161
108
3
10
Cat. No. | Product Name | ||
---|---|---|---|
L1010 | FDA上市及药典收录分子库 | 3157 compounds | |
3157 个上市及药典分子集合,可用于高通量筛选和高内涵筛选; | |||
L6800 | 中国药典收录天然产物库 | 2051 compounds | |
2051 种中国药典收录的天然产物,是药物开发、药理研究等领域的有力工具; | |||
L7830 | 高溶解性片段药效团化合物库 | 985 compounds | |
高溶解性片段药效团库包含985 个片段小分子。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T29612 | ACO Ser CNU | ||
ACO Ser CNU is a therapeutic agent. | |||
T35664 |
Tetracosactide acetate
|
Others | Others |
Tetracosactide acetate 是一种合成的多肽,可刺激肾上腺释放皮质类固醇 ,如皮质醇。Tetracosactide acetate 在溃疡性结肠炎和克罗恩病、青少年和成人类风湿性关节炎和骨关节病方面有研究的价值。 | |||
T77443 |
Racotumomab
|
Others | Others |
Racotumomab (Anti-Human NGcGM3 Recombinant Antibody) 是一种小鼠 γ 型抗独特型单克隆抗体,可特异性诱导针对在多种实体瘤中过表达的 Neu-glycolyl GM3 神经节苷脂 (NeuGcGM3) 的抗体反应。Racotumomab 可与含有 Neu-glycolyl (NeuGc) 的神经节苷脂、硫苷脂和肿瘤中表达的其他抗原发生反应。Racotumomab 具有抗癌活性,可用于肺癌的研究。 | |||
T21294 |
Polmacoxib
CG-100649,帕马考昔,CG100649,CG 100649 |
COX; Carbonic Anhydrase | Immunology/Inflammation; Metabolism; Neuroscience |
Polmacoxib (CG 100649) 是一流的 NSAID 候选药物,是碳酸酐酶 (CA) 和 COX-2 的双重抑制剂。它在小鼠模型中抑制大肠腺瘤和肿瘤生长。 | |||
T7725 |
Albaconazole
W 0027,UR-9825,UR9825,W-0027 |
P450; Antifungal | Metabolism; Microbiology/Virology |
Albaconazole (W-0027)是一种小分子真菌细胞色素P450家族成员51 (fungal CYP51A1)抑制剂。它可用于治疗真菌感染、皮肤和肌肉骨骼疾病,可用于研究外阴阴道念珠菌病、Chagas病和泌尿生殖系统疾病。 | |||
TN6963 |
Hentriacontane
|
NF-κB | NF-κB |
Hentriacontane 是一种天然产物,具有多种药理作用,包括抗炎、抗肿瘤和抗菌活性。 | |||
T0484 |
Deracoxib
SC 46,SC 046,地拉考昔,SC 59046 |
Apoptosis; COX | Apoptosis; Immunology/Inflammation; Neuroscience |
Deracoxib (SC 46) 是非甾体、非麻醉性抗炎药。 它也是选择性 cyclooxygenase-2 抑制剂,IC50 值:70 至 150 μM,抑制 3 种骨肉瘤细胞系。 | |||
T50005 |
Sertaconazole
|
Antifungal | Microbiology/Virology |
Sertaconazole 是一种广谱抗真菌药。 | |||
T11864 |
Iptacopan
LNP023 |
Others | Others |
Iptacopan (LNP023) 是一种与factor B 亲和力较高的抑制剂。 | |||
TP1031 |
Tetracosactide
Tetracosactrin,替可克肽 |
Others | Others |
Tetracosactide (Tetracosactrin) 是一种肾上腺皮质激素 (ACTH) 的类似物,能够刺激肾上腺皮质激素分泌。 | |||
T29328 |
21-deacetyldeflazacort
|
Others | Others |
21-deacetyldeflazacort 是 Deflazacort 的代谢物,它是一种全身性皮质类固醇和泼尼松龙的衍生物。 | |||
T5377 |
Dimethyl itaconate
|
Others | Others |
Dimethyl itaconate 是一种化学试剂,用于合成功能化 2-异恶唑啉,用于基于片段的药物发现。 | |||
T9511 |
Monoethyl itaconate
|
Others | Others |
Monoethyl itaconate 是一种可用于聚合反应的自由基。 | |||
T26109 |
Robenacoxib
Onsior |
COX | Immunology/Inflammation; Neuroscience |
Robenacoxib (Onsior) 是一种对环氧化酶-2 有很强的选择性的非甾体化合物,具有抗炎活性。 | |||
T7670 |
Mavacoxib
|
COX | Immunology/Inflammation; Neuroscience |
Mavacoxib 是口服长效环氧合酶 2 选择性抑制剂,是长效的非甾体类抗炎药,用于犬退化性关节病相关的炎疼及痛症的研究。 | |||
T10239 |
Acolbifene
阿考比芬,EM-652,SCH 57068 |
Estrogen Receptor/ERR | Endocrinology/Hormones |
Acolbifene (SCH 57068) 是一种选择性雌激素受体拮抗剂,对雌二醇诱导的 ERα 和 ERβ 转录活性的 IC50 分别为 2 nM 和 0.4 nM。 Acolbifene 显示出抗癌特性。 | |||
T2319 |
Acotiamide monohydrochloride trihydrate
Acotiamide hydrochloride,YM-443 HCl,盐酸阿考替胺,Z-338 HCl |
AChE | Neuroscience |
Acotiamide monohydrochloride trihydrate (Z-338 HCl) 是一种首创的、具有口服活性的胃肠动力药。它通过促毒蕈碱受体拮抗作用和乙酰胆碱酯酶(AChE)抑制作用增强肠神经元释放的乙酰胆碱,从而增强胃排空和胃部适应性,有潜力用于功能性消化不良的研究。 | |||
T6211 |
Posaconazole
泊沙康唑,SCH 56592,POS |
Antifungal | Microbiology/Virology |
Posaconazole (POS) 是一种甾醇 C14ɑ 去甲基化酶的三唑类广谱抑制剂,IC50值为 0.25 nM,具有抗真菌作用。 | |||
T76883 |
Talacotuzumab
CSL 362,JNJ 56022473 |
Immunology/Inflammation related; Interleukin | Immunology/Inflammation |
Talacotuzumab (JNJ 56022473) 是一种含有修饰的 Fc 结构的IgG1 型完全人源化的 CD123 中和单克隆抗体。Talacotuzumab 对 CD123、CD32b/c、CD16-158F、CD16-158V 具有很高的亲和力, KD 分别为 0.43 nM、188 nM、46 nM、16.8 nM。Talacotuzumab 通过抑制 IL-3 与 CD123 结合进而抑制靶细胞中的 IL-3 信号传导。Talacotuzumab 诱导 Fc 区发生突变以增加对 CD16 (FcγRIIIa) 的亲和力,从而加强抗体依赖性细胞介导的细胞毒性 (ADCC)。Talacotuzumab 急性髓性白血病 (AML) 异种移植小鼠模型中抑制白血病细胞生长。 | |||
T40042 |
Evifacotrep
|
TRP/TRPV Channel | Membrane transporter/Ion channel |
Evfacotrep 是一种有效的短期瞬态受体电位通道5 拮抗剂。Evfacotrep 可用于神经系统疾病的研究。 | |||
T16727 |
Relacorilant
CORT 125134 |
Glucocorticoid Receptor | Endocrinology/Hormones |
Relacorilant 是一种选择性和口服生物可利用的糖皮质激素受体拮抗剂(HepG2 TAT 试验中的 Kis 为 7.2 nM,在基于细胞的试验中对大鼠、人和猴糖皮质激素受体的 Kis 分别为 12、81.2、210 nM)。 它具有治疗库欣综合征的潜力。 | |||
T5966 |
Hexaconazole
己唑醇,(-)-Hexaconazol |
Reactive Oxygen Species; Antifungal | Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB |
Hexaconazole ((-)-Hexaconazol) 是一种广谱三唑类杀菌剂,通过抑制羊毛甾醇的细胞色素 P450 依赖性 14α-去甲基化来抑制麦角甾醇的生物合成,从而导致真菌细胞膜的破坏和细胞死亡。 | |||
T4580 |
4-Octyl itaconate
4-辛基衣康酸,衣康酸盐 |
Nrf2 | Immunology/Inflammation |
4-Octyl Itaconate 是 Itaconate 衍生物,具有细胞渗透性,Itaconate 是一种抗炎代谢产物。4-Octyl Itaconate 可通过 KEAP1 的烷基化而活化 Nrf2,还可抑制 STING 的磷酸化。 | |||
T69467 |
Azacosterol
IMD760,Diazasterol |
Others | Others |
Azacosterol (Diazasterol) 是一种DHCR24抑制剂。Azacosterol 口服或腹腔注射后会在皮质神经元中发生一系列反应。 | |||
T5321 |
Itaconic anhydride
|
Others | Others |
Itaconic anhydride 是一种从可再生资源中获得的生物基材料。广泛用于金属助粘剂、合成树脂改良剂、酯化剂、除草剂、杀虫剂。 | |||
T19805 |
Benoxacor
BRN-4190275,解草酮,BRN 4190275,BRN4190275 |
Others | Others |
Benoxacor (BRN-4190275) 是一种惰性农业化学品。它作为一种除草剂安全剂,可保护作物免受除草剂毒性。 | |||
T26892 |
Braco-19
|
Apoptosis; HIV Protease; Telomerase | Apoptosis; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome |
Braco-19 是一种端粒酶/端粒抑制剂,具有抗 HIV-1活性。Braco-19 是一种四联体 (GQ) 结合配体,可抑制肿瘤生长,抑制细胞凋亡。Braco-19 也是一种 HAdV 病毒复制抑制剂,可用于研究 HIV 感染和人疱疹病毒感染。 | |||
T9189 |
Iptacopan hydrochloride
Iptacopan HCl,LNP023 hydrochloride |
Complement System | Immunology/Inflammation |
Iptacopan hydrochloride (LNP023 hydrochloride) 是一种可口服、高效和高选择性的因子 B 抑制剂,IC50 为 10 nM。 LNP023 显示与人因子 B 的直接、可逆和高亲和力结合,KD 为 7.9 nM。 | |||
T12017 |
Methyllycaconitine citrate
MLA |
AChR | Neuroscience |
Methyllycaconitine citrate (MLA) 是一种可穿过血脑屏障的 α7 神经元烟碱乙酰胆碱受体(α7nAChR)拮抗剂,可用于研究神经系统疾病。 | |||
T12092 |
Monacolin J
Antibiotic MB 530A,Lovastatin diol lactone,辛伐他汀内酯二醇 |
HMG-CoA Reductase; Autophagy | Autophagy; Metabolism |
Monacolin J (Antibiotic MB 530A) 是一种胆固醇生物合成抑制剂,抑制 HMG-CoA 还原酶的活性。 | |||
T3510 |
Olumacostat Glasaretil
|
Acetyl-CoA Carboxylase | Metabolism |
Olumacostat glasaretil 是乙酰辅酶A 羧化酶的有效抑制剂。 | |||
T41302 |
Itaconate-alkyne
ITalk |
Others | Others |
Itaconate-alkyne (ITalk) 是一种生物正交探针,用于对炎症性巨噬细胞中的衣康酸进行定量和位点特异性化学蛋白质组学分析,并能够对其直接靶标进行生化评估和蛋白质组学分析。 | |||
T67152 |
Dacomitinib Intermediate 2
N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-nitroquinazolin-4-amine |
Others | Others |
Dacomitinib Intermediate 2 (N-(3-Chloro-4-fluorophenyl)-7-methoxy-6-nitroquinazolin-4-amine) 具有抗癌活性,可用于研究肺癌。 | |||
T39740 |
Acoramidis hydrochloride
AG10 hydrochloride,Alxn2060 hydrochloride |
Others | Others |
Acoramidis hydrochloride (Alxn2060 hydrochloride) 是具有口服活性的、选择性的甲状腺素转运蛋白 (TTR (transthyretin)) 的稳定剂,对野生型和 V1221 突变型均有效。Acoramidis hydrochloride 可用于转体甲状腺素淀粉样变性的研究。 | |||
T2333 |
Efinaconazole
KP-103,艾氟康唑 |
Antifungal | Microbiology/Virology |
Efinaconazole (KP-103) 是一种三唑类抗真菌剂,抑制T. mentagrophytesSM-110和C. albicansATCC 10231菌株的MIC 值分别为 0.0039 μg/mL 和 0.00098 μg/mL | |||
T5336 |
Zacopride hydrochloride
|
Potassium Channel; 5-HT Receptor | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Zacopride hydrochloride 是5-HT3受体拮抗剂 (Ki:0.38 nM),也是5-HT4受体激动剂 (Ki:373 nM),具有抗焦虑作用。它对精神分裂症具有潜在的研究价值。 | |||
T6665 |
Sertaconazole nitrate
FI-7045,Ginedermofix,FI7056,Ertaczo,硝酸舍他康唑 |
Antibiotic; Antifungal | Microbiology/Virology |
Sertaconazole nitrate (FI-7045) 是一种局部广谱抗真菌药,可用于治疗浅表皮肤和粘膜感染。 | |||
T2483 |
Dacomitinib
达克替尼,PF-299804,PF-00299804,PF299 |
Apoptosis; EGFR | Angiogenesis; Apoptosis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Dacomitinib (PF299) 是一种不可逆的特异性ERBB 家族抑制剂,作用于EGFR、ERBB2和ERBB4的IC50分别为 6 nM、45.7 nM 和 73.7 nM。 | |||
T21907 |
PACOCF3
1,1,1-trifluoroheptadecan-2-one,Palmityltrifluoromethylketone |
Phospholipase | Metabolism |
PACOCF3 (Palmityltrifluoromethylketone) (Palmityltrifluoromethylketone) 是一种钙非依赖性的磷脂酶 A2 (phospholipase A2) 抑制剂,IC50为 3.8 μM。PACOCF3 改变肾小管细胞中的 Ca2+信号传导。 | |||
T23819 |
Braco-19 trihydrochloride
BRAC-O19,BRACO19 hydrochloride,BRACO19 3HCl,BRACO 19,BRACO19 HCl |
Telomerase | DNA Damage/DNA Repair |
Braco-19 trihydrochloride (BRACO19 3HCl) 是一种端粒酶抑制剂,可阻止端粒酶的加帽和催化作用。 Braco-19 trihydrochloride 抑制 HAdV 病毒复制。 | |||
T3583 |
Macozinone
PBTZ169 |
Antibacterial; DprE1 | Microbiology/Virology; Others |
Macozinone (PBTZ169) 是具有杀菌作用的苯并噻嗪酮,也有抗结核作用。它也是一种 DprE1有效抑制剂,可通过与活性位点 Cys387 残基形成共价键来抑制必需的黄素蛋白 DprE1。 | |||
T0284 |
Sulfogaiacol
guaiacolsulfonate,愈创木酚磺酸钾 |
Others; Antibacterial | Microbiology/Virology; Others |
Sulfogaiacol (guaiacolsulfonate) 是一种镇咳剂,可研究急性呼吸道感染。 | |||
T3267 |
Potassium guaiacolsulfonate hemihydrate
愈创木酚磺酸钾水合物,Potassium guaiacolsulfonate,Potassium 4-guaiacolsulfonate hemihydrate,愈创木酚磺酸钾 |
Antibacterial; Antibiotic | Microbiology/Virology |
Potassium guaiacolsulfonate hemihydrate (Potassium guaiacolsulfonate) 是一种芳香族磺酸,在医药中用作祛痰剂,可治疗急性呼吸道感染。它可松弛粘液,与其他药物合用,可治疗普通感冒、感染或过敏引起的咳嗽。 | |||
T6574 |
Lumiracoxib
Prexige,罗美昔布,COX-189 |
COX | Immunology/Inflammation; Neuroscience |
Lumiracoxib (Prexige) 是强选择性有口服活性的 COX-2抑制剂,Ki 值为 0.06 μM。它是非选择性非甾体抗炎试剂,具有抗炎和解热活性,可用于骨关节炎和骨癌研究。 | |||
T12654 |
(Rac)-Acolbifene
(Rac)-EM-652,EM-343,阿考比芬 |
Estrogen Receptor/ERR | Endocrinology/Hormones |
(Rac)-Acolbifene (EM-343) 是 Acolbifene 的外消旋形式。Acolbifene 是一种 estrogen receptor 拮抗剂。(Rac)-Acolbifene 显示出抗雌激素和雌激素活性。 (Rac)-Acolbifene 包含哌啶环,显示出良好的药理作用,RBA=380。 | |||
T20503 |
Elfacos EHP
2-ethylhexyl palmitate,棕榈酸辛酯 |
Others | Others |
Elfacos EHP (2-ethylhexyl palmitate) 是一种衍生自 2-乙基己醇和棕榈酸的脂肪酸酯,可用作化妆品配方。 | |||
T68145 |
Stacofylline
|
||
Stacofylline 是一种黄嘌呤衍生物,可用于治疗偏头疼。 | |||
T19965 |
Dacomitinib hydrate
PF 299804,:达克替尼一水合物,PF00299804,PF 00299804,PF-00299804,PF299804,PF-299804 |
EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Dacomitinib hydrate (PF 299804) 是泛表皮生长因子受体家族酪氨酸激酶的高选择性第二代小分子抑制剂。 Dacomitinib 特异性且不可逆地结合并抑制人 EGFR 亚型,从而抑制表达 EGFR 的肿瘤细胞的增殖和诱导细胞凋亡。 | |||
T20152 |
Tetraconazole
M 14360,氟醚唑 |
||
Tetraconazole is an agent of pesticides. | |||
T124583 | 26-Desglucoavenacoside A | ||
26-Desglucoavenacoside A 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124583,CAS号为 59795-21-0。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1923 |
Mesaconine
|
IL Receptor; NF-κB | Immunology/Inflammation; NF-κB |
Mesaconine 是来自 Aconitum carmichaelii Debx 的一种成分。Mesaconine 具有心脏作用和抗 NF-κB 活性。 Mesaconine 可能是麻黄附子细辛汤抗炎和免疫抑制的部分物质基础。 | |||
T3761 |
1-Octacosanol
n-Octacosanol,二十八烷醇,Montanyl alcohol,Cluytyl alcohol,Octacosanol,Octacosyl alcohol,Octanosol |
Others | Others |
1-Octacosanol (Octanosol) 是直链脂肪族 28 碳脂肪醇,具有抗疲劳作用。 | |||
T8111 |
Triacontanoic Acid
蜂花酸,Melissic acid A |
Others | Others |
Triacontanoic Acid (Melissic acid A) 是一种超长链脂肪酸。 | |||
T5S1891 |
Flaconitine
乙酰乌头碱,3-Acetylaconitine,Acetylaconitine |
Others; NF-κB | NF-κB; Others |
Flaconitine (Acetylaconitine) 是一种 NF-κB 抑制剂,是一种生物碱。 | |||
T6S1884 |
Benzoylhypaconine
苯甲酰次乌头碱,Benzoylhypacoitine,苯甲酰次乌头原碱 |
Others | Others |
Benzoylhypaconine (Benzoylhypacoitine) 是来自 Aconitum 中的一种单酯生物碱,也是Aconitum 的主要药理和毒性成分。 | |||
T4525 |
Citraconic acid
2-Methylmaleic Acid,柠康酸,Cis-Methylbutenedioic Acid |
Endogenous Metabolite | Metabolism |
Citraconic acid (2-Methylmaleic Acid) 是由马来酸在2-位具有甲基取代基的二羧酸。 | |||
T20880 |
Mesaconic acid
中康酸,Methylfumaric acid,Mesaconate,Kyselina mesakonova |
Others | Others |
Mesaconic acid (Methylfumaric acid) 被用作阻燃剂,因为最近的研究表明这种酸是富马酸盐还原的竞争性抑制剂。 | |||
T7936 |
Benzopinacole
|
Others | Others |
Benzopinacole 是一种抗阿米巴药物,可作为中间体合成多种化合物。 | |||
TN1725 |
Hederacolchiside E
革叶常春藤皂苷E |
Beta Amyloid; ROS | Immunology/Inflammation; Neuroscience |
Hederacolchiside E 具有抗氧化活性,并通过调节氧化应激在阿尔茨海默病 (AD) 模型中显示神经保护作用。 Hederacolchiside E 对亚油酸乳液的脂质过氧化具有抑制作用。 Hederacolchiside E 可能通过阻断缓激肽或其他炎症介质发挥其抗炎作用。 | |||
T6S1880 |
Benzoylaconine
苯甲酰乌头原碱,Pikraconitin,Isaconitine,Benzoylaconitine |
Others | Others |
Benzoylaconine (Isaconitine) 是一种中药附子生物碱。 | |||
TN7017 |
Tetracosane
|
Others | Others |
Tetracosane 是从孟加拉国药用植物 Acrostichum aureum 中分离出来的天然产物。 | |||
T5765 |
ranaconitine
羟基高乌碱,7-羟基高乌甲素 |
Apoptosis; Others | Apoptosis; Others |
Ranaconitine 是从高乌头中分离得到的一种二萜生物碱,具有心脏毒性。 | |||
T4S1881 |
Aconine
乌头原碱,Jesaconine |
Others; NF-κB | NF-κB; Others |
Aconine (Jesaconine) 是一种退热药,有胃麻醉作用,能够抑制核因子 κB 受体活化剂配体诱导的 NF-κB 激活。 | |||
T8166 |
Pennogenin 3-O-beta-chacotrioside
偏诺皂苷元-3-O-Α-L-吡喃鼠李糖-(1→4)[Α-L-吡喃鼠李糖基](1→2)-Β-D-葡萄糖苷 |
Autophagy | Autophagy |
Pennogenin 3-O-beta-chacotrioside 是从七叶一枝花中分离得到的一种天然产物,具有抗结肠癌活性。它可以调节自噬,增加自噬相关蛋白 LC3 和 Beclin-1 的表达。 | |||
TN1754 |
Hypaconine
|
Others | Others |
Hypaconine 是一种 C19-二萜生物碱,从乌头和飞燕草属中分离出来得到。 它表现出强烈的心脏活性。 | |||
T7095 |
Hexacosanoic acid
二十六酸,Cerotic acid |
Endogenous Metabolite | Metabolism |
Hexacosanoic acid 是长链脂肪酸,与多种疾病有关(如肾上腺脑白质营养不良,肾上腺髓鞘病和动脉粥样硬化)。 | |||
TN1833 |
Karacoline
|
NF-κB | NF-κB |
Karacoline 是发现于植物Aconitum kusnezoffii 中的一种二萜生物碱,通过 NF-κB 信号通路,抑制椎间盘退变中细胞外基质的降解。 | |||
T7986 |
Methyl tetracosanoate
|
Others | Others |
Methyl tetracosanoate 常作为一种标准品,用于色谱分析实验中。 | |||
T8137 |
(Z)-Aconitic acid
顺乌头酸,顺式乌头酸,Cls-Aconitic acid |
Others; Endogenous Metabolite | Metabolism; Others |
(Z)-Aconitic acid 是 Aconitic acid 的顺式异构体。它是三羧酸循环中柠檬酸盐异构化为异柠檬酸盐的中间产物。 | |||
T8379 |
Aconitic Acid
|
Others | Others |
Aconitic acid 是一种有机酸。 | |||
T1011 |
Itraconazole
伊曲康唑,R51211 |
P450; Hedgehog/Smoothened; Antibiotic; Autophagy; Antifungal | Autophagy; GPCR/G Protein; Metabolism; Microbiology/Virology; Stem Cells |
Itraconazole (R51211) 是三唑类抗真菌药,也是口服活性的Hedgehog 信号通路拮抗剂,IC50约为 800 nM。它也是 oxysterol-binding protein 抑制剂。它抑制羊毛甾醇 14α-脱甲基酶,从而抑制羊毛甾醇向麦角固醇的氧化转化。它有抗癌和抗血管作用。 | |||
T2806 |
Lappaconitine
高乌甲素,(+)-Lappaconitine |
P2X Receptor; Sodium Channel | Membrane transporter/Ion channel; Neuroscience |
Lappaconitine ((+)-Lappaconitine) 是从高乌头中分离得到的一种天然产物,可用于缓解疼痛的研究。 | |||
T3372 |
Dipsacoside B
|
Others | Others |
Dipsacoside B 是主要的具有生物活性的皂素,可用作标志物。 | |||
T1716 |
Echinacoside
|
Reactive Oxygen Species; Wnt/beta-catenin | Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells |
Echinacoside 是一种从Cistanche salsa 中分离的苯乙醇类化合物,抑制Wnt/β-catenin 信号通路。它能够激活 Trk 受体及其下游信号通路而起到神经保护作用,还具有显著的抗骨质疏松作用。 | |||
TN3273 | 8-Deacetylyunaconitine | Others | Others |
8-Deacetylyunaconitine 是一种源自乌头的二萜生物碱。 | |||
T3764 |
1-Triacontanol
Myricyl alcohol,1-Triacontanol,三十烷醇,Melissyl alcohol,Well-Bloom,Miraculan,Lithospermoside,triacontan-1-ol |
Others | Others |
1-Triacontanol (Melissyl alcohol) 是天然存在的植物生长调节剂。它是饱和长链醇,能够促进许多植物的生长。 | |||
T2P2937 |
Nonacosane
|
Others; Antibacterial | Microbiology/Virology; Others |
Nonacosane 是从Baphia massaiensis 分离的,是一种由 29 个碳原子组成的直链烷烃,具有植物代谢物和挥发油成分的作用。 | |||
T8192 |
Pentacosanoic acid
|
Others; Endogenous Metabolite | Metabolism; Others |
Pentacosanoic acid 是戊酸的共轭酸,是 25 碳长链饱和脂肪酸。 | |||
TN1421 |
Bacopaside II
|
Apoptosis | Apoptosis |
Bacopaside II 是药用植物Bacopa monnieri 的提取物,可阻断Aquaporin-1 (AQP1)水通道并阻碍表达 AQP1 的细胞迁移,还诱导细胞周期停滞和细胞凋亡。 | |||
T5805 |
Guvacoline hydrochloride
1,2,5,6-四氢吡啶-3-甲酸甲酯盐酸盐,Norarecoline hydrochloride,去甲槟榔碱 |
AChR | Neuroscience |
Guvacoline hydrochloride (Norarecoline hydrochloride) 是从三药槟榔中发现的一种吡啶生物碱,可作为心房和回肠的毒蕈碱激动剂。 | |||
TN1420 |
Bacopaside I
|
Others | Others |
Bacopaside I 是一种皂苷,分离自 Bacopa monniera 中,具有抗氧化活性和清除自由基的功能,有抗抑郁作用。 | |||
T41078 |
Lipopolysaccharides, Escherichiacoli
Lipopolysaccharide, E. coli O111:B4 |
Others | Others |
Lipopolysaccharides, Escherichiacoli (E. coli O111:B4)是革兰阴性菌外膜的大分子成分,由脂质a、寡糖核心和o -特异性多糖(O-antigen) 3个区域组成。 | |||
T3790 |
Hederacoside D
常春藤苷 D,常春藤苷D;常春藤皂苷D |
TNF | Apoptosis |
Hederacoside D 是从常春藤中分离到的皂苷,具有很高的生物活性。 | |||
T3021 |
Bulleyaconitine A
草乌甲素,Bulleyaconi cine A |
Sodium Channel | Membrane transporter/Ion channel |
Bulleyaconitine A (Bulleyaconi cine A) 是一种分离自乌头属植物的抗炎活性化合物,也可用于缓解疼痛的研究。 | |||
T4837 |
Itaconic acid
methylene-butanedioicaci,衣康酸 |
Others; Endogenous Metabolite | Metabolism; Others |
Itaconic acid (methylene-butanedioicaci) 是聚合物,化学物质和燃料的合成前体。Itaconic acid 可由真菌合成。它也是巨噬细胞特异性代谢产物。它介导巨噬细胞代谢和腹膜肿瘤之间的串扰。 | |||
T4861 |
trans-Aconitic acid
|
ATPase; Endogenous Metabolite | Membrane transporter/Ion channel; Metabolism |
trans-Aconitic acid 是反式丙酮酸2-甲基转移酶的底物,存在于正常人尿液中,大量存在于 Reye 综合征和有机酸尿症。 | |||
T2P2806 |
Hederacolchiside A1
黑海常春藤苷A1,革叶常春藤皂苷 A1,Raddeanoside R13 |
Apoptosis; ERK; MEK; Akt; PI3K; Parasite; mTOR | Apoptosis; Cytoskeletal Signaling; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling |
Hederacolchiside A1 (Raddeanoside R13) 是从白头翁中分离的一种有抗利什曼原虫和抗肿瘤增殖活性的天然产物。 | |||
T2S2043 |
Dracorhodin perchlorate
Dracorhodin perochlorate,血竭素高氯酸盐,Dracohodin perochlorate |
Apoptosis; Others | Apoptosis; Others |
Dracorhodin perchlorate 是来源于中药血竭的一种天然产物。它抑制细胞生长,并以剂量和时间依赖性方式诱导成纤维细胞凋亡,将细胞周期阻滞在 G1 期,可作为抗乳腺癌的候选药物。 | |||
T6S0630 |
Hypaconitine
|
P450; TNF | Apoptosis; Metabolism |
Hypaconitine 是从乌头属种分离的一种高毒性成分,可研究风湿病。 | |||
T6560 |
Lappaconitine hydrobromide
氢溴酸高乌甲素,Lappaconite HBr,Allapinine |
Others | Others |
Lappaconitine hydrobromide (Allapinine) 是天然生物碱类化合物,具有抗心律失常作用。 | |||
T3426 |
Bacoside A
|
MMP; Others; TNF; Dopamine Receptor; NOS; ROS | Apoptosis; GPCR/G Protein; Immunology/Inflammation; Neuroscience; Others; Proteases/Proteasome |
Bacoside A has a possible anticancer activity that could be inducing cell cycle arrest and apoptosis through Notch pathway in GBM in vitro. It exerts cytoprotective efficacy by attenuation of ROS generated through oxidative stress by an increase in the concentration of antioxidant enzymes and sustain membrane integrity which leads to restoring the damage caused by tBHP. Bacoside A can able to inhibit the progression of Experimental Autoimmune Encephalomyelitis (EAE) may be by the inhibition of i... | |||
TN6753 |
1-TETRACOSANOL
二十四醇,Tetracosanol,LIGNOCERYL ALCOHOL |
Others | Others |
1-Tetracosanol (LIGNOCERYL ALCOHOL) 是从多根火龙果 Hylocereus polyrhizus 中提取的天然成分。 | |||
T8121 |
Octacosanoic acid
|
Anti-infection | Microbiology/Virology |
Octacosanoic acid 具有抗血小板和抗血栓作用。 | |||
TN6751 |
1-HEXACOSANOL
|
NPC1L1; AMPK | Chromatin/Epigenetic; Membrane transporter/Ion channel; PI3K/Akt/mTOR signaling |
1-HEXACOSANOL 激活 AMPK 和肝脏自噬并抑制 SREBP2,导致降胆固醇活性和肝脏脂肪变性的改善。 | |||
TN1425 |
Bacoside A3
苦艾素A3,白花猪母菜甙 A3 |
ATPase; ROS; P-gp | Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience |
Bacoside A3 是一种天然的三萜皂苷,是Bacopa monnieri 的主要活性成分之一,显示出神经保护活性。 | |||
T4S1876 |
3-Deoxyaconitine
|
Sodium Channel | Membrane transporter/Ion channel |
3-Deoxyaconitine 是一种二萜类生物碱,对钠离子通道有激活作用。 | |||
T5S1889 |
Yunaconitine
Guayewuanine B,滇乌头碱 |
Others | Others |
Yunaconitine (Guayewuanine B) 是一种乌头类生物碱,具有剧毒。 | |||
T32570 |
Lappaconine
20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol,O(sup 1)-Methyllappaconidine |
Others | Others |
Lappaconine (20-ethyl-1,14,16-trimethoxyaconitane-4,6,8-triol) 衍生自去甲二萜生物碱。 | |||
TN7026 |
Acorus gramineus, ext.
|
Others | Others |
Acorus gramineus, ext. | |||
T6S1885 |
Benzoylmesaconine
Mesaconine 14-benzoate,苯甲酰新乌头原碱 |
Others | Others |
Benzoylmesaconine (Mesaconine 14-benzoate) 是乌头汤最丰富的组分。其中乌头汤可用于研究类风湿性关节炎。 | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-00491 |
Kallikrein 15/KLK15 Protein, Human, Recombinant (hFc)
ACO,kallikrein-related peptidase 15,HSRNASPH |
Human | HEK293 Cells |
Kallikrein 15/KLK15 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 53.1 kDa and the accession number is Q9H2R5-1. | |||
TMPY-05289 |
Kallikrein 15/KLK15 Protein, Human, Recombinant (His)
ACO,HSRNASPH,kallikrein-related peptidase 15 |
Human | HEK293 Cells |
Kallikrein 15/KLK15 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 27.8 kDa and the accession number is Q9H2R5-1. | |||
TMPY-02787 |
Aconitase 2 Protein, Mouse, Recombinant (His & GST)
Aco-2,D10Wsu183e,aconitase 2, mitochondria... |
Mouse | Baculovirus Insect Cells |
Aconitase 2 Protein, Mouse, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 110 kDa and the accession number is Q99KI0. | |||
TMPY-02481 |
ACOX1 Protein, Human, Recombinant (His)
PALMCOX,ACOX,SCOX,acyl-CoA oxidase 1, palmitoyl |
Human | Baculovirus Insect Cells |
Peroxisomal acyl-coenzyme A oxidase 1(ACOX1 or AOX) is the first enzyme of the fatty acid beta-oxidation pathway and belongs to the Acyl-CoA oxidase family. Human liver peroxisomes contain two acyl-CoA oxidases, namely, palmitoyl-CoA oxidase (ACOX1/AOX) and a branched chain acyl-CoA oxidase. The palmitoyl-CoA oxidase (ACOX1/AOX) oxidizes the CoA esters of straight chain fatty acids and prostaglandins and donates electrons directly to molecular oxygen, thereby producing H2O2. Human ACOX1/AOX is a... | |||
TMPH-02585 |
ACOD1 Protein, Mouse, Recombinant (His & Myc)
Cis-aconitate decarboxylase,Cis-aconitic a... |
Mouse | Baculovirus Insect Cells |
Cis-aconitate decarboxylase that catalyzes production of itaconate and is involved in the inhibition of the inflammatory response. Acts as a negative regulator of the Toll-like receptors (TLRs)-mediated inflammatory innate response by stimulating the tumor necrosis factor alpha-induced protein TNFAIP3 expression via reactive oxygen species (ROS) in LPS-tolerized macrophages. Involved in antimicrobial response of innate immune cells; ACOD1-mediated itaconic acid production contributes to the anti... | |||
TMPY-01140 |
ACOT13/THEM2 Protein, Human, Recombinant (His)
THEM2,HT012,ACOT13,PNAS-27,acyl-CoA thioesterase 13 |
Human | E. coli |
The metabolites of fatty acyl-Coenzyme A (CoA) and metabolic enzymes contribute to lipid biosynthesis, signal transduction, and gene transcription. Members of the acyl-CoA thioesterase (Acot) gene family hydrolyze fatty acyl-CoAs, but their biological functions remain incompletely understood. Thioesterase superfamily member 2 (Them2; synonym Acot13) is enriched in oxidative tissues, associated with mitochondria, and relatively specific for long chain fatty acyl-CoA substrates. Using Them2(-/-) m... | |||
TMPY-02482 |
Aconitase 1 Protein, Human, Recombinant (His)
HEL60,IRP1,ACONS,aconitase 1, soluble,IREB... |
Human | Baculovirus Insect Cells |
Aconitase 1(ACO1) or IRP1 is one member of the aconitase family that contains a diverse group of iron-sulphur(Fe-S) isomerases and two types of iron regulatory protein. Aconitase exits in two forms: one is soluble and the other is mitochondrial. ACO1 is the soluble existing form, and the mitochondrial form is ACO2. Residues from all three N-terminal domains and the larger C-terminal domain contribute to the active site region. When the enzyme is activated, it gains an additional iron atom. ACO1 ... | |||
TMPH-02825 |
ACOX1 Protein, Mouse, Recombinant (Myc)
AOX,Peroxisomal fatty acyl-CoA oxidase,EC:1.3.3.6,Peroxisoma... |
Mouse | E. coli |
Catalyzes the desaturation of acyl-CoAs to 2-trans-enoyl-CoAs. First enzyme of the fatty acid beta-oxidation pathway.; Shows highest activity against medium-chain fatty acyl-CoAs and activity decreases with increasing chain length.; Is active against a much broader range of substrates and shows activity towards very long-chain acyl-CoAs. Is twice as active as isoform 1 against 16-hydroxy-palmitoyl-CoA and is 25% more active against 1,16-hexadecanodioyl-CoA. | |||
TMPH-01098 |
ACOD1 Protein, Human, Recombinant (His)
Aconitate decarboxylase 1,IRG1,Cis-aconita... |
Human | E. coli |
ACOD1 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 58.6 kDa and the accession number is A6NK06. | |||
TMPY-02545 |
Aconitase 2 Protein, Human, Recombinant (His & GST)
ACONM,ICRD,aconitase 2, mitochondrial |
Human | Baculovirus Insect Cells |
Aconitase 2 Protein, Human, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag. The predicted molecular weight is 110 kDa and the accession number is Q99798. |