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138

抑制剂 & 化合物

75

天然产物

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Cat. No. Product Name Target Signaling Pathways
T81091 Steroid sulfatase-IN-5

Steroid sulfatase-IN-5 (compound 10b) 是一种高效的STS抑制剂,具有0.32 nM的IC50值。该化合物还能显著抑制T-47D细胞增殖,其IC50为35.7 μM,常用于乳腺癌相关的研究领域。
T62237 Steroid sulfatase-IN-4

Steroid sulfatase-IN-4 (Compound 16) 是一种类固醇硫酸酯酶 (STS) 的不可逆抑制剂,能够作用于人 STS (IC50: 25 nM)。Steroid sulfatase-IN-4 能够用于研究子宫内膜异位。
T61212 Steroid sulfatase-IN-2

Steroid sulfatase-IN-2 is an active inhibitor of steroid sulfatase (STS), demonstrating an IC50 value of 109.5 nM. Its potential application lies in hormone-dependent cancer research, specifically estrogen-dependent breast and endometrial cancer [1].
T81090 Steroid sulfatase-IN-6

Steroid sulfatase-IN-6 (Compound 10c) 是一种针对类固醇硫酸酯酶 (STS) 的不可逆抑制剂,对人胎盘 STS 的 Ki 值达到 0.4 nM。该化合物适用于肿瘤疾病研究。
T83752 Biotin-SRC-1 (676–700) TFA

Biotin-Steroid Receptor Coactivator 1 (676-700)

Biotin-SRC-1 (676–700)是一种生物素化且缩短的类固醇受体辅助激活蛋白1 (SRC-1)。它已在基于亲和力的报告试验中使用,包括时间分辨荧光共振能量转移 (TR-FRET) 和增强型近距离发光均匀检测法 (ΑLPHASCREEN™)。
T81089 Steroid sulfatase-IN-7

Steroid sulfatase-IN-7是一种具有高度选择性的不可逆STS抑制剂,表现出0.05 nM的强效对人胎盘STS抑制能力,常被用于癌症方面的科学研究。
T61687 Steroid sulfatase-IN-1

Steroid sulfatase-IN-1 is a highly potent and orally active inhibitor of the enzyme Steroid sulfatase, with an impressive IC50 value of 1.71 μM. This compound exhibits notable antitumor activity, achieving a TGI (tumor growth inhibition) of 51% in vivo. Therefore, Steroid sulfatase-IN-1 holds great promise in the field of breast cancer research [1].
T61686 Steroid sulfatase-IN-3

Steroid sulfatase-IN-3 (compound 1q) is a highly effective Steroid sulfatase (STS) inhibitor, exhibiting an IC 50 value of 25.8 nM. This compound also demonstrates antiproliferative properties against T-47D estrogen-dependent breast cancer cells, with an IC 50 of 1.04 μM [1].
T61716 Steroid sulfatase/17β-HSD1-IN-1

Steroid sulfatase/17β-HSD1-IN-1 is a highly effective inhibitor of both steroid sulfatase and 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) activities, displaying an IC50 value of 28 nM against cellular human steroid sulfatase. This compound holds significant potential for investigating estrogen-dependent diseases [1].
T81092 Steroid sulfatase/17β-HSD1-IN-5

Steroid sulfatase/17β-HSD1-IN-5 是一种不可逆抑制剂,针对类固醇硫酸酯酶(STS),同时也是17β-羟甾类固醇脱氢酶1型(17β-HSD1)的可逆且选择性抑制剂,表现出对17β-HSD1的IC50为43 nM,对17β-HDS1为6.2 μM。该化合物主要用于研究代谢性疾病,特别是子宫内膜异位症。
T61979 Steroid sulfatase/17β-HSD1-IN-4

Steroid sulfatase/17β-HSD1-IN-4 (compound 37) 是一种类固醇硫酸酯酶 (STS) 和 17β-羟基类固醇脱氢酶 1 型 (17β HSD1) 双重抑制剂。Steroid sulfatase/17β-HSD1-IN-4 对 hSTS 的活性抑制作用不可逆,IC50为 63 nM。Steroid sulfatase/17β-HSD1-IN-4 在子宫内膜异位症及其他雌激素依赖性疾病方面有研究价值。
T62236 Steroid sulfatase/17β-HSD1-IN-3

Steroid sulfatase/17β-HSD1-IN-3 (compound 19) 是一种双重的类固醇硫酸酯酶 (STS) 和 17β-羟基类固醇脱氢酶 1 型 (17β HSD1) 抑制剂。Steroid sulfatase/17β-HSD1-IN-3 对 hSTS 的活性具有不可逆的抑制作用 (IC50: 27 nM)。Steroid sulfatase/17β-HSD1-IN-3 能够用于研究子宫内膜异位症及其他雌激素依赖性疾病。
T0181 Loteprednol etabonate

Lotemax,Alrex,氯替泼诺

Glucocorticoid Receptor; Antibacterial; Antibiotic Endocrinology/Hormones; Microbiology/Virology
Loteprednol etabonate (Lotemax) 是具有抗炎活性的皮质类固醇,用于眼科。
T0166 Pancuronium dibromide

Pancuronium bromide,Pavulon,泮库溴铵

AChR Neuroscience
Pancuronium dibromide (Pavulon) 是一种双季基类固醇,是一种神经肌肉松弛剂。它通过与乙酰胆碱竞争 nACh 受体上的结合位点来抑制神经肌肉传递。它还可抑制心脏毒蕈碱受体并具有拟交感神经作用。
T0094 Budesonide

Entocort,Pulmicort,布地奈德,Rhinocort

Glucocorticoid Receptor Endocrinology/Hormones
Budesonide (Pulmicort) 是吸入型糖皮质类固醇,是一种口服具有活性的糖皮质激素受体激动剂。它能够减小肺部肿瘤的体积,逆转 DNA 低度甲基化,调节基因的 mRNA 表达。它是能够用于哮喘的抗炎药。
T1531 Mometasone furoate

糠酸莫美他松,糠酸莫米松,Sch32088

Glucocorticoid Receptor Endocrinology/Hormones
Mometasone furoate (Sch32088) 是糖皮质激素受体激动剂,具有抗炎和抗过敏作用。它是皮质固醇类试剂,动物模型中,可局部应用于气道炎症、慢性皮肤湿疹、哮喘。
T1167 Cyproterone acetate

Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮

Androgen Receptor Endocrinology/Hormones
Cyproterone acetate (Cyproterone 17-O-acetate) 是能够抗雄激素(IC50=7.1 nM) 和孕激素合成的类固醇。它与 progesteron 和糖皮质激素受体有亲和力。
T61444 Nonsteroidal aromatase inhibitor 1

Nonsteroidal aromatase inhibitor 1 (Compound 13h) effectively inhibits the enzyme CYP19A1 with an IC50 value of 0.09 nM. Due to its potent inhibitory activity, Nonsteroidal aromatase inhibitor 1 holds promise for research in the field of breast cancer [1].
T76147 3α-Hydroxysteroid dehydrogenase

3α-Hydroxysteroid dehydrogenase(3α-HSD) 是一种由 AKR1C4 基因编码的酶,可以催化 3-酮类甾体转化为 3α-羟基化合物。3α-Hydroxysteroid dehydrogenase 在雄激素 DHT 的失活中起重要作用,可以将 DHT 转化成雄激素活性很弱的 3α-雄烷二醇,可用于多毛症研究。
T4464 Irosustat

667-Coumate,BN83495,STX64

Others Others
Irosustat (667-Coumate) 是类固醇硫酸酯酶抑制剂(IC50:8 nM),具有抗乳腺癌作用。
T33414 MK 0434

MK0434,MK434,MK 434,MK-0434,MK-434

MK 0434 is a steroid 5α-reductase inhibitor and hormone antagonist associated with a significant reduction in DHT.
T0293 Metyrapone

美替拉酮,甲吡酮,NSC-25265,Su-4885

Others; P450; Dehydrogenase; Autophagy Autophagy; Metabolism; Others
Metyrapone (NSC-25265) 是 STEROID 11-BETA-MONOOXYGENASE 酶抑制剂。 它被用作库欣综合征诊断中下丘脑-垂体反馈机制的测试。
T19213 Boldenone Cypionate

Others; Androgen Receptor Endocrinology/Hormones; Others
Boldenone Cypionate 是一种雄激素合成代谢类固醇,常被休闲健美运动员和普通健身房成员使用。
T0870 Altrenogest

R2267,RU2267,Allyltrenbolone,A35957,烯丙孕素

Estrogen/progestogen Receptor; Progesterone Receptor Endocrinology/Hormones; Others
Altrenogest (Allyltrenbolone) 是一种结构与trenbolone 相关的孕激素,能作用于孕激素受体。
T3137 Boldenone Undecylenate

Parenabol,Ba 29038,Vebonol,十一碳烯酸去甲睾酮

Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Boldenone Undecylenate (Parenabol) 十一碳烯酸盐一种是人工合成的甾体,作用与天然的睾酮相似。
T83615 S5A1

Others Others
S5A1 是一种合成的类固醇,可用于研究糖尿病。
T60929 Brassinazole

(2S,3R)-Brassinazole

Others Others
Brassinazole 是一种选择性的三唑型类固醇 (BR)生物合成抑制剂。Brassinazole 可用于调节油芸素类固醇 (BR) 信号转导通路,用于调节植物木质部的生长和发育。
T21452 Anecortave Acetate

Retaane,Al 3789,NSC 24345,NSC 15475,Anecortave

Others Others
Anecortave Acetate (NSC-24345) 是一种血管抑制类固醇,用于蛋白质组学研究。
T27478 GSK3987

Liver X Receptor Metabolism
GSK3987 是广谱LXRα/β激动剂,EC50分别为 50 nM 和 40 nM。GSK3987增加 ABCA1 和 SREBP-1c 蛋白的表达,诱导细胞甘油三酯的积累和胆固醇流出。
T11235 Estradiol 3-sulfamate

雌二醇 3-氨基磺酸,ES-J 995,E2MATE,BLE 00084

Others Others
.Estradiol 3-sulfamate inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor.
T5326 Sugammadex sodium

Org25969,Sugammadex (sodium),舒更葡糖钠

Others Others
Sugammadex sodium (Org25969) 是合成的 γ 环糊精衍生物,是一种新型的神经肌肉阻断逆转剂。
T6465 Dexamethasone Sodium Phosphate

Dexadreson,地塞米松磷酸钠,Dexagro,Dalalone

IL Receptor; COX Immunology/Inflammation; Neuroscience
Dexamethasone Sodium Phosphate (Dexadreson) 是一种白细胞介素受体调节剂,具有抗炎和免疫抑制作用。它属于类固醇合成药物的强效糖皮质激素类。
T0384 Estradiol benzoate

Benzoestrofol,Benzhormovarine,苯甲酸雌二醇,Benovocylin

Estrogen Receptor/ERR; Estrogen/progestogen Receptor Endocrinology/Hormones
Estradiol benzoate (Benzhormovarine) 是一种类固醇性激素,是一种雌二醇的前体药物。它表现出轻微的合成代谢特性,增加血液凝固性。
T6502 Fluocinonide

醋酸氟轻松,Lidex,Metosyn,氟轻松,Topsyn

Glucocorticoid Receptor Endocrinology/Hormones
Fluocinonide (Topsyn) 是一种糖皮质激素类固醇,具有抗炎作用,可作用于皮肤疾病的研究。
T6503 Fluorometholone Acetate

NSC 47438,Flarex,Eflone,氟米龙醋酸酯,Oxylone acetate

Glucocorticoid Receptor; Carbonic Anhydrase Endocrinology/Hormones; Metabolism
Fluorometholone Acetate (Oxylone acetate) 是合成的糖皮质激素皮质类固醇及皮质类固醇酯。它有效抑制碳酸酐酶 (CA) 对 hCA-I(IC50:2.18 μM)和 hCA-II(IC50:17.5 μM)。它具有抗炎活性,可用于研究外部眼部炎症。
T2199 Myclobutanil

Systhane,腈菌唑

Antifungal Microbiology/Virology
Myclobutanil (Systhane) 是康唑类抗真菌剂,可用作农药。
T13684 Equilin

7-Dehydroestrone

Calcium Channel Membrane transporter/Ion channel; Metabolism
Equilin (7-Dehydroestrone) 是神经营养性雌激素类固醇,具有血管扩张活性,通过 NF-κB 信号传导增加单核细胞-内皮粘附。Equilin 通过阻断Ca(2+)进入平滑肌来同样放松肠系膜动脉的阻力。
T1594 Vecuronium bromide

ORG NC 45,维库溴铵

AChR Neuroscience
Vecuronium bromide (ORG NC 45) 是一种合成的中效单季铵盐类固醇和非去极化神经肌肉阻滞剂,具有肌肉松弛活性。
T15000 Cort108297

Glucocorticoid Receptor Endocrinology/Hormones
Cort108297是一种选择性糖皮质激素受体调节剂,也是一种对其他类固醇受体无亲和力的选择性GR 拮抗剂。Cort108297对gr 具有较高的亲和力(Ki: 0.45 nM)。
T6215 Abiraterone Acetate

Zytiga,乙酸阿比特龙酯,CB7630

P450 Metabolism
Abiraterone Acetate (CB7630) 是一种具有口服活性的、不可逆的 CYP17A1选择性抑制剂,具有抗雄激素作用。它是 Abiraterone 的前药。
T23549 YM 511

P450; Aromatase Endocrinology/Hormones; Metabolism
YM 511 是一种高度特异性的非甾体芳香酶 (aromatase) 抑制剂。YM 511 竞争性抑制大鼠卵巢和人胎盘微粒体中的芳香酶活性 (IC50 分别为 0.4 和 0.12 nM)。YM 511 轻微抑制其他类固醇激素的产生。YM 511 具有用于抑制雌激素依赖性作用研究,不会影响其他类固醇激素的血清水平的潜力。
T6886 MCB-613

MCB 613

Src Angiogenesis; Tyrosine Kinase/Adaptors
MCB-613 是类固醇受体共激活因子 (SRC) 小分子“刺激物” (SMS),超刺激 SRCs 的转录活性。它促进 SRC 与其他共激活因子发生相互作用,并显著诱导 ER 应激与活性氧的产生相结合。它是一种 SMS,能够过度刺激 SRC 致癌程序,靶向癌基因用作抗癌药物。
T67901 SRD5A1-IN-1

Others Others
SRD5A1-IN-1 是类固醇 5α-还原酶 1 型的抑制剂(SRD5A1,IC50 = 1.44 µM)。 SRD5A1-IN-1 可降低二氢睾酮的产生并显着降低 SRD5A1 蛋白表达。
T0947 Dexamethasone acetate

Dexamethasone 21-acetate,醋酸地塞米松,Dexamethason acetate,NSC 39471

Glucocorticoid Receptor; Mitophagy; IL Receptor; Annexin A; NOS; Antibacterial; Autophagy Autophagy; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology
Dexamethasone acetate (NSC 39471) 是一种糖皮质素类甾体,有抗炎和免疫抑制活性。它可研究眼部感染。
T3316 Fluorometholone

氟米龙,Fluoromethalone,Cortilet,Oxylone,Delmeson

Glucocorticoid Receptor Endocrinology/Hormones
Fluorometholone (Fluoromethalone) 是合成糖皮质激素,具有抗炎和抗过敏作用。它可用作糖皮质激素受体激动剂,能够用于干眼症的研究。
T72470 Estrone O-sulfamate

Estrone 3-O-sulfamate

Others Others
Estrone O-sulfamate (Estrone 3-O-sulfamate) 是一种高效的的类固醇硫酸酯酶 (STS) 抑制剂。Estrone O-sulfamate 是一种胎盘微粒体抑制剂 (P.M.) ,IC50 值分别为 18 nM。Estrone O-sulfamate 在 MCF-7 细胞中对 STS 显示出抑制作用,IC50 值分别为 0.83 nM。Estrone O-sulfamate 可用于研究癌症。
T60924 Verosudil

AR-12286

ROCK Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells
Verosudil (AR-12286) 是一种高效的 Rho 激酶 (ROCK) 抑制剂,对 ROCK1 和 ROCK2 的 Ki 分别为 2 和 2 nM。AR-12286 可逆转类固醇诱导的小鼠眼内压,可通过增加眼房水通过小梁网流出来减缓眼压。
T2556 Nandrolone decanoate

癸酸诺龙,19-Nortestosterone decanoate

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Nandrolone decanoate (19-Nortestosterone decanoate) 是一种合成代谢雄激素,通过涉及谷氨酸诱导的 N-甲基-D-天冬氨酸受体过度兴奋的机制诱导攻击性行为表征。
T1438 Butoconazole nitrate

RS 35887,硝酸布康唑

Estrogen/progestogen Receptor; Antifungal Endocrinology/Hormones; Microbiology/Virology
Butoconazole nitrate (RS 35887) 是一种咪唑类抗真菌药物,可治疗由白色念珠菌引起的阴道感染。它可通过抑制类固醇合成起到抗菌作用。
T28773 SI-2

SI2,EPH 116,EPH116,EPH-116

Others Others
SI-2是类固醇受体辅激活因子-3(SRC-3或 AIB1)的抑制剂(SMI)。SI-2可选择性降低细胞中 SRC-3的转录活性和蛋白浓度,并选择性诱导低纳摩尔范围(3-20 nM)内的乳腺癌症细胞死亡,但不影响正常细胞存活率。

化合物

Steroid sulfatase-IN-5
Cat.No: T81091
Synonym:
Target:
Steroid sulfatase-IN-4
Cat.No: T62237
Synonym:
Target:
Steroid sulfatase-IN-2
Cat.No: T61212
Synonym:
Target:
Steroid sulfatase-IN-6
Cat.No: T81090
Synonym:
Target:
Biotin-SRC-1 (676–700) TFA
Cat.No: T83752
Synonym: Biotin-Steroid Receptor Coactivator 1 (676-700)
Target:
Steroid sulfatase-IN-7
Cat.No: T81089
Synonym:
Target:
Steroid sulfatase-IN-1
Cat.No: T61687
Synonym:
Target:
Steroid sulfatase-IN-3
Cat.No: T61686
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-1
Cat.No: T61716
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-5
Cat.No: T81092
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-4
Cat.No: T61979
Synonym:
Target:
Steroid sulfatase/17β-HSD1-IN-3
Cat.No: T62236
Synonym:
Target:
Loteprednol etabonate
Cat.No: T0181
Synonym: Lotemax,Alrex,氯替泼诺
Target: Glucocorticoid Receptor, Antibacterial, Antibiotic
Pancuronium dibromide
Cat.No: T0166
Synonym: Pancuronium bromide,Pavulon,泮库溴铵
Target: AChR
Budesonide
Cat.No: T0094
Synonym: Entocort,Pulmicort,布地奈德,Rhinocort
Target: Glucocorticoid Receptor
Mometasone furoate
Cat.No: T1531
Synonym: 糠酸莫美他松,糠酸莫米松,Sch32088
Target: Glucocorticoid Receptor
Cyproterone acetate
Cat.No: T1167
Synonym: Androcur,醋酸环丙氯地孕酮,Cyproterone 17-O-acetate,醋酸环丙孕酮
Target: Androgen Receptor
Nonsteroidal aromatase inhibitor 1
Cat.No: T61444
Synonym:
Target:
3α-Hydroxysteroid dehydrogenase
Cat.No: T76147
Synonym:
Target:
Irosustat
Cat.No: T4464
Synonym: 667-Coumate,BN83495,STX64
Target: Others
MK 0434
Cat.No: T33414
Synonym: MK0434,MK434,MK 434,MK-0434,MK-434
Target:
Metyrapone
Cat.No: T0293
Synonym: 美替拉酮,甲吡酮,NSC-25265,Su-4885
Target: Others, P450, Dehydrogenase, Autophagy
Boldenone Cypionate
Cat.No: T19213
Synonym:
Target: Others, Androgen Receptor
Altrenogest
Cat.No: T0870
Synonym: R2267,RU2267,Allyltrenbolone,A35957,烯丙孕素
Target: Estrogen/progestogen Receptor, Progesterone Receptor
Boldenone Undecylenate
Cat.No: T3137
Synonym: Parenabol,Ba 29038,Vebonol,十一碳烯酸去甲睾酮
Target: Androgen Receptor, Endogenous Metabolite
S5A1
Cat.No: T83615
Synonym:
Target: Others
Brassinazole
Cat.No: T60929
Synonym: (2S,3R)-Brassinazole
Target: Others
Anecortave Acetate
Cat.No: T21452
Synonym: Retaane,Al 3789,NSC 24345,NSC 15475,Anecortave
Target: Others
GSK3987
Cat.No: T27478
Synonym:
Target: Liver X Receptor
Estradiol 3-sulfamate
Cat.No: T11235
Synonym: 雌二醇 3-氨基磺酸,ES-J 995,E2MATE,BLE 00084
Target: Others
Sugammadex sodium
Cat.No: T5326
Synonym: Org25969,Sugammadex (sodium),舒更葡糖钠
Target: Others
Dexamethasone Sodium Phosphate
Cat.No: T6465
Synonym: Dexadreson,地塞米松磷酸钠,Dexagro,Dalalone
Target: IL Receptor, COX
Estradiol benzoate
Cat.No: T0384
Synonym: Benzoestrofol,Benzhormovarine,苯甲酸雌二醇,Benovocylin
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor
Fluocinonide
Cat.No: T6502
Synonym: 醋酸氟轻松,Lidex,Metosyn,氟轻松,Topsyn
Target: Glucocorticoid Receptor
Fluorometholone Acetate
Cat.No: T6503
Synonym: NSC 47438,Flarex,Eflone,氟米龙醋酸酯,Oxylone acetate
Target: Glucocorticoid Receptor, Carbonic Anhydrase
Myclobutanil
Cat.No: T2199
Synonym: Systhane,腈菌唑
Target: Antifungal
Equilin
Cat.No: T13684
Synonym: 7-Dehydroestrone
Target: Calcium Channel
Vecuronium bromide
Cat.No: T1594
Synonym: ORG NC 45,维库溴铵
Target: AChR
Cort108297
Cat.No: T15000
Synonym:
Target: Glucocorticoid Receptor
Abiraterone Acetate
Cat.No: T6215
Synonym: Zytiga,乙酸阿比特龙酯,CB7630
Target: P450
YM 511
Cat.No: T23549
Synonym:
Target: P450, Aromatase
MCB-613
Cat.No: T6886
Synonym: MCB 613
Target: Src
SRD5A1-IN-1
Cat.No: T67901
Synonym:
Target: Others
Dexamethasone acetate
Cat.No: T0947
Synonym: Dexamethasone 21-acetate,醋酸地塞米松,Dexamethason acetate,NSC 39471
Target: Glucocorticoid Receptor, Mitophagy, IL Receptor, Annexin A, NOS, Antibacterial, Autophagy
Fluorometholone
Cat.No: T3316
Synonym: 氟米龙,Fluoromethalone,Cortilet,Oxylone,Delmeson
Target: Glucocorticoid Receptor
Estrone O-sulfamate
Cat.No: T72470
Synonym: Estrone 3-O-sulfamate
Target: Others
Verosudil
Cat.No: T60924
Synonym: AR-12286
Target: ROCK
Nandrolone decanoate
Cat.No: T2556
Synonym: 癸酸诺龙,19-Nortestosterone decanoate
Target: Others, HIV Protease
Butoconazole nitrate
Cat.No: T1438
Synonym: RS 35887,硝酸布康唑
Target: Estrogen/progestogen Receptor, Antifungal
SI-2
Cat.No: T28773
Synonym: SI2,EPH 116,EPH116,EPH-116
Target: Others
Cat. No. Product Name Target Signaling Pathways
T19470 Nandrolone propionate

Others; Androgen Receptor Endocrinology/Hormones; Others
Nandrolone propionate 是合成代谢类固醇,主要由雄激素和保氮剂组成,具有作用时间相对较长的特点。
T8709 Nandrolone phenylpropionate

Nandrolone phenpropionate,苯丙酸诺龙

Androgen Receptor Endocrinology/Hormones
Nandrolone phenylpropionate (Nandrolone phenpropionate) 是一种合成代谢类固醇,是一种 19-nortestosterone 的衍生物。它能够促进蛋白质合成,用于缓解组织分解代谢,可以用于骨质疏松症和特纳综合征的研究。
T5S1982 Periplocin

Periplocoside,杠柳毒苷

Apoptosis; Others Apoptosis; Others
Periplocin (Periplocoside) 是从黑龙骨中分离出的一种强心类固醇。它可促进肿瘤细胞凋亡并抑制肿瘤生长。它通过激活 Na/K-ATPase 介导的 Src/ERK 和 PI3K/Akt 途径,具有促进伤口愈合的潜力。
TN3270 (R)-3β-Hydroxy steroid sulfotransferase-IN-11

Others Others
T8117 Metenolone acetate

Methenolone acetate,美替诺龙醋酸酯

Others; Androgen Receptor Endocrinology/Hormones; Others
Metenolone acetate (Methenolone acetate) 是一种合成代谢类固醇(AAS) 药物,是一种雄激素,主要用于治疗由于骨髓衰竭引起的贫血。
T2207 Adrenosterone

肾上腺甾酮,11-ketoandrostenedione,11-oxoandrostenedione,Reichstein's substance G

Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Adrenosterone (11-ketoandrostenedione) 是一种人内源性代谢物,由肾上腺皮质产生。Adrenosterone 是一种竞争性羟基类固醇脱氢酶 1 抑制剂。它是一种的类固醇激素,具有较弱的雄激素特性。它是一种膳食补充剂,能够减少脂肪并提高肌肉质量。它能够抑制人类癌细胞的转移进展。
TMA0984 Cerevisterol

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Cerevisterol 是一种细胞毒性类固醇,提取于Agaricus blazei 子实体,对 DNA 聚合酶 α 的活性具有抑制作用。
T36857 Estrone sulfate sodium

雌酮3-硫酸钠,Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate

Endogenous Metabolite Metabolism
Estrone sulfate sodium (17β-Estrone 3-sulfate) 是一种主要的循环血浆雌激素,无生物活性,通过类固醇硫酸酯酶(STS) 转化为生物活性雌激素雌酮。
T1048 Estradiol

雌二醇,E2,17β-Estradiol,17β-Oestradiol,β-Estradiol

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Estradiol (E2) 是一种天然的类固醇性激素,对于女性生育能力和第二性征的维持至关重要。Estradiol 通过雌激素受体 β (ERβ) 上调 IL-6 表达。
T14001 11-Beta-hydroxyandrostenedione

4-雄烯-11β-醇-3,17-二酮,NSC-17102,4-Androsten-11β-ol-3,17-dione

Endogenous Metabolite Metabolism
11-Beta-hydroxyandrostenedione (NSC-17102) 是主要存在于肾上腺的类固醇,也是 11β-羟基类固醇脱氢酶同工酶抑制剂。随着 4-androstenedione 的提高,通过测量血浆中的11-Beta-hydroxyandrostenedione,能够区分高雄激素血症的肾上腺或卵巢起源。
TN3910 Ecdysone

Apoptosis; ATPase; Glucocorticoid Receptor; Potassium Channel; Sodium Channel; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; Membrane transporter/Ion channel; Metabolism
Ecdysone 是存在于昆虫和草药中的主要类固醇激素,可以激活盐皮质激素受体并诱导细胞凋亡。Ecdysone 的活性代谢物 20-羟基蜕皮激素在协调发育过渡和体内稳态睡眠调节中起重要作用。
T3220 Euphorbiasteroid

Euphobiasteroid,Euphorbia factor L1,千金子甾醇

Others; AMPK Chromatin/Epigenetic; Others; PI3K/Akt/mTOR signaling
Euphorbiasteroid (Euphobiasteroid) 是续随子中的一种三环二萜,可抑制酪氨酸酶活性,增强AMPK 的磷酸化。它通过减少细胞内甘油三酯的积累来降低 3T3-L1 细胞的分化,具有抗癌、抗病毒、抗肥胖及多重耐药调节作用。
TN7130 Chlorogenin

Others Others
Chlorogenin 是一种源自 Agave americana 草本植物的天然类固醇。
T13500 3-O-Acetyl-20-Hydroxyecdysone

Others Others
3-O-Acetyl-20-Hydroxyecdysone 是分离自Cyanotis arachnoidea C.B.Clark 根中的类固醇。
T8043 5α-Cholestane

Endogenous Metabolite Metabolism
5α-Cholestane 属于胆甾烷类固醇类化合物。
T20302 Deoxycorticosterone

Desoxycorticosterone,去氧皮质酮,Desoxycorticosteronum,Desoxycortone

Endogenous Metabolite Metabolism
Deoxycorticosterone (Desoxycortone) 是由肾上腺产生的类固醇代谢物。 Deoxycorticosterone 是醛固酮前体,具有盐皮质激素活性。
T10048 17a-Hydroxypregnenolone

Endogenous Metabolite Metabolism
17a-Hydroxypregnenolone 是一种孕烷类固醇, 是形成脱氢表雄酮的激素原。
TC0026 Testosterone benzoate

Others Others
Testosterone benzoate 是一种合成的注射合成代谢雄激素类固醇 (AAS) 和一种雄激素酯。
TN1075 Adynerin

Others Others
Adynerin 是一种发现于夹竹桃中的天然类固醇。
T0856 Dehydroisoandrosterone 3-acetate

Dehydroepiandrosterone 3-acetate,Dehydroepiandrosterone acetate,Prasterone acetate,DHEA acetate,醋酸去氢表雄酮,androstenolone acetate

Androgen Receptor Endocrinology/Hormones
Dehydroisoandrosterone 3-acetate (Prasterone acetate) 是一种雄性激素/雌性激素的前体物质,是一种由肾上腺皮质产生的主要 C19 类固醇,能够调节脊椎动物的攻击性行为。
T2748 Cortodoxone

可托多松,11-Deoxycortisol,cortexolone,17α,21-dihydroxyprogesterone,Reichstein's substance S,11-Desoxycortisol

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Cortodoxone (11-Desoxycortisol) 是糖皮质类固醇激素,能够氧化为皮质醇。
T3130 Testosterone phenylpropionate

Testosterone hydrocinnamate,苯丙酸睾酮,Retandrol,Testosterone 17-phenylpropionate

Others Others
Testosterone phenylpropionate (Testosterone 17-phenylpropionate) 是一种长效雄激素。d3-Testosterone phenylpropionate 可用作内标物。
T2912 Ergosterol

麦角固醇,Provitamin D,Ergosterin,Provitamin D2

Others; Endogenous Metabolite Metabolism; Others
Ergosterol (Provitamin D2) 是真菌中的主要固醇类,具有抗炎,抗氧化和抗增殖的作用。
T73772 Estrone sulfate potassium

Endogenous Metabolite Metabolism
Estrone sulfate potassium 是一种雌激素酯和共轭物,是一种天然内源性类固醇。
T6S1842 Tenacissoside G

Tenacissimoside A,通关藤苷G

Others Others
Tenacissoside G 是一种 C21 甾体,来自于Marsdenia tenacissima 茎部。它可逆转 P-糖蛋白过度表达的多药耐药癌细胞的多药耐药。
T7024 Qingyangshengenin

青阳参甙元,Qingyangshengenin A,Cynanchagenin

Others Others
Qingyangshengenin (Cynanchagenin) 是一种孕烷糖苷,是一种分离自Cychuchumot ophyllum(Asclepiadaceae) 的根中的 C21 类固醇糖苷配基。它具有抗癌作用。
T12536 Pregnenolone monosulfate

3β-Hydroxy-5-pregnen-20-one monosulfate

NMDAR Neuroscience
Pregnenolone monosulfate (3β-Hydroxy-5-pregnen-20-one monosulfate) 是一种强效神经类固醇,可正向调节 NMDA 记录,可用于研究神经分裂和抑郁症。
T3033 Deoxycorticosterone acetate

醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮

Glucocorticoid Receptor; Endogenous Metabolite; Adrenergic Receptor Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience
Deoxycorticosterone acetate (Cortexone acetate) 是肾上腺产生的类固醇激素,具有盐皮质激素活性,并作为醛固酮的前体。
T9171 Methenolone enanthate

Others Others
Methenolone enanthate 是一种雄激素和合成代谢类固醇 (AAS) 药物,主要用于治疗由于骨髓衰竭引起的贫血。
TC0019 Pregnenolone acetate

孕烯醇酮醋酸酯,3β-Hydroxy-5-pregnen-20-one acetate

Cannabinoid Receptor; Endogenous Metabolite GPCR/G Protein; Metabolism
Pregnenolone acetate 是一种强大的神经类固醇,是各种类固醇激素(包括类固醇酮)的主要前体。它作为大麻素 CB1 受体的信号特异性抑制剂,抑制由 CB1 受体介导的四氢大麻酚 (THC) 的作用。它可以保护大脑免受大麻中毒。
T2822 Ginsenoside Rb1

Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III

ATPase; Mitophagy; IRAK; NF-κB; Autophagy; HSV Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Ginsenoside Rb1 (Gypenoside Ⅲ) 是中药人参的成分,可能具有抑制或阻止肿瘤生长的特性。
TN7099 antcin A

NOD Immunology/Inflammation; NF-κB
antcin A 是一种类固醇类植物化学物质,从珍贵的食用菌牛樟芝子实体中分离出来,具有很强的抗炎和抗肿瘤作用。
T3S0895 Spirostan-3-ol

剑麻皂苷元,Sarsaponin

Others Others
Spirostan-3-ol (Sarsaponin) 是 Sarsasapogenin 的立体异构体,是从植物材料中分离出来的类固醇糖苷,具有潜在的通过细胞凋亡的抗肿瘤活性。它可驱赶蜜蜂。
T8040 Cholesterol myristate

胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate

Others; Potassium Channel; GABA Receptor; Endogenous Metabolite; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
Cholesterol myristate (Cholesteryl myristate) 是粗吻海龙中的一种类固醇,可与多种离子通道结合,例如nAChR、GABAA 受体和内向整流钾离子通道。
T7990 9-hydroxy-4-androstene-3,17-dione

Others Others
9-hydroxy-4-androstene-3,17-dione 是一种类固醇激素,具有抗肿瘤活性,可以抑制多种癌症细胞的生长,包括乳腺癌、前列腺癌和肺癌细胞。
T6654 Saponins

Sapogenins Glycosides,皂素,Saponin

Others Others
Saponins (Sapogenins Glycosides) 是一种苷类的化合物,多发现于多种植物中,可保护植物免受微生物和真菌的破坏。
T0948L Corticosterone

皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)

Glucocorticoid Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Corticosterone (Kendall's compound B) 是一种肾上腺皮质类固醇,有盐皮质激素和糖皮质激素的活性,具有口服活性。Corticosterone 参与体内能量、免疫反应和应激反应的调节。
T0851 Pregnenolone

3β-Hydroxy-5-pregnen-20-one,Arthenolone,孕烯醇酮

Cannabinoid Receptor; Endogenous Metabolite; TRP/TRPV Channel; AChR; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Pregnenolone (Arthenolone) 是一种由胆固醇合成的内源性类固醇激素,用于治疗阿尔茨海默病。它是大麻素 CB1受体的信号传导特异性抑制剂,抑制由 CB1受体介导的四氢大麻酚 的作用。它也是 TRPM3通道激活剂,也可弱激活 TRPM1通道。
T5751 Tigogenin

Others Others
Tigogenin 是甾体皂甙元,普遍用于甾体类药物的合成。它能够阻碍小鼠骨髓基质细胞脂肪细胞分化,促使成骨细胞的分化。
T1429 17α-Hydroxyprogesterone

Hydroxyprogesterone,17-OHP,羟孕酮,17-Hydroxyprogesterone,17α-羟孕酮

Estrogen/progestogen Receptor; Progesterone Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
17α-Hydroxyprogesterone (17-OHP) 是一种内源性孕激素,其他类固醇激素(包括糖皮质激素,雌激素,和雄激素)生物合成的化学中间体。
T2777 Ginsenoside Rg1

Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2

Apoptosis; Beta Amyloid; NF-κB Apoptosis; Neuroscience; NF-κB
Ginsenoside Rg1 (Panaxoside Rg1) 是人参的主要活性成分之一,可减少NF-κB 核易位。它改善认知功能受损,通过降低大脑Aβ水平来发挥作用。
T5574 Guggulsterone

Guggulsterone E&Z,香胶甾酮

Apoptosis; FXR; Akt; Caspase; JNK; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; MAPK; Metabolism; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Guggulsterone (Guggulsterone E&Z) E&Z 是来自Commiphora wightii 树中树胶脂的植物甾醇。 它通过下调抗细胞凋亡基因产物 ,调节细胞周期蛋白,激活caspases,JNK,抑制Akt,抑制多种肿瘤细胞的生长并诱导细胞凋亡。它是法尼醇 X 受体拮抗剂,可降低 CDCA 诱导的 FXR 活化。
T2881 Crustecdysone

Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,β-蜕皮甾酮,Hydroxyecdysone,羟基蜕皮激素

Others; Caspase; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism; Others; Proteases/Proteasome
Crustecdysone (Hydroxyecdysone) 是来源于露水草的一种蜕皮激素,可调节昆虫的蜕皮或蜕皮过程。它是 Ecdysone 的活性代谢物,通过 20E 核受体复合物 EcR-USP 抑制半胱天冬酶活性并诱导自噬,在心血管系统中具有调节或保护作用。
T4878 Hecogenin

海柯吉宁,Hocogenin

Others; Antifungal Microbiology/Virology; Others
Hecogenin(Hocogenin),一种从Agave sisalana提取的甾体皂苷,作为人类UDP-glucuronosyltransferases的特异性抑制剂。它具有广泛的药理活性,包括抗炎、抗真菌和胃保护作用[1]。
T0478 Progesterone

孕酮,Pregn-4-ene-3,20-dione

Estrogen/progestogen Receptor; Progesterone Receptor; Opioid Receptor; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience; Others
Progesterone (Pregn-4-ene-3,20-dione) 是类固醇激素,能够调节月经周期。
T19124 3-​Oxocholic acid

3-Ketocholic acid

Endogenous Metabolite Metabolism
3-​Oxocholic acid(3-Ketocholic acid) 是胆汁酸的代谢产物,也是产气荚膜梭菌在肠道中由胆汁降解的主要产物。33-​Oxocholic acid 是一种主要存在于哺乳动物的胆汁中类固醇酸。
T2733 Sarsasapogenin

Parigenin,知母皂苷元,Sarsagenin

Apoptosis; NF-κB; Endogenous Metabolite Apoptosis; Metabolism; NF-κB
Sarsasapogenin (Parigenin) 是一种甾体皂苷元,从中草药知母中分离到,具有抗糖尿病、抗氧化、抗癌、抗炎等作用。
T4717 25-Hydroxycholesterol

25-羟基胆固醇,25-羟基胆甾醇

Others; Endogenous Metabolite; HMG-CoA Reductase Metabolism; Others
25-Hydroxycholesterol 是胆固醇的代谢产物,由巨噬细胞响应 Toll 样受体激活而分泌。它有效抑制 B 细胞产生 IgA,EC50约为 65 nM。
T1009 Estrone

Oestrone,雌酮,Fluoroethyl,Aquacrine

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Estrone (Aquacrine) 是内源性雌激素的主要代表,由多种组织产生,尤其是脂肪组织。它是脂肪细胞中雄烯二酮芳构化过程的结果。
T3674 Hydroxysafflor yellow A

藏红花,羟基红花黄色素A,HSYA,Safflomin A

TGF-beta/Smad Stem Cells
Hydroxysafflor yellow A (Safflomin A) 是一种黄酮类天然产物,从中药红花中分离得到,具有抗癌作用。
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天然产物

Nandrolone propionate
Cat.No: T19470
Synonym:
Target: Others, Androgen Receptor
Nandrolone phenylpropionate
Cat.No: T8709
Synonym: Nandrolone phenpropionate,苯丙酸诺龙
Target: Androgen Receptor
Periplocin
Cat.No: T5S1982
Synonym: Periplocoside,杠柳毒苷
Target: Apoptosis, Others
(R)-3β-Hydroxy steroid sulfotransferase-IN-11
Cat.No: TN3270
Synonym:
Target: Others
Metenolone acetate
Cat.No: T8117
Synonym: Methenolone acetate,美替诺龙醋酸酯
Target: Others, Androgen Receptor
Adrenosterone
Cat.No: T2207
Synonym: 肾上腺甾酮,11-ketoandrostenedione,11-oxoandrostenedione,Reichstein's substance G
Target: Androgen Receptor, Endogenous Metabolite
Cerevisterol
Cat.No: TMA0984
Synonym:
Target: DNA/RNA Synthesis
Estrone sulfate sodium
Cat.No: T36857
Synonym: 雌酮3-硫酸钠,Estrone 3-sulfate (sodium salt),17β-Estrone 3-sulfate
Target: Endogenous Metabolite
Estradiol
Cat.No: T1048
Synonym: 雌二醇,E2,17β-Estradiol,17β-Oestradiol,β-Estradiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
11-Beta-hydroxyandrostenedione
Cat.No: T14001
Synonym: 4-雄烯-11β-醇-3,17-二酮,NSC-17102,4-Androsten-11β-ol-3,17-dione
Target: Endogenous Metabolite
Ecdysone
Cat.No: TN3910
Synonym:
Target: Apoptosis, ATPase, Glucocorticoid Receptor, Potassium Channel, Sodium Channel, Endogenous Metabolite, Autophagy
Euphorbiasteroid
Cat.No: T3220
Synonym: Euphobiasteroid,Euphorbia factor L1,千金子甾醇
Target: Others, AMPK
Chlorogenin
Cat.No: TN7130
Synonym:
Target: Others
3-O-Acetyl-20-Hydroxyecdysone
Cat.No: T13500
Synonym:
Target: Others
5α-Cholestane
Cat.No: T8043
Synonym:
Target: Endogenous Metabolite
Deoxycorticosterone
Cat.No: T20302
Synonym: Desoxycorticosterone,去氧皮质酮,Desoxycorticosteronum,Desoxycortone
Target: Endogenous Metabolite
17a-Hydroxypregnenolone
Cat.No: T10048
Synonym:
Target: Endogenous Metabolite
Testosterone benzoate
Cat.No: TC0026
Synonym:
Target: Others
Adynerin
Cat.No: TN1075
Synonym:
Target: Others
Dehydroisoandrosterone 3-acetate
Cat.No: T0856
Synonym: Dehydroepiandrosterone 3-acetate,Dehydroepiandrosterone acetate,Prasterone acetate,DHEA acetate,醋酸去氢表雄酮,androstenolone acetate
Target: Androgen Receptor
Cortodoxone
Cat.No: T2748
Synonym: 可托多松,11-Deoxycortisol,cortexolone,17α,21-dihydroxyprogesterone,Reichstein's substance S,11-Desoxycortisol
Target: Glucocorticoid Receptor, Endogenous Metabolite
Testosterone phenylpropionate
Cat.No: T3130
Synonym: Testosterone hydrocinnamate,苯丙酸睾酮,Retandrol,Testosterone 17-phenylpropionate
Target: Others
Ergosterol
Cat.No: T2912
Synonym: 麦角固醇,Provitamin D,Ergosterin,Provitamin D2
Target: Others, Endogenous Metabolite
Estrone sulfate potassium
Cat.No: T73772
Synonym:
Target: Endogenous Metabolite
Tenacissoside G
Cat.No: T6S1842
Synonym: Tenacissimoside A,通关藤苷G
Target: Others
Qingyangshengenin
Cat.No: T7024
Synonym: 青阳参甙元,Qingyangshengenin A,Cynanchagenin
Target: Others
Pregnenolone monosulfate
Cat.No: T12536
Synonym: 3β-Hydroxy-5-pregnen-20-one monosulfate
Target: NMDAR
Deoxycorticosterone acetate
Cat.No: T3033
Synonym: 醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮
Target: Glucocorticoid Receptor, Endogenous Metabolite, Adrenergic Receptor
Methenolone enanthate
Cat.No: T9171
Synonym:
Target: Others
Pregnenolone acetate
Cat.No: TC0019
Synonym: 孕烯醇酮醋酸酯,3β-Hydroxy-5-pregnen-20-one acetate
Target: Cannabinoid Receptor, Endogenous Metabolite
Ginsenoside Rb1
Cat.No: T2822
Synonym: Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III
Target: ATPase, Mitophagy, IRAK, NF-κB, Autophagy, HSV
antcin A
Cat.No: TN7099
Synonym:
Target: NOD
Spirostan-3-ol
Cat.No: T3S0895
Synonym: 剑麻皂苷元,Sarsaponin
Target: Others
Cholesterol myristate
Cat.No: T8040
Synonym: 胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate
Target: Others, Potassium Channel, GABA Receptor, Endogenous Metabolite, AChR
9-hydroxy-4-androstene-3,17-dione
Cat.No: T7990
Synonym:
Target: Others
Saponins
Cat.No: T6654
Synonym: Sapogenins Glycosides,皂素,Saponin
Target: Others
Corticosterone
Cat.No: T0948L
Synonym: 皮质酮,17-Deoxycortisol,11β,21-Dihydroxyprogesterone,Kendall's compound B,肾上腺酮,Corticosterone (From plants)
Target: Glucocorticoid Receptor, Endogenous Metabolite
Pregnenolone
Cat.No: T0851
Synonym: 3β-Hydroxy-5-pregnen-20-one,Arthenolone,孕烯醇酮
Target: Cannabinoid Receptor, Endogenous Metabolite, TRP/TRPV Channel, AChR, Autophagy
Tigogenin
Cat.No: T5751
Synonym:
Target: Others
17α-Hydroxyprogesterone
Cat.No: T1429
Synonym: Hydroxyprogesterone,17-OHP,羟孕酮,17-Hydroxyprogesterone,17α-羟孕酮
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Endogenous Metabolite
Ginsenoside Rg1
Cat.No: T2777
Synonym: Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2
Target: Apoptosis, Beta Amyloid, NF-κB
Guggulsterone
Cat.No: T5574
Synonym: Guggulsterone E&Z,香胶甾酮
Target: Apoptosis, FXR, Akt, Caspase, JNK, Autophagy
Crustecdysone
Cat.No: T2881
Synonym: Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,β-蜕皮甾酮,Hydroxyecdysone,羟基蜕皮激素
Target: Others, Caspase, Endogenous Metabolite, Autophagy
Hecogenin
Cat.No: T4878
Synonym: 海柯吉宁,Hocogenin
Target: Others, Antifungal
Progesterone
Cat.No: T0478
Synonym: 孕酮,Pregn-4-ene-3,20-dione
Target: Estrogen/progestogen Receptor, Progesterone Receptor, Opioid Receptor, Endogenous Metabolite
3-​Oxocholic acid
Cat.No: T19124
Synonym: 3-Ketocholic acid
Target: Endogenous Metabolite
Sarsasapogenin
Cat.No: T2733
Synonym: Parigenin,知母皂苷元,Sarsagenin
Target: Apoptosis, NF-κB, Endogenous Metabolite
25-Hydroxycholesterol
Cat.No: T4717
Synonym: 25-羟基胆固醇,25-羟基胆甾醇
Target: Others, Endogenous Metabolite, HMG-CoA Reductase
Estrone
Cat.No: T1009
Synonym: Oestrone,雌酮,Fluoroethyl,Aquacrine
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
Hydroxysafflor yellow A
Cat.No: T3674
Synonym: 藏红花,羟基红花黄色素A,HSYA,Safflomin A
Target: TGF-beta/Smad
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