购物车

搜索结果

Search Results for " nse "
Targets Recommended: TGF-beta/Smad

93

抑制剂 & 化合物

83

天然产物

12

重组蛋白

如果没找到您满意的产品或者您对产品有其他要求,可以联系我们专业顾问为您提供针对性的合理建议。     QQ咨询       网站留言咨询

提交您的定制咨询

点击图片重新获取验证码
Cat. No. Product Name Target Signaling Pathways
T76774 Ponsegromab

PF 06946860

TGF-beta/Smad Stem Cells
Ponsegromab (PF 06946860) 是一种具有选择性和有效性的人源化抗 GDF15 抗体抑制剂。 Ponsegromab 具有抗恶病质活性,通过与 GDF15 结合来阻止其与 GFRAL 结合,从而中断 GDF15/GFRAL 介导的信号传导。 Ponsegromab 具有潜在的抗癌活性,可用于治疗患有癌症厌食-恶病质综合征的癌症患者。
T3467 Miransertib

ARQ-092,AKT inhibitor 2

Akt; Parasite Cytoskeletal Signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling
Miransertib (ARQ-092) 是一种具有口服活性的,选择性和变构性Akt 抑制剂。它有效抑制利什曼原虫,还是 AKT1-E17K 突变蛋白抑制剂,可研究PI3K/AKT 驱动的肿瘤和 Proteus 综合征。
T68141 Seganserin

5-HT Receptor GPCR/G Protein; Neuroscience
Seganserin 是一种非选择性5-羟色胺2-HT 受体拮抗剂,可逆转了氟西汀和喹帕嗪对黄体酮诱导的食欲亢进,抑郁和痛觉的抑制作用,逆转氟西汀和喹帕嗪诱导的抗抑郁和镇痛作用。
T1066 Ketanserin

R41468,凯他色林,Ketanserin tartrate,酮色林,Ketanserinum

Potassium Channel; 5-HT Receptor; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Ketanserin (Ketanserinum) 是一种喹唑啉衍生物和 5-羟色胺受体亚型 2 拮抗剂,具有潜在的抗高血压和抗血小板活性。它也浓度依赖性抑制 hERG 电流,IC50为 0.11 μM。
T7350 Nelotanserin

1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲,APD125

5-HT Receptor GPCR/G Protein; Neuroscience
Nelotanserin (APD125) 是5-HT2A 强完全逆向激动剂,5-HT2C 中等强度的部分反向激动剂和5-HT2B 的弱反向激动剂,IC50s 值分别为 1.7、79 和 791 nM。
T6946 Pimavanserin tartrate

ACP-103,ACP-103 tartrate,Nuplazid,Pimavanserin,匹莫范色林

5-HT Receptor GPCR/G Protein; Neuroscience
Pimavanserin tartrate (Nuplazid) 是一种有效的5-HT 2A 受体反向激动剂,pIC50和 pKi 值分别为8.73和9.3,用于治疗与帕金森病相关的精神病。
T6247 Onvansertib

NMS-P937,NMS-1286937

Apoptosis; PLK Apoptosis; Cell Cycle/Checkpoint
Onvansertib (NMS-1286937) 是一种可口服的高选择性PLK1抑制剂,IC50值为 2 nM。
T16759 Ritanserin

利坦丝林,R 55667

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ritanserin (R 55667) 是一种长效、高效、相对选择性、可口服的5-HT2受体拮抗剂,IC50值为 0.9 nM。
T1478 Ondansetron hydrochloride dihydrate

盐酸昂丹司琼,SN 307,NSC 665799,GR 38032,Ondansetron hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Ondansetron hydrochloride dihydrate (GR 38032) 是5- HT3受体拮抗剂,可治疗化疗后的恶心和呕吐,有抗焦虑和抗精神病作用。
T5389 Volinanserin

M 100907,MDL100907,氟利色林

5-HT Receptor GPCR/G Protein; Neuroscience
Volinanserin (MDL100907) 是选择性的5-HT2受体拮抗剂,Ki 值为 0.36 nM,可用于精神疾病的研究。它对 5-HT2 受体的选择性比 5-HT1c、α-1 肾上腺素能受体和 σ 受体高 300 倍。
T22964 Glemanserin

MDL11939

5-HT Receptor GPCR/G Protein; Neuroscience
Glemanserin (MDL11939) 是一种特异性 5-HT2A 拮抗剂,对兔、人和大鼠 5-HT2A 的 Ki 值为 0.54 nM、2.5 nM 和 2.89 nM。
T37979 N-Desmethyl Pimavanserin

AC-279

5-HT Receptor GPCR/G Protein; Neuroscience
N-Desmethyl Pimavanserin (AC-279) 是 Pimavanserin (一种 5-HT2A 受体反向激动剂)的活性代谢物,可用于治疗失眠等睡眠障碍。
T8451 Tropanserin

MDL 72422

5-HT Receptor GPCR/G Protein; Neuroscience
Tropanserin (MDL 72422) 是一种 5-羟色胺受体拮抗剂,抑制5-HT3受体活性。Tropanserin 具有抗焦虑活性,可用于治疗抑郁症和认知障碍。
T62083 Camonsertib

ATR inhibitor 4,RP-3500

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Camonsertib (RP-3500) 是一种选择性的、口服具有活力的 ATR 激酶抑制剂 (ATRi),在生化试验中的 IC50: 1.00 nM,表现出有效的抗肿瘤作用。RP-3500 对 ATR 的选择性是 mTOR 的 30 倍 (IC50: 120 nM),是 ATM、DNA-PK 和 PI3Kα 激酶的 2,000 倍以上。
T23445 Anxiolytic/nonsedative agent-1

TCS 1205

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Anxiolytic/nonsedative agent-1 (TCS 1205) 是一种有效的选择性 GABAA 激动剂。Anxiolytic/nonsedative agent-1 对牛脑膜中的 BzR 显示出明显的亲和力,对 α1β2γ2、α2β2γ2、α5β3γ2 的 Kis 分别为 14、121、239 nM。Anxiolytic/nonsedative agent-1 在体外表现出 α2 选择性功效,在体内表现出抗焦虑选择性作用。
T14968 Cinanserin hydrochloride

SQ 10643

Influenza Virus; 5-HT Receptor GPCR/G Protein; Microbiology/Virology; Neuroscience
Cinanserin hydrochloride (SQ 10643) 是一种高亲和力拮抗剂,对 5-HT2 受体的Ki 值为 41 nM。它也是严重急性呼吸综合征冠状病毒的 3C 样蛋白酶抑制剂。
T1517 Benserazide hydrochloride

Benserazide HCl,盐酸苄丝肼,Serazide,Ro 4-4602

Dopamine Receptor GPCR/G Protein; Neuroscience
Benserazide hydrochloride (Ro 4-4602) 是一种芳香族 L-氨基酸脱羧酶(AADC)的抑制剂,常用于帕金森病。
T23631 Adatanserin

WY-50324,WY 50324,WAY SEB 324,WY50324

5-HT Receptor GPCR/G Protein; Neuroscience
Adatanserin (WY 50324) 是一种混合型 5-HT1A 受体部分激动剂,也是一种 5-HT2A 和 5-HT2C 受体拮抗剂,具有潜在的神经保护活性,可用于研究焦虑和抑郁症。
T67914 Insecticidal agent 364

mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Insecticidal agent 364是一种雷帕霉素激酶靶蛋白的选择性小分子抑制剂。Insecticidal agent 364具有抗肿瘤活性,通过抑制mTOR, Insecticidal agent 364旨在破坏参与癌细胞生长和存活的信号通路,从而潜在地抑制肿瘤生长。
T3350 Selonsertib

GS-4997

Apoptosis; ASK; MAPK Apoptosis; MAPK
Selonsertib (GS-4997) 是一种选择性的,具有生物口服可利用的凋亡信号调节激酶1 抑制剂,pIC50为 8.3。它具有潜在的抗炎、抗肿瘤和抗纤维化活性。
T21428 Mianserin

Lantanon,Lumin,Norval,Lerivon,Depnon

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mianserin 是H1受体反向激动剂,是四环抗抑郁药(TeCA)治疗家族中的一种精神活性化合物,具有抗抑郁、抗焦虑、止吐、促氧、催眠和抗组胺作用,可作为去甲肾上腺素和特定的血清素联合用药能治疗抑郁症。
T1180 Blonanserin

布南色林,AD-5423

Dopamine Receptor; Sigma receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Blonanserin (AD-5423) 是一种有效的5-HT2A 和多巴胺 D2 受体拮抗剂,Ki 为 0.812 和 0.142 nM,是一种非典型的抗精神病试剂。
T2076 Pimavanserin

ACP-103,匹莫范色林

5-HT Receptor GPCR/G Protein; Neuroscience
Pimavanserin (ACP-103) 是特异性的 5-HT2A 受体反向激动剂,在基于细胞的功能测定中,平均 pIC50值为8.7。它是非典型抗精神病药,用于治疗帕金森病患者的幻觉和精神病。
T15270 Fananserin

RP 62203,法南色林

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Fananserin 是一种有效的、特异性的、口服活性的 5-HT2 拮抗剂(大鼠 5-HT2A 的 Ki = 0.37 nM)。 Fananserin 是人 D4 受体的拮抗剂 (Ki = 2.93 nM)。
T6615 Ondansetron

GR-C507/75,GR 38032,昂丹司琼,GR 38032F,SN 307,恩丹西酮

5-HT Receptor GPCR/G Protein; Neuroscience
Ondansetron (GR 38032) 是一种血清素 5-HT3 受体拮抗剂,主要用作止吐剂。
T27020 Cilansetron

KC-9946,KC9946,DU-123265,DU123265

5-HT Receptor GPCR/G Protein; Neuroscience
Cilansetron 是一种具有有效性和选择性的 5-HT3 受体拮抗剂,可用于结肠炎引发的相关疾病。
T6616 Ondansetron hydrochloride

SN 307,盐酸昂丹司琼,帕罗西汀杂质A,Ondansetron HCl,Emeset,GR 38032 HCl,NSC 665799,Zofran

5-HT Receptor GPCR/G Protein; Neuroscience
Ondansetron hydrochloride (Zofran) 是5-HT3受体的拮抗剂,可用作化疗后止吐剂。
T4297 Flibanserin

BIMT-17BS,氟立班丝氨,Girosa,BIMT-17

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Flibanserin (Girosa) 一种具有口服活性的 5-HT1A 受体激动剂和 5-HT2A 受体拮抗剂,Ki 值分别为 1 和 49 nM。它与多巴胺 D4 受体结合,Ki 值在 4 到 24 nM 之间。它是一种血清素能抗抑郁药,用于治疗性欲减退症。
T9833 Opiranserin hydrochloride

P2X Receptor; GlyT; 5-HT Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Opiranserin hydrochloride 是甘氨酸转运蛋白 2 型 (GlyT2) 和 5-羟色胺受体 2A (5HT2A) 的双重拮抗剂,IC50 分别为 0.86 和 1.3 μM。它显示对 rP2X3 的拮抗活性 (IC50=0.87 μM)。它正在开发为用于治疗术后疼痛的注射剂。
T1066L Ketanserin tartrate

KJK 945 tartrate,KJK-945 tartrate,KJK945 tartrate

5-HT Receptor; Serotonin Transporter; Adrenergic Receptor GPCR/G Protein; Neuroscience
Ketanserin tartrate (KJK-945 tartrate) 是 5-HT2A 受体和α1-肾上腺素能受体拮抗剂,具有抗高血压活性,抑制血清素诱导的血管收缩和血小板活化,可用于研究系统性硬化症。
T29645 Adatanserin hydrochloride

WY50324 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Adatanserin hydrochloride (WY50324 hydrochloride) 是一种新型 5-HT(1A)/5-HT(2) 受体配体,具有潜在的神经保护作用,抑制内源性氨基酸缺血性外排,可用于研究抑郁症和焦虑症。
T22243 Anserine

L-鹅肌肽,L-Anserine

Endogenous Metabolite Metabolism
Anserine (L-Anserine) 是 Carnosine 的甲基化形式,是口服具有活性的天然二肽,存在于脊椎动物的骨骼肌。它不会被血清肌肽酶裂解,能够作为生化缓冲液,螯合剂,抗糖化剂和抗氧化剂。它能够改善阿尔茨海默氏病模型小鼠的记忆功能。
T12477 Uzansertib phosphate

INCB053914 phosphate

Pim Chromatin/Epigenetic; JAK/STAT signaling
Uzansertib phosphate (INCB053914 phosphate) 是一种可口服的 ATP 竞争性泛-PIM 激酶抑制剂,对多种血液肿瘤细胞系具有广泛的抗增殖活性,对 PIM1、PIM2 和 PIM3 的 IC50分别为 0.24 、30 和 0.12 nM。
T11217 Eplivanserin

依利色林,SR-46349

5-HT Receptor GPCR/G Protein; Neuroscience
Eplivanserin (SR-46349) 是一种有效和特异性的 5-HT2A 受体拮抗剂,Kd 值为 1.14 nM,在大鼠皮质膜中 IC50 值为 5.8 nM。
T27020L isomer-Cilansetron

Others Others
isomer-Cilansetron 是 Cilansetron 的异构体。
T29913 Altanserin

R-53200,R53200,R 53200

Altanserin can binds to the 5-HT2A receptor. Labeled with the isotope fluorine-18 it is used as a radioligand in positron emission tomography (PET) studies of the brain.
T12446 Phenserine

(-)-Eseroline phenylcarbamate,(-)-Phenserine

AChR Neuroscience
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
T39090 Uzansertib

INCB053914

Uzansertib (INCB053914) is a potent ATP-competitive pan-PIM kinase inhibitor. It exhibits exceptional inhibitory activity against PIM1, PIM2, and PIM3 with IC50 values of 0.24 nM, 30 nM, and 0.12 nM, respectively. Furthermore, Uzansertib demonstrates significant anti-proliferative effects against an assorted range of hematologic tumor cell lines.
T39126 Zunsemetinib

CDD-450,ATI-450

Zunsemetinib (CDD-450) is a potent and specific inhibitor of the p38α-MK2 pathway, exerting its effects through oral administration. It has proven activity against immuno-inflammatory diseases, making it a valuable tool for research in this area.
T26768 Benanserin HCl

Benanserin Hydrochloride,BAS,Benanserin,Benzyl antiserotonin

Benanserin HCl is a serotonin antagonist. It causes psychotropic effects in humans.
T34918 Trelanserin

SL650472,SL-650472,SL 650472

Trelanserin (SL-650472) is an antagonist of the serotonin receptor.
T1517L Benserazide

Ro-44602,Ro44602,Ro 44602,Serazide

Benserazide is an inhibitor of dopa decarboxylase. It is often given with levodopa in the treatment of Parkinson's to prevent the conversion of levodopa to dopamine in the periphery, thereby increasing the amount that reaches the central nervous system an
T9901A-011 Lunsekimig

SAR443765

Lunsekimig (SAR443765) 是一种 IL-13/TSLP 双抗,将靶向 IL-13 和靶向 TSLP 的重链可变区 (VHH) 连接在一起的纳米抗体,可用于哮喘研究。
T16399 Opiranserin

P2X Receptor; GlyT; 5-HT Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Opiranserin 是一种非阿片类和非 NSAID 镇痛候选药物,是 2 型甘氨酸转运蛋白 (GlyT2) 和 5-羟色胺受体 2A (5HT2A) 的双重拮抗剂,IC50分别为 0.86 和 1.3 μM。它可用于术后疼痛的研究,对 rP2X3 有拮抗作用,IC50为0.87 μM。
T82064 Insecticidal agent 6

Parasite Microbiology/Virology
Insecticidal agent 6(化合物 Im)是昆虫兰尼碱受体(RyRs)的抑制剂,该化合物对 S. frugiperda RyRs 具有强效的抑制作用,其 EC50 值为0.6308 µM。该化合物在鳞翅目害虫中展现出卓越的杀虫效果,适用于病虫害研究。
T25568 Ketanserinol

Reduced ketanserin

Ketanserinol is the metabolite of ketanserin. Ketanserin is a hypotensive drug with 5-HT2 receptor antagonism, used to reverse pulmonary hypertension caused by protamine.
T83106 Anselamimab

Anselamimab (CAEL-101) 为一种靶向血清淀粉样蛋白 A1 (SAA1) 的人源 IgG1-κ 抗淀粉样蛋白原纤维抗体。
T30936 Cilansetron Hydrochloride

KC-9946,KC9946,KC 9946

Cilansetron Hydrochloride can be used for irritable Bowel Syndrome (IBS) with Diarrhea Predominance.
T70439 Galdansetron hydrochloride

Galdansetron hydrochloride is a serotonin antagonist and anti-emetic.
T71292 Rivipansel sodium

Rivipansel sodium is a glycomimetic drug candidate that acts as a pan-selectin antagonist and reverses acute vascular occlusions in sickle cell mice.

化合物

Ponsegromab
Cat.No: T76774
Synonym: PF 06946860
Target: TGF-beta/Smad
Miransertib
Cat.No: T3467
Synonym: ARQ-092,AKT inhibitor 2
Target: Akt, Parasite
Seganserin
Cat.No: T68141
Synonym:
Target: 5-HT Receptor
Ketanserin
Cat.No: T1066
Synonym: R41468,凯他色林,Ketanserin tartrate,酮色林,Ketanserinum
Target: Potassium Channel, 5-HT Receptor, Autophagy
Nelotanserin
Cat.No: T7350
Synonym: 1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲,APD125
Target: 5-HT Receptor
Pimavanserin tartrate
Cat.No: T6946
Synonym: ACP-103,ACP-103 tartrate,Nuplazid,Pimavanserin,匹莫范色林
Target: 5-HT Receptor
Onvansertib
Cat.No: T6247
Synonym: NMS-P937,NMS-1286937
Target: Apoptosis, PLK
Ritanserin
Cat.No: T16759
Synonym: 利坦丝林,R 55667
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Ondansetron hydrochloride dihydrate
Cat.No: T1478
Synonym: 盐酸昂丹司琼,SN 307,NSC 665799,GR 38032,Ondansetron hydrochloride
Target: 5-HT Receptor
Volinanserin
Cat.No: T5389
Synonym: M 100907,MDL100907,氟利色林
Target: 5-HT Receptor
Glemanserin
Cat.No: T22964
Synonym: MDL11939
Target: 5-HT Receptor
N-Desmethyl Pimavanserin
Cat.No: T37979
Synonym: AC-279
Target: 5-HT Receptor
Tropanserin
Cat.No: T8451
Synonym: MDL 72422
Target: 5-HT Receptor
Camonsertib
Cat.No: T62083
Synonym: ATR inhibitor 4,RP-3500
Target: ATM/ATR
Anxiolytic/nonsedative agent-1
Cat.No: T23445
Synonym: TCS 1205
Target: GABA Receptor
Cinanserin hydrochloride
Cat.No: T14968
Synonym: SQ 10643
Target: Influenza Virus, 5-HT Receptor
Benserazide hydrochloride
Cat.No: T1517
Synonym: Benserazide HCl,盐酸苄丝肼,Serazide,Ro 4-4602
Target: Dopamine Receptor
Adatanserin
Cat.No: T23631
Synonym: WY-50324,WY 50324,WAY SEB 324,WY50324
Target: 5-HT Receptor
Insecticidal agent 364
Cat.No: T67914
Synonym:
Target: mTOR, Autophagy
Selonsertib
Cat.No: T3350
Synonym: GS-4997
Target: Apoptosis, ASK, MAPK
Mianserin
Cat.No: T21428
Synonym: Lantanon,Lumin,Norval,Lerivon,Depnon
Target: Histamine Receptor
Blonanserin
Cat.No: T1180
Synonym: 布南色林,AD-5423
Target: Dopamine Receptor, Sigma receptor, 5-HT Receptor, Adrenergic Receptor
Pimavanserin
Cat.No: T2076
Synonym: ACP-103,匹莫范色林
Target: 5-HT Receptor
Fananserin
Cat.No: T15270
Synonym: RP 62203,法南色林
Target: Dopamine Receptor, 5-HT Receptor
Ondansetron
Cat.No: T6615
Synonym: GR-C507/75,GR 38032,昂丹司琼,GR 38032F,SN 307,恩丹西酮
Target: 5-HT Receptor
Cilansetron
Cat.No: T27020
Synonym: KC-9946,KC9946,DU-123265,DU123265
Target: 5-HT Receptor
Ondansetron hydrochloride
Cat.No: T6616
Synonym: SN 307,盐酸昂丹司琼,帕罗西汀杂质A,Ondansetron HCl,Emeset,GR 38032 HCl,NSC 665799,Zofran
Target: 5-HT Receptor
Flibanserin
Cat.No: T4297
Synonym: BIMT-17BS,氟立班丝氨,Girosa,BIMT-17
Target: Dopamine Receptor, 5-HT Receptor
Opiranserin hydrochloride
Cat.No: T9833
Synonym:
Target: P2X Receptor, GlyT, 5-HT Receptor
Ketanserin tartrate
Cat.No: T1066L
Synonym: KJK 945 tartrate,KJK-945 tartrate,KJK945 tartrate
Target: 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor
Adatanserin hydrochloride
Cat.No: T29645
Synonym: WY50324 hydrochloride
Target: 5-HT Receptor
Anserine
Cat.No: T22243
Synonym: L-鹅肌肽,L-Anserine
Target: Endogenous Metabolite
Uzansertib phosphate
Cat.No: T12477
Synonym: INCB053914 phosphate
Target: Pim
Eplivanserin
Cat.No: T11217
Synonym: 依利色林,SR-46349
Target: 5-HT Receptor
isomer-Cilansetron
Cat.No: T27020L
Synonym:
Target: Others
Altanserin
Cat.No: T29913
Synonym: R-53200,R53200,R 53200
Target:
Phenserine
Cat.No: T12446
Synonym: (-)-Eseroline phenylcarbamate,(-)-Phenserine
Target: AChR
Uzansertib
Cat.No: T39090
Synonym: INCB053914
Target:
Zunsemetinib
Cat.No: T39126
Synonym: CDD-450,ATI-450
Target:
Benanserin HCl
Cat.No: T26768
Synonym: Benanserin Hydrochloride,BAS,Benanserin,Benzyl antiserotonin
Target:
Trelanserin
Cat.No: T34918
Synonym: SL650472,SL-650472,SL 650472
Target:
Benserazide
Cat.No: T1517L
Synonym: Ro-44602,Ro44602,Ro 44602,Serazide
Target:
Lunsekimig
Cat.No: T9901A-011
Synonym: SAR443765
Target:
Opiranserin
Cat.No: T16399
Synonym:
Target: P2X Receptor, GlyT, 5-HT Receptor
Insecticidal agent 6
Cat.No: T82064
Synonym:
Target: Parasite
Ketanserinol
Cat.No: T25568
Synonym: Reduced ketanserin
Target:
Anselamimab
Cat.No: T83106
Synonym:
Target:
Cilansetron Hydrochloride
Cat.No: T30936
Synonym: KC-9946,KC9946,KC 9946
Target:
Galdansetron hydrochloride
Cat.No: T70439
Synonym:
Target:
Rivipansel sodium
Cat.No: T71292
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN2245 Sunset Yellow FCF

Food Yellow 3,Orange Yellow S,Sunset yellow,CI 15985

Androgen Receptor Endocrinology/Hormones
Sunset Yellow FCF (Sunset yellow) 是一种橙色偶氮染料,吸光度具有pH 依赖性。Sunset Yellow FCF 可在食品,化妆品和药品中使用,在许多食品中用作着色剂食品添加剂,它们可能具有细胞毒性和遗传毒性,因此在使用这些材料作为食品添加剂时必须小心。
T3829 Ginsenoside F3

人参皂苷F3

Others; IFNAR; Interleukin Immunology/Inflammation; Others
Ginsenoside F3 是一种皂苷,提取自Panax ginseng 叶片。它能够调节1 型 (IL-2, IFN-γ) 及 2 型细胞因子(IL-4 and IL-10) 的产生和表达,有免疫增强的作用。
T11398 Ginsenoside Ra3

人参皂苷 RA3,人参皂苷RA3

Others Others
Ginsenoside Ra3 是分离自人参中,具有抗癌作用。
T3918 Ginsenoside Rb3

人参皂苷 Rb3,Gypenoside IV,人参皂苷Rb3

NF-κB; COX; NO Synthase Immunology/Inflammation; Neuroscience; NF-κB
Ginsenoside Rb3 (Gypenoside IV) 是从三七中提取的一种天然产物。它在 293T 细胞系中抑制 TNFα 诱导的NF-κB 转录活性,IC50为 8.2 μM。它还抑制COX-2和iNOSmRNA 的诱导。
T2822 Ginsenoside Rb1

Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III

ATPase; Mitophagy; IRAK; NF-κB; Autophagy; HSV Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Ginsenoside Rb1 (Gypenoside Ⅲ) 是中药人参的成分,可能具有抑制或阻止肿瘤生长的特性。
T2873 Ginsenoside Rg2

Chikusetsusaponin I,Panaxoside Rg2,人参皂苷Rg2,Prosapogenin C2,(20S)Ginsenoside Rg2,人参皂苷 Rg2

Beta Amyloid; GSK-3; NF-κB Neuroscience; NF-κB; PI3K/Akt/mTOR signaling; Stem Cells
Ginsenoside Rg2 (Chikusetsusaponin I) 是一种人参的主要活性成分。它能够降低Aβ1-42积聚,抑制脂多糖介导的VCAM-1和ICAM-1表达的增加。
T3830 20(R)-Ginsenoside Rg2

20R-Ginsenoside Rg2,20R-人参皂苷Rg2,20(R)-人参皂苷 Rg2

IL Receptor Immunology/Inflammation
20(R)-Ginsenoside Rg2 (20R-Ginsenoside Rg2) 是一种人参皂苷。它能够抑制肺癌 NCI-H1650 细胞,具有抗癌作用。
T6S1485 Ginsenoside Rh4

人参皂苷Rh4

Others Others
Ginsenoside Rh4 可以安全地用作佐剂,具有低溶血作用或无溶血作用。它具有细胞毒活性,其苷元对癌细胞系具有杀伤作用。
T2959 Ginsenoside Rh2

20(S)-Rh2,20S-Ginsenoside Rh2,人参皂苷Rh2,20(S)-Ginsenoside Rh2,人参皂苷 Rh2

Apoptosis; EGFR; Caspase; Endogenous Metabolite Angiogenesis; Apoptosis; JAK/STAT signaling; Metabolism; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Ginsenoside Rh2 (20(S)-Ginsenoside Rh2) 诱导caspase-8和caspase-9活化。它以多途径方式诱导癌细胞凋亡。
T4S1519 Pseudoginsenoside RT5

拟人参皂苷RT5

Others Others
Pseudoginsenoside RT5 分离于 Panax quinquefolium 中。它通过促进神经生长和提高认知能力,具有抗癫痫、抗抑郁活性,还具有抗菌、抗肿瘤、抗疟疾等活性。
T6S1487 Ginsenoside Rg5

人参皂苷Rg5,人参皂甙 Rg5

NF-κB; COX; IGF-1R Immunology/Inflammation; Neuroscience; NF-κB; Tyrosine Kinase/Adaptors
Ginsenoside Rg5 是红参的主要成分,可阻断IGF-1与其受体的结合,IC50约为90 nM。它还通过抑制NF-κB p65的 DNA 结合活性来抑制COX-2的 mRNA 表达。它可促进血管生成和改善高血压,具有抗炎和治疗阿尔茨海默病的潜力。
T3919 Ginsenoside Rb2

Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2

GPR; Others; Influenza Virus; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Microbiology/Virology; Others
Ginsenoside Rb2 (Ginsenoside C) 是人参提取物中的一种主要生物活性成分,具有抗病毒活性,可上调 GPR120 基因表达。
T2878 Ginsenoside Rd

Panaxoside Rd,Sanchinoside Rd,人参皂苷Rd,人参皂苷 Rd,Gypenoside VIII

P450; Calcium Channel; NF-κB; COX; Endogenous Metabolite Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
Ginsenoside Rd (Gypenoside VIII) 抑制 TNFα 诱导的NF-κB 转录活性,还抑制COX-2和iNOSmRNA 的表达。它抑制CYP2D6、CYP1A2、CYP3A4和CYP2C9,也抑制Ca2+内流,有可能抑制或阻止肿瘤生长。
TN1096 Ginsenoside Ra1

人参皂苷 Ra1,人参皂苷Ra1

Others; Tyrosine Kinases Others; Tyrosine Kinase/Adaptors
Ginsenoside Ra1 是来自人参的成分。 Ginsenoside Ra1 对缺氧/复氧诱导的蛋白酪氨酸激酶 (PTK) 活化具有显着抑制作用。
TN1686 Ginsenoside Rg4

人参皂苷 RG4

Antibacterial Microbiology/Virology
Ginsenoside Rg4 是分离自Panax ginsengC. A. Meyer 叶子中的一种人参三醇型人参皂苷。人参三醇型人参皂苷具有多种生物活性,包括防腐,抗糖尿病,伤口愈合,免疫刺激和抗氧化活性等。
T2872 Ginsenoside Re

人参皂苷 Re,Ginsenoside B2,Panaxoside Re,Chikusetsusaponin Ivc,Sanchinoside Re,人参皂苷Re

Beta Amyloid; NF-κB; Endogenous Metabolite; JNK MAPK; Metabolism; Neuroscience; NF-κB
Ginsenoside Re (Ginsenoside B2) 是一种人参提取物,可降低 β-淀粉样蛋白 (Aβ),还通过抑制 JNK 和 NF-κB 发挥抗炎作用。
T3916 Ginsenoside F2

人参皂苷F2

Apoptosis; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism
Ginsenoside F2 是 Ginsenoside Rb1 的代谢物,通过激活内在的凋亡途径和线粒体功能障碍来诱导乳腺的凋亡,对乳腺癌干细胞具有抗增殖活性。
TN1997 Notoginsenoside FP2

三七皂苷FP2

Others Others
Notoginsenoside FP2 是从三七 Panax notoginseng 果实花梗中分离得到的天然产物,可用于治疗心血管疾病的研究。
T3849 Kinsenoside

金线莲苷,(+)-Kinsenoside

Apoptosis; Nrf2 Apoptosis; Immunology/Inflammation
Kinsenoside ((+)-Kinsenoside) 是从金盏花属植物中分离得到的主要活性成分,以 Nrf2 依赖的方式保护髓核细胞在氧化应激下的生存能力,防止细胞凋亡、衰老和线粒体功能障碍。它显示出显着的抗肝毒性和抗炎活性。
T4S1518 Pseudoginsenoside RT1

拟人参皂苷 RT1,假人参皂苷RT1

Others Others
Pseudoginsenoside RT1 是分离自 Randia siamensis 中,具有鱼毒素作用。它可导致血压下降、心率加快和子宫自发收缩力增加。
T3401 Ginsenoside F1

人参皂苷 F1,20(S)-Ginsenoside F1

P450; Endogenous Metabolite Metabolism
Ginsenoside F1 (20(S)-Ginsenoside F1) 是一种 Ginsenoside Rg1 的酶促修饰衍生物,它竞争性抑制CYP3A4,对 CYP2D6 具有较弱的抑制作用。
TN7110 Ginsenoside Rs2

人参皂苷Rs2

Others Others
Ginsenoside Rs2 是从人参Panax japonicus var.叶中分离得到的天然产物。
T2932 Ginsenoside Rh1

Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1

IL Receptor; TNF; Endogenous Metabolite; PPAR; Interleukin Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism
Ginsenoside Rh1 (Sanchinoside B2) 是人参的一种主要成分,具有抗炎作用,抑制PPAR-γ,TNF-α,IL-6和IL-1β的表达。
T2S0223 Isosinensetin

异橙黄酮,6-Demethoxynobiletin

Antioxidant; HIV Protease; Antibacterial; P-gp Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; oxidation-reduction; Proteases/Proteasome
Isosinensetin (6-Demethoxynobiletin) 是从青皮中提取的一种甲氧基黄酮,具有抗氧化和抑制 HIV-1 蛋白酶的活性。
T5S1590 Notoginsenoside Fe

三七皂苷Fe,Notoginseng triterpenes,Ginsenoside Mb

Others Others
Notoginsenoside Fe (Ginsenoside Mb) 是一种分离自珠子参变种中的天然化合物。
T3811 Ginsenoside C-K

20(S)-人参皂苷 C-K,Ginsenoside compound K,Ginsenoside K,人参皂苷 C-K

P450; cell cycle arrest; COX; NO Synthase Cell Cycle/Checkpoint; Immunology/Inflammation; Metabolism; Neuroscience
Ginsenoside C-K (Ginsenoside K) 是 Ginsenoside Rb1 的细菌代谢物,可通过抑制诱生型一氧化氮合酶和COX-2来发挥抗炎作用。它在人肝微粒体中抑制CYP2C9和CYP2A6活性,IC50分别为 32.0±3.6 和 63.6±4.2 μM。
TN2296 Vinaginsenoside R4

越南参皂苷R4

Others Others
Vinaginsenoside R4 是分离自水培人参的叶子中。它能够抑制黑色素的生物合成,并增强斑马鱼的色素沉着,对 melan-a 细胞没有任何细胞毒性作用。
T2777 Ginsenoside Rg1

Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2

Apoptosis; Beta Amyloid; NF-κB Apoptosis; Neuroscience; NF-κB
Ginsenoside Rg1 (Panaxoside Rg1) 是人参的主要活性成分之一,可减少NF-κB 核易位。它改善认知功能受损,通过降低大脑Aβ水平来发挥作用。
TN6930 5-Desmethylsinensetin

Others Others
5-desmethylsinensetin 是分离自Stevia satureiifoliavar.satureiifolia 的天然产物,显示出抗原生动物的活性,抑制T. cruzi epimastigotes 和trypomastigotes 的IC50分别为 0.4 μg/mL 和75.1 μg/mL。
TN2100 Pratensein

红车轴草素,三叶草

Others; NF-κB NF-κB; Others
Pratensein 是黄酮类化合物,能够减少氧化损伤和恢复突触和 BDNF 水平,改善 β-淀粉样蛋白诱导的大鼠认知障碍。
T4704 L-Anserine nitrate

L-鹅肌肽硝酸盐,L-Anserine nitrate salt

Others; Endogenous Metabolite Metabolism; Others
L-Anserine nitrate (L-Anserine nitrate salt) 是一种存在于大多数动物组织中的二肽。在模型系统中,它是一种有效的抗氧化剂和羟基自由基清除剂。该化合物抑制醛糖和酮糖还原糖诱导的非酶蛋白糖基化。
T3812 (20R)-Ginsenoside Rg3

人参皂甙 RG3,(20R)-人参皂苷Rg3,20(R)-Ginsenoside Rg3,(20R)Ginsenoside Rg3,20(R)-Propanaxadiol

Others Others
(20R)-Ginsenoside Rg3 (20(R)-Propanaxadiol) 是一种人参根中的化合物,具有抑制血管内皮细胞增生(IC50= 10 nM)和抗肿瘤作用。
T0783 Mianserin hydrochloride

Mianserin HCl,Org GB 94,盐酸米安色林,ORG GB-94 HCl

Dopamine Receptor; 5-HT Receptor; Opioid Receptor; Adrenergic Receptor; Histamine Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mianserin hydrochloride (Org GB 94) 是一种有抗抑郁活性的 H1 受体反向激动剂。
T13626 Cottonseed oil

Others Others
Cottonseed oil 是一种提取自棉花种子中的食用油,是一种植物油中杀虫能力极强的油。
T3920 Pseudoginsenoside F11

Ginsenoside A1,拟人参皂苷 F11,拟人参皂苷F11

Others; Endogenous Metabolite Metabolism; Others
Pseudoginsenoside F11 (Ginsenoside A1) 从人参根和叶中分离得到。PF11在一系列心血管和中枢神经系统疾病中具有广泛的保护作用。
T3402 20(S)-Ginsenoside Rg3

20(S)-人参皂苷 Rg3,人参皂苷 Rg3,20(S)-Ginsenoside-Rg3,Rg3,20S-Ginsenoside Rg3,Ginsenoside Rg3,S-Ginsenoside Rg3

EGFR; Beta Amyloid; Potassium Channel; NF-κB; COX; Sodium Channel; Endogenous Metabolite Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Tyrosine Kinase/Adaptors
20(S)-Ginsenoside Rg3 (Rg3) 是红参的主要成分,通过抑制肿瘤细胞的粘附和侵袭来抑制肿瘤细胞肺转移。它抑制Na+和hKv1.4通道,IC50分别为 32.2±4.5 和 32.6±2.2 μM。它还抑制Aβ,NF-κB 活性和COX-2表达,抑制人脐静脉内皮细胞的增殖并具有抗血管生成活性。
T6S1495 Ginsenoside Rk3

人参皂苷Rk3,人参皂甙 Rk3

Others; NF-κB NF-κB; Others
Ginsenoside Rk3 是存在于 Panax notoginseng 的根中。它能够抑制 HepG2 细胞中 TNF-α 诱导的 NF-κB 转录活性,IC50=14.24±1.30 μM。
T3813 20(R)-Ginsenoside Rh2

20(R)-人参皂苷 RH2,(20R)Ginsenoside Rh2,Ginsenoside Rh2,20(R)-人参皂苷Rh2

Apoptosis; MMP; HSV Apoptosis; Microbiology/Virology; Proteases/Proteasome
20(R)-Ginsenoside Rh2 (Ginsenoside Rh2) 是人参皂苷 Rh2 的次要立体异构体,具有基质金属蛋白酶抑制作用。它有抗癌、抗炎和抗氧化活性。
T3915 Ginsenoside Ro

人参皂苷Ro,Chikusetsusaponin 5,Polysciasaponin P3,人参皂苷 Ro,Chikusetsusaponin V

Calcium Channel; Reductase; Prostaglandin Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism
Ginsenoside Ro (Chikusetsusaponin V) 能降低 TXA2产量,较弱降低 COX-1 和 TXAS 活性,具有 Ca2+拮抗剂的抗血小板作用,IC50为 155 μM。
T4S0227 Sinensetin

Pedalitin permethyl ether,甜橙素

TNF; PGE Synthase Apoptosis; Immunology/Inflammation
Sinensetin (Pedalitin permethyl ether) 是从水果中发现的一种甲基化黄酮,有很强的抗血管和抗炎症的能力。
T3S1589 Notoginsenoside Fa

Others Others
Notoginsenoside Fa 是一种原人参二醇型皂苷,从P. notoginseng 提取出来得到,有激活和恢复退化脑功能的潜能。
T2961 Notoginsenoside R1

Sanqi glucoside R1,Sanchinoside R1,三七皂苷R1

Apoptosis; ERK; Beta Amyloid Apoptosis; MAPK; Neuroscience
Notoginsenoside R1 (Sanchinoside R1) 是一种从三七中分离出来的皂苷,具有抗氧化、抗炎、抗血管生成和抗凋亡的活性。它有神经保护和抗缺血/再灌注损伤的心脏保护作用。
T6S1587 Notoginsenoside R2

三七皂苷R2,20(S)-Notoginsenoside R2,Ginsenoside Ng-R2

Others; Nrf2 Immunology/Inflammation; Others
Notoginsenoside R2 (20(S)-Notoginsenoside R2) 是一种新分离三七皂苷,表现出对6-OHDA 诱导的氧化应激及细胞凋亡的保护作用。
T3S1591 Notoginsenoside Fc

三七皂苷 FC,三七皂苷Fc

Others; Autophagy Autophagy; Others
Notoginsenoside Fc 是从三七叶中分离得到的原卟啉二醇型皂苷,可通过促进自噬促进糖尿病大鼠血管损伤后的内皮细胞再生,具有抗血小板聚集的作用。
TN1684 Ginsenoside F5

人参皂苷 F5,人参皂苷F5

Apoptosis Apoptosis
Ginsenoside F5 是从人参中提取的一种天然产物,通过凋亡途径显着抑制 HL-60 细胞的生长。
T5761 Notoginsenoside Ft1

三七皂苷FT1,三七皂甙 Ft1

Others; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; Metabolism; Others
Notoginsenoside Ft1 是一种植物分离的三七皂苷,具有刺激血管生成的作用。
T6S1500 Ginsenoside Rf

人参皂苷 Rf,Ginsenoside-Rf,Panaxoside Rf

Calcium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
Ginsenoside Rf (Panaxoside Rf) 是人参根的微量成分,可抑制 N 型 Ca2+通道。
T3793 (20R)-Ginsenoside Rh1

20(R)-Ginsenoside Rh1,人参皂苷 R-RH1,人参皂苷R-RH1

Others Others
(20R)-Ginsenoside Rh1 (20(R)-Ginsenoside Rh1) 是 Ginsenoside Rh1 的 R 型异构体,分离自 Panax Ginseng 中,能够阻碍凝血酶诱导的纤维蛋白原向纤维蛋白的转化。
T2720 Ginsenoside Rc

Panaxoside Rc,人参皂苷Rc,人参皂苷 Rc

Others; TNF; GABA Receptor; Interleukin Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; Others
Ginsenoside Rc (Panaxoside Rc) 是人参中的一种人参皂苷,可抑制 TNF-α 和 IL-1β 的表达。它增强 GABA 受体 A 介导的离子通道电流。
TN2802 20-O-Glucoginsenoside Rf

Others Others
20-O-Glucoginsenoside Rf 是从人参 Panax ginseng C. A. Mey 中提取的天然产物。
------------------------ 更多 ------------------------

天然产物

Sunset Yellow FCF
Cat.No: TN2245
Synonym: Food Yellow 3,Orange Yellow S,Sunset yellow,CI 15985
Target: Androgen Receptor
Ginsenoside F3
Cat.No: T3829
Synonym: 人参皂苷F3
Target: Others, IFNAR, Interleukin
Ginsenoside Ra3
Cat.No: T11398
Synonym: 人参皂苷 RA3,人参皂苷RA3
Target: Others
Ginsenoside Rb3
Cat.No: T3918
Synonym: 人参皂苷 Rb3,Gypenoside IV,人参皂苷Rb3
Target: NF-κB, COX, NO Synthase
Ginsenoside Rb1
Cat.No: T2822
Synonym: Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III
Target: ATPase, Mitophagy, IRAK, NF-κB, Autophagy, HSV
Ginsenoside Rg2
Cat.No: T2873
Synonym: Chikusetsusaponin I,Panaxoside Rg2,人参皂苷Rg2,Prosapogenin C2,(20S)Ginsenoside Rg2,人参皂苷 Rg2
Target: Beta Amyloid, GSK-3, NF-κB
20(R)-Ginsenoside Rg2
Cat.No: T3830
Synonym: 20R-Ginsenoside Rg2,20R-人参皂苷Rg2,20(R)-人参皂苷 Rg2
Target: IL Receptor
Ginsenoside Rh4
Cat.No: T6S1485
Synonym: 人参皂苷Rh4
Target: Others
Ginsenoside Rh2
Cat.No: T2959
Synonym: 20(S)-Rh2,20S-Ginsenoside Rh2,人参皂苷Rh2,20(S)-Ginsenoside Rh2,人参皂苷 Rh2
Target: Apoptosis, EGFR, Caspase, Endogenous Metabolite
Pseudoginsenoside RT5
Cat.No: T4S1519
Synonym: 拟人参皂苷RT5
Target: Others
Ginsenoside Rg5
Cat.No: T6S1487
Synonym: 人参皂苷Rg5,人参皂甙 Rg5
Target: NF-κB, COX, IGF-1R
Ginsenoside Rb2
Cat.No: T3919
Synonym: Ginsenoside C,人参皂苷 Rb2,人参皂苷Rb2
Target: GPR, Others, Influenza Virus, Endogenous Metabolite
Ginsenoside Rd
Cat.No: T2878
Synonym: Panaxoside Rd,Sanchinoside Rd,人参皂苷Rd,人参皂苷 Rd,Gypenoside VIII
Target: P450, Calcium Channel, NF-κB, COX, Endogenous Metabolite
Ginsenoside Ra1
Cat.No: TN1096
Synonym: 人参皂苷 Ra1,人参皂苷Ra1
Target: Others, Tyrosine Kinases
Ginsenoside Rg4
Cat.No: TN1686
Synonym: 人参皂苷 RG4
Target: Antibacterial
Ginsenoside Re
Cat.No: T2872
Synonym: 人参皂苷 Re,Ginsenoside B2,Panaxoside Re,Chikusetsusaponin Ivc,Sanchinoside Re,人参皂苷Re
Target: Beta Amyloid, NF-κB, Endogenous Metabolite, JNK
Ginsenoside F2
Cat.No: T3916
Synonym: 人参皂苷F2
Target: Apoptosis, Endogenous Metabolite, Autophagy
Notoginsenoside FP2
Cat.No: TN1997
Synonym: 三七皂苷FP2
Target: Others
Kinsenoside
Cat.No: T3849
Synonym: 金线莲苷,(+)-Kinsenoside
Target: Apoptosis, Nrf2
Pseudoginsenoside RT1
Cat.No: T4S1518
Synonym: 拟人参皂苷 RT1,假人参皂苷RT1
Target: Others
Ginsenoside F1
Cat.No: T3401
Synonym: 人参皂苷 F1,20(S)-Ginsenoside F1
Target: P450, Endogenous Metabolite
Ginsenoside Rs2
Cat.No: TN7110
Synonym: 人参皂苷Rs2
Target: Others
Ginsenoside Rh1
Cat.No: T2932
Synonym: Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1
Target: IL Receptor, TNF, Endogenous Metabolite, PPAR, Interleukin
Isosinensetin
Cat.No: T2S0223
Synonym: 异橙黄酮,6-Demethoxynobiletin
Target: Antioxidant, HIV Protease, Antibacterial, P-gp
Notoginsenoside Fe
Cat.No: T5S1590
Synonym: 三七皂苷Fe,Notoginseng triterpenes,Ginsenoside Mb
Target: Others
Ginsenoside C-K
Cat.No: T3811
Synonym: 20(S)-人参皂苷 C-K,Ginsenoside compound K,Ginsenoside K,人参皂苷 C-K
Target: P450, cell cycle arrest, COX, NO Synthase
Vinaginsenoside R4
Cat.No: TN2296
Synonym: 越南参皂苷R4
Target: Others
Ginsenoside Rg1
Cat.No: T2777
Synonym: Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2
Target: Apoptosis, Beta Amyloid, NF-κB
5-Desmethylsinensetin
Cat.No: TN6930
Synonym:
Target: Others
Pratensein
Cat.No: TN2100
Synonym: 红车轴草素,三叶草
Target: Others, NF-κB
L-Anserine nitrate
Cat.No: T4704
Synonym: L-鹅肌肽硝酸盐,L-Anserine nitrate salt
Target: Others, Endogenous Metabolite
(20R)-Ginsenoside Rg3
Cat.No: T3812
Synonym: 人参皂甙 RG3,(20R)-人参皂苷Rg3,20(R)-Ginsenoside Rg3,(20R)Ginsenoside Rg3,20(R)-Propanaxadiol
Target: Others
Mianserin hydrochloride
Cat.No: T0783
Synonym: Mianserin HCl,Org GB 94,盐酸米安色林,ORG GB-94 HCl
Target: Dopamine Receptor, 5-HT Receptor, Opioid Receptor, Adrenergic Receptor, Histamine Receptor
Cottonseed oil
Cat.No: T13626
Synonym:
Target: Others
Pseudoginsenoside F11
Cat.No: T3920
Synonym: Ginsenoside A1,拟人参皂苷 F11,拟人参皂苷F11
Target: Others, Endogenous Metabolite
20(S)-Ginsenoside Rg3
Cat.No: T3402
Synonym: 20(S)-人参皂苷 Rg3,人参皂苷 Rg3,20(S)-Ginsenoside-Rg3,Rg3,20S-Ginsenoside Rg3,Ginsenoside Rg3,S-Ginsenoside Rg3
Target: EGFR, Beta Amyloid, Potassium Channel, NF-κB, COX, Sodium Channel, Endogenous Metabolite
Ginsenoside Rk3
Cat.No: T6S1495
Synonym: 人参皂苷Rk3,人参皂甙 Rk3
Target: Others, NF-κB
20(R)-Ginsenoside Rh2
Cat.No: T3813
Synonym: 20(R)-人参皂苷 RH2,(20R)Ginsenoside Rh2,Ginsenoside Rh2,20(R)-人参皂苷Rh2
Target: Apoptosis, MMP, HSV
Ginsenoside Ro
Cat.No: T3915
Synonym: 人参皂苷Ro,Chikusetsusaponin 5,Polysciasaponin P3,人参皂苷 Ro,Chikusetsusaponin V
Target: Calcium Channel, Reductase, Prostaglandin Receptor
Sinensetin
Cat.No: T4S0227
Synonym: Pedalitin permethyl ether,甜橙素
Target: TNF, PGE Synthase
Notoginsenoside Fa
Cat.No: T3S1589
Synonym:
Target: Others
Notoginsenoside R1
Cat.No: T2961
Synonym: Sanqi glucoside R1,Sanchinoside R1,三七皂苷R1
Target: Apoptosis, ERK, Beta Amyloid
Notoginsenoside R2
Cat.No: T6S1587
Synonym: 三七皂苷R2,20(S)-Notoginsenoside R2,Ginsenoside Ng-R2
Target: Others, Nrf2
Notoginsenoside Fc
Cat.No: T3S1591
Synonym: 三七皂苷 FC,三七皂苷Fc
Target: Others, Autophagy
Ginsenoside F5
Cat.No: TN1684
Synonym: 人参皂苷 F5,人参皂苷F5
Target: Apoptosis
Notoginsenoside Ft1
Cat.No: T5761
Synonym: 三七皂苷FT1,三七皂甙 Ft1
Target: Others, HIF/HIF Prolyl-Hydroxylase
Ginsenoside Rf
Cat.No: T6S1500
Synonym: 人参皂苷 Rf,Ginsenoside-Rf,Panaxoside Rf
Target: Calcium Channel, Endogenous Metabolite
(20R)-Ginsenoside Rh1
Cat.No: T3793
Synonym: 20(R)-Ginsenoside Rh1,人参皂苷 R-RH1,人参皂苷R-RH1
Target: Others
Ginsenoside Rc
Cat.No: T2720
Synonym: Panaxoside Rc,人参皂苷Rc,人参皂苷 Rc
Target: Others, TNF, GABA Receptor, Interleukin
20-O-Glucoginsenoside Rf
Cat.No: TN2802
Synonym:
Target: Others
--------- 更多 ---------
Cat. No. Product Name Species Expression System
TMPY-02646 NSE/ENO2 Protein, Human, Recombinant (His)

enolase 2 (γ, neuronal),NSE,HEL-S-279,enolase 2 (ga...

Human E. coli
The combination of silencing ENO2 and 2-deoxyglucose (2-DG) synergistically inhibited leukemia cell survival. ENO2 may be a biological marker for monitoring chemotherapeutic efficacy and relapse in ALL. Reduced ENO2 expression may be a biomarker for a subset of autistic children. Neuron specific enolase (ENO2, gamma-enolase) has been used as a biomarker to help identify neuroendocrine differentiation in breast cancer.
TMPH-03617 Miraculin Protein, Synsepalum dulcificum, Recombinant (His)

Synsepalum dulcificum P. pastoris (Yeast)
Miraculin has the property of modifying a sour taste into a sweet taste. This alteration of taste perception persists for many minutes. Miraculin Protein, Synsepalum dulcificum, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 23.4 kDa and the accession number is P13087.
TMPY-06016 Phl p 5 Protein, Phleum pratense, Recombinant

Phleum pratense E. coli
Phl p 5 Protein, Phleum pratense, Recombinant is expressed in E. coli expression system. The predicted molecular weight is 28.7 kDa and the accession number is Q40960-1.
TMPH-03095 Phl p 6 Protein, Phleum pratense, Recombinant (His & Myc)

Phleum pratense E. coli
Phl p 6 Protein, Phleum pratense, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 19.2 kDa and the accession number is P43215.
TMPH-03093 Phl p 5a Protein, Phleum pratense, Recombinant (His & SUMO)

Phleum pratense E. coli
N/A. Phl p 5a Protein, Phleum pratense, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 44.5 kDa and the accession number is Q40962.
TMPY-06015 Phl p 2 Protein, Phleum pratense, Recombinant (His)

Phleum pratense HEK293 Cells
Phl p 2 Protein, Phleum pratense, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 13.1 kDa and the accession number is P43214-1.
TMPH-03094 Phl p 5b Protein, Phleum pratense, Recombinant (His & SUMO)

Phleum pratense E. coli
Has ribonuclease activity. May be involved in host-pathogen interactions. Phl p 5b Protein, Phleum pratense, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 42.1 kDa and the accession number is Q40963.
TMPY-06149 Phl p 5 Protein, Phleum pratense, Recombinant (His)

Phleum pratense HEK293 Cells
Phl p 5 Protein, Phleum pratense, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 30.9 kDa and the accession number is Q40960-1.
TMPH-03616 Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His)

Synsepalum dulcificum E. coli
Miraculin has the property of modifying a sour taste into a sweet taste. This alteration of taste perception persists for many minutes. Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 24.9 kDa and the accession number is P13087.
TMPH-03096 Profilin 2 Protein, Phleum pratense, Recombinant (His & Myc)

Phleum pratense E. coli
Binds to actin and affects the structure of the cytoskeleton. At high concentrations, profilin prevents the polymerization of actin, whereas it enhances it at low concentrations. By binding to PIP2, it inhibits the formation of IP3 and DG. Profilin 2 Protein, Phleum pratense, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 21.5 kDa and the accession number is O24650.
TMPH-03626 Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (His & Myc)

Toxin II-11,Beta-like toxin Ts1,Ts7,Beta-mammal/inse

Tityus serrulatus Baculovirus Insect Cells
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (His & Myc) is expressed in Baculovirus insect cells with N-10xHis and C-Myc tag. The predicted molecular weight is 10.8 kDa and the accession number is P15226.
TMPH-03627 Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (E. coli, His & Myc)

Ts VII,Beta-like toxin Ts1,Toxin II-11,Ts7,Tityustoxin VII,P...

Tityus serrulatus E. coli
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (E. coli, His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 14.3 kDa and the accession number is P15226.

重组蛋白

NSE/ENO2 Protein, Human, Recombinant (His)
Cat.No: TMPY-02646
Species: Human
Expression System: E. coli
Miraculin Protein, Synsepalum dulcificum, Recombinant (His)
Cat.No: TMPH-03617
Species: Synsepalum dulcificum
Expression System: P. pastoris (Yeast)
Phl p 5 Protein, Phleum pratense, Recombinant
Cat.No: TMPY-06016
Species: Phleum pratense
Expression System: E. coli
Phl p 6 Protein, Phleum pratense, Recombinant (His & Myc)
Cat.No: TMPH-03095
Species: Phleum pratense
Expression System: E. coli
Phl p 5a Protein, Phleum pratense, Recombinant (His & SUMO)
Cat.No: TMPH-03093
Species: Phleum pratense
Expression System: E. coli
Phl p 2 Protein, Phleum pratense, Recombinant (His)
Cat.No: TMPY-06015
Species: Phleum pratense
Expression System: HEK293 Cells
Phl p 5b Protein, Phleum pratense, Recombinant (His & SUMO)
Cat.No: TMPH-03094
Species: Phleum pratense
Expression System: E. coli
Phl p 5 Protein, Phleum pratense, Recombinant (His)
Cat.No: TMPY-06149
Species: Phleum pratense
Expression System: HEK293 Cells
Miraculin Protein, Synsepalum dulcificum, Recombinant (E. coli, His)
Cat.No: TMPH-03616
Species: Synsepalum dulcificum
Expression System: E. coli
Profilin 2 Protein, Phleum pratense, Recombinant (His & Myc)
Cat.No: TMPH-03096
Species: Phleum pratense
Expression System: E. coli
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (His & Myc)
Cat.No: TMPH-03626
Species: Tityus serrulatus
Expression System: Baculovirus Insect Cells
Beta-mammal/insect toxin Ts1 Protein, Tityus serrulatus, Recombinant (E. coli, His & Myc)
Cat.No: TMPH-03627
Species: Tityus serrulatus
Expression System: E. coli
TargetMol Loading
联系我们
400-820-0310

上海市静安区江场三路238号8楼