Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Others |
Ginsenoside Rb2 (Ginsenoside C) 是人参提取物中的一种主要生物活性成分,具有抗病毒活性,可上调 GPR120 基因表达。 | |||
T2878 |
Ginsenoside Rd
Panaxoside Rd,Sanchinoside Rd,人参皂苷Rd,人参皂苷 Rd,Gypenoside VIII |
P450; Calcium Channel; NF-κB; COX; Endogenous Metabolite | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB |
Ginsenoside Rd (Gypenoside VIII) 抑制 TNFα 诱导的NF-κB 转录活性,还抑制COX-2和iNOSmRNA 的表达。它抑制CYP2D6、CYP1A2、CYP3A4和CYP2C9,也抑制Ca2+内流,有可能抑制或阻止肿瘤生长。 | |||
TN1096 |
Ginsenoside Ra1
人参皂苷 Ra1,人参皂苷Ra1 |
Others; Tyrosine Kinases | Others; Tyrosine Kinase/Adaptors |
Ginsenoside Ra1 是来自人参的成分。 Ginsenoside Ra1 对缺氧/复氧诱导的蛋白酪氨酸激酶 (PTK) 活化具有显着抑制作用。 | |||
TN1686 |
Ginsenoside Rg4
人参皂苷 RG4 |
Antibacterial | Microbiology/Virology |
Ginsenoside Rg4 是分离自Panax ginsengC. A. Meyer 叶子中的一种人参三醇型人参皂苷。人参三醇型人参皂苷具有多种生物活性,包括防腐,抗糖尿病,伤口愈合,免疫刺激和抗氧化活性等。 | |||
T2872 |
Ginsenoside Re
人参皂苷 Re,Ginsenoside B2,Panaxoside Re,Chikusetsusaponin Ivc,Sanchinoside Re,人参皂苷Re |
Beta Amyloid; NF-κB; Endogenous Metabolite; JNK | MAPK; Metabolism; Neuroscience; NF-κB |
Ginsenoside Re (Ginsenoside B2) 是一种人参提取物,可降低 β-淀粉样蛋白 (Aβ),还通过抑制 JNK 和 NF-κB 发挥抗炎作用。 | |||
T3916 |
Ginsenoside F2
人参皂苷F2 |
Apoptosis; Endogenous Metabolite; Autophagy | Apoptosis; Autophagy; Metabolism |
Ginsenoside F2 是 Ginsenoside Rb1 的代谢物,通过激活内在的凋亡途径和线粒体功能障碍来诱导乳腺的凋亡,对乳腺癌干细胞具有抗增殖活性。 | |||
TN1997 |
Notoginsenoside FP2
三七皂苷FP2 |
Others | Others |
Notoginsenoside FP2 是从三七 Panax notoginseng 果实花梗中分离得到的天然产物,可用于治疗心血管疾病的研究。 | |||
T3849 |
Kinsenoside
金线莲苷,(+)-Kinsenoside |
Apoptosis; Nrf2 | Apoptosis; Immunology/Inflammation |
Kinsenoside ((+)-Kinsenoside) 是从金盏花属植物中分离得到的主要活性成分,以 Nrf2 依赖的方式保护髓核细胞在氧化应激下的生存能力,防止细胞凋亡、衰老和线粒体功能障碍。它显示出显着的抗肝毒性和抗炎活性。 | |||
T4S1518 |
Pseudoginsenoside RT1
拟人参皂苷 RT1,假人参皂苷RT1 |
Others | Others |
Pseudoginsenoside RT1 是分离自 Randia siamensis 中,具有鱼毒素作用。它可导致血压下降、心率加快和子宫自发收缩力增加。 | |||
T3401 |
Ginsenoside F1
人参皂苷 F1,20(S)-Ginsenoside F1 |
P450; Endogenous Metabolite | Metabolism |
Ginsenoside F1 (20(S)-Ginsenoside F1) 是一种 Ginsenoside Rg1 的酶促修饰衍生物,它竞争性抑制CYP3A4,对 CYP2D6 具有较弱的抑制作用。 | |||
TN7110 |
Ginsenoside Rs2
人参皂苷Rs2 |
Others | Others |
Ginsenoside Rs2 是从人参Panax japonicus var.叶中分离得到的天然产物。 | |||
T2932 |
Ginsenoside Rh1
Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1 |
IL Receptor; TNF; Endogenous Metabolite; PPAR; Interleukin | Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism |
Ginsenoside Rh1 (Sanchinoside B2) 是人参的一种主要成分,具有抗炎作用,抑制PPAR-γ,TNF-α,IL-6和IL-1β的表达。 | |||
T2S0223 |
Isosinensetin
异橙黄酮,6-Demethoxynobiletin |
Antioxidant; HIV Protease; Antibacterial; P-gp | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; oxidation-reduction; Proteases/Proteasome |
Isosinensetin (6-Demethoxynobiletin) 是从青皮中提取的一种甲氧基黄酮,具有抗氧化和抑制 HIV-1 蛋白酶的活性。 | |||
T5S1590 |
Notoginsenoside Fe
三七皂苷Fe,Notoginseng triterpenes,Ginsenoside Mb |
Others | Others |
Notoginsenoside Fe (Ginsenoside Mb) 是一种分离自珠子参变种中的天然化合物。 | |||
T3811 |
Ginsenoside C-K
20(S)-人参皂苷 C-K,Ginsenoside compound K,Ginsenoside K,人参皂苷 C-K |
P450; cell cycle arrest; COX; NO Synthase | Cell Cycle/Checkpoint; Immunology/Inflammation; Metabolism; Neuroscience |
Ginsenoside C-K (Ginsenoside K) 是 Ginsenoside Rb1 的细菌代谢物,可通过抑制诱生型一氧化氮合酶和COX-2来发挥抗炎作用。它在人肝微粒体中抑制CYP2C9和CYP2A6活性,IC50分别为 32.0±3.6 和 63.6±4.2 μM。 | |||
TN2296 |
Vinaginsenoside R4
越南参皂苷R4 |
Others | Others |
Vinaginsenoside R4 是分离自水培人参的叶子中。它能够抑制黑色素的生物合成,并增强斑马鱼的色素沉着,对 melan-a 细胞没有任何细胞毒性作用。 | |||
T2777 |
Ginsenoside Rg1
Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2 |
Apoptosis; Beta Amyloid; NF-κB | Apoptosis; Neuroscience; NF-κB |
Ginsenoside Rg1 (Panaxoside Rg1) 是人参的主要活性成分之一,可减少NF-κB 核易位。它改善认知功能受损,通过降低大脑Aβ水平来发挥作用。 | |||
TN6930 |
5-Desmethylsinensetin
|
Others | Others |
5-desmethylsinensetin 是分离自Stevia satureiifoliavar.satureiifolia 的天然产物,显示出抗原生动物的活性,抑制T. cruzi epimastigotes 和trypomastigotes 的IC50分别为 0.4 μg/mL 和75.1 μg/mL。 | |||
TN2100 |
Pratensein
红车轴草素,三叶草 |
Others; NF-κB | NF-κB; Others |
Pratensein 是黄酮类化合物,能够减少氧化损伤和恢复突触和 BDNF 水平,改善 β-淀粉样蛋白诱导的大鼠认知障碍。 | |||
T4704 |
L-Anserine nitrate
L-鹅肌肽硝酸盐,L-Anserine nitrate salt |
Others; Endogenous Metabolite | Metabolism; Others |
L-Anserine nitrate (L-Anserine nitrate salt) 是一种存在于大多数动物组织中的二肽。在模型系统中,它是一种有效的抗氧化剂和羟基自由基清除剂。该化合物抑制醛糖和酮糖还原糖诱导的非酶蛋白糖基化。 | |||
T3812 |
(20R)-Ginsenoside Rg3
人参皂甙 RG3,(20R)-人参皂苷Rg3,20(R)-Ginsenoside Rg3,(20R)Ginsenoside Rg3,20(R)-Propanaxadiol |
Others | Others |
(20R)-Ginsenoside Rg3 (20(R)-Propanaxadiol) 是一种人参根中的化合物,具有抑制血管内皮细胞增生(IC50= 10 nM)和抗肿瘤作用。 | |||
T0783 |
Mianserin hydrochloride
Mianserin HCl,Org GB 94,盐酸米安色林,ORG GB-94 HCl |
Dopamine Receptor; 5-HT Receptor; Opioid Receptor; Adrenergic Receptor; Histamine Receptor | Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Mianserin hydrochloride (Org GB 94) 是一种有抗抑郁活性的 H1 受体反向激动剂。 | |||
T13626 |
Cottonseed oil
|
Others | Others |
Cottonseed oil 是一种提取自棉花种子中的食用油,是一种植物油中杀虫能力极强的油。 | |||
T3920 |
Pseudoginsenoside F11
Ginsenoside A1,拟人参皂苷 F11,拟人参皂苷F11 |
Others; Endogenous Metabolite | Metabolism; Others |
Pseudoginsenoside F11 (Ginsenoside A1) 从人参根和叶中分离得到。PF11在一系列心血管和中枢神经系统疾病中具有广泛的保护作用。 | |||
T3402 |
20(S)-Ginsenoside Rg3
20(S)-人参皂苷 Rg3,人参皂苷 Rg3,20(S)-Ginsenoside-Rg3,Rg3,20S-Ginsenoside Rg3,Ginsenoside Rg3,S-Ginsenoside Rg3 |
EGFR; Beta Amyloid; Potassium Channel; NF-κB; COX; Sodium Channel; Endogenous Metabolite | Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Tyrosine Kinase/Adaptors |
20(S)-Ginsenoside Rg3 (Rg3) 是红参的主要成分,通过抑制肿瘤细胞的粘附和侵袭来抑制肿瘤细胞肺转移。它抑制Na+和hKv1.4通道,IC50分别为 32.2±4.5 和 32.6±2.2 μM。它还抑制Aβ,NF-κB 活性和COX-2表达,抑制人脐静脉内皮细胞的增殖并具有抗血管生成活性。 | |||
T6S1495 |
Ginsenoside Rk3
人参皂苷Rk3,人参皂甙 Rk3 |
Others; NF-κB | NF-κB; Others |
Ginsenoside Rk3 是存在于 Panax notoginseng 的根中。它能够抑制 HepG2 细胞中 TNF-α 诱导的 NF-κB 转录活性,IC50=14.24±1.30 μM。 | |||
T3813 |
20(R)-Ginsenoside Rh2
20(R)-人参皂苷 RH2,(20R)Ginsenoside Rh2,Ginsenoside Rh2,20(R)-人参皂苷Rh2 |
Apoptosis; MMP; HSV | Apoptosis; Microbiology/Virology; Proteases/Proteasome |
20(R)-Ginsenoside Rh2 (Ginsenoside Rh2) 是人参皂苷 Rh2 的次要立体异构体,具有基质金属蛋白酶抑制作用。它有抗癌、抗炎和抗氧化活性。 | |||
T3915 |
Ginsenoside Ro
人参皂苷Ro,Chikusetsusaponin 5,Polysciasaponin P3,人参皂苷 Ro,Chikusetsusaponin V |
Calcium Channel; Reductase; Prostaglandin Receptor | Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism |
Ginsenoside Ro (Chikusetsusaponin V) 能降低 TXA2产量,较弱降低 COX-1 和 TXAS 活性,具有 Ca2+拮抗剂的抗血小板作用,IC50为 155 μM。 | |||
T4S0227 |
Sinensetin
Pedalitin permethyl ether,甜橙素 |
TNF; PGE Synthase | Apoptosis; Immunology/Inflammation |
Sinensetin (Pedalitin permethyl ether) 是从水果中发现的一种甲基化黄酮,有很强的抗血管和抗炎症的能力。 | |||
T3S1589 |
Notoginsenoside Fa
|
Others | Others |
Notoginsenoside Fa 是一种原人参二醇型皂苷,从P. notoginseng 提取出来得到,有激活和恢复退化脑功能的潜能。 | |||
T2961 |
Notoginsenoside R1
Sanqi glucoside R1,Sanchinoside R1,三七皂苷R1 |
Apoptosis; ERK; Beta Amyloid | Apoptosis; MAPK; Neuroscience |
Notoginsenoside R1 (Sanchinoside R1) 是一种从三七中分离出来的皂苷,具有抗氧化、抗炎、抗血管生成和抗凋亡的活性。它有神经保护和抗缺血/再灌注损伤的心脏保护作用。 | |||
T6S1587 |
Notoginsenoside R2
三七皂苷R2,20(S)-Notoginsenoside R2,Ginsenoside Ng-R2 |
Others; Nrf2 | Immunology/Inflammation; Others |
Notoginsenoside R2 (20(S)-Notoginsenoside R2) 是一种新分离三七皂苷,表现出对6-OHDA 诱导的氧化应激及细胞凋亡的保护作用。 | |||
T3S1591 |
Notoginsenoside Fc
三七皂苷 FC,三七皂苷Fc |
Others; Autophagy | Autophagy; Others |
Notoginsenoside Fc 是从三七叶中分离得到的原卟啉二醇型皂苷,可通过促进自噬促进糖尿病大鼠血管损伤后的内皮细胞再生,具有抗血小板聚集的作用。 | |||
TN1684 |
Ginsenoside F5
人参皂苷 F5,人参皂苷F5 |
Apoptosis | Apoptosis |
Ginsenoside F5 是从人参中提取的一种天然产物,通过凋亡途径显着抑制 HL-60 细胞的生长。 | |||
T5761 |
Notoginsenoside Ft1
三七皂苷FT1,三七皂甙 Ft1 |
Others; HIF/HIF Prolyl-Hydroxylase | Chromatin/Epigenetic; Metabolism; Others |
Notoginsenoside Ft1 是一种植物分离的三七皂苷,具有刺激血管生成的作用。 | |||
T6S1500 |
Ginsenoside Rf
人参皂苷 Rf,Ginsenoside-Rf,Panaxoside Rf |
Calcium Channel; Endogenous Metabolite | Membrane transporter/Ion channel; Metabolism |
Ginsenoside Rf (Panaxoside Rf) 是人参根的微量成分,可抑制 N 型 Ca2+通道。 | |||
T3793 |
(20R)-Ginsenoside Rh1
20(R)-Ginsenoside Rh1,人参皂苷 R-RH1,人参皂苷R-RH1 |
Others | Others |
(20R)-Ginsenoside Rh1 (20(R)-Ginsenoside Rh1) 是 Ginsenoside Rh1 的 R 型异构体,分离自 Panax Ginseng 中,能够阻碍凝血酶诱导的纤维蛋白原向纤维蛋白的转化。 | |||
T2720 |
Ginsenoside Rc
Panaxoside Rc,人参皂苷Rc,人参皂苷 Rc |
Others; TNF; GABA Receptor; Interleukin | Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; Others |
Ginsenoside Rc (Panaxoside Rc) 是人参中的一种人参皂苷,可抑制 TNF-α 和 IL-1β 的表达。它增强 GABA 受体 A 介导的离子通道电流。 | |||
TN2802 |
20-O-Glucoginsenoside Rf
|
Others | Others |
20-O-Glucoginsenoside Rf 是从人参 Panax ginseng C. A. Mey 中提取的天然产物。 | |||
------------------------ 更多 ------------------------ |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-02646 |
NSE/ENO2 Protein, Human, Recombinant (His)
enolase 2 (γ, neuronal),NSE,HEL-S-279,enolase 2 (ga... |
Human | E. coli |
The combination of silencing ENO2 and 2-deoxyglucose (2-DG) synergistically inhibited leukemia cell survival. ENO2 may be a biological marker for monitoring chemotherapeutic efficacy and relapse in ALL. Reduced ENO2 expression may be a biomarker for a subset of autistic children. Neuron specific enolase (ENO2, gamma-enolase) has been used as a biomarker to help identify neuroendocrine differentiation in breast cancer. | |||
TMPH-03617 |
Miraculin Protein, Synsepalum dulcificum, Recombinant (His)
|
Synsepalum dulcificum | P. pastoris (Yeast) |
Miraculin has the property of modifying a sour taste into a sweet taste. This alteration of taste perception persists for many minutes. Miraculin Protein, Synsepalum dulcificum, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 23.4 kDa and the accession number is P13087. | |||
TMPY-06016 |
Phl p 5 Protein, Phleum pratense, Recombinant
|
Phleum pratense | E. coli |
Phl p 5 Protein, Phleum pratense, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 28.7 kDa and the accession number is Q40960-1. | |||
TMPH-03095 |
Phl p 6 Protein, Phleum pratense, Recombinant (His & Myc)
|
Phleum pratense | E. coli |
Phl p 6 Protein, Phleum pratense, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 19.2 kDa and the accession number is P43215. | |||
TMPH-03093 |
Phl p 5a Protein, Phleum pratense, Recombinant (His & SUMO)
|
Phleum pratense | E. coli |
N/A. Phl p 5a Protein, Phleum pratense, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 44.5 kDa and the accession number is Q40962. | |||
TMPY-06015 |
Phl p 2 Protein, Phleum pratense, Recombinant (His)
|
Phleum pratense | HEK293 Cells |
Phl p 2 Protein, Phleum pratense, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 13.1 kDa and the accession number is P43214-1. | |||
TMPH-03094 |
Phl p 5b Protein, Phleum pratense, Recombinant (His & SUMO)
|
Phleum pratense | E. coli |
Has ribonuclease activity. May be involved in host-pathogen interactions. Phl p 5b Protein, Phleum pratense, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 42.1 kDa and the accession number is Q40963. | |||
TMPY-06149 |
Phl p 5 Protein, Phleum pratense, Recombinant (His)
|
Phleum pratense | HEK293 Cells |
Phl p 5 Protein, Phleum pratense, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 30.9 kDa and the accession number is Q40960-1. | |||
TMPH-03616 |
Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His)
|
Synsepalum dulcificum | E. coli |
Miraculin has the property of modifying a sour taste into a sweet taste. This alteration of taste perception persists for many minutes. Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 24.9 kDa and the accession number is P13087. | |||
TMPH-03096 |
Profilin 2 Protein, Phleum pratense, Recombinant (His & Myc)
|
Phleum pratense | E. coli |
Binds to actin and affects the structure of the cytoskeleton. At high concentrations, profilin prevents the polymerization of actin, whereas it enhances it at low concentrations. By binding to PIP2, it inhibits the formation of IP3 and DG. Profilin 2 Protein, Phleum pratense, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 21.5 kDa and the accession number is O24650. | |||
TMPH-03626 |
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (His & Myc)
Toxin II-11,Beta-like toxin Ts1,Ts7,Beta-mammal/inse |
Tityus serrulatus | Baculovirus Insect Cells |
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 10.8 kDa and the accession number is P15226. | |||
TMPH-03627 |
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (E. coli, His & Myc)
Ts VII,Beta-like toxin Ts1,Toxin II-11,Ts7,Tityustoxin VII,P... |
Tityus serrulatus | E. coli |
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (E. coli, His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 14.3 kDa and the accession number is P15226. |