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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T21618L Myelin Basic Protein (87-99) Acetate

Myelin Basic Protein (87-99) Acetate (118506-26-6 Free base)

Others Others
Myelin Basic Protein (87-99) Acetate (Myelin Basic Protein (87-99) Acetate (118506-26-6 Free base)) 是一种致脑炎肽,可诱导碱性蛋白特异性 T 细胞增殖。 它导致外周血单核细胞中的 Th1 极化,这与多发性硬化症 (MS) 有牵连。
TP1786L Amyloid β-Protein 10-20 acetate

Amyloid β-Protein 10-20 acetate(152286-31-2 free base)

Beta Amyloid Neuroscience
Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) 是 Amyloid-β 肽的片段,可能用于神经系统疾病的研究。Amyloid β 蛋白片段含有 α-分泌酶加工位点(Lys16-Leu17 键)。它还包含负责与小胶质细胞结合的 HHQK 结构域(残基 13-16)。
TP1053L Protein Kinase C 19-31 acetate

Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Protein Kinase C 19-31 acetate(121545-65-1 free base) 是一种蛋白激酶 C (PKC) 的肽抑制剂,源自 PKCa 的假底物调节结构域(残基 19-31),在 25 位用丝氨酸取代野生型丙氨酸作为蛋白激酶 C 底物肽,用于测试蛋白激酶 C 活性。
T9892 JAMM protein inhibitor 2 

Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]-

Others Others
JAMM protein inhibitor 2 (Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]-) 是 JAMM 蛋白酶的抑制剂,可用于抗癌的研究。 对thrombin、Rpn11 和 MMP2 的 IC50 分别为 10 μM、46 μM 和 89 μM。
TP1271L Calmodulin-Dependent Protein Kinase II 290-309 acetate

Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base)

CaMK Neuroscience
Calmodulin-Dependent Protein Kinase II 290-309 acetate 是 Ca2+/calmodulin-dependent protein kinase II 的有效拮抗剂(IC50 = 52 nM)。
TP1453 Tau protein (592-597), Human TFA

Others Others
Tau protein (592-597), Human TFA 是人 Tau 蛋白的肽片段。
T67755 Protein kinase G inhibitor-1

PKA Tyrosine Kinase/Adaptors
Protein kinase G inhibitor-1是有效的蛋白激酶G 抑制剂,IC50= 0.9 uM。
T9779 Protein kinase inhibitor 6

Protein kinase inhibitor 6 是一种蛋白激酶抑制剂。
T9940 Protein kinase G inhibitor-2

Others Others
Protein kinase G inhibitor-2 具有抗菌、抗病毒和抗肿瘤活性。
T4207 (S,R,S)-AHPC hydrochloride

VHL Ligand 1 hydrochloride,ULM-1,Protein degrader 1 hydrochloride

Others; Ligand for E3 Ligase Others; PROTAC
(S,R,S)-AHPC hydrochloride (Protein degrader 1 hydrochloride) 是基于 VH032 的 VHL 配体,可用于募集 von Hippel-Lindau (VHL) 蛋白。它能够利用 linker 与靶蛋白配体连接,得到 PROTAC 分子。
T9631 IRAK-4 protein kinase inhibitor 2

IRAK Immunology/Inflammation; NF-κB
IRAK-4 protein kinase inhibitor 2 是有效的白介素 1 受体相关激酶 4 抑制剂,IC50为 4 μM。它在与炎症和免疫相关的疾病领域有研究价值。
T4692 Protein kinase inhibitors 1 hydrochlorid

Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))

Others Others
Protein kinase inhibitors 1 hydrochlorid (Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))) 是一种新型 HIPK2 抑制剂,IC50 为 74 nM,Kd 为 9.5 nM。
TP1051L Protein Kinase C Peptide Substrate acetate

Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)

Others Others
Protein Kinase C Peptide Substrate acetate(120253-69-2 free base) 以依赖于第二信使和特定衔接蛋白的方式靶向特定细胞间隔物,以响应激活 g 蛋白偶联受体、酪氨酸激酶受体或酪氨酸激酶偶联受体的细胞外信号。
TP1628L Activated Protein C (390-404), human acetate

Activated Protein C (390-404), human acetate(146340-20-7 Free base)

APC Cell Cycle/Checkpoint
Activated Protein C (390-404), human acetate (Activated Protein C ) 抑制 APC 抗凝活性。
TP1676L C-Reactive Protein (CRP) 201-206 acetate

C-Reactive Protein (CRP) 201-206 acetate(130348-99-1 free base)

Others Others
C-Reactive Protein (CRP) 201-206 acetate (C-Reactive Protein )(130348-99-1 free base) 是 C-反应蛋白的 201-206 片段。 C-反应蛋白 (CRP) 醋酸盐是炎症的原型标志物,是心血管风险标志物,可能促进动脉粥样硬化形成。
TP1516L C-Reactive Protein (CRP) 77-82 acetate

C-Reactive Protein (CRP) 77-82 acetate(130349-01-8 free base)

Others Others
C-Reactive Protein (CRP) 77-82 acetate(130349-01-8 free base) 是 C-反应蛋白的 77-82 片段。 C-反应蛋白 (CRP) 是炎症的原型标志物,是心血管风险标志物,可能促进动脉粥样硬化。C-反应蛋白 (CRP) 是一种环状(环状)五聚体蛋白,存在于血浆中,其循环浓度炎症反应而升高。它是一种肝脏来源的急性期蛋白,在巨噬细胞和 T 细胞分泌 IL-6 后会增加。
TP1592L C-Reactive Protein (CRP) 174-185 acetate

C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base)

Others Others
C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base) 是一种急性期血清蛋白,可响应炎性细胞因子而合成,在动物中产生抗肿瘤作用。片段 CRP (174-185) (RS-83277) 通过显着增强体外人单核细胞和肺泡巨噬细胞的杀肿瘤活性显示出相似的活性。
TP1270L 2:PN:US20040072744 SEQID:2 claimed protein acetate

2:PN:US20040072744 SEQID:2 claimed protein acetate(389572-87-6 free base)

Others Others
2:PN:US20040072744 SEQID:2 claimed protein acetate 是一种合成肽,用于唐氏综合症和精神分裂症的研究。
T40250 SHP2 protein degrader-1

SHP2 protein degrader-1

SHP2 protein degrader-1 is a highly efficient allosteric inhibitor targeting SHP2. It effectively induces degradation of SHP2 protein, resulting in cell apoptosis. This compound shows promising potential for studying diseases associated with SHP2.
T38919 Protein E7(43-62)

Protein E7(43-62)

Protein E7(43-62) is a peptide derived from the E7 protein. The peptide spans the 43rd to 62nd amino acid residues and exhibits anti-tumor effects.
TP1902L1 G-Protein antagonist peptide acetate

Adrenergic Receptor GPCR/G Protein; Neuroscience
G-Protein antagonist peptide acetate 是一种 substance P 相关肽,可抑制 G 蛋白与其受体的结合。G-Protein antagonist peptide acetate 竞争性和可逆性地抑制毒蕈碱型乙酰胆碱受体 M2 (M2 muscarinic receptor) 对 Gi 或 Go 的激活,并通过 β-肾上腺素受体抑制 Gs 的激活。
TP1229 β-Amyloid (1-15)

Amyloid β-Protein (1-15)

Beta Amyloid Neuroscience
β-Amyloid (1-15) (Amyloid β-Protein (1-15)) 是 β-淀粉样蛋白片段,可用于研究阿尔茨海默病。
T3201 WDR5-0103

WD-Repeat Protein 5-0103

Histone Methyltransferase; JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
WDR5-0103 (WD-Repeat Protein 5-0103) 是一种有效且特异性的 WD 重复蛋白 5 (WDR5) 拮抗剂,Kd 值为450 nM。
TP1676 C-Reactive Protein (CRP) (201-206)

C-Reactive Protein (CRP) 201-206

Others Others
C-Reactive Protein (CRP) (201-206) 是 C-反应蛋白的 201-206 片段。其中C-反应蛋白 (CRP) 是炎症的原型标志物,是心血管风险标志物,可能促进动脉粥样硬化形成。
T40719 (Cys47)-HIV-1 tat Protein (47-57)

(Cys47)-HIV-1 tat Protein (47-57)

(Cys47)-HIV-1 tat Protein (47-57) possesses membrane translocation functionality and can serve as a surface derivatization agent for magnetic pharmaceuticals, thereby enhancing their uptake into specific target cells.
T2444 KNK437

Heat Shock Protein Inhibitor I

HSP Cytoskeletal Signaling; Metabolism
KNK437 (Heat Shock Protein Inhibitor I) 是一种 HSP 抑制剂,抑制 HSP40,HSP70 和 HSP105 的活化。
T38964 Peripheral Myelin P0 Protein (180-199), mouse

Peripheral Myelin P0 Protein (180-199), mouse

Peripheral Myelin P0 Protein (180-199), derived from mice, is a purified component of the myelin found in the peripheral nerves. This protein serves as a neuritogenic peptide, initiating the growth of neuronal processes.
T40925 Peripheral Myelin Protein P2 (53-78), bovine

Peripheral Myelin Protein P2 (53-78), bovine

Bovine Peripheral Myelin Protein P2 (53-78) is a derivative composed of amino acid residues 53 to 78 from the peripheral myelin P2 protein of bovine origin. It acts as a T cell epitope and is used to induce experimental autoimmune neuritis (EAN) in Lewis rats.
T40272 KRAS mutant protein inhibitor 1

KRAS mutant protein inhibitor 1 is a KRAS mutant protein inhibitor for potential treatment in cancer.
T39860 Protein kinase inhibitors 1 hydrochloride

Protein Kinase Inhibitors 1 Hydrochloride effectively inhibits HIPK2, demonstrating high potency with IC50 values of 136 nM for HIPK1 and 74 nM for HIPK2, alongside a dissociation constant (Kd) of 9.5 nM for HIPK2.
T38687 Influenza Matrix Protein (61-72)

Influenza Matrix Protein (61-72) is a peptide derived from the matrix protein of influenza viruses and encompasses amino acids 61-72. This specific epitope, Influenza Matrix Protein (61-72), has the ability to elicit a CD4+ T-cell response.
T41099 EGFR Protein Tyrosine Kinase Substrate

EGFR Protein Tyrosine Kinase Substrate is a EGFR protein tyrosine kinase substrate.
TP1092 Myelin Basic Protein (MBP) (68-82), guinea pig

MBP (68-82), guinea pig,豚鼠髓磷脂碱性蛋白片段68-82

Others Others
Myelin Basic Protein (MBP) (68-82), guinea pig 是一种髓鞘碱性蛋白 (MBP) 的片段。
T36865 Heat Shock Protein Inhibitor II

Heat shock protein (Hsp) inhibitor II is the active form of Hsp inhibitor I and a benzylidene lactam compound that prevents the synthesis of inducible Hsps, such as Hsp105, Hsp72, and Hsp40. Hsp inhibitor II decreases Hsp72 synthesis in vivo and reduces thermotolerance of tumors in SCC VII tumor-containing mice. At 100 μM, it inhibits the development of thermotolerance in COLO 320 DM cells. Inhibition of Hsp70 with Hsp inhibitor II in combination with amphotericin B increases susceptibility of A...
T22831 Protein kinase inhibitor H-7 dihydrochloride

H-7 dihydrochloride

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Protein kinase inhibitor H-7 dihydrochloride(H-7 dihydrochloride0) 是一种有效的蛋白激酶 C(PKC)抑制剂。Protein kinase inhibitor H-7 dihydrochloride(100 μM)显著抑制 TPA (皮肤肿瘤启动子,12-O-tetradecanoylphorbol-13-acetate) 和磷脂酶 C 促使的 ODC (鸟氨酸脱羧酶),抑制 PMA 诱导的混杂细胞溶解活性。
TP1120L IRBP acetate(211426-18-5 free base)

Interphotoreceptor Retinoid Binding Protein Fragment IRBP

Others Others
IRBP acetate(211426-18-5 free base) (Interphotoreceptor Retinoid Binding Protein Fragment IRBP) 是一种含有 20 个残基的肽,是一种主要的致病表位。它存在于间质视觉色素结合蛋白肽(IRBP 161-180)的第一个同源重复序列中,可诱导葡萄膜炎后(EAU)。
T4636 Protein kinase inhibitors 1

Others; DYRK Cell Cycle/Checkpoint; Others; Tyrosine Kinase/Adaptors
Protein kinase inhibitors 1 是新型的 HIPK2 抑制剂,其 IC50=74 nM,Kd=9.5 nM。
T6250 H-89 dihydrochloride

Protein kinase inhibitor H-89 dihydrochloride,H 89 2HCl,5-Isoquinolinesulfonamide

PKA; S6 Kinase; Autophagy Autophagy; MAPK; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
H-89 dihydrochloride (5-Isoquinolinesulfonamide) 是一种选择性 cAMP 依赖性蛋白激酶A(PKA) 抑制剂,IC50值为 48 nM。也可轻微抑制 PKG、PKC 和酪蛋白激酶活性。
TP1650 Myelin Basic Protein

Myelin Basic Protein MBP

Myelin basic protein (MBP) is a protein believed to be important in the process of myelination of nerves in the nervous system.
TP2465 PHYD protein, Arabidopsis

Phyd gene product,Phyd protein

PHYD protein, Arabidopsis belongs to the phytochrome apoprotein family in Arabidopsis.
T5140 WDR5-0103 hydrochloride[890190-22-4(free base)]

WD-Repeat Protein 5-0103,WDR5-0103盐酸盐

JAK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
WDR5-0103 hydrochloride[890190-22-4(free base)] (WD-Repeat Protein 5-0103) 是一种有效且特异性的 WD 重复蛋白 5 (WDR5) 拮抗剂 (Kd: 450 nM)。
T40400 Enhanced Green Fluorescent Protein (EGFP) (200-208)

Enhanced Green Fluorescent Protein (EGFP) (200-208) is a reporter protein obtained from Aequorea Victoria jellyfish. EGFP is widely used as a marker gene product due to its strong fluorescence properties, making it easily detectable.
TP1149 HIV-1 Rev (34-50)

HIV-1 Rev 34-50,HIV-1 rev Protein (34-50)

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) 是一种具有抗 HIV-1 活性的 17 个氨基酸多肽。 HIV-1 Rev (34-50) 源自 HIV-1 中 Rev 的 Rev 响应元件结合域。
TP1503 Protein Kinase C (19-36)

Protein Kinase C 19-36

Protein Kinase C (19-36) is a pseudosubstrate peptide inhibitor of protein kinase C (PKC), with an IC50 of 0.18 μM.
TP1507 CEF14, EBV Rta Protein (28-37)

CEF14, EBV Rta Protein 28-37

CEF14, EBV Rta Protein (28-37) is the HLA a24-restricted epitope from the epstein-barr virus Rta Protein (28-37).
TP1053 Protein Kinase C (19-31)

Protein Kinase C 19-31,PKC (19-31)

Protein Kinase C (19-31), a peptide inhibitor of protein kinase C (PKC), derived from the pseudo-substrate regulatory domain of PKCa (residues 19-31) with a serine at position 25 replacing the wild-type alanine, is used as protein kinase C substrate pepti
T39311 Tyrosinase-related Protein 2 (TRP-2) (181-188)

Tyrosinase-related Protein 2 (TRP-2) (181-188) is a peptide derived from the tyrosinase-related protein 2 (TRP-2), specifically corresponding to residues 180-188. It is the primary epitope within TRP-2 that is recognized by anti-B16 CTLs. Moreover, It is a peptide that conforms to the binding motif of the MHC class I H2-Kb.
TP1516 C-Reactive Protein (CRP) (77-82)

C-Reactive Protein (CRP) 77-82

C-Reactive Protein (CRP) 77-82 is the 77-82 fragment of C-Reactive Protein. C-Reactive Protein (CRP), the prototypic marker of inflammation, is a cardiovascular risk marker and may promote atherogenesis.C-reactive protein (CRP) is an annular (ring-shaped)
TP1592 C-Reactive Protein (CRP) (174-185)

C-Reactive Protein (CRP) 174-185

CRP, an acute phase serum protein synthesized in response to inflammatory cytokines, produces antitumor effects in animals. The fragment CRP (174-185) (RS-83277) shows similar activity by significantly enhancing the tumoricidal activity of human monocytes
TP1837 Acyl Carrier Protein (ACP) (65-74)

Acyl Carrier Protein (ACP) 65-74

Acyl Carrier Protein (ACP) (65-74) is an active acyl carrier protein (ACP) fragment.Acyl Carrier Protein (ACP) is a component of plastid-located plant fatty acid synthetase. It binds acyl groups covalently via the prosthetic group, 4-phosphopantetheine, d

化合物

Myelin Basic Protein (87-99) Acetate
Cat.No: T21618L
Synonym: Myelin Basic Protein (87-99) Acetate (118506-26-6 Free base)
Target: Others
Amyloid β-Protein 10-20 acetate
Cat.No: TP1786L
Synonym: Amyloid β-Protein 10-20 acetate(152286-31-2 free base)
Target: Beta Amyloid
Protein Kinase C 19-31 acetate
Cat.No: TP1053L
Synonym: Protein Kinase C 19-31 acetate(121545-65-1 free base),PKC (19-31) acetate
Target: PKC
JAMM protein inhibitor 2 
Cat.No: T9892
Synonym: Acetamide, 2-(2-ethylphenoxy)-N-[2-methyl-4-(1-pyrrolidinyl)phenyl]-
Target: Others
Calmodulin-Dependent Protein Kinase II 290-309 acetate
Cat.No: TP1271L
Synonym: Calmodulin-Dependent Protein Kinase II 290-309 acetate (115044-69-4 Free base)
Target: CaMK
Tau protein (592-597), Human TFA
Cat.No: TP1453
Synonym:
Target: Others
Protein kinase G inhibitor-1
Cat.No: T67755
Synonym:
Target: PKA
Protein kinase inhibitor 6
Cat.No: T9779
Synonym:
Target:
Protein kinase G inhibitor-2
Cat.No: T9940
Synonym:
Target: Others
(S,R,S)-AHPC hydrochloride
Cat.No: T4207
Synonym: VHL Ligand 1 hydrochloride,ULM-1,Protein degrader 1 hydrochloride
Target: Others, Ligand for E3 Ligase
IRAK-4 protein kinase inhibitor 2
Cat.No: T9631
Synonym:
Target: IRAK
Protein kinase inhibitors 1 hydrochlorid
Cat.No: T4692
Synonym: Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base))
Target: Others
Protein Kinase C Peptide Substrate acetate
Cat.No: TP1051L
Synonym: Protein Kinase C Peptide Substrate acetate(120253-69-2 free base)
Target: Others
Activated Protein C (390-404), human acetate
Cat.No: TP1628L
Synonym: Activated Protein C (390-404), human acetate(146340-20-7 Free base)
Target: APC
C-Reactive Protein (CRP) 201-206 acetate
Cat.No: TP1676L
Synonym: C-Reactive Protein (CRP) 201-206 acetate(130348-99-1 free base)
Target: Others
C-Reactive Protein (CRP) 77-82 acetate
Cat.No: TP1516L
Synonym: C-Reactive Protein (CRP) 77-82 acetate(130349-01-8 free base)
Target: Others
C-Reactive Protein (CRP) 174-185 acetate
Cat.No: TP1592L
Synonym: C-Reactive Protein (CRP) 174-185 acetate(160369-86-8 free base)
Target: Others
2:PN:US20040072744 SEQID:2 claimed protein acetate
Cat.No: TP1270L
Synonym: 2:PN:US20040072744 SEQID:2 claimed protein acetate(389572-87-6 free base)
Target: Others
SHP2 protein degrader-1
Cat.No: T40250
Synonym: SHP2 protein degrader-1
Target:
Protein E7(43-62)
Cat.No: T38919
Synonym: Protein E7(43-62)
Target:
G-Protein antagonist peptide acetate
Cat.No: TP1902L1
Synonym:
Target: Adrenergic Receptor
β-Amyloid (1-15)
Cat.No: TP1229
Synonym: Amyloid β-Protein (1-15)
Target: Beta Amyloid
WDR5-0103
Cat.No: T3201
Synonym: WD-Repeat Protein 5-0103
Target: Histone Methyltransferase, JAK
C-Reactive Protein (CRP) (201-206)
Cat.No: TP1676
Synonym: C-Reactive Protein (CRP) 201-206
Target: Others
(Cys47)-HIV-1 tat Protein (47-57)
Cat.No: T40719
Synonym: (Cys47)-HIV-1 tat Protein (47-57)
Target:
KNK437
Cat.No: T2444
Synonym: Heat Shock Protein Inhibitor I
Target: HSP
Peripheral Myelin P0 Protein (180-199), mouse
Cat.No: T38964
Synonym: Peripheral Myelin P0 Protein (180-199), mouse
Target:
Peripheral Myelin Protein P2 (53-78), bovine
Cat.No: T40925
Synonym: Peripheral Myelin Protein P2 (53-78), bovine
Target:
KRAS mutant protein inhibitor 1
Cat.No: T40272
Synonym:
Target:
Protein kinase inhibitors 1 hydrochloride
Cat.No: T39860
Synonym:
Target:
Influenza Matrix Protein (61-72)
Cat.No: T38687
Synonym:
Target:
EGFR Protein Tyrosine Kinase Substrate
Cat.No: T41099
Synonym:
Target:
Myelin Basic Protein (MBP) (68-82), guinea pig
Cat.No: TP1092
Synonym: MBP (68-82), guinea pig,豚鼠髓磷脂碱性蛋白片段68-82
Target: Others
Heat Shock Protein Inhibitor II
Cat.No: T36865
Synonym:
Target:
Protein kinase inhibitor H-7 dihydrochloride
Cat.No: T22831
Synonym: H-7 dihydrochloride
Target: PKC
IRBP acetate(211426-18-5 free base)
Cat.No: TP1120L
Synonym: Interphotoreceptor Retinoid Binding Protein Fragment IRBP
Target: Others
Protein kinase inhibitors 1
Cat.No: T4636
Synonym:
Target: Others, DYRK
H-89 dihydrochloride
Cat.No: T6250
Synonym: Protein kinase inhibitor H-89 dihydrochloride,H 89 2HCl,5-Isoquinolinesulfonamide
Target: PKA, S6 Kinase, Autophagy
Myelin Basic Protein
Cat.No: TP1650
Synonym: Myelin Basic Protein MBP
Target:
PHYD protein, Arabidopsis
Cat.No: TP2465
Synonym: Phyd gene product,Phyd protein
Target:
WDR5-0103 hydrochloride[890190-22-4(free base)]
Cat.No: T5140
Synonym: WD-Repeat Protein 5-0103,WDR5-0103盐酸盐
Target: JAK
Enhanced Green Fluorescent Protein (EGFP) (200-208)
Cat.No: T40400
Synonym:
Target:
HIV-1 Rev (34-50)
Cat.No: TP1149
Synonym: HIV-1 Rev 34-50,HIV-1 rev Protein (34-50)
Target: HIV Protease
Protein Kinase C (19-36)
Cat.No: TP1503
Synonym: Protein Kinase C 19-36
Target:
CEF14, EBV Rta Protein (28-37)
Cat.No: TP1507
Synonym: CEF14, EBV Rta Protein 28-37
Target:
Protein Kinase C (19-31)
Cat.No: TP1053
Synonym: Protein Kinase C 19-31,PKC (19-31)
Target:
Tyrosinase-related Protein 2 (TRP-2) (181-188)
Cat.No: T39311
Synonym:
Target:
C-Reactive Protein (CRP) (77-82)
Cat.No: TP1516
Synonym: C-Reactive Protein (CRP) 77-82
Target:
C-Reactive Protein (CRP) (174-185)
Cat.No: TP1592
Synonym: C-Reactive Protein (CRP) 174-185
Target:
Acyl Carrier Protein (ACP) (65-74)
Cat.No: TP1837
Synonym: Acyl Carrier Protein (ACP) 65-74
Target:
Cat. No. Product Name Target Signaling Pathways
T23927 Cylindrin

Hollow cylinder protein complex

Cylindrin is a six-stranded antiparallel beta-barrel that induces cell toxicity through an unknown mechanism.
TN1433 Batatasin III

FAK; Others; Akt Angiogenesis; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Batatasin III 通过抑制上皮间质转化和 FAK-AKT 信号来抑制癌症迁移和侵袭,并具有抗癌活性。 Batatasin III 对整株生长有长期抑制作用,显示出抑制萌发活性。
T2851 Daphnetin

7,8-Dihydroxycoumarin,Daphnetol,瑞香素

EGFR; PKA; PKC; Parasite; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物,有抗氧化、抗炎、抗疟疾和解热作用,可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。
TN1557 Decursinol angelate

ERK; VEGFR; PKC; JNK Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Tyrosine Kinase/Adaptors
Decursinol angelate 是从朝鲜当归根部分离得到的一种天然产物,是 PKC 激酶的激活剂,有细胞毒性,抗肿瘤和抗炎活性。
TN1828 Kahweol

Apoptosis; NF-κB; AMPK Apoptosis; Chromatin/Epigenetic; NF-κB; PI3K/Akt/mTOR signaling
Kahweol 是小果咖啡的成分之一,可诱导细胞凋亡,具有抗炎、抗血管生成和抗癌活性。它通过激酶的活化抑制的脂肪生成和增加葡萄糖摄取。
T2S2215 Crebanine

Apoptosis; Others; Akt Apoptosis; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling
Crebanine 是来自于韦诺萨千金藤的一种生物碱,通过抑制 MAPKs 和 Akt 信号通路表现出抗炎活性,还具有抗心律失常的作用。它可诱导人类癌细胞的 G1阻滞和凋亡。
T3889 Platycodin D

Prostaglandin Receptor; AMPK Chromatin/Epigenetic; GPCR/G Protein; Immunology/Inflammation; PI3K/Akt/mTOR signaling
Platycodin D 是从桔梗中分离得到的一种皂苷类天然产物,是AMPKα的激活剂,具有抗肥胖活性。它可刺激 TNF-α 合成或抑制 TNF-α mRNA 的降解。
T7846 Aegeline

Others; Antifungal Microbiology/Virology; Others
Aegeline 是从 Aegle marmelos 的叶子中分离出来的一种生物碱酰胺,有抗高血糖和抗血脂异常的活性。
TN1100 Nepodin

transporter; COX; AMPK; Parasite Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling
Nepodin 是从Rumex crispus 中分离的一种醌氧化还原酶抑制剂,具有抗糖尿病和抗疟疾的作用。。它通过激活 AMPK 刺激 GLUT4 向质膜的转运。
T7190 Actein

Apoptosis; Akt; JNK; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
Actein 是从升麻的根茎中分离的一种三萜糖苷,通过促进ROS/JNK 活化和钝化人膀胱癌中的AKT 途径来抑制细胞增殖,诱导自噬和凋亡。
T5771 Hypocrellin A

Antibacterial; PKC; Parasite Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
Hypocrellin A 是一种天然的PKC 抑制剂,具有光诱导的抗肿瘤、抗真菌和抗病毒活性,还对 MHC 限制性抗原呈递发挥免疫调节作用。
TN1305 Ethoxysanguinarine

乙氧基血根碱,6-Ethoxydihydrosanguinarine

Apoptosis; AChR Apoptosis; Neuroscience
Ethoxysanguinarine (6-Ethoxydihydrosanguinarine) 是存在于龙葵中的一种苯并菲啶生物碱天然产物,通过抑制蛋白磷酸酶 2A,可抑制结直肠癌细胞活力,诱导细胞凋亡。
T5077 Deoxycholic acid sodium salt

脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid sodium salt (Sodium deoxycholate) 是 G 蛋白偶联胆汁酸受体TGR5的激活剂。
T7327 7-Methoxyisoflavone

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
7-Methoxyisoflavone 是单磷酸腺苷活化蛋白激酶 (AMPK) 的激活剂,是异黄酮衍生物。
T2965 Deoxycholic acid

Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。
T4S0800 Demethyleneberberine

P450; NOS; NF-κB; HIF; AMPK Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Demethyleneberberine 是从黄连中提取的一种天然产物,是线粒体靶向抗氧化剂。它也可作为AMPK 激活剂,用于非酒精性脂肪性肝病的研究。它通过抑制NF-κB 通路和调节 Th 细胞的平衡来减轻小鼠结肠炎并抑制炎症反应。
TN2268 Tetrahydromagnolol

Cannabinoid Receptor; GPR; GABA Receptor Endocrinology/Hormones; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Tetrahydromagnolol 是 Magnolol 的主要代谢产物,是一种弱的GPR55受体拮抗剂。它是选择性大麻素CB2受体激动剂,EC50为 170 nM,Ki 为 416 nM,对CB2受体的选择性比 CB1 受体高 20 倍。
T6677 Sophocarpine

ERK; p38 MAPK; NF-κB; TLR; COX; HER; JNK; STAT Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; MAPK; Neuroscience; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Sophocarpine 是一种从传统草药苦参中提取的重要生物碱。苦参具有抗病毒、抗肿瘤和抗炎等多种药理作用。它通过多种机制显著抑制癌细胞的生长,具有抗肿瘤活性。
T3904 Gomisin J

Calcium Channel; AMPK Chromatin/Epigenetic; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling
Gomisin J 是在五味子中发现的小分子量木脂素,具有血管舒张活性,在非酒精性脂肪性肝病方面有研究潜力。 它通过激活 AMPK、LKB1 和 Ca2+/钙调蛋白依赖性蛋白激酶 II 以及抑制 HepG2 细胞中的胎球蛋白 A 来调节脂肪生成酶和脂肪分解酶以及炎症分子的表达,从而抑制脂质积累。
T3881 Vaccarin

Integrin; Akt; PERK; AMPK Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Vaccarin 是从王不留行中提取的一种黄酮糖苷,可显著促进伤口愈合以及伤口部位的内皮和成纤维细胞增殖。它通过激活 AMPK 信号通路改善胰岛素抵抗和脂肪变性。
T5497 AMAROGENTIN

苦杏苷,苦龙胆酯苷

Apoptosis; AMPK Apoptosis; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Amarogentin 是要从 Swertia 和 Gentiana 根中提取的裂环烯醚萜苷,有抗氧化、抗肿瘤和抗糖尿病活性,具有保肝和免疫调节作用。它通过激活 AMPK 发挥有益的血管代谢作用。它促进细胞凋亡,阻止 G2/M 细胞周期和下调 PI3K/Akt/mTOR 信号通路。
T5S0896 Loureirin A

龙血素 A,龙血素A

Akt; PI3K Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Loureirin A 是一种黄酮类物质,从龙血树中分离得到,能够降低Akt 的磷酸化,具有抗血小板聚集作用。
T13265 Urolithin B

尿石素B,3-羟基-6H-苯并[C]苯并吡喃-6-酮

ERK; NF-κB; Akt; Endogenous Metabolite; JNK; AMPK Chromatin/Epigenetic; Cytoskeletal Signaling; MAPK; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Urolithin B 是一种 ellagitannins 的肠道微生物代谢产物,具有抗炎和抗氧化作用。它也是骨骼肌质量的调节因子,通过减少 IκBα 的磷酸化和降解来抑制 NF-κB 活性,并抑制 JNK、ERK 和 Akt 的磷酸化,并增强 AMPK 的磷酸化。
T5S2017 Ingenol

(-)-Ingenol,巨大戟二萜醇,巨大戟醇

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Ingenol ((-)-Ingenol) 是一种PKC 激活剂,Ki 值为 30 μM,具有抗肿瘤活性。 从 Ingenol 酯中配制新的衍生物可能是开发新的先导化合物以重新激活潜伏 HIV 的创新方法。Ingenol mebutate 是治疗光化性角化病的有效方法。
TN1877 Lonicerin

忍冬苦苷,金银花

Apoptosis; Antibacterial Apoptosis; Microbiology/Virology
Lonicerin 是一种抗藻酸盐分泌蛋白的黄酮类化合物,对铜绿假单胞菌有抑制作用。它可预防脂多糖诱导的急性肺损伤的炎症和细胞凋亡。
T3844 Deltonin

三角叶薯蓣皂苷

ERK; Others; Akt; Endogenous Metabolite Cytoskeletal Signaling; MAPK; Metabolism; Others; PI3K/Akt/mTOR signaling
Deltonin 是从盾叶薯蓣中得到的一种甾体皂苷,抑制ERK1/2和AKT 的活化,具有抗肿瘤活性。
T4S1335 Daphnoretin

Dephnoretin,西瑞香素,Thymelol

Influenza Virus; Caspase; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
Daphnoretin (Thymelol) 是从了哥王中提取得到的一种天然产物,具有抗癌和抗病毒活性。它通过在 G2/M 期连续阻断细胞并激活 caspase-3 通路导致 HOS 细胞死亡。
T4S2128 Bilobetin

白果双黄酮,白果素

PKA; PPAR DNA Damage/DNA Repair; Metabolism; Tyrosine Kinase/Adaptors
Bilobetin 是银杏的活性成分,可改善胰岛素抵抗,增加肝脏对脂质的吸收和氧化,降低极低密度脂蛋白甘油三酯分泌和血液甘油三酯水平,增强组织中 β-氧化的酶的表达和活性,并减弱甘油三酯及其代谢产物的积累。它还增加了 PPARα的磷酸化,核转位和活性,并伴随着 cAMP 水平和 PKA 活性的升高。
T0700 Ursodeoxycholic acid

熊去氧胆酸,UDCA,Ursodiol

Potassium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
Ursodeoxycholic acid (UDCA)是一种有效的肝脏特异性脂肪酸转运蛋白 5 (FATP5) 抑制剂,通过 FATP5 依赖性方式抑制原代肝细胞摄取长链脂肪酸。Ursodeoxycholic acid 能够抑制胆固醇的吸收,用于溶解胆结石,并具有研究与肥胖相关的脂肪肝疾病的潜力。
TN1637 Eurycomalactone

Anti-infection; NF-κB Microbiology/Virology; NF-κB
Eurycomalactone 是一种NF-κB 抑制剂,IC50=0.5 μM,是一种天然产物。它可抑制蛋白合成,降低 cyclin D1 蛋白水平,但对 TNFα 诱导的 IκBα 降解或 IKKα/β 和 IκBα 的磷酸化水平没有作用。
T13803 N-Oleoyl glycine

Cannabinoid Receptor; Akt; Endogenous Metabolite; PPAR Cytoskeletal Signaling; DNA Damage/DNA Repair; GPCR/G Protein; Metabolism; PI3K/Akt/mTOR signaling
N-Oleoyl glycine 是一种脂氨酸。在 3T3-L1 脂肪细胞中,N-Oleoyl glycine 通过激活CB1受体和Akt 信号通路来刺激脂肪形成。
T17280 (Z)-Guggulsterone

Apoptosis; VEGFR; Akt Angiogenesis; Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
(Z)-Guggulsterone 是印度阿育吠陀药用植物Commiphora mukul 的成分,可通过引起细胞凋亡来抑制人前列腺癌细胞的生长,还可通过抑制VEGF-VEGF-R2-Akt 信号传导轴来抑制血管生成。
TQ0183 Narciclasine

水仙环素,Lycoricidinol

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
Narciclasine (Lycoricidinol) 是一种植物生长调节剂。它通过调节Rho/Rho 激酶/LIM 激酶/cofilin 信号传导途径,大大增加GTP 酶RhoA 活性以及以RhoA 依赖性方式诱导肌动蛋白应力纤维形成。
T2968 Hyodeoxycholic acid

NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA

FXR; Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Hyodeoxycholic acid (NSC 60672) 是由肠道菌群在小肠中形成的次级胆汁酸,是TGR5(GPCR19)的激动剂, CHO 细胞中的EC50=31.6 µM。它已用于研究高胆固醇血症的治疗。
T5654 Musk ketone

Others Others
Musk ketone 可诱导癌细胞生长抑制和凋亡。它增加谷胱甘肽 S-转移酶的活性,因此可能被证明是有用的癌症化学保护剂。
T5S0246 Pseudoprotodioscin

山药

Others; Fatty Acid Synthase Metabolism; Others
Pseudoprotodioscin 是一种呋喃葡糖苷,抑制SREBP1/2和microRNA 33a/b 水平,降低胆固醇和甘油三酯合成相关的基因表达。
TN1651 Furanodiene

Apoptosis; PARP; Reactive Oxygen Species; Caspase; CDK; P-gp Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Proteases/Proteasome
Furanodiene 是从姜黄中提取的一种萜类天然产物,可抑制外排转运蛋白Pgp 功能并降低 Pgp 蛋白水平。它通过抗血管生成和诱导ROS 产生,DNA 链断裂和细胞凋亡发挥抗癌作用。
T6S0781 Phellodendrine

黄柏碱,Phallodendrin

Others; NF-κB; Akt Cytoskeletal Signaling; NF-κB; Others; PI3K/Akt/mTOR signaling
Phellodendrine (Phallodendrin) 是异喹啉生物碱,是黄柏皮层中的重要特征成分之一。它具有良好的抗氧化,抗炎作用。它通过调节AKT/NF-κB 途径抵抗 AAPH 诱导的氧化应激。
TQ0302 Thapsigargin

毒胡萝卜素

Apoptosis; SARS-CoV; Calcium Channel Apoptosis; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Thapsigargin 属于天然产物,是一种肌/内质网 Ca2+ ATP 酶 (SERCA) 的抑制剂,也是一种内质网应激诱导剂。Thapsigargin 通过阻断细胞将钙泵入肌浆和内质网的能力来提高胞浆钙浓度。
T2S0820 Karanjin

干华豆晶 4,水黄皮素

Apoptosis; AMPK Apoptosis; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Karanjin 是干花豆中的主要活性呋喃黄酮醇成分,可通过细胞周期阻滞诱导癌细胞死亡,促进细胞凋亡,还通过提高AMPK 的方式诱导骨骼肌细胞 GLUT4 易位。
T3861 Isobavachalcone

Corylifolinin,Isobacachalcone,补骨脂乙素

Apoptosis; Others; Reactive Oxygen Species; Akt; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; Others; PI3K/Akt/mTOR signaling
Isobavachalcone (Corylifolinin) 是来源于补骨脂的一种Akt 信号通路抑制剂,可诱导人类癌细胞凋亡,以IC50值为 7.92 μM 抑制 OVCAR-8 癌细胞生长,具有抗癌和抗增殖活性。它还能诱导 OVCAR-8 细胞中活性氧的产生。
T6817 Deguelin

鱼藤素,(-)-Deguelin,(-)-cis-Deguelin,魚藤素

Apoptosis; Akt; PI3K; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Deguelin ((-)-Deguelin) 是一种 PI3K/AKT 抑制剂,从 Mundulea sericea 家族植物中分离出来的鱼藤酮类天然产物。
T6S0052 Chelerythrine

Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine (Broussonpapyrine) 是一种天然生物碱,为有效、选择性的 Ca2+/磷脂依赖性PKC 拮抗剂,IC50值为 0.7 μM。它具有抗肿瘤、抗糖尿病、抗炎的活性。它抑制BclXL-Bak BH3肽结合,IC50为 1.5 μM,并从 BclXL 取代了 Bax。它诱导细胞凋亡和自噬。
T3405 [6]-Gingerol

6-Gingerol,gingerol,(S)-(+)-[6]Gingerol,6-姜酚

Apoptosis; AMPK Apoptosis; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
[6]-Gingerol ((S)-(+)-[6]Gingerol) 是一种从生姜中分离的活性物质,具有抗癌,抗炎和抗氧化活性。
T3S0012 coniferyl ferulate

P-gp; GST Membrane transporter/Ion channel; Neuroscience; oxidation-reduction
Coniferyl ferulate 是从川芎中提取的一种天然产物,是强效的谷胱甘肽 S-转移酶抑制剂,强抑制人胎盘型谷胱甘肽 S-转移酶,IC50为 0.3 μM。它还可逆转多药耐药性并下调 P-糖蛋白。
T3419 Chelerythrine chloride

白屈菜红碱,盐酸白屈菜红碱

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine chloride 是一种可渗透细胞的蛋白激酶 C 抑制剂,对磷酸盐受体具有竞争性,而对 ATP 是非竞争性的。它诱导细胞凋亡和自噬。
T5S0506 Rotundic acid

Rutundic acid,铁冬青酸

Apoptosis; Others; p38 MAPK; Akt; mTOR Apoptosis; Cytoskeletal Signaling; MAPK; Others; PI3K/Akt/mTOR signaling
Rotundic acid (Rutundic acid) 是一种从圆形肠球菌中获得的三萜类天然产物,具有抗炎和保护心脏的能力。它可通过 AKT/mTOR 和 MAPK 途径在肝细胞癌中诱导 DNA 损伤和细胞凋亡。
T1032 Erythromycin

红霉素,E-Mycin

ribosome; Antibacterial; Antibiotic Microbiology/Virology
Erythromycin (E-Mycin) 是由放线菌产生的大环内酯类抗生素。它结合细菌的 50S 核糖体亚基,通过阻断转肽和易位反应来抑制 RNA 依赖性蛋白的合成。
T0950 Neomycin sulfate

Framycin sulfate,硫酸新霉素

Phospholipase; ribosome; Antibacterial; Antibiotic Metabolism; Microbiology/Virology
Neomycin sulfate (Framycin sulfate) 是一种广谱的氨基糖苷类抗生素。Neomycin sulfate 可以阻断细菌蛋白质的合成以发挥抗菌活性。Neomycin sulfate 常用于筛选具有 Neo 抗性基因的原核和真核细胞。
T6680 Staurosporine

Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素

Apoptosis; PKA; Antibacterial; Antibiotic; Src; PKC; Antifungal Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Staurosporine (AM-2282) 是一种蛋白激酶抑制剂,对 PKC、PKA、c-Fgr、Phosphorylase kinase 和 TAOK2 均有抑制活性 (IC50=6/15/2/3/3000 nM),具有 ATP 竞争性和非选择性。Staurosporine 也可以诱导凋亡。
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天然产物

Cylindrin
Cat.No: T23927
Synonym: Hollow cylinder protein complex
Target:
Batatasin III
Cat.No: TN1433
Synonym:
Target: FAK, Others, Akt
Daphnetin
Cat.No: T2851
Synonym: 7,8-Dihydroxycoumarin,Daphnetol,瑞香素
Target: EGFR, PKA, PKC, Parasite, Autophagy
Decursinol angelate
Cat.No: TN1557
Synonym:
Target: ERK, VEGFR, PKC, JNK
Kahweol
Cat.No: TN1828
Synonym:
Target: Apoptosis, NF-κB, AMPK
Crebanine
Cat.No: T2S2215
Synonym:
Target: Apoptosis, Others, Akt
Platycodin D
Cat.No: T3889
Synonym:
Target: Prostaglandin Receptor, AMPK
Aegeline
Cat.No: T7846
Synonym:
Target: Others, Antifungal
Nepodin
Cat.No: TN1100
Synonym:
Target: transporter, COX, AMPK, Parasite
Actein
Cat.No: T7190
Synonym:
Target: Apoptosis, Akt, JNK, Autophagy
Hypocrellin A
Cat.No: T5771
Synonym:
Target: Antibacterial, PKC, Parasite
Ethoxysanguinarine
Cat.No: TN1305
Synonym: 乙氧基血根碱,6-Ethoxydihydrosanguinarine
Target: Apoptosis, AChR
Deoxycholic acid sodium salt
Cat.No: T5077
Synonym: 脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate
Target: Endogenous Metabolite, GPCR19
7-Methoxyisoflavone
Cat.No: T7327
Synonym:
Target: AMPK
Deoxycholic acid
Cat.No: T2965
Synonym: Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
Demethyleneberberine
Cat.No: T4S0800
Synonym:
Target: P450, NOS, NF-κB, HIF, AMPK
Tetrahydromagnolol
Cat.No: TN2268
Synonym:
Target: Cannabinoid Receptor, GPR, GABA Receptor
Sophocarpine
Cat.No: T6677
Synonym:
Target: ERK, p38 MAPK, NF-κB, TLR, COX, HER, JNK, STAT
Gomisin J
Cat.No: T3904
Synonym:
Target: Calcium Channel, AMPK
Vaccarin
Cat.No: T3881
Synonym:
Target: Integrin, Akt, PERK, AMPK
AMAROGENTIN
Cat.No: T5497
Synonym: 苦杏苷,苦龙胆酯苷
Target: Apoptosis, AMPK
Loureirin A
Cat.No: T5S0896
Synonym: 龙血素 A,龙血素A
Target: Akt, PI3K
Urolithin B
Cat.No: T13265
Synonym: 尿石素B,3-羟基-6H-苯并[C]苯并吡喃-6-酮
Target: ERK, NF-κB, Akt, Endogenous Metabolite, JNK, AMPK
Ingenol
Cat.No: T5S2017
Synonym: (-)-Ingenol,巨大戟二萜醇,巨大戟醇
Target: PKC
Lonicerin
Cat.No: TN1877
Synonym: 忍冬苦苷,金银花
Target: Apoptosis, Antibacterial
Deltonin
Cat.No: T3844
Synonym: 三角叶薯蓣皂苷
Target: ERK, Others, Akt, Endogenous Metabolite
Daphnoretin
Cat.No: T4S1335
Synonym: Dephnoretin,西瑞香素,Thymelol
Target: Influenza Virus, Caspase, PKC
Bilobetin
Cat.No: T4S2128
Synonym: 白果双黄酮,白果素
Target: PKA, PPAR
Ursodeoxycholic acid
Cat.No: T0700
Synonym: 熊去氧胆酸,UDCA,Ursodiol
Target: Potassium Channel, Endogenous Metabolite
Eurycomalactone
Cat.No: TN1637
Synonym:
Target: Anti-infection, NF-κB
N-Oleoyl glycine
Cat.No: T13803
Synonym:
Target: Cannabinoid Receptor, Akt, Endogenous Metabolite, PPAR
(Z)-Guggulsterone
Cat.No: T17280
Synonym:
Target: Apoptosis, VEGFR, Akt
Narciclasine
Cat.No: TQ0183
Synonym: 水仙环素,Lycoricidinol
Target: ROCK
Hyodeoxycholic acid
Cat.No: T2968
Synonym: NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA
Target: FXR, Endogenous Metabolite, GPCR19
Musk ketone
Cat.No: T5654
Synonym:
Target: Others
Pseudoprotodioscin
Cat.No: T5S0246
Synonym: 山药
Target: Others, Fatty Acid Synthase
Furanodiene
Cat.No: TN1651
Synonym:
Target: Apoptosis, PARP, Reactive Oxygen Species, Caspase, CDK, P-gp
Phellodendrine
Cat.No: T6S0781
Synonym: 黄柏碱,Phallodendrin
Target: Others, NF-κB, Akt
Thapsigargin
Cat.No: TQ0302
Synonym: 毒胡萝卜素
Target: Apoptosis, SARS-CoV, Calcium Channel
Karanjin
Cat.No: T2S0820
Synonym: 干华豆晶 4,水黄皮素
Target: Apoptosis, AMPK
Isobavachalcone
Cat.No: T3861
Synonym: Corylifolinin,Isobacachalcone,补骨脂乙素
Target: Apoptosis, Others, Reactive Oxygen Species, Akt, Autophagy
Deguelin
Cat.No: T6817
Synonym: 鱼藤素,(-)-Deguelin,(-)-cis-Deguelin,魚藤素
Target: Apoptosis, Akt, PI3K, Autophagy
Chelerythrine
Cat.No: T6S0052
Synonym: Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine
Target: Apoptosis, BCL, PKC, Autophagy
[6]-Gingerol
Cat.No: T3405
Synonym: 6-Gingerol,gingerol,(S)-(+)-[6]Gingerol,6-姜酚
Target: Apoptosis, AMPK
coniferyl ferulate
Cat.No: T3S0012
Synonym:
Target: P-gp, GST
Chelerythrine chloride
Cat.No: T3419
Synonym: 白屈菜红碱,盐酸白屈菜红碱
Target: Apoptosis, BCL, PKC, Autophagy
Rotundic acid
Cat.No: T5S0506
Synonym: Rutundic acid,铁冬青酸
Target: Apoptosis, Others, p38 MAPK, Akt, mTOR
Erythromycin
Cat.No: T1032
Synonym: 红霉素,E-Mycin
Target: ribosome, Antibacterial, Antibiotic
Neomycin sulfate
Cat.No: T0950
Synonym: Framycin sulfate,硫酸新霉素
Target: Phospholipase, ribosome, Antibacterial, Antibiotic
Staurosporine
Cat.No: T6680
Synonym: Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素
Target: Apoptosis, PKA, Antibacterial, Antibiotic, Src, PKC, Antifungal
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