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377

抑制剂 & 化合物

118

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Cat. No. Product Name Target Signaling Pathways
T24656 PQ-10

A844337,PQ 10,A-844337,A 844337

PDE Metabolism
PQ-10 (A-844337) 是磷酸二酯酶 10A 抑制剂,其IC50=4.6 nM,ED50=13 mg/kg。它能够诱导大脑葡萄糖代谢模式,这可能是潜在的转化生物标志物。它对精神分裂症等精神疾病具有研究潜力。
T1674 Nateglinide

那格列奈,A4166,Senaglinide

Potassium Channel; Proteasome; PPAR DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome; Ubiquitination
Nateglinide (Senaglinide) 是 D-苯丙氨酸的一种衍生物,是口服有效的、短效促胰岛素释放化合物,也是 DPP IV 抑制剂。 Nateglinide 抑制胰岛 β 细胞中 ATP 敏感的 K+通道。Nateglinide 在 2 型糖尿病中具有研究价值。
T37898 UDP-α-D-Glucose (sodium salt hydrate)

UDP-α-D-Glucose is an endogenous nucleotide sugar involved in glycosyltransferase reactions in metabolism. It has been shown to bind the P2Y14receptor (EC50= 0.35 μM), an atypical P2Y receptor involved in the activation of dendritic cells and glial cells.1It can also bind to and activate GPR17, inducing oligodendrocyte differentiation at a maximal concentration of 100 μM.2 1.Jacobson, K.A., Ivanov, A.A., de Castro, S., et al.Development of selective agonists and antagonists of P2Y receptorsPurin...
T35416 α-D-Glucose-1-phosphate (sodium salt hydrate)

α-D-Glucose-1-phosphate is an intermediate in glycogen metabolism.1,2It is a precursor in the biosynthesis of UDP-glucose, the glucose donor in glycogen biosynthesis.2α-D-Glucose-1-phosphate can be formed during glycogen breakdownviaphosphorolytic cleavage of glycogen by glycogen phosphorylase.1It can be converted to glucose-6-phosphate by phosphoglucomutase. α-D-Glucose-1-phosphate is combined with CTP by α-D-glucose-1-phosphate cytidylyltransferase to form CDP-glucose in the first step of CDP-...
T19261 D-Glucose-13C6

D-(+)-Glucose-13C6,Glucose-13C6,Dextrose-13C6

Endogenous Metabolite Metabolism
D-Glucose-13C6 (Dextrose-13C6) 是一种 D-Glucose 的同位素标记物,可作为代谢示踪剂,可用于研究机体代谢相关疾病和部分物质的代谢过程。
T20839 Kojibiose

a-葡糖-a-葡糖苷,Kojibiose

Others Others
Kojibiose (Kojibiose) 是蜂蜜中的一种二糖。 Kojibiose 是葡萄糖焦糖化的产物。
T20029 Buformin hydrochloride

NSC528218,NSC-528218,盐酸丁双胍,NSC 528218

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
Buformin hydrochloride (NSC-528218) 是一种有效的 AMPK 激活剂,是一种双胍类的口服抗糖尿病药物。Buformin 延缓胃肠道对葡萄糖的吸收,增加胰岛素敏感性和葡萄糖对细胞的吸收,并抑制肝脏对葡萄糖的合成。Buformin 也具有抗癌活性,可用于各种癌症研究。
T0582 Fructooligosaccharides

Others Others
Fructooligosaccharides 是一种左旋单糖,是葡萄糖的异构体。
T22317 DRB18

transporter Metabolism
DRB18 is a highly effective pan-class inhibitor of glucose transporter proteins (GLUT). It significantly modulates energy-related metabolism in A549 cells by inducing alterations in the abundance of metabolites associated with glucose-related pathways. DRB18 exerts its effects by promoting G1/S phase arrest, increasing oxidative stress, and prompting necrotic cell death, ultimately displaying notable anti-tumor activity [1].
T33412 MitoPQ

MitoParaquat

Glucokinase; transporter Metabolism
MitoPQ (MitoParaquat) 是一个线粒体靶向的小分子化合物。MitoPQ 选择性加强线粒体超氧化物和过氧化氢的含量,抑制胰岛素刺激的葡萄糖摄取和葡萄糖转运蛋白 4 (GLUT4) 向脂肪细胞和肌管中质膜的易位。MitoPQ 可用于研究线粒体氧化应激与调节的 GLUT4 转运。
T30142 ARRY-403

AMG-151,ARRY 403,ARRY403,ARRY-403,AMG151,AMG 151

Glucokinase Metabolism
ARRY-403 是一种新型葡萄糖激酶激活剂,可降低 2 型糖尿病患者的空腹和餐后血糖,可用于治疗糖尿病。
T37985 D-Fructose-6-phosphate (sodium salt hydrate)

D-Fructose-6-phosphate (sodium salt hydrate) (643-13-0 free base)

D-Fructose-6-phosphate (sodium salt hydrate) 是由磷酸葡萄糖异构酶将 6-磷酸葡萄糖异构化产生的糖酵解途径的糖中间体,可用于研究癌症。
T22520 5-Carboxamidotryptamine maleate

5-CT maleate

5-HT Receptor GPCR/G Protein; Neuroscience
5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) 是一种 受体激动剂,具有降压和升血糖的作用。
T6551 Isosorbide

Devicoran,Isobide,异山梨酯,异山梨醇,Hydronol,Dianhydro-D-glucitol,D-Isosorbide

Others Others
Isosorbide (Devicoran) 是一种血管舒张剂,也是一种高渗利尿剂,口服具有活性。可用于研究心力衰竭和心绞痛(胸痛)。
T19211 BM152054

Others Others
BM152054 是一种有效的 PPARγ配体,可以通过加强胰岛素作用来诱导外周组织对葡萄糖的利用。
T6455 CP-91149

Phosphorylase Metabolism
CP91149 是GP (糖原磷酸化酶)的抑制剂,能够促进糖原的重新合成,但不会造成糖原的过度积累。它对2型糖尿病具有潜在的研究价值。
T4460 Dapagliflozin ((2S)-1,2-propanediol, hydrate)

BMS-512148 (2S)-1,2-propanediol, hydrate,达格列净 (2S)-1,2-丙二醇水合物,Dapagliflozin propanediol monohydrate

SGLT GPCR/G Protein
Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) 是 Dapagliflozin 1,2-propanediol, hydrate 的 S 型异构体,是竞争性葡萄糖协同转运蛋白2 抑制剂,可促进尿液中葡萄糖的排泄,可用于糖尿病的研究。它诱导 HIF1表达并减轻肾脏 IR 损伤。
T1782L Canagliflozin hemihydrate

JNJ28431754,TA 7284,TA7284,TA-7284,JNJ 28431754,JNJ-28431754

SGLT GPCR/G Protein
Canagliflozin hemihydrate (TA 7284) (JNJ28431754 hemihydrate) 是一种选择性的 SGLT2 抑制剂,作用于表达 mSGLT2,rSGLT2 和 hSGLT2 的 CHO 细胞,IC50 分别为 2 nM,3.7 nM 和 4.4 nM。
T14017 2-NBDG

2-(N-7-硝基-2,1,3-苯并恶二唑-4-氨基)-2-脱氧-D-葡萄糖

Others Others
2-NBDG 是一种荧光指示剂 (λex=467 nm,λem=542 nm),是一种荧光 D-葡萄糖类似物,可用于监测活细胞中的葡萄糖吸收。
T0050 Ampyrone

Minoazophene,Aminoantipyrin,NSC 60242,4-Aminoantipyrine,4-氨基安替比林,Solnapyrin-A

COX; Drug Metabolite Immunology/Inflammation; Metabolism; Neuroscience
Ampyrone (4-Aminoantipyrine) 是一种检测试剂,在过氧化物酶与苯酚存在时,用于葡萄糖测定。
T22708 Darglitazone

CP-86325

PPAR DNA Damage/DNA Repair; Metabolism
Darglitazone (CP-86325) 是一种噻唑烷二酮,是口服有效的PPAR-γ选择性激动剂。Darglitazone 可以有效控制血糖和脂质代谢,在 II 型糖尿病中有研究价值。
T32237 Isoxaben

EL 107,NA 8318,Isoxaben; EL 107; NA 8318

Cell wall Immunology/Inflammation
Isoxaben (EL 107) 是一种细胞壁生物合成的特异性抑制剂,常作为除草剂使用,可抑制放射性标记的葡萄糖掺入酸不溶性细胞壁部分。
T11765 KPLH1130

Dehydrogenase; PDK Metabolism; PI3K/Akt/mTOR signaling
KPLH1130,一种选择性丙酮酸脱氢酶激酶(PDK)抑制剂,在高脂饮食(HFD)喂养的小鼠中提高了糖耐量。KPLH1130 抑制巨噬细胞极化并减轻了炎症反应。
T2608 CHIR-98014

CHIR 98014,CT98014,CHIR98014

FGFR; GSK-3; Src; S6 Kinase Angiogenesis; MAPK; PI3K/Akt/mTOR signaling; Stem Cells; Tyrosine Kinase/Adaptors
CHIR-98014 (CT98014) 是有效的,细胞通透的GSK-3抑制剂,可抑制 GSK-3α (IC50:0.65 nM) 和 GSK-3β (IC50:0.58 nM) 的活性,对 cdc2 和 erk2 的作用较弱。
T1782 Canagliflozin

卡格列净,JNJ 24831754ZAE,JNJ 28431754AAA,TA 7284,JNJ 28431754

SGLT GPCR/G Protein
Canagliflozin (JNJ 28431754AAA) 是SGLT2的选择性抑制剂,在表达 mSGLT2,rSGLT2 和 hSGLT2 的 CHO 细胞上,IC50分别为 2 nM,3.7 nM 和 4.4 nM。
T37958 Acetyl Coenzyme A trisodium

Acetyl-CoA trisodium

OXPHOS; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism
Acetyl Coenzyme A trisodium (Acetyl-CoA trisodium) 是糖代谢和脂代谢的重要化合物,参与三羧酸循环。
T16083 Mizagliflozin

GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base

SGLT GPCR/G Protein
Mizagliflozin (GSK-1614235 free base) 是口服有效的、选择性的 SGLT1抑制剂,对人 SGLT1 的 Ki 值为 27 nM。Mizagliflozin 对 SGLT1 的选择性是 SGLT2的303 倍。它是抗糖尿病药物,可以改善餐后血糖波动。它在改善慢性便秘方面具有潜在的作用。
T7814 Alloxan monohydrate

Proteasome Proteases/Proteasome; Ubiquitination
Alloxan Monohydrate 是一种能够引起糖尿病的致糖尿病药物。它作为蛋白酶体抑制剂,破坏胰腺中能够分泌胰岛素的B 细胞,导致实验动物患糖尿病。
T67728 α-Glucosidase-IN-23

Glucosidase Metabolism
α-Glucosidase-IN-23 是具有口服活性的 α-Glucosidase 抑制剂。α-Glucosidase-IN-23 通过抑制 a-glucosidase 降低血糖 (IC50= 4.48 μM)。α-Glucosidase-IN-23 可用于糖尿病的研究。
T13867 RH01386

Others Others
RH01386是可以预防 ER 应激诱导的β细胞功能障碍和死亡、抑制促凋亡基因表达的小分子。它恢复内质网应激受损的葡萄糖刺激的胰岛素分泌反应。对2型糖尿病具有潜在的研究价值。
T67893 PTP1B-IN-22

Phosphatase Metabolism
PTP1B-IN-22是一种蛋白酪氨酸磷酸酶1B (PTP1B)抑制剂,可抑制骨骼肌 L6肌管的葡萄糖摄取。
T37891L GLP-1(32-36)amide acetate

GLP-1(32-36)amide 醋酸盐,GLP-1(32-36)amide acetate(1417302-71-6 Free base)

Others Others
GLP-1(32-36)amide acetate 是一种五肽,衍生自糖调节激素 GLP-1 的 C 末端。GLP-1(32-36)amide acetate 可抑制糖尿病小鼠的体重增加并调节全身葡萄糖代谢。
T14212 AMG-1694

Glucokinase Metabolism
AMG-1694 是一种强效的葡萄糖激酶-葡萄糖激酶调节蛋白(GK-GKRP)干扰物,能促进 GK-GKRP 复合物的解离,其 IC50 值为 7 nM,从而间接提高 GK 酶的活性。AMG-1694 可使几种啮齿动物糖尿病模型的血糖水平恢复正常,并降低糖尿病动物而非正常血糖动物的血糖。AMG-1694 能有效逆转 GKRP 对 GK 活性的抑制作用,并促进 GK 转位。
T1781 GW9508

GW 9508

GPR; Potassium Channel Endocrinology/Hormones; GPCR/G Protein; Membrane transporter/Ion channel
GW 9508 是一种选择性 G 蛋白偶联受体FFA1(GPR40) 和GPR120激动剂。它是一种葡萄糖敏感性胰岛素促分泌剂和 ATP 敏感性钾通道开放剂,具有抗炎和抗动脉粥样硬化活性。
T19596 UDP-GlcNAc Disodium Salt

Uridine 5′-diphospho-N-acetylglucosamine,5′-二磷酸尿嘧啶核苷-N-乙酰半乳糖胺二钠盐,UDP-α-D-N-Acetylglucosamine Disodium Salt

Others Others
UDP-GlcNAc Disodium Salt (UDP-α-D-N-Acetylglucosamine Disodium Salt) 是一种 O-GlcNAc 转移酶 (OGT) 的供体底物。
T4999 Ertugliflozin

埃格列净,MK-8835,PF-04971729

SGLT GPCR/G Protein
Ertugliflozin (PF-04971729) 是选择性的、口服有效的钠离子依赖的葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,对h-SGLT2 的IC50值为 0.877 nM。Ertugliflozin 在2型糖尿病中有研究价值。
T22459 Xanthinol Nicotinate

Angioamin,烟酸占替诺,Complamin

Others Others
Xanthinol Nicotinate (Complamin) 是血管扩张剂,可直接作用于小动脉和毛细血管的平滑肌,能够扩大血管,改善血液流变学并降低外周血管阻力。
T5195 Alrestatin

阿瑞司他丁,AY-22284

Reductase Endocrinology/Hormones; Metabolism
Alrestatin (AY-22284) 是醛糖还原酶的特异性抑制剂,能够在体外减弱大鼠血管平滑肌中葡萄糖诱导的血管紧张素 II 的产生。
T2389 Dapagliflozin

达格列净,BMS-512148

SGLT; HIF Angiogenesis; Chromatin/Epigenetic; GPCR/G Protein
Dapagliflozin (BMS-512148) 竞争性的葡萄糖协同转运蛋白2 (SGLT2) 抑制剂,可促进尿液中葡萄糖的排泄,在糖尿病 (DM) 研究中具有价值。Dapagliflozin 诱导 HIF1表达并减轻肾脏 IR 损伤。
T15810 LY2922470

GPR Endocrinology/Hormones; GPCR/G Protein
LY2922470 是选择性口服有效的GPR40激动剂,作用于 人 GPR40、小鼠 GPR40、大鼠 GPR40 的EC50值分别为 7 nM、1 nM、3 nM。它可降低血糖水平,同时显著增加胰岛素和 GLP-1,有潜力用于 2 型糖尿病的研究。
T7018 WZB117

transporter Metabolism
WZB117 是葡萄糖转运蛋白 1 抑制剂,可下调糖酵解,诱导细胞周期停滞,有抗癌细胞生长的作用。
T14327 AS1949490

Phosphatase Metabolism
AS1949490 是选择性SHIP-2抑制剂,其IC50=620 nM。它能够通过上调L6肌管GLUT1基因激活葡萄糖代谢。
T40514 2,2,14,14-Tetramethyl-8-oxopentadecanedioic acid

Others Others
2,2,14,14-Tetramethyl-8-oxopentadecanedioic acid 属于酮类化合物,化合物 II-9。它在心血管疾病、血脂异常、蛋白异常和糖代谢紊乱方面具有研究的价值。
T24793 SIRT6-IN-5

SIRT6 inhibitor5,SIRT6 IN 5,SIRT6 inhibitor-5,SIRT6 inhibitor 5

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
SIRT6-IN-5(SIRT6 inhibitor 5) 是一种具有有效性和选择性的 SIRT6 抑制剂 ,IC50 值为 34 μM。SIRT6-IN-5 具有免疫抑制和化疗增敏作用,可增加 H3K9 的乙酰化并增加培养细胞中的葡萄糖摄取,减少 T 细胞增殖。
T62238 AMPK activator 4

AMPK Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
AMPK activator 4 是一种有效且具有选择性的AMPK激活剂,不抑制线粒体复合物 I。AMPK activator 4 选择性地激活肌肉组织中的 AMPK且剂量依赖性地改善正常小鼠的糖耐量,显著降低 db/db 糖尿病小鼠的空腹血糖水平和改善胰岛素抵抗。AMPK activator 4 具有降血糖作用。
T63166 LSN3318839

LSN-3318839,LSN 3318839

Glucagon Receptor GPCR/G Protein
LSN3318839 是一种有效且可口服的胰高血糖素样肽-1受体(GLP-1R)变构调节剂。LSN3318839可增强GLP-1R的G蛋白偶联信号传导,可用来降低血糖。
T6646 Rosiglitazone hydrochloride

盐酸罗格列酮,BRL-49653 HCl,Rosiglitazone HCl

Ferroptosis; TRP/TRPV Channel; PPAR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Metabolism
Rosiglitazone hydrochloride (BRL-49653 HCl) 是一种降血糖药物,通过与脂肪细胞中的 PPAR 受体结合来刺激胰岛素分泌。它对 PPARγ1、PPARγ2 和 PPARγ 的EC50值分别为 30 nM、100 nM 和 60 nM。它也是TRPC5的激活剂和TRPM3的抑制剂。
T8818 TC-G 1005

(4-环丙基-3,4-二氢-1(2H)-喹喔啉基)[4-(2,5-二甲基苯氧基)-3-吡啶基]甲酮

GPCR19 GPCR/G Protein
TC-G 1005 是具有口服活性的TGR5选择性激动剂,能够激活 hTGR5 (EC50:0.72 nM)和 mTGR5 (EC50:6.2 nM)。它能够减少小鼠体内葡萄糖水平。
T7217 Bexagliflozin

THR-1442,EGT1442,EGT0001442

SGLT GPCR/G Protein
Bexagliflozin (EGT1442) 是一种选择性的,口服有效的钠葡萄糖协同转运蛋白-2 (SGLT2) 抑制剂,对人 SGLT2 和 SGLT1 作用的 IC50值分别为 2 nM 和 5.6 μM。EGT1442在 2 型糖尿病中有研究价值。
T40542 Sinbaglustat

ACT-519276,Sinbaglustat,OGT2378

Transferase Metabolism
Sinbaglustat (OGT2378) (OGT2378) 是葡萄糖神经酰胺合成酶 (GCS) 和非溶酶体葡萄糖神经酰胺酶 (GBA2) 的双重抑制剂。Sinbaglustat 是一种可透过血脑屏障的的口服N-烷基亚氨基糖。Sinbaglustat 可用于治疗溶酶体贮积症和研究溶酶体功能障碍相关的中枢神经退行性疾病。

化合物

PQ-10
Cat.No: T24656
Synonym: A844337,PQ 10,A-844337,A 844337
Target: PDE
Nateglinide
Cat.No: T1674
Synonym: 那格列奈,A4166,Senaglinide
Target: Potassium Channel, Proteasome, PPAR
UDP-α-D-Glucose (sodium salt hydrate)
Cat.No: T37898
Synonym:
Target:
α-D-Glucose-1-phosphate (sodium salt hydrate)
Cat.No: T35416
Synonym:
Target:
D-Glucose-13C6
Cat.No: T19261
Synonym: D-(+)-Glucose-13C6,Glucose-13C6,Dextrose-13C6
Target: Endogenous Metabolite
Kojibiose
Cat.No: T20839
Synonym: a-葡糖-a-葡糖苷,Kojibiose
Target: Others
Buformin hydrochloride
Cat.No: T20029
Synonym: NSC528218,NSC-528218,盐酸丁双胍,NSC 528218
Target: AMPK
Fructooligosaccharides
Cat.No: T0582
Synonym:
Target: Others
DRB18
Cat.No: T22317
Synonym:
Target: transporter
MitoPQ
Cat.No: T33412
Synonym: MitoParaquat
Target: Glucokinase, transporter
ARRY-403
Cat.No: T30142
Synonym: AMG-151,ARRY 403,ARRY403,ARRY-403,AMG151,AMG 151
Target: Glucokinase
D-Fructose-6-phosphate (sodium salt hydrate)
Cat.No: T37985
Synonym: D-Fructose-6-phosphate (sodium salt hydrate) (643-13-0 free base)
Target:
5-Carboxamidotryptamine maleate
Cat.No: T22520
Synonym: 5-CT maleate
Target: 5-HT Receptor
Isosorbide
Cat.No: T6551
Synonym: Devicoran,Isobide,异山梨酯,异山梨醇,Hydronol,Dianhydro-D-glucitol,D-Isosorbide
Target: Others
BM152054
Cat.No: T19211
Synonym:
Target: Others
CP-91149
Cat.No: T6455
Synonym:
Target: Phosphorylase
Dapagliflozin ((2S)-1,2-propanediol, hydrate)
Cat.No: T4460
Synonym: BMS-512148 (2S)-1,2-propanediol, hydrate,达格列净 (2S)-1,2-丙二醇水合物,Dapagliflozin propanediol monohydrate
Target: SGLT
Canagliflozin hemihydrate
Cat.No: T1782L
Synonym: JNJ28431754,TA 7284,TA7284,TA-7284,JNJ 28431754,JNJ-28431754
Target: SGLT
2-NBDG
Cat.No: T14017
Synonym: 2-(N-7-硝基-2,1,3-苯并恶二唑-4-氨基)-2-脱氧-D-葡萄糖
Target: Others
Ampyrone
Cat.No: T0050
Synonym: Minoazophene,Aminoantipyrin,NSC 60242,4-Aminoantipyrine,4-氨基安替比林,Solnapyrin-A
Target: COX, Drug Metabolite
Darglitazone
Cat.No: T22708
Synonym: CP-86325
Target: PPAR
Isoxaben
Cat.No: T32237
Synonym: EL 107,NA 8318,Isoxaben; EL 107; NA 8318
Target: Cell wall
KPLH1130
Cat.No: T11765
Synonym:
Target: Dehydrogenase, PDK
CHIR-98014
Cat.No: T2608
Synonym: CHIR 98014,CT98014,CHIR98014
Target: FGFR, GSK-3, Src, S6 Kinase
Canagliflozin
Cat.No: T1782
Synonym: 卡格列净,JNJ 24831754ZAE,JNJ 28431754AAA,TA 7284,JNJ 28431754
Target: SGLT
Acetyl Coenzyme A trisodium
Cat.No: T37958
Synonym: Acetyl-CoA trisodium
Target: OXPHOS, Endogenous Metabolite, Autophagy
Mizagliflozin
Cat.No: T16083
Synonym: GSK-1614235 free base,KGA-3235 free base,DSP-3235 free base
Target: SGLT
Alloxan monohydrate
Cat.No: T7814
Synonym:
Target: Proteasome
α-Glucosidase-IN-23
Cat.No: T67728
Synonym:
Target: Glucosidase
RH01386
Cat.No: T13867
Synonym:
Target: Others
PTP1B-IN-22
Cat.No: T67893
Synonym:
Target: Phosphatase
GLP-1(32-36)amide acetate
Cat.No: T37891L
Synonym: GLP-1(32-36)amide 醋酸盐,GLP-1(32-36)amide acetate(1417302-71-6 Free base)
Target: Others
AMG-1694
Cat.No: T14212
Synonym:
Target: Glucokinase
GW9508
Cat.No: T1781
Synonym: GW 9508
Target: GPR, Potassium Channel
UDP-GlcNAc Disodium Salt
Cat.No: T19596
Synonym: Uridine 5′-diphospho-N-acetylglucosamine,5′-二磷酸尿嘧啶核苷-N-乙酰半乳糖胺二钠盐,UDP-α-D-N-Acetylglucosamine Disodium Salt
Target: Others
Ertugliflozin
Cat.No: T4999
Synonym: 埃格列净,MK-8835,PF-04971729
Target: SGLT
Xanthinol Nicotinate
Cat.No: T22459
Synonym: Angioamin,烟酸占替诺,Complamin
Target: Others
Alrestatin
Cat.No: T5195
Synonym: 阿瑞司他丁,AY-22284
Target: Reductase
Dapagliflozin
Cat.No: T2389
Synonym: 达格列净,BMS-512148
Target: SGLT, HIF
LY2922470
Cat.No: T15810
Synonym:
Target: GPR
WZB117
Cat.No: T7018
Synonym:
Target: transporter
AS1949490
Cat.No: T14327
Synonym:
Target: Phosphatase
2,2,14,14-Tetramethyl-8-oxopentadecanedioic acid
Cat.No: T40514
Synonym:
Target: Others
SIRT6-IN-5
Cat.No: T24793
Synonym: SIRT6 inhibitor5,SIRT6 IN 5,SIRT6 inhibitor-5,SIRT6 inhibitor 5
Target: Sirtuin
AMPK activator 4
Cat.No: T62238
Synonym:
Target: AMPK
LSN3318839
Cat.No: T63166
Synonym: LSN-3318839,LSN 3318839
Target: Glucagon Receptor
Rosiglitazone hydrochloride
Cat.No: T6646
Synonym: 盐酸罗格列酮,BRL-49653 HCl,Rosiglitazone HCl
Target: Ferroptosis, TRP/TRPV Channel, PPAR, Autophagy
TC-G 1005
Cat.No: T8818
Synonym: (4-环丙基-3,4-二氢-1(2H)-喹喔啉基)[4-(2,5-二甲基苯氧基)-3-吡啶基]甲酮
Target: GPCR19
Bexagliflozin
Cat.No: T7217
Synonym: THR-1442,EGT1442,EGT0001442
Target: SGLT
Sinbaglustat
Cat.No: T40542
Synonym: ACT-519276,Sinbaglustat,OGT2378
Target: Transferase
Cat. No. Product Name Target Signaling Pathways
T4884 alpha-D-glucose

α-D-Glucose,α-葡萄糖,alpha-Glucose,α-Dextrose

Others; Endogenous Metabolite Metabolism; Others
alpha-D-glucose (α-Dextrose) 是内源性代谢产物的一种。
T4924 α-D-Glucose-1-phosphate disodium

A-D-葡萄糖-1-磷酸-二钠盐,α-D-Glucose 1-phosphate disodium salt hy,α-D-Glucopyranose 1-phosphate

Others; Endogenous Metabolite Metabolism; Others
α-D-Glucose 1-phosphate disodium salt hydrate 是合成葡萄糖醛酸的起始原料。它可用作心脏病研究所必需的细胞抑制剂、抗生素、免疫抑制剂和循环系统研究材料。
T4004 Concanavalin A

Apoptosis Apoptosis
Concanavalin A 是 Ca2+/Mn2+依赖性和甘露糖/葡萄糖结合植物凝集素。它能够促使程序性细胞死亡。
T0581 Isomaltose

D-Isomaltose,6-O-α-D-Glucopyranosyl-D-glucose,低聚异麦芽糖900

Others; Endogenous Metabolite Metabolism; Others
Isomaltose (D-Isomaltose) 是由两个葡萄糖组成的麦芽糖类似物,能够作为蔗糖的替代物,适合于糖尿病患者及有糖尿病倾向的人群。
T4743 Uridine 5′-diphosphoglucose disodium salt

二磷酸尿苷葡萄糖二钠盐,UDP-Glucose sodium salt,UDPG sodium salt,UDP-α-D-Glucose sodium salt,Uridine 5'-diphosphoglucose disodium sal

Endogenous Metabolite; P2Y Receptor GPCR/G Protein; Metabolism; Neuroscience
Uridine 5′-diphosphoglucose disodium salt (UDP-Glucose sodium salt) 是一种内源性核苷酸糖,参与代谢中的糖基转移酶反应。它是 P2Y14 受体的激动剂,EC50为 0.35 μM。
T72172 4,6-O-Ethylidene-α-D-glucose

Ethylidene-glucose

4,6-O-ethylidene-α-D-glucose (Ethylidene-glucose) 是一种葡萄糖衍生物,是竞争性的葡萄糖转运蛋白 1 (GLUT1) 面部结合部位抑制剂,对野生型 2-脱氧-D-葡萄糖转运的 Ki 值为 12 mM。
T35415 α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)

α-D-Glucose-1,6-bisphosphate is abis-phosphorylated derivative of α-D-glucose that has roles in carbohydrate metabolism.1It is the product of the reaction of glucose-1- or 6-phosphate with glucose-1,6-bisphosphate synthase (PGM2LI) in the conversion of 1,3-bisphosphoglycerate to 3-phosphoglycerate.2It is also a cofactor for the bacterial enzyme phosphopentomutase.3,4α-D-Glucose-1,6-bisphosphate has been used in the study of carbohydrate metabolism. 1.Beitner, R.Regulation of carbohydrate metabol...
TN1033 Sennidin A

HCV Protease; transporter; Akt; PI3K Cytoskeletal Signaling; Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Sennidin A 是从狭叶番泻分离得到的一种天然产物,能够抑制 HCV NS3 解旋酶,其 IC50值为0.8 μM。它诱导 Akt 和葡萄糖转运蛋白4的磷酸化,刺激葡萄糖掺入。
T19262 D-Glucose 6-phosphate disodium salt

D-​Glucose ​6-​phosphate disodium salt

Endogenous Metabolite Metabolism
D-Glucose 6-phosphate disodium salt 广泛存在于生物提内的化合物,是葡萄糖第 6 号碳经过磷酸化后生成的分子,参与磷酸戊糖途径与糖酵解途径等体内多种多种代谢调节途径。
T7997 β-D-Glucose pentaacetate

β-D-葡萄糖五乙酸酯,Penta-O-acetyl-β-D-glucopyranose,1,2,3,4,6-beta-D-葡萄糖五乙酸酯

Others Others
β-D-Glucose pentaacetate (Penta-O-acetyl-β-D-glucopyranose) 一种能够用于生化反应的物质。
T5S0669 Bergamottin

5-Geranoxypsoralen,Bergamotine,Bergaptin,佛手柑素

P450 Metabolism
Bergamottin (5-Geranoxypsoralen) 是竞争性CYP1A1抑制剂(Ki:10.703 nM)。
T4S0758 Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden

槲皮素-3-O-Β-D-葡萄糖-7-O-Β-D-龙胆双糖苷,Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside

Others Others
Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden (Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside) 是一种黄酮,来源于 Quercetin 中。
T2880 D-(+)-Cellobiose

Cellose,Beta-Cellobiose,D-纤维二糖,D-Cellobiose,Cellobiose

Others; Endogenous Metabolite Metabolism; Others
D-(+)-Cellobiose (Cellobiose) 是一种双糖,一种还原糖,由两个β-葡萄糖分子通过β(1→4)键连接而成。它可以被酶或酸水解成葡萄糖。
TN1166 1,3,6-Tri-O-galloyl-beta-D-glucose

1,3,6-三没食子酰葡萄糖,1,3,6-Tri-O-galloyl-β-D-glucose,1,3,6-Tri-O-galloylglucose,1,3,6-三-O-3,4,5-三羟基苯甲酰-BETA-D-葡萄糖

Immunology/Inflammation related Immunology/Inflammation
1,3,6-Tri-O-galloyl-beta-D-glucose (1,3,6-Tri-O-galloylglucose) 是一种酚类化合物,分离自Black Walnut Kernels 中。
T20255 L-Galactose

Galactose, L-

Endogenous Metabolite Metabolism
L-Galactose (Galactose, L-) 是一种天然产物,广泛存在动植物体内。L-Galactose 在Pistia stratiotes 中被证明是D-葡萄糖转化为草酸的分子途径中的关键中间体。
TN7217 4,6-Benzilidine-D-Glucose

4,6-Benzilidine-D-Glucose 是一种临床抗肿瘤化合物,在化学诱导肝细胞癌大鼠中显示出抗肿瘤活性。
T0887 D-Glucose

Dextrose,D-无水葡萄糖,Glucopyranose,Grape sugar,葡萄糖,D(+)-Glucose

Endogenous Metabolite Metabolism
D-Glucose (Glucopyranose) 是一种单糖。D-Glucose 是甜味剂,是一般代谢的关键组成部分,并作为与细胞代谢状态以及生物和非生物应激反应有关的关键信号分子。
T4733 Sucrose

D(+)-Sucrose,D-(+)-Saccharose,蔗糖

Others; Endogenous Metabolite Metabolism; Others
Sucrose (D-(+)-Saccharose) 是一种二糖,由果糖和葡萄糖组成。Sucrose 能够应用于一些动物模型,包括代谢性疾病、偏食、肥胖、糖尿病等。
T0800 Danthron

Dantron,1,8-Dihydroxyanthraquinone,1,8-二羟基蒽醌,丹蒽醌,Chrysazin,Antrapurol

Virus Protease; Antibacterial; AMPK; Autophagy Autophagy; Chromatin/Epigenetic; Microbiology/Virology; PI3K/Akt/mTOR signaling
Danthron (Antrapurol) 是一种从中药 rhubarb 中提取的天然产物,可通过激活 AMPK 来调节葡萄糖和脂质代谢。
T3794 Pentagalloylglucose

Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose,1,2,3,4,6-五没食子酰葡萄糖

Influenza Virus Microbiology/Virology
1,2,3,4,6-O-Pentagalloylglucose (Penta-O-galloyl-β-D-glucose) 存在于多种植物中,具有重要的药理作用。Pentagalloylglucose 表现出显著的抗狂犬病病毒 (RABV) 活性。
T3675 1-Deoxynojirimycin

Duvoglustat,Moranoline,1-脱氧野尻霉素,moranolin

PI3K; Glucosidase Metabolism; PI3K/Akt/mTOR signaling
1-Deoxynojirimycin (Moranoline) 是一种口服具有活性的 α-葡萄糖苷酶抑制剂。它具有降血糖、减肥和抗病毒的活性。它抑制餐后血糖,预防糖尿病。
T0586 Lactose

Others; Endogenous Metabolite Metabolism; Others
Lactose 是半乳糖和葡萄糖衍生的二糖,是大多数物种乳汁中的主要糖分,能够调节人类肠道的微生物菌群。
T19117 3-Deoxyglucosone

3-Deoxy-D-glucosone,2-keto-3-Deoxyglucose

GPX; Glucagon Receptor GPCR/G Protein; oxidation-reduction
3-Deoxyglucosone(3-Deoxy-D-glucosone) 是美拉德反应和多元醇反应的中间体途径合成。3-Deoxyglucosone 与蛋白质氨基快速反应形成晚期糖基化末端蛋白 (AGEs)。3-Deoxyglucosone 可使谷胱甘肽过氧化物酶失活,可与低葡萄糖协同作用以增强 GLP-1 分泌,可以作为糖尿病生物学检测的标志物。
T3386 Kaempferitrin

Lespedin,Kaempferol,Lespenephryl,Lespenefril,Kaempferol 3,7-dirhamnoside,山奈苷

cell cycle arrest; Glucokinase; IGF-1R Cell Cycle/Checkpoint; Metabolism; Tyrosine Kinase/Adaptors
Kaempferitrin (Lespenephryl) 是天然黄酮苷类化合物,具有缓解疼痛、抗糖尿病、消炎、抗肿瘤和化疗作用,可激活胰岛素信号传导。
T0592 D-Mannopyranose

Mannose,D-甘露糖

Others Others
D-Mannopyranose (Mannose) 是一种己糖或可发酵单糖,是甘露糖、水曲柳和相关植物的葡萄糖异构体。
T19615 α-Amylase

Amylase Metabolism
α-Amylase 是一种能够催化淀粉中 α-1,4-糖苷键水解的水解酶,使淀粉产生葡萄糖、麦芽糖等产物。
T3145 D-(+)-Trehalose dihydrate

Trehalose dihydrate,α,α-Trehalose dihydrate,alpha,alpha-Trehalose dihydrate,D-Trehalose dihydrate,二水合海藻糖

Others Others
D-(+)-Trehalose dihydrate (α,α-Trehalose dihydrate) 是分离自 Saccharomyces cerevisiae 中,可用作食品成分和药物赋形剂。
T5735 Methyl deacetylasperulosidate

Deacetyl asperulosidic acid methyl ester,6α-Hydroxygeniposide,去乙酰车叶草苷酸甲酯

Others Others
Methyl deacetylasperulosidate (6α-Hydroxygeniposide) 是环烯醚萜类化合物,能够降低正常小鼠的血糖水平,对小鼠具有通便作用。
T2914 D-Melibiose

Galalpha1-6Glcbeta,蜜二糖,Melibiose

Others; Endogenous Metabolite Metabolism; Others
D-Melibiose (Galalpha1-6Glcbeta) 是一种还原性二糖,由一个半乳糖和一个糖基组成 (1-6) 糖苷链构成的。
T3403 Glabridin

光甘草定,Q-100692,KB-289522,LS-176045

Reactive Oxygen Species; Tyrosinase; GABA Receptor; Antibacterial; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome
Glabridin (KB-289522) 能够结合并激活PPARγ,EC50值为 6115 nM,是一种从Glycyrrhiza glabra 中分到的异黄烷类天然产物。它具有抗炎、抗菌、抗肾炎、抗氧化、抗肿瘤、抗糖尿病、抗骨质疏松、保护神经、保护心血管、清除自由基等作用。
TN1740 Homoeriodictyol

高胜草酚,高圣草酚

5-HT Receptor; transporter; Sodium Channel; Drug Metabolite GPCR/G Protein; Membrane transporter/Ion channel; Metabolism; Neuroscience
Homoeriodictyol 是 Eriocitrin 的代谢物,属于黄酮类。Eriocitrin 是强效抗氧化剂。
T4514 N-Acetyl-D-Glucosamine

N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc

Endogenous Metabolite Metabolism
N-Acetyl-D-Glucosamine (NAG) 是葡萄糖的单糖衍生物。
T4929 L-2-Phosphoglyceric acid

L-GLYCERATE 3-PHOSPHATE 二钠盐,L-2-Phosphoglyceric acid disodium salt h

Others; Endogenous Metabolite Metabolism; Others
L-2-Phosphoglyceric acid (L-2-Phosphoglyceric acid disodium salt) 是内源性代谢产物的一种。
T2713 Stachyose tetrahydrate

Stachyose,D-Stachyose tetrahydrate,水苏糖

Apoptosis; Others Apoptosis; Others
Stachyose tetrahydrate (D-Stachyose tetrahydrate) 是一种功能性低聚糖,可在肠道内产生有益物质或通过促进益生菌的增殖,间接防止结肠癌细胞生长,可作为益生元。
T0591 D-Galactose

D-(+)-Galactose,alpha-D-半乳糖,D-半乳糖,D-Galactopyranose,Alpha-D-galactose

Endogenous Metabolite Metabolism
D-Galactose (Alpha-D-galactose) 是一种天然的己糖,是葡萄糖的C-4差向异构体。
T3S0309 D(+)-Raffinose pentahydrate

D-Raffinose pentahydrate,Raffinose,D(+)-五水棉子糖,五水棉子糖

Others; Endogenous Metabolite Metabolism; Others
D(+)-Raffinose pentahydrate (D-Raffinose pentahydrate) 是果糖,半乳糖和葡萄糖组成的三糖,天然存在于各种蔬菜和谷物中。D(+)-Raffinose pentahydrate 是一种功能性低聚糖。
T8144 Raffinose

Melitose,Melitriose,棉子糖

Others; Endogenous Metabolite Metabolism; Others
Raffinose (Melitriose) 是不能够消化的短链寡糖,是由半乳糖,葡萄糖和果糖组成的三糖,能够在许多植物中找到。它能够被 α-半乳糖苷酶 (α-GAL) 水解为 D-半乳糖和蔗糖。
T4785 Oxfenicine

4-羟基-L-苯甘氨酸,4-Hydroxy-L-phenylglycine

Others Others
Oxfenicine (4-Hydroxy-L-phenylglycine) 是具有口服活性的肉碱棕榈酰转移酶-1 抑制剂。它在缺血期间保护心脏免受坏死组织的损害。它可抑制心脏中脂肪酸的氧化。
T2P2919 (2S,3R,4S)-4-Hydroxyisoleucine

(4S)-4-Hydroxy-L-isoleucine,(4S)4-羟基异亮氨酸,Hydroxyisoleucine

PI3K PI3K/Akt/mTOR signaling
(2S,3R,4S)-4-Hydroxyisoleucine (Hydroxyisoleucine) 是分离自胡芦巴中的一种可口服的有效成分,具有抗糖尿病、抗糖尿病肾病的作用。
T5250 Levoglucosan

1,6-anhydro-b-D-Glucose,1,6-脱水-β-D-葡萄糖

Others; Endogenous Metabolite Metabolism; Others
Levoglucosan (1,6-anhydro-b-D-Glucose) 是一种无水己糖,是 β -D-葡萄糖的 1,6-无水衍生物。它是由碳水化合物,如淀粉和纤维素的热解形成的。左旋葡聚糖还可用于手性聚合物如不可水解葡萄糖聚合物的合成。左旋葡聚糖也可以通过糖的焦糖化产生。食用焦糖或含焦糖的甜食可导致尿中左旋葡聚糖水平短期增加5倍(从20 μm /mM肌酐增加到100 μm /mM肌酐)。
TN1275 p-Hydroxyphenethyl anisate

4-Hydroxyphenethylanisate

Others Others
p-Hydroxyphenethyl anisate (4-Hydroxyphenethylanisate) 是一种来自 Notopterygium forbe-siiBoiss 的天然产品,是一种新型聚合物缓释材料,与 AAPBA 嵌段共聚后, 制备的纳米颗粒具有良好的 Ph 敏感性、葡萄糖敏感性、胰岛素负载速率和稳定性。
T3332 Isosteviol

异甜菊醇,(-)-Isosteviol

IL Receptor; Potassium Channel; TNF; NF-κB; Reactive Oxygen Species; COX; Topoisomerase Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB
Isosteviol ((-)-Isosteviol) 是一种常见的天然甜味剂,属于四环二萜糖苷,是甜菊糖苷通过酸催化水解产生的。它抑制 DNA 聚合酶和 DNA 拓扑异构酶,具有抗菌、抗癌和抗结核作用。
TN6745 PALATINOSE

TNP-470,帕拉金糖水合物,Isomaltulose

Others Others
PALATINOSE (TNP-470) 是一种天然存在的二糖,由α-1,6-连接的葡萄糖和果糖组成。PALATINOSE 对肝脏代谢功能具有有益的影响,因此可能是蔗糖甜味剂的良好替代品。
TN1051 1-Caffeoylquinic acid

金银花,1-咖啡酰奎宁酸

NF-κB NF-κB
1-Caffeoylquinic acid 是一种有效的NF-κB 抑制剂,对 p105 的 RH 结构域显示高结合亲和力,Ki= 0.002 μM,结合能为 1.50 Kcal/mol。它抑制PD-1/PD-L1相互作用。它具有抗氧化应激能力。
T4875 Palatinose hydrate

6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物

Others; Endogenous Metabolite Metabolism; Others
Palatinose hydrate (6-O-α-D-Glucopyranosyl-D-fructose, Isoma) 是内源性代谢产物的一种。
TN1003 DL-Alanine

DL-2-Aminopropionic acid

Endogenous Metabolite Metabolism
DL-Alanine (DL-2-Aminopropionic acid) 是一种氨基酸,是L-和D-丙氨酸的外消旋化合物。DL-Alanine 与硝酸银水溶液一起用于纳米颗粒生成时常作为还原剂和封端剂。DL-Alanine 是一种甜味剂,可把它位与甘氨酸和糖精钠归为一类。DL-Alanine 在组织和肝脏之间的葡萄糖-丙氨酸循环中起重要作用。DL-Alanine 可用于研究 Cu、Zn、Cd 等过渡金属螯合。
T5S0384 Rhapontin

Ponticin,土大黄苷,Rhaponiticin,Rhaponticin,Rhapontigenin glucoside

Apoptosis; Others Apoptosis; Others
Rhapontin (Ponticin) 是药用大黄的一种成分,可减轻KK/Ay 糖尿病小鼠肝脏脂肪变性,改善血糖和血脂,表明其具有显着的降糖作用,有望成为治疗2型糖尿病及其并发症的新药。
TN2111 Prunin

Naringenin 7-0-glucoside,柚皮素-7-O-葡萄糖苷

Phosphatase; Anti-infection; Virus Protease Metabolism; Microbiology/Virology
Prunin (Naringenin 7-0-glucoside) 是一种人肠道病毒 A71 抑制剂。它抑制蛋白酪氨酸磷酸酶 1B,IC50值为 5.5 μM。
T13979 (S)-3-Hydroxybutanoic acid

L-β-Hydroxybutyric acid,(S)-β-Hydroxybutanoic acid,L-(+)-3-Hydroxybutyric acid,(S)-3-羟基丁酸

Endogenous Metabolite Metabolism
(S)-3-Hydroxybutanoic acid (L-(+)-3-Hydroxybutyric acid) 是一种正常的人体代谢产物,在患有抑郁症的老年患者中升高。它在人类的肝脏中由乙酰-CoA 合成,当血糖低时能够被脑用作能量来源。
T0332 D-Sorbitol

山梨醇,Glucitol,Sorbitol,D-Glucitol

Others; Endogenous Metabolite Metabolism; Others
D-Sorbitol (Sorbitol) 是一种六碳糖醇,能够用作糖的替代品。D-Sorbitol 能够用作稳定的赋形剂和/或等渗剂,保湿剂,增稠剂,甜味剂和膳食补充剂。
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天然产物

alpha-D-glucose
Cat.No: T4884
Synonym: α-D-Glucose,α-葡萄糖,alpha-Glucose,α-Dextrose
Target: Others, Endogenous Metabolite
α-D-Glucose-1-phosphate disodium
Cat.No: T4924
Synonym: A-D-葡萄糖-1-磷酸-二钠盐,α-D-Glucose 1-phosphate disodium salt hy,α-D-Glucopyranose 1-phosphate
Target: Others, Endogenous Metabolite
Concanavalin A
Cat.No: T4004
Synonym:
Target: Apoptosis
Isomaltose
Cat.No: T0581
Synonym: D-Isomaltose,6-O-α-D-Glucopyranosyl-D-glucose,低聚异麦芽糖900
Target: Others, Endogenous Metabolite
Uridine 5′-diphosphoglucose disodium salt
Cat.No: T4743
Synonym: 二磷酸尿苷葡萄糖二钠盐,UDP-Glucose sodium salt,UDPG sodium salt,UDP-α-D-Glucose sodium salt,Uridine 5'-diphosphoglucose disodium sal
Target: Endogenous Metabolite, P2Y Receptor
4,6-O-Ethylidene-α-D-glucose
Cat.No: T72172
Synonym: Ethylidene-glucose
Target:
α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)
Cat.No: T35415
Synonym:
Target:
Sennidin A
Cat.No: TN1033
Synonym:
Target: HCV Protease, transporter, Akt, PI3K
D-Glucose 6-phosphate disodium salt
Cat.No: T19262
Synonym: D-​Glucose ​6-​phosphate disodium salt
Target: Endogenous Metabolite
β-D-Glucose pentaacetate
Cat.No: T7997
Synonym: β-D-葡萄糖五乙酸酯,Penta-O-acetyl-β-D-glucopyranose,1,2,3,4,6-beta-D-葡萄糖五乙酸酯
Target: Others
Bergamottin
Cat.No: T5S0669
Synonym: 5-Geranoxypsoralen,Bergamotine,Bergaptin,佛手柑素
Target: P450
Quercetin-3-O-β-D-glucose-7-O-β-D-gentiobiosiden
Cat.No: T4S0758
Synonym: 槲皮素-3-O-Β-D-葡萄糖-7-O-Β-D-龙胆双糖苷,Quercetin-3-O-beta-D-glucose-7-O-beta-D-gentiobioside
Target: Others
D-(+)-Cellobiose
Cat.No: T2880
Synonym: Cellose,Beta-Cellobiose,D-纤维二糖,D-Cellobiose,Cellobiose
Target: Others, Endogenous Metabolite
1,3,6-Tri-O-galloyl-beta-D-glucose
Cat.No: TN1166
Synonym: 1,3,6-三没食子酰葡萄糖,1,3,6-Tri-O-galloyl-β-D-glucose,1,3,6-Tri-O-galloylglucose,1,3,6-三-O-3,4,5-三羟基苯甲酰-BETA-D-葡萄糖
Target: Immunology/Inflammation related
L-Galactose
Cat.No: T20255
Synonym: Galactose, L-
Target: Endogenous Metabolite
4,6-Benzilidine-D-Glucose
Cat.No: TN7217
Synonym:
Target:
D-Glucose
Cat.No: T0887
Synonym: Dextrose,D-无水葡萄糖,Glucopyranose,Grape sugar,葡萄糖,D(+)-Glucose
Target: Endogenous Metabolite
Sucrose
Cat.No: T4733
Synonym: D(+)-Sucrose,D-(+)-Saccharose,蔗糖
Target: Others, Endogenous Metabolite
Danthron
Cat.No: T0800
Synonym: Dantron,1,8-Dihydroxyanthraquinone,1,8-二羟基蒽醌,丹蒽醌,Chrysazin,Antrapurol
Target: Virus Protease, Antibacterial, AMPK, Autophagy
Pentagalloylglucose
Cat.No: T3794
Synonym: Penta-O-galloyl-β-D-glucose,1,2,3,4,6-O-Pentagalloylglucose,1,2,3,4,6-Penta-O-galloyl-beta-D-glucopyranose,1,2,3,4,6-五没食子酰葡萄糖
Target: Influenza Virus
1-Deoxynojirimycin
Cat.No: T3675
Synonym: Duvoglustat,Moranoline,1-脱氧野尻霉素,moranolin
Target: PI3K, Glucosidase
Lactose
Cat.No: T0586
Synonym:
Target: Others, Endogenous Metabolite
3-Deoxyglucosone
Cat.No: T19117
Synonym: 3-Deoxy-D-glucosone,2-keto-3-Deoxyglucose
Target: GPX, Glucagon Receptor
Kaempferitrin
Cat.No: T3386
Synonym: Lespedin,Kaempferol,Lespenephryl,Lespenefril,Kaempferol 3,7-dirhamnoside,山奈苷
Target: cell cycle arrest, Glucokinase, IGF-1R
D-Mannopyranose
Cat.No: T0592
Synonym: Mannose,D-甘露糖
Target: Others
α-Amylase
Cat.No: T19615
Synonym:
Target: Amylase
D-(+)-Trehalose dihydrate
Cat.No: T3145
Synonym: Trehalose dihydrate,α,α-Trehalose dihydrate,alpha,alpha-Trehalose dihydrate,D-Trehalose dihydrate,二水合海藻糖
Target: Others
Methyl deacetylasperulosidate
Cat.No: T5735
Synonym: Deacetyl asperulosidic acid methyl ester,6α-Hydroxygeniposide,去乙酰车叶草苷酸甲酯
Target: Others
D-Melibiose
Cat.No: T2914
Synonym: Galalpha1-6Glcbeta,蜜二糖,Melibiose
Target: Others, Endogenous Metabolite
Glabridin
Cat.No: T3403
Synonym: 光甘草定,Q-100692,KB-289522,LS-176045
Target: Reactive Oxygen Species, Tyrosinase, GABA Receptor, Antibacterial, PPAR
Homoeriodictyol
Cat.No: TN1740
Synonym: 高胜草酚,高圣草酚
Target: 5-HT Receptor, transporter, Sodium Channel, Drug Metabolite
N-Acetyl-D-Glucosamine
Cat.No: T4514
Synonym: N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc
Target: Endogenous Metabolite
L-2-Phosphoglyceric acid
Cat.No: T4929
Synonym: L-GLYCERATE 3-PHOSPHATE 二钠盐,L-2-Phosphoglyceric acid disodium salt h
Target: Others, Endogenous Metabolite
Stachyose tetrahydrate
Cat.No: T2713
Synonym: Stachyose,D-Stachyose tetrahydrate,水苏糖
Target: Apoptosis, Others
D-Galactose
Cat.No: T0591
Synonym: D-(+)-Galactose,alpha-D-半乳糖,D-半乳糖,D-Galactopyranose,Alpha-D-galactose
Target: Endogenous Metabolite
D(+)-Raffinose pentahydrate
Cat.No: T3S0309
Synonym: D-Raffinose pentahydrate,Raffinose,D(+)-五水棉子糖,五水棉子糖
Target: Others, Endogenous Metabolite
Raffinose
Cat.No: T8144
Synonym: Melitose,Melitriose,棉子糖
Target: Others, Endogenous Metabolite
Oxfenicine
Cat.No: T4785
Synonym: 4-羟基-L-苯甘氨酸,4-Hydroxy-L-phenylglycine
Target: Others
(2S,3R,4S)-4-Hydroxyisoleucine
Cat.No: T2P2919
Synonym: (4S)-4-Hydroxy-L-isoleucine,(4S)4-羟基异亮氨酸,Hydroxyisoleucine
Target: PI3K
Levoglucosan
Cat.No: T5250
Synonym: 1,6-anhydro-b-D-Glucose,1,6-脱水-β-D-葡萄糖
Target: Others, Endogenous Metabolite
p-Hydroxyphenethyl anisate
Cat.No: TN1275
Synonym: 4-Hydroxyphenethylanisate
Target: Others
Isosteviol
Cat.No: T3332
Synonym: 异甜菊醇,(-)-Isosteviol
Target: IL Receptor, Potassium Channel, TNF, NF-κB, Reactive Oxygen Species, COX, Topoisomerase
PALATINOSE
Cat.No: TN6745
Synonym: TNP-470,帕拉金糖水合物,Isomaltulose
Target: Others
1-Caffeoylquinic acid
Cat.No: TN1051
Synonym: 金银花,1-咖啡酰奎宁酸
Target: NF-κB
Palatinose hydrate
Cat.No: T4875
Synonym: 6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物
Target: Others, Endogenous Metabolite
DL-Alanine
Cat.No: TN1003
Synonym: DL-2-Aminopropionic acid
Target: Endogenous Metabolite
Rhapontin
Cat.No: T5S0384
Synonym: Ponticin,土大黄苷,Rhaponiticin,Rhaponticin,Rhapontigenin glucoside
Target: Apoptosis, Others
Prunin
Cat.No: TN2111
Synonym: Naringenin 7-0-glucoside,柚皮素-7-O-葡萄糖苷
Target: Phosphatase, Anti-infection, Virus Protease
(S)-3-Hydroxybutanoic acid
Cat.No: T13979
Synonym: L-β-Hydroxybutyric acid,(S)-β-Hydroxybutanoic acid,L-(+)-3-Hydroxybutyric acid,(S)-3-羟基丁酸
Target: Endogenous Metabolite
D-Sorbitol
Cat.No: T0332
Synonym: 山梨醇,Glucitol,Sorbitol,D-Glucitol
Target: Others, Endogenous Metabolite
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