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513

抑制剂 & 化合物

49

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Cat. No. Product Name Target Signaling Pathways
T22124 Oleoyl Serotonin

TRP/TRPV Channel Membrane transporter/Ion channel
Oleoyl Serotonin 是 hTRPV1 的拮抗剂,IC50(Human TRPV1) 为 2.57 μM。
T34617 Serotonin adipinate

Serotonin adipinate can be used to treat serotonin insufficiency for surgical patients.
T22582 Arachidonyl serotonin

Others Others
Dual FAAH inhibitor/TRPV1 antagonist
T23086 NPEC-caged-serotonin

Others Others
5-HT receptor agonist
T8441 Lerisetron

5-HT Receptor GPCR/G Protein; Neuroscience
Lerisetron 是5-HT3拮抗剂,与 5-HT3受体具有高亲和力(pKi:9.2)。它对尿烷麻醉大鼠的 5-HT 引发的反射性心率过缓具有抑制作用。
T8708 Paroxetine

Serotonin Transporter Neuroscience
Paroxetine 是选择性血清素再摄取抑制剂,是苯基哌啶的衍生物。 它对于甲肾上腺素摄取抑制功能较弱,但比该位点其他SSRIs 更有效。
T21629 Loxapine

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Loxapine 是 D2DR 和 D4DR 抑制剂和5-羟色胺能受体拮抗剂,是一种抗精神病药物,主要用于治疗精神分裂症。
T22453 Venlafaxine

Wy 45030,文拉法辛

Serotonin Transporter Neuroscience
Venlafaxine (Wy 45030) 是一种口服有效的 5-羟色胺 (5-HT)/去甲肾上腺素 (NE) 重摄取的双重抑制剂,具有抗抑郁活性。
T11075 Donitriptan

5-HT Receptor GPCR/G Protein; Neuroscience
Donitriptan 是一种 5-HT 受体激动剂,对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。
T37015 Iprindole

5-HT Receptor GPCR/G Protein; Neuroscience
Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].
T1566 Aripiprazole

阿立哌唑,OPC-14597

5-HT Receptor GPCR/G Protein; Neuroscience
Aripiprazole (OPC-14597) 是血清素受体 5-HT1A 和多巴胺 D2 受体的部分激动剂,还用作突触后拮抗剂和血清素受体 5-HT2A 的拮抗剂。
T1092 Zolmitriptan

佐米曲普坦,311C90,BW-311C90

5-HT Receptor GPCR/G Protein; Neuroscience
Zolmitriptan (311C90) 是一种5-HT1B/1D 受体部分激动剂,可用于偏头痛的研究,对 5-HT1B、5-HT1D、5-HT1F 受体的Ki 分别为 5.01、0.63 和 63.09 nM。
T12232 Nitroxazepine

CIBA 2330Go

Serotonin Transporter Neuroscience
Nitroxazepine (CIBA 2330Go) 是三环抗抑郁化合物,是一种 5-羟色胺去甲肾上腺素再摄取抑制剂,可用于抗抑郁的研究。
T8666 Naratriptan

5-HT Receptor GPCR/G Protein; Neuroscience
Naratriptan 是一种5-HT1受体选择性激动剂,可作用于偏头疼。
T28531 Facinicline hydrochloride

RG3487

5-HT Receptor; AChR GPCR/G Protein; Neuroscience
Facinicline hydrochloride (RG3487) 是一种口服有效的烟碱α7 receptor 部分激动剂,对人 nAChR 的 Ki 值为 6 nM。它可改善啮齿类动物的认知和感觉运动门控。它与5-HT3受体结合的 Ki 为 1.2 nM。
T37197 5-HT1A modulator 2 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
5-HT1A modulator 2 hydrochloride 是 8-OH-DPAT 的一种衍生物,是5-HT1A 的调节剂,Ki 为 53 nM。
T2395 Vortioxetine

沃替西汀,Lu AA 21004

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Vortioxetine (Lu AA 21004) 是5-HT1A、5-HT1B、5-HT3A、5-HT7受体和 5-羟色胺转运体抑制剂,Ki 值分别为 15、33、3.7、19 和 1.6 nM。它作为抗抑郁药,用于治疗重度抑郁症。
T0031L2 Ziprasidone

齐拉西酮,Geodon,Zeldox,CP-88059

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ziprasidone (Geodon) 是一种联合的 5-HT(5-羟色胺)和多巴胺受体拮抗剂,具有强大的抗精神病活性。它是去甲肾上腺素再摄取抑制剂,对大鼠和人的5-HT1A,5-HT2A 和多巴胺 D2 受体有很高的亲和力。
T0472 Venlafaxine hydrochloride

Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Venlafaxine hydrochloride (Wy 45030 hydrochloride) 是一种口服有效的 5-羟色胺 (5-HT)/去甲肾上腺素 (NE) 重摄取的双重抑制剂,具有抗抑郁活性。
T5179 AVN-492

AVN492

5-HT Receptor GPCR/G Protein; Neuroscience
AVN-492 是一种有效的选择性 5-HT6R 拮抗剂,Ki 为 91 pM。
T11720 JNJ-18038683

5-HT Receptor GPCR/G Protein; Neuroscience
JNJ-18038683 是 5-羟色胺受体 7 拮抗剂,HEK293 细胞中检测出其对大鼠和人类 5-羟色胺受体 7 的pKi 值分别为 8.19和8.20。
T1279 Vilazodone

维拉佐酮,SB659746A,EMD 68843

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Vilazodone (SB659746A) 是一种可口服的选择性 5 -羟色胺再摄取抑制剂 (SSRI) 和部分5-HT1A 受体激动剂。它有抗抑郁作用,可用于抑郁症和情绪性疾病的研究。
T2459 BRL 54443

BRL54443

5-HT Receptor GPCR/G Protein; Neuroscience
BRL 54443 是一种有效的 5-HT1E/1F 受体激动剂,pKi 值分别为 8.7 和 8.9。
T2599 Pirenperone

5-HT Receptor GPCR/G Protein; Neuroscience
Pirenperone 是5-HT2血清素受体拮抗剂,具有一定抗焦虑作用。
T4274 Melitracen hydrochloride

盐酸美利曲辛,盐酸美力他欣,Thymeol hydrochloride,Melixeran

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Melitracen hydrochloride (Thymeol hydrochloride) 是一种可口服的双相抗抑郁药和抗焦虑药。它可以通过突触前膜抑制去甲肾上腺素和5-羟色胺(5-HT)的吸收,从而诱导突触空间中单胺递质的增加。
T6232 Vilazodone Hydrochloride

盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl

Others; 5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience; Others
Vilazodone Hydrochloride (EMD 68843) 是 5-HT1A 受体和特异性 5-羟色胺再摄取抑制剂(SSRI) 的部分激动剂,用于治疗重度抑郁症。
T14049 5-FAM SE

Others Others
5-FAM SE 是单一异构体,是用于标记肽、蛋白质和核苷酸的荧光标记试剂。它能够与胺反应,产生稳定的胺结合物。
T16669 PRX-08066

5-HT Receptor GPCR/G Protein; Neuroscience
PRX-08066是5-HT 受体2B 拮抗剂,IC50为3.4 nM,可诱​​导肺动脉的选择性血管舒张。
T5387 LP-211

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
LP-211 是一种可透过血脑屏障的选择性5-HT7受体激动剂,Ki 值为 0.58 nM,选择性高于 5-HT1A 受体和 D2受体,Ki 分别为188 和 142 nM。
T2428 TG6-10-1

5-HT Receptor; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
TG6-10-1 是一种 EP2 拮抗剂。
T5336 Zacopride hydrochloride

Potassium Channel; 5-HT Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Zacopride hydrochloride 是5-HT3受体拮抗剂 (Ki:0.38 nM),也是5-HT4受体激动剂 (Ki:373 nM),具有抗焦虑作用。它对精神分裂症具有潜在的研究价值。
T21029 Norfluoxetine Hydrochloride

Norfluoxetine HCl,去甲氟西汀

Others Others
Norfluoxetine Hydrochloride (Norfluoxetine HCl) 是氟西汀的活性代谢物。氟西汀是一种抗抑郁药。
T1412 Loxapine succinate

Daxolin,Loxapac,Cloxazepin,Loxapine succinate salt,丁二酸洛沙平,琥珀酸洛沙平

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Loxapine succinate (Loxapac) 是D2/D4多巴胺受体,5-羟色胺受体抑制剂,用于精神分裂症。
T22671 CJ 033466

5-HT Receptor GPCR/G Protein; Neuroscience
CJ 033466 是 5-HT4 受体 (EC50 = 9 nM) 的特异性部分激动剂,具有促胃动力作用。
T22921 LE 300

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
LE 300 是选择性多巴胺 D1 样受体拮抗剂,作用于人多巴胺 D1 和 D5 受体的Kis 分别为 1.9 nM 和 7.5 nM。在大鼠尾动脉实验中,它作用于5-HT2A 受体的pA2 为 8.32。
T3179 Eptapirone

F 11440

5-HT Receptor GPCR/G Protein; Neuroscience
Eptapirone (F 11440) 是一种高效且选择性的 5-HT1A 受体激动剂,具有显着的抗抑郁和抗焦虑潜力。
T17033 Temanogrel

APD791

5-HT Receptor GPCR/G Protein; Neuroscience
Temanogrel (APD791) 是一种高度选择性的 5-HT2A 受体拮抗剂,Ki 值为 4.9 nM。
T19680 Zotepine

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Zotepine 是一种抗精神病剂,是有效的5-HT2A、5-HT2C、组胺H1、α1-肾上腺素能和多巴胺D2受体拮抗剂,Kd 值分别为 2.6、3.2、3.3、7.3 和 8 nM。它在体内表现出抗抑郁和抗焦虑作用。
T8946 Indophagolin

P2X Receptor; 5-HT Receptor; Autophagy Autophagy; GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Indophagolin 是一种有效的含有二氢吲哚的自噬抑制剂,IC50 为 140 nM。它拮抗 Gq 蛋白偶联的 P2Y4、P2Y6和 P2Y11受体。它还拮抗嘌呤能受体 P2X4 以及 P2X1 和 P2X3,IC50 分别为 2.71、2.40 和 3.49 μM。
T7061 Duloxetine

Serotonin Transporter Neuroscience
Duloxetine 是一种 5 羟色胺-去甲肾上腺素重吸收 (serotonin-norepinephrine reuptake) 抑制剂,Ki=4.6 nM,可作用于广泛性焦虑症的研究。
T12847 SB-616234-A

SB-616234A

5-HT Receptor GPCR/G Protein; Neuroscience
SB-616234-A 是选择性的,口服有效的5-HT1B receptor 拮抗剂。SB-616234-A 具有抗焦虑和抗抑郁活性。
T12489 Pimethixene

Calmixen,匹美噻吨,Pimetixene

Dopamine Receptor; 5-HT Receptor; AChR; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Pimethixene (Calmixen) 是抗组胺和抗血清素剂,用作抗偏头疼剂。它是高效多靶点拮抗剂。
T0031 Ziprasidone hydrochloride monohydrate

齐拉西酮盐酸盐一水合物,盐酸齐拉西酮水合物,CP 88059

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ziprasidone hydrochloride monohydrate (CP 88059) 是一种联合 5-HT(5-羟色胺)和多巴胺受体拮抗剂,具有抗精神病活性的强效作用。它也是去甲肾上腺素再摄取抑制剂。
T3648 Hypidone hydrochloride

YL0919

5-HT Receptor GPCR/G Protein; Neuroscience
Hypidone hydrochloride (YL0919) 是一种新型抗抑郁候选药物,具有作为 5-HT1A 受体激动剂和选择性 5-羟色胺再摄取抑制剂的双重活性。
T0450 Fluoxetine

氟西汀,LY-110140

5-HT Receptor; Serotonin Transporter; MRP; Autophagy Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Fluoxetine (LY-110140) 是一种高度特异性的血清素摄取抑制剂,是选择性 5-羟色胺 (5-HT) 再吸收抑制剂。Fluoxetine 具有抗抑郁活性。
T22514 4F 4PP oxalate

5-HT Receptor GPCR/G Protein; Neuroscience
4F 4PP oxalate 是一种选择性5-HT2A 拮抗剂。
T7281 F-15599

5-HT Receptor GPCR/G Protein; Neuroscience
F-15599 是一种高度选择性的 G 蛋白偏向 5-HT1A 受体激动剂,Ki 值为 3.4 nM。
T22987 MK 212 hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
MK 212 monohydrochloride 是一种5-HT1C/5-HT2激动剂。它具有中枢作用,可刺激大脑皮层中的磷酸肌醇水解。
T2688 LY310762

LY310762 HCl

5-HT Receptor GPCR/G Protein; Neuroscience
LY310762 是 5-HT1D 受体拮抗剂,Ki 为 249 nM。
T21946 BIMU 8

5-HT Receptor GPCR/G Protein; Neuroscience
BIMU 8 是 5-HT4 的选择性激动剂,对野生型 5HT4 受体、T3.36A 和 W6.48A 突变体 5-HT4 的 EC50 分别为 18 nM、77 nM 和 540 nM。

化合物

Oleoyl Serotonin
Cat.No: T22124
Synonym:
Target: TRP/TRPV Channel
Serotonin adipinate
Cat.No: T34617
Synonym:
Target:
Arachidonyl serotonin
Cat.No: T22582
Synonym:
Target: Others
NPEC-caged-serotonin
Cat.No: T23086
Synonym:
Target: Others
Lerisetron
Cat.No: T8441
Synonym:
Target: 5-HT Receptor
Paroxetine
Cat.No: T8708
Synonym:
Target: Serotonin Transporter
Loxapine
Cat.No: T21629
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
Venlafaxine
Cat.No: T22453
Synonym: Wy 45030,文拉法辛
Target: Serotonin Transporter
Donitriptan
Cat.No: T11075
Synonym:
Target: 5-HT Receptor
Iprindole
Cat.No: T37015
Synonym:
Target: 5-HT Receptor
Aripiprazole
Cat.No: T1566
Synonym: 阿立哌唑,OPC-14597
Target: 5-HT Receptor
Zolmitriptan
Cat.No: T1092
Synonym: 佐米曲普坦,311C90,BW-311C90
Target: 5-HT Receptor
Nitroxazepine
Cat.No: T12232
Synonym: CIBA 2330Go
Target: Serotonin Transporter
Naratriptan
Cat.No: T8666
Synonym:
Target: 5-HT Receptor
Facinicline hydrochloride
Cat.No: T28531
Synonym: RG3487
Target: 5-HT Receptor, AChR
5-HT1A modulator 2 hydrochloride
Cat.No: T37197
Synonym:
Target: 5-HT Receptor
Vortioxetine
Cat.No: T2395
Synonym: 沃替西汀,Lu AA 21004
Target: 5-HT Receptor, Serotonin Transporter
Ziprasidone
Cat.No: T0031L2
Synonym: 齐拉西酮,Geodon,Zeldox,CP-88059
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Norepinephrine, Histamine Receptor
Venlafaxine hydrochloride
Cat.No: T0472
Synonym: Venlafaxine HCl,盐酸文拉法辛,Wy 45030 hydrochloride
Target: 5-HT Receptor, Serotonin Transporter
AVN-492
Cat.No: T5179
Synonym: AVN492
Target: 5-HT Receptor
JNJ-18038683
Cat.No: T11720
Synonym:
Target: 5-HT Receptor
Vilazodone
Cat.No: T1279
Synonym: 维拉佐酮,SB659746A,EMD 68843
Target: 5-HT Receptor, Serotonin Transporter
BRL 54443
Cat.No: T2459
Synonym: BRL54443
Target: 5-HT Receptor
Pirenperone
Cat.No: T2599
Synonym:
Target: 5-HT Receptor
Melitracen hydrochloride
Cat.No: T4274
Synonym: 盐酸美利曲辛,盐酸美力他欣,Thymeol hydrochloride,Melixeran
Target: Dopamine Receptor, 5-HT Receptor
Vilazodone Hydrochloride
Cat.No: T6232
Synonym: 盐酸维拉佐酮,SB659746A,EMD 68843,Vilazodone HCl
Target: Others, 5-HT Receptor, Serotonin Transporter
5-FAM SE
Cat.No: T14049
Synonym:
Target: Others
PRX-08066
Cat.No: T16669
Synonym:
Target: 5-HT Receptor
LP-211
Cat.No: T5387
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
TG6-10-1
Cat.No: T2428
Synonym:
Target: 5-HT Receptor, Prostaglandin Receptor
Zacopride hydrochloride
Cat.No: T5336
Synonym:
Target: Potassium Channel, 5-HT Receptor
Norfluoxetine Hydrochloride
Cat.No: T21029
Synonym: Norfluoxetine HCl,去甲氟西汀
Target: Others
Loxapine succinate
Cat.No: T1412
Synonym: Daxolin,Loxapac,Cloxazepin,Loxapine succinate salt,丁二酸洛沙平,琥珀酸洛沙平
Target: Dopamine Receptor, 5-HT Receptor
CJ 033466
Cat.No: T22671
Synonym:
Target: 5-HT Receptor
LE 300
Cat.No: T22921
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
Eptapirone
Cat.No: T3179
Synonym: F 11440
Target: 5-HT Receptor
Temanogrel
Cat.No: T17033
Synonym: APD791
Target: 5-HT Receptor
Zotepine
Cat.No: T19680
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Indophagolin
Cat.No: T8946
Synonym:
Target: P2X Receptor, 5-HT Receptor, Autophagy
Duloxetine
Cat.No: T7061
Synonym:
Target: Serotonin Transporter
SB-616234-A
Cat.No: T12847
Synonym: SB-616234A
Target: 5-HT Receptor
Pimethixene
Cat.No: T12489
Synonym: Calmixen,匹美噻吨,Pimetixene
Target: Dopamine Receptor, 5-HT Receptor, AChR, Histamine Receptor
Ziprasidone hydrochloride monohydrate
Cat.No: T0031
Synonym: 齐拉西酮盐酸盐一水合物,盐酸齐拉西酮水合物,CP 88059
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Norepinephrine, Histamine Receptor
Hypidone hydrochloride
Cat.No: T3648
Synonym: YL0919
Target: 5-HT Receptor
Fluoxetine
Cat.No: T0450
Synonym: 氟西汀,LY-110140
Target: 5-HT Receptor, Serotonin Transporter, MRP, Autophagy
4F 4PP oxalate
Cat.No: T22514
Synonym:
Target: 5-HT Receptor
F-15599
Cat.No: T7281
Synonym:
Target: 5-HT Receptor
MK 212 hydrochloride
Cat.No: T22987
Synonym:
Target: 5-HT Receptor
LY310762
Cat.No: T2688
Synonym: LY310762 HCl
Target: 5-HT Receptor
BIMU 8
Cat.No: T21946
Synonym:
Target: 5-HT Receptor
Cat. No. Product Name Target Signaling Pathways
TN2437 Serotonin

5-羟基色胺,5-hydroxytryptamine,血清素,五羟色胺,5-HT

Others; 5-HT Receptor; Endogenous Metabolite; Transferase GPCR/G Protein; Metabolism; Neuroscience; Others
Serotonin (5-hydroxytryptamine) 是 CNS 中的单胺神经递质和内源性5-HT 受体激动剂。它也是儿茶酚 O-甲基转移酶(COMT) 的抑制剂,Ki 值为 44 μM。
T2209 Serotonin hydrochloride

5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride

5-HT Receptor; Endogenous Metabolite; Transferase GPCR/G Protein; Metabolism; Neuroscience
Serotonin hydrochloride (Serotonin HCl) 是一种内源性 5-HT 受体激动剂、CNS 中的单胺神经递质和儿茶酚 O-甲基转移酶 (COMT) 抑制剂,Ki 值为 44 μM。
TN1969 N-(p-Coumaroyl) serotonin

PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
N-(p-Coumaroyl) Serotonin 是从红花种子中分离出来的多酚,具有抗氧化、抗动脉粥样硬化和抗炎作用,常用于动脉粥样硬化的研究。它可改善动脉粥样硬化和主动脉壁膨大。它可降低肌浆网中 PDGF 诱导的对中PDGFR 酪氨酸磷酸化和 Ca2+释放的作用。
T4860 5-Hydroxytryptamine creatinine sulfate monohydrate

Serotonin creatinine sulfate monohydrate,5-Hydroxytryptamine creatinine sulfate complex,5-五羟色胺肌酸酐

Others; Endogenous Metabolite Metabolism; Others
5-Hydroxytryptamine creatinine sulfate monohydrate (Serotonin creatinine sulfate monohydrate) 是内源性代谢产物的一种。
T19931 Gentisein

NSC 329491,NSC329491,NSC-329491

Serotonin Transporter Neuroscience
Gentisein (NSC-329491) 是 Mangiferin 的主要代谢物,有效抑制 5-HT 的摄取,IC50为 4.7 µM。
T2815 Puerarin

葛根素,Kakonein

5-HT Receptor GPCR/G Protein; Neuroscience
Puerarin (Kakonein) 是从葛根中提取的一种异黄酮,是一种5-HT2C 受体拮抗剂。
T0525 Flopropione

夫洛丙酮,Phloropropiophenone

5-HT Receptor; Transferase GPCR/G Protein; Metabolism; Neuroscience
Flopropione (Phloropropiophenone) 是一种解痉剂,用作 5-HT1A 受体拮抗剂,也是儿茶酚-O-甲基转移酶抑制剂。
T9113 Myristicin

Myristicine,肉豆蔻醚

IL Receptor; Anti-infection; BCL; P450; PARP; 5-HT Receptor; Caspase; GABA Receptor; NO Synthase Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Myristicin (Myristicine) 是一种在香料和伞形植物中发现的天然产物。肉豆蔻素具有抗胆碱能、抗菌和肝保护作用,还具有抗炎作用,其通过钙途径抑制dsrna 刺激的巨噬细胞中的NO、细胞因子、趋化因子和生长因子。Myristicin 可以诱导细胞凋亡,其特征是改变线粒体膜电位、细胞色素c 释放、Caspase-3激活、parp 切割和DNA 断裂。
T6S0654 Isocorynoxeine

7-Isocorynoxeine,异去氢钩藤碱

5-HT Receptor GPCR/G Protein; Neuroscience
Isocorynoxeine (7-Isocorynoxeine) 是钩藤中的一种生物碱,剂量依赖性抑制5-HT2A 受体介导的电流反应,IC50为 72.4 μM。
TN1032 Geissoschizine methyl ether

缝籽木嗪甲醚,缝籽嗪甲醚

5-HT Receptor GPCR/G Protein; Neuroscience
Geissoschizine methyl ether 是从钩藤中发现的一种生物碱,是 Yokukansan 的主要活性成分,具有精神药物作用。它是一种有效的 5-羟色胺 A 受体激动剂,是 Yokukansan 改善攻击性和社交性的候选药物。
T4S1637 gamma-Mangostin

Normangostin,γ-倒捻子素

Others; 5-HT Receptor GPCR/G Protein; Neuroscience; Others
gamma-Mangostin (Normangostin) 是从药用植物山竹的果壳中提纯的一种天然产物,是一种竞争性5-HT2A 受体拮抗剂。它是运甲状腺素蛋白原纤维化抑制剂,与甲状腺素结合位点结合并稳定了 TTR 四聚体,具有抗高血压、预防结肠癌等作用。
T1045 Trimipramine maleate

Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐

Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂,对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。
T7521 Azaphen

Pipofezin hydrochloride,阿扎吩,Pipofezine hydrochloride,Azafen

5-HT Receptor; Serotonin Transporter GPCR/G Protein; Neuroscience
Azaphen (Pipofezin hydrochloride) 是一种 5-羟色胺重吸收抑制剂。
T6648 Rotundine

Gindarine,L-Tetrahydropalmatine,Caseanine,罗通定,(-)-Tetrahydropalmatine

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Rotundine (Gindarine) 是多巴胺D1、D2和D3受体的拮抗剂,IC50值分别为 166、1.4 和 3.3 μM。 它也是5-HT1A 的拮抗剂,IC50值为 370 nM。
TN1217 2'-O-Methylisoliquiritigenin

Dopamine Receptor; 5-HT Receptor; GABA Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
2'-O-Methylisoliquiritigenin 是从洋甘草中分离出来的一种天然产物,是由 NR 中特异性诱导的酶合成的。它上调 5-HT、NE、DA 和 GABA 途径,对 NE 通路有显著影响。
T1317 Cinchonidine

奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine

5-HT Receptor; Serotonin Transporter; Parasite GPCR/G Protein; Microbiology/Virology; Neuroscience
Cinchonidine (L-Cinchonidine) 是在金鸡纳和角蒿中发现的一种生物碱,有抗疟活性。 它是用于有机化学中不对称合成的砌块,是血清素转运蛋白的弱抑制剂。
T1711 Harmine

Telepathine,去氢骆驼蓬碱

MAO; 5-HT Receptor; DYRK Cell Cycle/Checkpoint; GPCR/G Protein; Metabolism; Neuroscience; Tyrosine Kinase/Adaptors
Harmine (Telepathine) 是一种从山茱萸种子中分离出来的生物碱,具有抗癌和抗炎活性。它是双特异性酪氨酸磷酸化调节激酶抑制剂,对5-HT2A 血清素受体具有高亲和力,Ki 值为 397 nM。
T3369 Nuciferine

(-)-Nuciferine,VLT 049,荷叶碱,Sanjoinine E

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Nuciferine ((-)-Nuciferine) 是一种在埃及蓝睡莲和水芙蓉中发现的生物碱,是5-HT2A、5-HT2B 和5-HT2C 拮抗剂,IC50分别为 478 nM、1 μM 和 131 nM。它也是5-HT7的反向激动剂,IC50为 150 nM。
TN1465 Cannabigerol

NOS; 5-HT Receptor; ROS GPCR/G Protein; Immunology/Inflammation; Neuroscience
Cannabigerol 是一种植物大麻素,是一种高亲和力 α2-肾上腺素能受体激动剂、中度亲和力 5-HT1A 受体拮抗剂和低亲和力 CB1/CB2受体拮抗剂。它可降低眼压,有潜力治疗青光眼。
T0076 Paliperidone

9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Paliperidone (9-hydroxyrisperidone) 是 Risperidone 的主要活性代谢产物,是多巴胺 D2 拮抗剂和5-HT2A 拮抗剂。它用作非典型抗精神病药,用于精神分裂症的急性及维持治疗。它对α1和α2肾上腺素能受体和 H1组胺能受体也有拮抗作用。
TN2865 (E)-3,4,5-Trimethoxycinnamic acid

O-Methylsinapic acid,3,4,5-三甲氧基肉桂酸,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid

Others Others
(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) 是一种来自羌活根和根茎的天然产物。
T2811 Harmine hydrochloride

telepathine hydrochloride,盐酸哈尔明碱

5-HT Receptor; DYRK; GluR Cell Cycle/Checkpoint; GPCR/G Protein; Neuroscience; Tyrosine Kinase/Adaptors
Harmine hydrochloride (telepathine hydrochloride) 是一种 DYRK 抑制剂,具有抗癌和抗炎活性。它对5-HT2A 血清素受体具有高亲和力,Ki 值为 397 nM。
T0185 Escitalopram

Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram

Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Adrenergic Receptor; AChR; Norepinephrine; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Escitalopram (Seroplex) 是一种外消旋 Citalopram 的 S-对映体,是一种选择性 5-羟色胺再摄取抑制剂,Ki=0.89 nM,比 R(-)-enantiomer 结合亲和力高 30 倍。它对多巴胺转运体和去甲肾上腺素转运体均有选择性,是一种研究抑郁症的抗抑郁药。
T3933 Jatrorrhizine

Yatrorizine,neprotin,药根碱

MAO; 5-HT Receptor; Antibacterial; AChE GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Jatrorrhizine (neprotin) 是一种从黄连中分离得到的生物碱,具有抗菌、抗氧化、抗疟原虫和神经保护活性。它通过抑制 uptake-2 transporter 的活性减少血清素和去甲肾上腺素的摄取。它是一种有口服活性的乙酰胆碱酯酶制剂。
T1156 Palonosetron hydrochloride

盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259

5-HT Receptor GPCR/G Protein; Neuroscience
Palonosetron hydrochloride (RS 25259) 是一种 5-HT3 拮抗剂,用于预防和治疗化疗引起的恶心和呕吐。
T4S1659 Xanthotoxol

8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,花椒毒酚,8-Hydroxypsoralene

Reactive Oxygen Species; 5-HT Receptor; Endogenous Metabolite GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB
Xanthotoxol (Psoralen) 是一种具有生物活性的线性呋喃香豆素,具有很强的抗炎、抗氧化、5-HT 拮抗和神经保护作用等药理活性。
T4912 Jatrorrhizine chloride

盐酸药根碱,Yatrorhizine chloride,Neprotine chloride

Others; 5-HT Receptor; OCT; Antibacterial; AChE GPCR/G Protein; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Others
Jatrorrhizine chloride (Neprotine chloride) 是从黄连中分离得到的生物碱,具有神经保护、抗菌、抗氧化和抗疟原虫活性。它通过抑制摄取2转运蛋白的活性减少血清素和去甲肾上腺素的摄取。它是具有口服活性的乙酰胆碱酯酶抑制剂。
TMA1122 N-Feruloylserotonin

(E/Z)-Moschamine,Moschamine

Antioxidant oxidation-reduction
N-Feruloylserotonin ((E/Z)-Moschamine) 是可从 Carthamus tinctorius L. 中分离得到的一种血清素衍生物,具有抗氧化活性,有用于动脉粥样硬化和主动脉壁膨胀研究的潜能。
T82808 Bufoserotonin C

Bufoserotonin C为蟾酥中新发现的吲哚生物碱,展现出对抗肿瘤的活性。其在A549细胞系中的IC50为34.3 μM。
T4744 5-HYDROXYINDOLE-3-ACETIC ACID

5-羟基吲哚-3-乙酸,5-HIAA

Others; Endogenous Metabolite Metabolism; Others
5-Hydroxyindole-3-acetic acid (5-HIAA) 是 甲氧基肾上腺素或5-羟色胺的主要代谢产物,被用作神经内分泌肿瘤的生物标志物。它是血清素的分解产物,能够从尿液中排出。
T0783 Mianserin hydrochloride

Mianserin HCl,Org GB 94,盐酸米安色林,ORG GB-94 HCl

Dopamine Receptor; 5-HT Receptor; Opioid Receptor; Adrenergic Receptor; Histamine Receptor Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mianserin hydrochloride (Org GB 94) 是一种有抗抑郁活性的 H1 受体反向激动剂。
T3003 5-hydroxytryptophan

5-羟基色氨酸,NSC-92523

Others; Endogenous Metabolite Metabolism; Others
5-hydroxytryptophan (NSC-92523) 是色氨酸的代谢物,是5-羟色胺直接的前体,是芳香氨基酸脱羧酶底物。
T4761 Pyridoxal hydrochloride

Others; Endogenous Metabolite Metabolism; Others
Pyridoxal hydrochloride 是内源性代谢产物的一种。
T1354 N-Acetyl-5-hydroxytryptamine

Normelatonin,N-乙酰-5-羟色胺,O-Demethylmelatonin,N-Acetylserotonin

Trk receptor; Endogenous Metabolite Metabolism; Tyrosine Kinase/Adaptors
N-Acetyl-5-hydroxytryptamine (O-Demethylmelatonin) 是褪黑激素的直接前体,能够有效激活TrkB 受体。
T13515 5-Methoxytryptophol

2-(5-Methoxy-1H-indol-3-yl)ethanol,Methoxytryptophol,5-甲氧基色醇

Endogenous Metabolite Metabolism
5-Methoxytryptophol (2-(5-Methoxy-1H-indol-3-yl)ethanol) 是衍生自血清素的松果体吲哚胺,在许多物种中都具有生物特性。
TN1740 Homoeriodictyol

高胜草酚,高圣草酚

5-HT Receptor; transporter; Sodium Channel; Drug Metabolite GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Homoeriodictyol 是 Eriocitrin 的代谢物,属于黄酮类。Eriocitrin 是强效抗氧化剂。
T0973L Pyridoxine hydrochloride

Pyridoxine HCl,吡哆醇盐酸盐,Pyridoxol (hydrochloride),吡哆醇盐酸盐(维生素B6),Vitamin B6 (hydrochloride),Vitamin B6

Nrf2; Endogenous Metabolite Immunology/Inflammation; Metabolism
Pyridoxine hydrochloride (Vitamin B6) 是一种吡啶衍生物。在于阿尔茨海默病细胞模型中,通过 Nrf-2/HO-1 途径发挥抗氧化作用。
T1379 L-5-Hydroxytryptophan

5-羟基色氨酸,L-oxitriptan,Oxitriptan,L-5-HTP

Amino Acids and Derivatives; Endogenous Metabolite Metabolism
L-5-Hydroxytryptophan (L-5-HTP) 是一种天然氨基酸和膳食补充剂,可以用作抗抑郁剂、食欲抑制剂和睡眠辅助剂,是神经递质血清素的前体,是利血平(reserpine) 的拮抗剂。它能够用于肌阵挛、纤维肌痛症、偏头痛和小脑共济失调的研究。
TN1370 Allura Red AC

Allura Red,CI 16035,FD&C RED NO. 40

Others; Estrogen/progestogen Receptor; Androgen Receptor Endocrinology/Hormones; Others
Allura Red AC (CI 16035) 是一种非常重要的食用偶氮染料,可用于食品、药品、造纸、化妆品和纺织行业。Allura Red AC 可通过小鼠肠道血清素促进实验性结肠炎的易感性。
T0439 L-Tryptophan

(S)-Tryptophan,Tryptophan,L-Tryptophane,Tryptophane,L-色氨酸

Amino Acids and Derivatives; Endogenous Metabolite Metabolism
L-Tryptophan (Tryptophane) 是一种必需氨基酸,是褪黑素、血清素和维生素B3的前体。
T0791 Reserpine

利血平,Serpalan,Serpasil,Serpivite

Others; Potassium Channel; MRP; Monoamine Transporter; Autophagy Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Others
Reserpine (Serpalan) 是一种从催吐萝芙木的根中发现的生物碱。它抑制去甲肾上腺素吸收到储存囊泡中,导致中枢和外周轴突末端的儿茶酚胺和血清素耗尽。它可作为抗高血压药和抗精神病药以及研究工具。
T4429 Rauwolscine hydrochloride

Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) 是一种高选择性的 α2 adrenergic 受体拮抗剂,Ki=12 nM。
T1311 4-aminobenzoic acid

PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸

Endogenous Metabolite Metabolism
4-aminobenzoic acid (para-Aminobenzoic acid) 是一种具有紫外线吸收和抗纤维化特性的有机酸。当暴露在光线下时,4-aminobenzoic acid 吸收紫外线并通过光化学反应释放多余的能量,这可能会对DNA造成损害。4-aminobenzoic acid 还可以增加组织水平的摄氧量,并可能增强单胺氧化酶(MAO)活性以促进血清素的降解,过量可能导致纤维化变化。
T6S1684 8-Gingerol

Antioxidant; Antibacterial; TRP/TRPV Channel Membrane transporter/Ion channel; Microbiology/Virology; oxidation-reduction
8-Gingerol 分离自姜的根状茎,是口服有效的 TRPV1激活剂,EC50值为5.0 µM。8-Gingerol 抑制 COX-2,还能抑制体外 H. pylori 的生长。
T28019 (-)-Mesembrine

Mesembrin,Mesembrine,Mesembranone

Mesembrine is a serotonin reuptake inhibitor and is also a weak inhibitor of the enzyme phosphodiesterase 4 (PDE4).
T19772 Mesembrenone

(+)-Mesembrenone

Mesembrenone is a selective the serotonin transporter (SERT) inhibitor. Mesembrenone is the main alkaloid of Sceletium tortuosum.
T36532 SCH 38519

SCH 38519 is an isochromanequinone fungal metabolite originally isolated from Thermomonospora. It inhibits aggregation induced by thrombin , as well as inhibits serotonin secretion in human platelets (IC50s = 68 and 61 μg/ml, respectively). It inhibits the growth of various Gram-negative and Gram-positive bacteria (mean MICs = 122.1 and 0.92 μg/ml, respectively).
TN1623 Escin IIB

Others; NOS Immunology/Inflammation; Others
Escin IIB has positive effects on acute inflammation in animals, it can inhibit the induced by serotonin in rats, the hind paw edema induced by carrageenin, and the scratching behavior induced by compound 48/80 in mice.
T75436 Jatrorrhizine hydroxide

Jatrorrhizine hydroxide, 一种从黄连中提取的生物碱,展现了神经保护、抗菌、抗疟原虫及抗氧化的活性。作为一种高效的乙酰胆碱酯酶(AChE)抑制剂(IC50=872 nM),其对BuChE的选择性高达115倍。此外,Jatrorrhizine hydroxide还能通过抑制uptake-2 transporter活性来减少血清素(5-HT)和去甲肾上腺素(NE)的摄取,表现出口服活性。

天然产物

Serotonin
Cat.No: TN2437
Synonym: 5-羟基色胺,5-hydroxytryptamine,血清素,五羟色胺,5-HT
Target: Others, 5-HT Receptor, Endogenous Metabolite, Transferase
Serotonin hydrochloride
Cat.No: T2209
Synonym: 5-HT hydrochloride,5-羟基色胺盐酸盐,5-HT HCl,Serotonin HCl,5-Hydroxytryptamine hydrochloride
Target: 5-HT Receptor, Endogenous Metabolite, Transferase
N-(p-Coumaroyl) serotonin
Cat.No: TN1969
Synonym:
Target: PDGFR
5-Hydroxytryptamine creatinine sulfate monohydrate
Cat.No: T4860
Synonym: Serotonin creatinine sulfate monohydrate,5-Hydroxytryptamine creatinine sulfate complex,5-五羟色胺肌酸酐
Target: Others, Endogenous Metabolite
Gentisein
Cat.No: T19931
Synonym: NSC 329491,NSC329491,NSC-329491
Target: Serotonin Transporter
Puerarin
Cat.No: T2815
Synonym: 葛根素,Kakonein
Target: 5-HT Receptor
Flopropione
Cat.No: T0525
Synonym: 夫洛丙酮,Phloropropiophenone
Target: 5-HT Receptor, Transferase
Myristicin
Cat.No: T9113
Synonym: Myristicine,肉豆蔻醚
Target: IL Receptor, Anti-infection, BCL, P450, PARP, 5-HT Receptor, Caspase, GABA Receptor, NO Synthase
Isocorynoxeine
Cat.No: T6S0654
Synonym: 7-Isocorynoxeine,异去氢钩藤碱
Target: 5-HT Receptor
Geissoschizine methyl ether
Cat.No: TN1032
Synonym: 缝籽木嗪甲醚,缝籽嗪甲醚
Target: 5-HT Receptor
gamma-Mangostin
Cat.No: T4S1637
Synonym: Normangostin,γ-倒捻子素
Target: Others, 5-HT Receptor
Trimipramine maleate
Cat.No: T1045
Synonym: Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐
Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor
Azaphen
Cat.No: T7521
Synonym: Pipofezin hydrochloride,阿扎吩,Pipofezine hydrochloride,Azafen
Target: 5-HT Receptor, Serotonin Transporter
Rotundine
Cat.No: T6648
Synonym: Gindarine,L-Tetrahydropalmatine,Caseanine,罗通定,(-)-Tetrahydropalmatine
Target: Dopamine Receptor, 5-HT Receptor
2'-O-Methylisoliquiritigenin
Cat.No: TN1217
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, GABA Receptor
Cinchonidine
Cat.No: T1317
Synonym: 奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine
Target: 5-HT Receptor, Serotonin Transporter, Parasite
Harmine
Cat.No: T1711
Synonym: Telepathine,去氢骆驼蓬碱
Target: MAO, 5-HT Receptor, DYRK
Nuciferine
Cat.No: T3369
Synonym: (-)-Nuciferine,VLT 049,荷叶碱,Sanjoinine E
Target: Dopamine Receptor, 5-HT Receptor
Cannabigerol
Cat.No: TN1465
Synonym:
Target: NOS, 5-HT Receptor, ROS
Paliperidone
Cat.No: T0076
Synonym: 9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
(E)-3,4,5-Trimethoxycinnamic acid
Cat.No: TN2865
Synonym: O-Methylsinapic acid,3,4,5-三甲氧基肉桂酸,3,4,5-Trimethoxy-trans-cinnamic acid,3,4,5-Trimethoxyphenylacrylic acid
Target: Others
Harmine hydrochloride
Cat.No: T2811
Synonym: telepathine hydrochloride,盐酸哈尔明碱
Target: 5-HT Receptor, DYRK, GluR
Escitalopram
Cat.No: T0185
Synonym: Seroplex,依他普仑,S-(+)-Citalopram,艾司西酞普兰,(S)-Citalopram
Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Adrenergic Receptor, AChR, Norepinephrine, Histamine Receptor
Jatrorrhizine
Cat.No: T3933
Synonym: Yatrorizine,neprotin,药根碱
Target: MAO, 5-HT Receptor, Antibacterial, AChE
Palonosetron hydrochloride
Cat.No: T1156
Synonym: 盐酸帕洛诺司琼,RS 25259 197,Palonosetron HCl,RS 25259
Target: 5-HT Receptor
Xanthotoxol
Cat.No: T4S1659
Synonym: 8-Hydroxypsoralen,8-Hydroxyfuranocoumarin,Psoralen,花椒毒酚,8-Hydroxypsoralene
Target: Reactive Oxygen Species, 5-HT Receptor, Endogenous Metabolite
Jatrorrhizine chloride
Cat.No: T4912
Synonym: 盐酸药根碱,Yatrorhizine chloride,Neprotine chloride
Target: Others, 5-HT Receptor, OCT, Antibacterial, AChE
N-Feruloylserotonin
Cat.No: TMA1122
Synonym: (E/Z)-Moschamine,Moschamine
Target: Antioxidant
Bufoserotonin C
Cat.No: T82808
Synonym:
Target:
5-HYDROXYINDOLE-3-ACETIC ACID
Cat.No: T4744
Synonym: 5-羟基吲哚-3-乙酸,5-HIAA
Target: Others, Endogenous Metabolite
Mianserin hydrochloride
Cat.No: T0783
Synonym: Mianserin HCl,Org GB 94,盐酸米安色林,ORG GB-94 HCl
Target: Dopamine Receptor, 5-HT Receptor, Opioid Receptor, Adrenergic Receptor, Histamine Receptor
5-hydroxytryptophan
Cat.No: T3003
Synonym: 5-羟基色氨酸,NSC-92523
Target: Others, Endogenous Metabolite
Pyridoxal hydrochloride
Cat.No: T4761
Synonym:
Target: Others, Endogenous Metabolite
N-Acetyl-5-hydroxytryptamine
Cat.No: T1354
Synonym: Normelatonin,N-乙酰-5-羟色胺,O-Demethylmelatonin,N-Acetylserotonin
Target: Trk receptor, Endogenous Metabolite
5-Methoxytryptophol
Cat.No: T13515
Synonym: 2-(5-Methoxy-1H-indol-3-yl)ethanol,Methoxytryptophol,5-甲氧基色醇
Target: Endogenous Metabolite
Homoeriodictyol
Cat.No: TN1740
Synonym: 高胜草酚,高圣草酚
Target: 5-HT Receptor, transporter, Sodium Channel, Drug Metabolite
Pyridoxine hydrochloride
Cat.No: T0973L
Synonym: Pyridoxine HCl,吡哆醇盐酸盐,Pyridoxol (hydrochloride),吡哆醇盐酸盐(维生素B6),Vitamin B6 (hydrochloride),Vitamin B6
Target: Nrf2, Endogenous Metabolite
L-5-Hydroxytryptophan
Cat.No: T1379
Synonym: 5-羟基色氨酸,L-oxitriptan,Oxitriptan,L-5-HTP
Target: Amino Acids and Derivatives, Endogenous Metabolite
Allura Red AC
Cat.No: TN1370
Synonym: Allura Red,CI 16035,FD&C RED NO. 40
Target: Others, Estrogen/progestogen Receptor, Androgen Receptor
L-Tryptophan
Cat.No: T0439
Synonym: (S)-Tryptophan,Tryptophan,L-Tryptophane,Tryptophane,L-色氨酸
Target: Amino Acids and Derivatives, Endogenous Metabolite
Reserpine
Cat.No: T0791
Synonym: 利血平,Serpalan,Serpasil,Serpivite
Target: Others, Potassium Channel, MRP, Monoamine Transporter, Autophagy
Rauwolscine hydrochloride
Cat.No: T4429
Synonym: Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
4-aminobenzoic acid
Cat.No: T1311
Synonym: PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸
Target: Endogenous Metabolite
8-Gingerol
Cat.No: T6S1684
Synonym:
Target: Antioxidant, Antibacterial, TRP/TRPV Channel
(-)-Mesembrine
Cat.No: T28019
Synonym: Mesembrin,Mesembrine,Mesembranone
Target:
Mesembrenone
Cat.No: T19772
Synonym: (+)-Mesembrenone
Target:
SCH 38519
Cat.No: T36532
Synonym:
Target:
Escin IIB
Cat.No: TN1623
Synonym:
Target: Others, NOS
Jatrorrhizine hydroxide
Cat.No: T75436
Synonym:
Target:
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