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453

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
TQ0146 Ac-DEVD-CHO

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Ac-DEVD-CHO 是一种特异性 Caspase-3 抑制剂(Ki: 230 pM)。Ac-DEVD-CHO在 SLNT 诱导的细胞凋亡中有抑制作用。
TQ0146L Ac-DEVD-CHO acetate

Caspase-3 Inhibitor I,N-acetyl-asp-glu-val-asp-al,Ac-DEVD-CHO acetate (169332-60-9 free base),乙酰基-天冬氨酰-谷氨酰-缬氨酰-天冬氨醛

Caspase Apoptosis; Proteases/Proteasome
Caspase-3 Inhibitor I (N-acetyl-asp-glu-val-asp-al) 是 Caspase-3 的特异性抑制剂。
T41069 CHO-C-PEG2-C-CHO

CHO-C-PEG2-C-CHO

CHO-C-PEG2-C-CHO is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T80624 Ac-VAD-CHO

Ac-Val-Ala-Asp-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-VAD-CHO (Ac-Val-Ala-Asp-CHO)是一款caspase抑制剂,能够阻止缺氧细胞内MMP的降解以及细胞色素c的释出。
T80531 Ac-AAVALLPAVLLALLAP-DEVD-CHO

DEVD-CHO-CPP 32

Caspase Apoptosis; Proteases/Proteasome
DEVD-CHO-CPP 32(Ac-AAVALLPAVLLALLAP-DEVD-CHO)是一种高效且可逆的caspase-3抑制剂。
T78640 Z-LLF-CHO

Z-Leu-Leu-Phe-CHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-LLF-CHO(Z-Leu-Leu-Phe-CHO)为垂体多催化蛋白酶复合物所具有的胰凝乳蛋白酶样活性提供有效抑制,具有Ki值为460 nM。此外,Z-LLF-CHO同样作为NF-κB核转位的抑制剂。
T39722 CHO-CH2-PEG1-CH2-Boc

CHO-CH2-PEG1-CH2-Boc

CHO-CH2-PEG1-CH2-Boc is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules. This linker enables selective protein degradation by leveraging the ubiquitin-proteasome system within cells.
T83205 Ac-DNLD-CHO

Ac-Asp-Asn-Leu-Asp-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-DNLD-CHO(Ac-Asp-Asn-Leu-Asp-CHO)是一种有效的Caspase-3/7抑制剂,具有较低的IC50(分别为9.89, 245 nM)和Kiapp(分别为0.68、55.7 nM)。该化合物在研究caspase介导的细胞凋亡过程中具有重要应用价值,适用于神经退行性疾病和病毒感染疾病的相关研究。
T21617 MG-115

Z-LL-Nva-CHO

Proteasome Proteases/Proteasome; Ubiquitination
MG-115 (Z-LL-Nva-CHO) 是一种有效且可逆的蛋白酶体抑制剂,对20S 和26S 蛋白酶体的 Ki 值分别为 21 nM 和 35 nM。MG-115 特异性抑制蛋白酶体的胰凝乳蛋白酶样活性,诱导 p53 依赖性细胞凋亡。
T80735 Z-Gly-Pro-Phe-Leu-CHO

Z-GPFL-CHO

Proteasome Proteases/Proteasome; Ubiquitination
Z-Gly-Pro-Phe-Leu-CHO(Z-GPFL-CHO)是一种具有高选择性和高效率的四肽醛类蛋白酶体抑制剂,优先抑制支链氨基酸(Ki为1.5 µM),对小中性氨基酸的Ki值为2.3 µM,胰凝乳蛋白酶样活性的Ki值为40.5 µM,对肽基-谷氨酰肽水解活性的IC50为3.1 µM。
T2154 MG-132

Z-LLL-al,Z-Leu-Leu-Leu-CHO

Apoptosis; Proteasome; Autophagy Apoptosis; Autophagy; Proteases/Proteasome; Ubiquitination
MG-132 (Z-Leu-Leu-Leu-al) 是一种 26S 蛋白酶体抑制剂 (IC50=100 nM),具有细胞渗透性、可逆性。MG-132 可作为自噬激活剂,可诱导凋亡。
T78586L Ac-IETD-CHO TFA

Ac-IETD-CHO TFA(191338-86-0 Free base )

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Ac-IETD-CHO TFA 是一种 granzyme B 和 caspase-8 抑制剂,通过阻断 caspase3 前体裂解抑制 caspase8 活性。Ac-IETD-CHO TFA 抑制 Fas 介导的细胞凋亡(Apoptosis)。
T36368 2H-Cho-Arg (trifluoroacetate salt)

2H-Cho-Arg is a steroid-based cationic lipid that contains a 2H-cholesterol skeleton coupled to an L-arginine head group and can be used to facilitate gene transfection. It forms a complex with plasmid DNA (pDNA) and decreases pDNA migration in an electrophoretic mobility shift assay at +/- charge ratios of 4 or higher. 2H-Cho-Arg facilitates transfection of a luciferase gene into H1299 cells, an effect that is reversed by the lipid raft-mediated endocytosis inhibitor methyl-β-cyclodextrin and t...
T36350 Cho-Arg (trifluoroacetate salt)

Cho-Arg is a steroid-based cationic lipid that contains a cholesterol skeleton coupled to an L-arginine head group. It forms a complex with plasmid DNA and decreases plasmid DNA migration in an agarose-gel retardant assay at charge ratios greater than or equal to 4. Cho-Arg facilitates transfection of plasmid DNA into H1299 and HeLa cells in the presence or absence of fetal bovine serum, an effect that is reversed by the lipid raft-mediated endocytosis inhibitor methyl-β-cyclodextrin and the cav...
T41236 Z-FY-CHO

Z-FY-CHO (Z-Phe-Tyr-CHO) 是一种特异且有效的组织蛋白酶 L (CTSL) 抑制剂。
T29233 Z-LLNle-CHO

Z-LLNle-CHO is a cell permeable inhibitor of gamma-secretase. Z-LLNle-CHO induces apoptosis of human glioblastoma tumor-initiating cells by proteasome inhibition and mitotic arrest response.
T19883 Ac-YVAD-CHO

L 709049,L-709049,L709049

L 709049是一种生物活性化合物,它是白细胞介素-1β转化酶( Caspase-1)的选择性抑制剂。 Caspase 抑制剂可干扰细胞凋亡的启动,具有多种临床应用前景。
T6583 MG-101

ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I

Cysteine Protease; Proteasome Proteases/Proteasome; Ubiquitination
MG-101 (Calpain inhibitor I) 是一种有效的半胱氨酸蛋白酶抑制剂,能够抑制钙蛋白酶I (Ki:190 pM),钙蛋白酶II (Ki:220 pM),组织蛋白酶B (Ki:150 pM)和组织蛋白酶L (Ki:500 pM)。
T80513 YVAD-CHO

YVAD-CHO为白细胞介素-1β转换酶(ICE,caspase 1)的抑制剂,能够在一定程度上减缓面神经损伤小鼠运动神经元死亡速率。
T80467 Boc-AEVD-CHO

Caspase Apoptosis; Proteases/Proteasome
Boc-AEVD-CHO是一种Caspase 8抑制剂,适用于细胞凋亡以及免疫和炎症疾病研究。
T78622 Ac-VDVAD-CHO

Casein Kinase Metabolism; Stem Cells
Ac-VDVAD-CHO为caspase-2/3抑制剂,其IC50值分别为46 nM和15 nM。
T80093 IETD-CHO TFA

Caspase Apoptosis; Proteases/Proteasome
IETD-CHO TFA (Caspase-8-IN-1) 是一种高效的 caspase-8 抑制剂。
T80076 Ac-ESMD-CHO

Casein Kinase Metabolism; Stem Cells
Ac-ESMD-CHO是一种抑制caspase-3和caspase-7的化合物。该化合物能有效阻止caspase-3前体肽(CPP32)在Glu-Ser-Met-Asp(ESMD)位点发生的蛋白水解切割作用。
T78586 Ac-​IETD-​CHO

Apoptosis Apoptosis
Ac-IETD-CHO是一种针对granzyme B和caspase 8的有效可逆抑制剂,能够阻止Fas介导的(Apoptosis)、出血和肝衰竭,并且能够抑制细胞毒性T淋巴细胞引发的细胞死亡。
T80532 Ac-AAVALLPAVLLALLAP-YVAD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-YVAD-CHO为具备细胞穿透能力的caspase-1抑制剂,展现出抗肿瘤活性。
T80536 Ac-AAVALLPAVLLALLAP-LEVD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-LEVD-CHO是一caspase-4抑制剂,可穿透细胞膜,并表现出抗肿瘤特性。
T73852 Ac-YVAD-CHO acetate

Ac-YVAD-CHO(L-709049)醋酸盐是一种高效、可逆、特异的四肽白介素1β转化酶(ICE)抑制剂,小鼠和人类的Ki值分别为3.0 nM和0.76 nM。它同时也能抑制caspase-1,从而抑制成熟IL-lβ的产生。
T73683 AC-VEID-CHO TFA

AC-VEID-CHO (TFA) 是一种源自多肽的半胱天冬酶抑制剂,针对Caspase-6、Caspase-3和Caspase-7展示出优异的抑制效果,其IC50值分别为16.2 nM、13.6 nM和162.1 nM。该化合物常用于研究阿尔茨海默病、亨廷顿病等神经退行性疾病。
T80537 Ac-AAVALLPAVLLALLAP-LEHD-CHO

Caspase Apoptosis; Proteases/Proteasome
Ac-AAVALLPAVLLALLAP-LEHD-CHO 是半胱天冬酶4、5和9的抑制剂,能够对Neocarzinostatin处理的MCF-7细胞展现保护效果。
T78619 Z-Pro-Pro-CHO

Prolyl Endopeptidase (PREP) Metabolism; Proteases/Proteasome
Z-Pro-Pro-CHO为一种有效的脯氨酰寡肽酶抑制剂,其具有针对人类及曼氏血吸虫脯氨酰寡肽酶的较低半抑制浓度(IC50),分别为0.16 μM和0.01 μM。
T17281 Z-Ile-Leu-aldehyde

Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII

Others Others
Z-Ile-Leu-aldehyde is an effective and competitive peptide aldehyde inhibitor of γ-secretase and notch.
T8566 AA92593

Others Others
AA92593 是一种选择性的 OPN4 (melanopsin)竞争性拮抗剂。
T38240 2,6-Dichlorodiphenylamine

Antibacterial Microbiology/Virology
2,6-Dichlorodiphenylamine 是双氯芬酸钠的一种结构类似物,显示出抗白色念珠菌活性。2,6-Dichlorodiphenylamine 是非选择性抗炎剂,为COX 的抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50分别为 4 和 1.3 nM。
T3306 PF-04418948

PF 04418948,PF04418948

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
PF-04418948 是一种可口服的,选择性的前列腺素EP2受体拮抗剂,IC50为16 nM。
T0432 Diclofenac diethylamine

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac diethylamine 是非选择性抗炎剂,通过活化 caspase 级联反应来诱导神经干细胞凋亡。它是一种COX 抑制剂,在 CHO 细胞中,对人COX-1和COX-2的IC50值分别为 4 和 1.3 nM。它对绵羊COX-1和COX-2的IC50值分别为 5.1 μM 和0.84 μM。
T1671 Mirabegron

YM178,米拉贝隆

Adrenergic Receptor GPCR/G Protein; Neuroscience
Mirabegron (YM178) 是选择性的肾上腺素受体激动剂,EC50=22.4 nM。
T9927 Panitumumab

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Panitumumab 是一种重组全人源 IgG2 单克隆抗体,可与表皮生长因子(EGFR)结合,具有抗肿瘤活性。
T8991 BMS986187

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
BMS986187 是一种有效的δ-阿片受体选择性正变构调节剂 (PAM),其 EC50= 0.03 μM,pKB= 6.02 (~1 μM)。BMS986187 对 μ 受体无明显 PAM 活性 (EC50=3 μM)。
T2667 PIK-75

Apoptosis; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK75 是一种可逆的DNA-PK 和p110α-选择性的抑制剂,抑制 DNA-PK、p110α 和 p110γ,IC50分别为 2、5.8 和 76 nM。它诱导凋亡,抑制 p110α 效果比抑制 p110β 高 200 多倍,p110β的IC50为 1.3 μM。
T1555 Diclofenac sodium

GP 45840,双氯芬酸钠

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac sodium (GP 45840) 是一种非选择性抗炎剂,是 COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的 IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的 IC50值分别为 5.1 μM,0.84 μM。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。
T6470 Diclofenac Potassium

双氯芬酸钾,CGP-45840B,Cataflam,Voltfast

Apoptosis; Others; COX Apoptosis; Immunology/Inflammation; Neuroscience; Others
Diclofenac Potassium (CGP-45840B) 是一种非甾体抗炎药,用于减轻炎症并在某些情况下作为镇痛剂减轻疼痛。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。它是一种COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的IC50值分别为 5.1 μM 和0.84 μM。
T0196 Diclofenac

双氯芬酸,奥尔芬,Diclofenacum,Voltaren

Apoptosis; COX Apoptosis; Immunology/Inflammation; Neuroscience
Diclofenac (Diclofenacum) 是一种具有抗炎活性的非甾体苯乙酸衍生物,是 COX 抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的 IC50值分别为 4 和 1.3 nM。它对绵羊 COX-1 和 COX-2 的 IC50值分别为 5.1 μM,0.84 μM。它通过活化 caspase 级联反应来诱导神经干细胞凋亡。
T6905 Netupitant

Ro 67-31898/000,奈妥吡坦,CID 6451149

Neurokinin receptor GPCR/G Protein; Neuroscience
Netupitant (CID 6451149) 是一种高效选择性、可口服的神经激肽 1 受体 (NK1) 拮抗剂,具有止吐作用,在 CHO 细胞中对 hNK1的 Ki 值为 0.95 nM。
T1566 Aripiprazole

阿立哌唑,OPC-14597

5-HT Receptor GPCR/G Protein; Neuroscience
Aripiprazole (OPC-14597) 是血清素受体 5-HT1A 和多巴胺 D2 受体的部分激动剂,还用作突触后拮抗剂和血清素受体 5-HT2A 的拮抗剂。
T6140 SB-334867 free base

SB334867A free base,SB-334867,SB 334867,SB334867

OX Receptor GPCR/G Protein; Neuroscience
SB-334867 free base (SB334867A free base) 是一种选择性 orexin-1(OX1) 受体拮抗剂,对 OX2有选择性,pKb 为7.4,对 5-HT2B、5-HT2C 的选择性是 100 倍,pKi 值分别为 5.4 和 5.3。它减少乙醇消耗,还抑制吗啡诱导的体内运动活动敏感性的获得。
T23386 SR 142948

Neurotensin Receptor GPCR/G Protein
SR 142948 是一种神经降压素 (NT) 受体拮抗剂。
T2287 PIK-75 hydrochloride

PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75

Apoptosis; DNA-PK; PI3K Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PIK-75 hydrochloride (PIK-75 HCl) 是一种可逆的 DNA-PK 和 p110α-选择性抑制剂,抑制 DNA-PK,p110α和 p110γ,可诱导凋亡。
T6684 Succinylcholine Chloride Dihydrate

choline chloride succinate,Succinyldicholine dichloride,Suxamethonium Chloride Dihydrate,司可林

AChR Neuroscience
Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) 是一种烟碱型 AChR 激动剂,也可作为去极化神经肌肉阻滞剂。
TP2419 V-9-M Cholecystokinin nonapeptide

V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M

Beta Amyloid Neuroscience
V-9-M Cholecystokinin nonapeptide (Prepro CCK Fragment V-9-M) 是胆囊收缩素(CCK)的前体化合物。胆囊收缩素(CCK)是一种刺激胆囊收缩和胰腺外分泌的脑肠肽,可从狗和猫的小肠中提取的,可以引起胆囊收缩。
T2227 Hemicholinium 3

半胆碱基-3,Hemicholinium-3,Hemicholine

Others; AChE Neuroscience; Others
Hemicholinium 3 是一种竞争性的、高亲和力的胆碱转运蛋白 (HACU) 抑制剂,Ki=25 nM。它是一种神经肌肉阻滞剂,能够抑制乙酰胆碱 (ACh)的合成和释放。它抑制Epibatidine 诱发的收缩和 [3H] 乙酰胆碱释放,IC50分别为 897 nM 和 693 nM。

化合物

Ac-DEVD-CHO
Cat.No: TQ0146
Synonym:
Target: Apoptosis, Caspase
Ac-DEVD-CHO acetate
Cat.No: TQ0146L
Synonym: Caspase-3 Inhibitor I,N-acetyl-asp-glu-val-asp-al,Ac-DEVD-CHO acetate (169332-60-9 free base),乙酰基-天冬氨酰-谷氨酰-缬氨酰-天冬氨醛
Target: Caspase
CHO-C-PEG2-C-CHO
Cat.No: T41069
Synonym: CHO-C-PEG2-C-CHO
Target:
Ac-VAD-CHO
Cat.No: T80624
Synonym: Ac-Val-Ala-Asp-CHO
Target: Caspase
Ac-AAVALLPAVLLALLAP-DEVD-CHO
Cat.No: T80531
Synonym: DEVD-CHO-CPP 32
Target: Caspase
Z-LLF-CHO
Cat.No: T78640
Synonym: Z-Leu-Leu-Phe-CHO
Target: Proteasome
CHO-CH2-PEG1-CH2-Boc
Cat.No: T39722
Synonym: CHO-CH2-PEG1-CH2-Boc
Target:
Ac-DNLD-CHO
Cat.No: T83205
Synonym: Ac-Asp-Asn-Leu-Asp-CHO
Target: Caspase
MG-115
Cat.No: T21617
Synonym: Z-LL-Nva-CHO
Target: Proteasome
Z-Gly-Pro-Phe-Leu-CHO
Cat.No: T80735
Synonym: Z-GPFL-CHO
Target: Proteasome
MG-132
Cat.No: T2154
Synonym: Z-LLL-al,Z-Leu-Leu-Leu-CHO
Target: Apoptosis, Proteasome, Autophagy
Ac-IETD-CHO TFA
Cat.No: T78586L
Synonym: Ac-IETD-CHO TFA(191338-86-0 Free base )
Target: Apoptosis, Caspase
2H-Cho-Arg (trifluoroacetate salt)
Cat.No: T36368
Synonym:
Target:
Cho-Arg (trifluoroacetate salt)
Cat.No: T36350
Synonym:
Target:
Z-FY-CHO
Cat.No: T41236
Synonym:
Target:
Z-LLNle-CHO
Cat.No: T29233
Synonym:
Target:
Ac-YVAD-CHO
Cat.No: T19883
Synonym: L 709049,L-709049,L709049
Target:
MG-101
Cat.No: T6583
Synonym: ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I
Target: Cysteine Protease, Proteasome
YVAD-CHO
Cat.No: T80513
Synonym:
Target:
Boc-AEVD-CHO
Cat.No: T80467
Synonym:
Target: Caspase
Ac-VDVAD-CHO
Cat.No: T78622
Synonym:
Target: Casein Kinase
IETD-CHO TFA
Cat.No: T80093
Synonym:
Target: Caspase
Ac-ESMD-CHO
Cat.No: T80076
Synonym:
Target: Casein Kinase
Ac-​IETD-​CHO
Cat.No: T78586
Synonym:
Target: Apoptosis
Ac-AAVALLPAVLLALLAP-YVAD-CHO
Cat.No: T80532
Synonym:
Target: Caspase
Ac-AAVALLPAVLLALLAP-LEVD-CHO
Cat.No: T80536
Synonym:
Target: Caspase
Ac-YVAD-CHO acetate
Cat.No: T73852
Synonym:
Target:
AC-VEID-CHO TFA
Cat.No: T73683
Synonym:
Target:
Ac-AAVALLPAVLLALLAP-LEHD-CHO
Cat.No: T80537
Synonym:
Target: Caspase
Z-Pro-Pro-CHO
Cat.No: T78619
Synonym:
Target: Prolyl Endopeptidase (PREP)
Z-Ile-Leu-aldehyde
Cat.No: T17281
Synonym: Z-IL-CHO,GSI-XII,γ-Secretase inhibitor XII
Target: Others
AA92593
Cat.No: T8566
Synonym:
Target: Others
2,6-Dichlorodiphenylamine
Cat.No: T38240
Synonym:
Target: Antibacterial
PF-04418948
Cat.No: T3306
Synonym: PF 04418948,PF04418948
Target: Prostaglandin Receptor
Diclofenac diethylamine
Cat.No: T0432
Synonym:
Target: Apoptosis, COX
Mirabegron
Cat.No: T1671
Synonym: YM178,米拉贝隆
Target: Adrenergic Receptor
Panitumumab
Cat.No: T9927
Synonym:
Target: EGFR
BMS986187
Cat.No: T8991
Synonym:
Target: Opioid Receptor
PIK-75
Cat.No: T2667
Synonym:
Target: Apoptosis, DNA-PK, PI3K
Diclofenac sodium
Cat.No: T1555
Synonym: GP 45840,双氯芬酸钠
Target: Apoptosis, COX
Diclofenac Potassium
Cat.No: T6470
Synonym: 双氯芬酸钾,CGP-45840B,Cataflam,Voltfast
Target: Apoptosis, Others, COX
Diclofenac
Cat.No: T0196
Synonym: 双氯芬酸,奥尔芬,Diclofenacum,Voltaren
Target: Apoptosis, COX
Netupitant
Cat.No: T6905
Synonym: Ro 67-31898/000,奈妥吡坦,CID 6451149
Target: Neurokinin receptor
Aripiprazole
Cat.No: T1566
Synonym: 阿立哌唑,OPC-14597
Target: 5-HT Receptor
SB-334867 free base
Cat.No: T6140
Synonym: SB334867A free base,SB-334867,SB 334867,SB334867
Target: OX Receptor
SR 142948
Cat.No: T23386
Synonym:
Target: Neurotensin Receptor
PIK-75 hydrochloride
Cat.No: T2287
Synonym: PIK-75 HCl,2-甲基-5-硝基苯磺酸 [(6-溴咪唑并[1,2-a]吡啶-3-基)亚甲基]甲基肼盐酸盐,PIK-75
Target: Apoptosis, DNA-PK, PI3K
Succinylcholine Chloride Dihydrate
Cat.No: T6684
Synonym: choline chloride succinate,Succinyldicholine dichloride,Suxamethonium Chloride Dihydrate,司可林
Target: AChR
V-9-M Cholecystokinin nonapeptide
Cat.No: TP2419
Synonym: V 9 M,Prepro CCK Fragment V-9-M,Val-pro-val-glu-ala-val-asp-pro-met,Cholecystokinin Precursor (24-32),V9M,V-9-M
Target: Beta Amyloid
Hemicholinium 3
Cat.No: T2227
Synonym: 半胆碱基-3,Hemicholinium-3,Hemicholine
Target: Others, AChE
Cat. No. Product Name Target Signaling Pathways
T5214 Cholesteryl linoleate

CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯

Others; Endogenous Metabolite Metabolism; Others
Cholesteryl linoleate (Linoleic Acid cholesteryl ester) 是低密度脂蛋白和动脉粥样硬化病变中主要的胆固醇酯。它存在于 LDL 中的胆固醇酯,利用 LDL 受体相关蛋白转移到表达 15-脂氧合酶的巨噬细胞和 CHO 细胞的质膜,被氧化形成胆固醇亚油酸氢过氧化物。
T2968 Hyodeoxycholic acid

NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA

FXR; Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Hyodeoxycholic acid (NSC 60672) 是由肠道菌群在小肠中形成的次级胆汁酸,是TGR5(GPCR19)的激动剂, CHO 细胞中的EC50=31.6 µM。它已用于研究高胆固醇血症的治疗。
T6805 Choline bitartrate

2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium,酒石酸氢胆碱

Others; AChR Neuroscience; Others
Choline bitartrate (2-hydroxyethyl(trimethyl)azanium) 是一种存在于食物中的营养胆碱,可影响肝脏疾病、动脉粥样硬化和神经系统疾病等疾病。它是神经递质乙酰胆碱的前体,作为甲基供体参与各种代谢过程和脂质代谢。
T4717 25-Hydroxycholesterol

25-羟基胆固醇,25-羟基胆甾醇

Others; Endogenous Metabolite; HMG-CoA Reductase Metabolism; Others
25-Hydroxycholesterol 是胆固醇的代谢产物,由巨噬细胞响应 Toll 样受体激活而分泌。它有效抑制 B 细胞产生 IgA,EC50约为 65 nM。
T19124 3-​Oxocholic acid

3-Ketocholic acid

Endogenous Metabolite Metabolism
3-​Oxocholic acid(3-Ketocholic acid) 是胆汁酸的代谢产物,也是产气荚膜梭菌在肠道中由胆汁降解的主要产物。33-​Oxocholic acid 是一种主要存在于哺乳动物的胆汁中类固醇酸。
T6751 Acetylcholine iodide

Acetylcolina

Others Others
Acetylcholine iodide (Acetylcolina) 是一种在中枢和外周神经系统中常见的神经递质。
T5240 Cholestenone

胆甾烯酮,4-胆甾烯-3-酮,(+)-4-Cholesten-3-one

Others; Endogenous Metabolite Metabolism; Others
Cholestenone ((+)-4-Cholesten-3-one) 是胆固醇的中间氧化产物,主要在肝脏中代谢。它能够会导致细胞长期功能缺陷。它在膜中具有很高的流动性,会影响胆固醇的翻转和外排。
TN2349 Taurodeoxycholate sodium salt

Sodium taurodeoxylate,牛磺脱氧胆酸钠

Endogenous Metabolite Metabolism
Taurodeoxycholate sodium salt (Sodium taurodeoxylate) 是胆盐相关的阴离子洗涤剂,用于分离膜蛋白,包括线粒体内膜蛋白。它还可以抑制各种炎症反应。
TJA2398 Taurodeoxycholic acid sodium hydrate

Sodium taurodeoxycholate monohydrate,Taurodeoxychloic Acid sodium hydrate,Taurohyodeoxycholic acid sodium salt,牛磺猪去氧胆酸

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Taurodeoxycholic acid sodium hydrate (Sodium taurodeoxycholate monohydrate) 通过阻断钙介导的凋亡通路和 Caspase-12的活化来阻止细胞凋亡。它可用于原发性胆汁性肝硬化、胰岛素抵抗、淀粉样变性、囊性纤维化、胆汁淤积和肌萎缩侧索硬化症。
T3742 3-Methylcatechol

3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene

Others Others
3-Methylcatechol (2,3-Toluenediol) 是由 Pseudomonas putidaMC2 产生,能够用作化学合成中的分子砌块。
T40646 Lipoteichoic acid

Complement System Immunology/Inflammation
Lipoteichoic acid 是 Staphylococcus aureus 细胞壁的聚合物,通过诱导 C3 和抑制 CD55 来激活补体系统,通过 IGF-1 途径减少脂肪沉积。
TN2215 Taurochenodeoxycholic acid sodium

牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
Taurochenodeoxycholic acid sodium (Sodium taurochenodeoxycholate) 是动物胆汁酸的主要生物活性物质之一。它可诱导细胞凋亡,具有抗炎和免疫调节作用。
T2962 5α-Cholestan-3β-ol

Dihydrocholesterol,Zymostanol,5α-Cholestanol,5alpha-Cholestanol,NSC 18188,Beta-Cholestanol,二氢胆甾醇

Others; Endogenous Metabolite Metabolism; Others
5α-Cholestan-3β-ol (NSC 18188) 是衍生化的类固醇化合物的一种。
T7628 3b-Hydroxy-5-cholenoic acid

Endogenous Metabolite Metabolism
3b-Hydroxy-5-cholenoic acid 是内源性的单羟基胆酸的一种,大量崔乃在于患有肝胆管状发育不全的儿童体内。
TN3651 Cichoriin

Others Others
Cichoriin 对SARS-CoV-2有明显活性,是治疗重症COVID-19的潜在候选物质。
T4713 Phosphorylcholine chloride calcium salt tetrahydrate

Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate

Others; Endogenous Metabolite Metabolism; Others
Phosphorylcholine chloride calcium salt tetrahydrate (Phosphocholine chloride calcium salt tet) 是内源性代谢产物的一种。
T9510 1,2-Distearoyl-sn-glycero-3-phosphorylcholine

DSPC,L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL,1,2-Distearoyl-sn-glycero-3-PC,二硬脂酰磷脂酰胆碱

Others Others
1,2-Distearoyl-sn-glycero-3-phosphorylcholine (L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL) 是一种脂质纳米颗粒(LNP) 系统中的脂质成分,可用于合成脂质体。
T1317 Cinchonidine

奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine

5-HT Receptor; Serotonin Transporter; Parasite GPCR/G Protein; Microbiology/Virology; Neuroscience
Cinchonidine (L-Cinchonidine) 是在金鸡纳和角蒿中发现的一种生物碱,有抗疟活性。 它是用于有机化学中不对称合成的砌块,是血清素转运蛋白的弱抑制剂。
T5077 Deoxycholic acid sodium salt

脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid sodium salt (Sodium deoxycholate) 是 G 蛋白偶联胆汁酸受体TGR5的激活剂。
T4727 Taurolithocholic acid sodium salt

牛磺石胆酸钠,Sodium taurolithocholate

Others; Calcium Channel Membrane transporter/Ion channel; Metabolism; Others
Taurolithocholic acid sodium salt (Sodium taurolithocholate) 是抑胆剂和 Ca2+激动剂,可抑制放射性配体与毒蕈碱 M1 结合。
TQ0274 27-Hydroxycholesterol

27-羟基胆固醇,5,25R-胆甾烯-3BETA,26-二醇,25(R)-27-hydroxy Cholesterol

Estrogen/progestogen Receptor; Liver X Receptor Endocrinology/Hormones; Metabolism
27-Hydroxycholesterol (25(R)-27-hydroxy Cholesterol) 是一种有效的、选择性的雌激素受体调节剂和肝X 受体激动剂。
TN7235 4-methoxylonchocarpin

TNF; NF-κB Apoptosis; NF-κB
4-methoxylonchocarpin 是从Abrus precatorius 的根中分离出来的以一种有效的抗炎化合物。4-methoxylonchocarpin 通过抑制LPS 与巨噬细胞的TLR4结合来抑制NF-κB 激活TNF 表达,抑制TNBS 引起的小鼠结肠炎。
T19189 Allocholic acid

Others Others
Allocholic acid 是一种胆汁酸,在脊椎动物中发现,在肝脏再生和致癌过程中会重新出现,也是成熟嗅觉系统的特定性刺激物。
T4136 Lapachol

Bethabarra wood,CI75490,黄钟花醌,Greenhartin,Tecomin

Others; Influenza Virus; Antibacterial; Parasite; Antifungal Microbiology/Virology; Others
Lapachol (CI75490) 是从Tabebuia avellanedae 中分离得到的一种萘醌。它具有具有抗菌、抗炎、镇痛、抗肿瘤和抗生素特性。
T8092 Taurohyodeoxycholic acid sodium salt

Sodium taurohyodeoxycholate hydrate

Caspase Apoptosis; Proteases/Proteasome
Taurohyodeoxycholic acid sodium salt (Sodium taurohyodeoxycholate hydrate) 通过阻断钙介导的细胞凋亡途径以及 Caspase-12 活化来防止细胞凋亡
T8712 1-Palmitoyl-sn-glycero-3-phosphocholine

1-十六酰-SN-丙三醇-磷酸胆碱,1-Hexadecanoyl-sn-glycero-3-phosphocholine

Others Others
1-Palmitoyl-sn-glycero-3-phosphocholine (1-Hexadecanoyl-sn-glycero-3-phosphocholine) 是一种用于荧光探针设计的磷酸胆碱。
T5072 Glycocholic acid hydrate

Others; Endogenous Metabolite Metabolism; Others
Glycocholic acid hydrate 是内源性代谢产物的一种。
T6S0659 Rhynchophylline

钩藤碱,Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin

Calcium Channel; NF-κB Membrane transporter/Ion channel; Metabolism; NF-κB
Rhynchophylline (Mitrinermine) 是一种生物碱类化合物,从钩藤中分离得到,具有很高的生物活性,被广泛用于抗炎、神经保护等方面的研究。
T2S0142 4-Hydroxylonchocarpin

异补骨脂色烯查耳酮,Isobavachromene

Others Others
Isobavachromene is a natural product from Psoralea corylifolia
T5352 GLYCODEOXYCHOLIC ACID

Others; Endogenous Metabolite Metabolism; Others
Glycodeoxycholic Acid 是内源性代谢产物的一种。
T31964 Glycolithocholic acid

Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine

Others Others
Glycolithocholic acid (Lithocholic acid glycine conjugate) 属于内源性代谢产物,是甘氨酸结合的次级胆汁酸。它可用于诊断非酒精性脂肪性肝炎,溃疡性结肠炎和原发性硬化性胆管炎。
T75319 Taurodeoxycholic acid

Taurodeoxychloic acid

Apoptosis; Calcium Channel; Caspase Apoptosis; Membrane transporter/Ion channel; Metabolism; Proteases/Proteasome
Taurodeoxycholic acid (Taurodeoxychloic acid) 是脱氧胆酸的胆汁酸牛磺酸共轭物,是一种人体代谢物,可稳定线粒体膜,减少自由基形成。Taurodeoxycholic acid 通过阻断钙介导的凋亡通路以及 Caspase-12 激活来抑制凋亡 (apoptosis)。Taurodeoxycholic acid具有神经保护活性,可用于研究 3-硝基丙酸诱导或稳定遗传的亨廷顿舞蹈病 (HD) 。
T10085 20(S)-Hydroxycholesterol

20α-Hydroxycholesterol

Smo Stem Cells
20(S)-Hydroxycholesterol (20α-Hydroxycholesterol) 是平滑 (smo) 癌蛋白的变构激活剂。
T13505 3α,12β-Dihydroxycholanoic acid

Others Others
3α,12β-Dihydroxycholanoic acid, a bile acid, can be isolated from urine specimens of healthy humans.
TN7024 Hyocholic acid

Hyocholic acid 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN7024,CAS号为 547-75-1。
T2744 Methyl Cholate

胆酸甲酯,Cholic acid methyl ester

Others Others
Methyl Cholate (Cholic acid methyl ester) 是胆酸的甲酯形式。其中胆酸是一种由肝脏产生的主要胆汁酸,由胆固醇合成。
T2965 Deoxycholic acid

Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic

Endogenous Metabolite; GPCR19 GPCR/G Protein; Metabolism
Deoxycholic acid (Cholanoic Acid) 是 G 蛋白偶联胆汁酸受体 TGR5的激活剂。
T0760 Cholesterol

Cholesterin,Cholesteryl alcohol,胆固醇

Estrogen Receptor/ERR; MRP; Endogenous Metabolite; ROR Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Cholesterol (Cholesteryl alcohol) 属于天然产物,是哺乳动物中的主要固醇,是一种雌激素相关受体 α (ERRα) 的激动剂。Cholesterol 广泛存在于动物的细胞膜,也是合成几种重要荷尔蒙及胆酸的材料。
T2963 Cholic Acid

Cholanic acid,胆汁酸,Cholate,Colalin

Endogenous Metabolite Metabolism
Cholic Acid (Cholate) 是肝脏产生的主要胆汁酸,与牛磺酸或甘氨酸缀合,有助于脂肪吸收和胆固醇排泄。
T8714 1-Stearoyl-sn-glycero-3-phosphocholine

1-硬脂酰-SN-甘油-3-磷酰胆碱,1-stearoyl-lysophosphatidylcholine,L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY

Others Others
1-Stearoyl-sn-glycero-3-phosphocholine (L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY) 是一种用于脂质代谢研究的化学物质。
T36585 Isodeoxycholic Acid

isoDCA

Chloride channel; Antibacterial Membrane transporter/Ion channel; Microbiology/Virology
Isodeoxycholic Acid 是一种胆汁酸,由肠道细菌通过脱氧胆酸的表聚作用形成。Isodeoxycholic acid 的临界胶束浓度高于二氯苯甲醚,这表明它的去污活性降低了,而且在抑制七种肠道共生细菌生长方面的活性低于二氯苯甲醚。Isodeoxycholic Acid(0.1%)能抑制几种艰难梭菌菌株在牛磺胆酸诱导下的孢子萌发,并能降低艰难梭菌培养上清对 Vero 细胞的细胞毒性。在高脂饮食诱发肥胖的大鼠模型中,血浆中的Isodeoxycholic acid 水平比正常饮食的大鼠低。
TN1641 (-)-Fenchone

Others; Antioxidant; Antifungal Microbiology/Virology; Others; oxidation-reduction
(-)-Fenchone 是一种双环单萜类化合物,广泛分布于植物中,可从Foeniculum vulgare 和Peumus boldus 中提取。(-)-Fenchone 具有广泛的生物活性,包括抗氧化,伤口愈合,止泻,抗真菌,抗伤害感受和支气管扩张剂活性。(-)-Fenchone 是一种潜在的抗肿瘤化合物。
T1138 Taurocholic acid sodium salt hydrate

牛胆酸钠,牛磺胆酸钠水合物,Sodium taurocholate hydrate,Taurocholic Acid sodium hydrate

Others; Potassium Channel; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Others
Taurocholic acid sodium salt hydrate (Sodium taurocholate hydrate) 是一种胆汁酸钠盐水合物,作用是参与脂肪的乳化。
TN1274 4-Allylcatechol

2-羟基胡椒酚,4-Allylpyrocatechol,Hydroxychavicol

Others Others
4-Allylcatechol (Hydroxychavicol) 是合成黄樟素的一种中间体。
T10086 24-Hydroxycholesterol

Cholest-5-ene-3beta,24-diol

Liver X Receptor; NMDAR Metabolism; Neuroscience
24-Hydroxycholesterol (Cholest-5-ene-3beta,24-diol) 是一种氧甾醇化合物,是一种 n-甲基-d-天门冬氨酸受体 (NMDA) 和转录因子 LXR 的激活剂,可用于研究心血管生成和胰腺癌。
T1039 Choline chloride

Biocolina,Biocoline,Hepacholine,氯化胆碱

AChR Neuroscience
Choline chloride (Biocoline) 是一种必需营养素,可激活 α7 烟碱受体,具有抗炎、镇痛的活性。对动脉粥样硬化、神经系统疾病和肝脏疾病等具有影响。
T22293 Chondroitine sulfate

Chondroitine sulfate (From cattle)

Others Others
Chondroitine sulfate 是软骨的重要结构成分,已被用作治疗关节不适的膳食补充剂。
T8040 Cholesterol myristate

胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate

Others; Potassium Channel; GABA Receptor; Endogenous Metabolite; AChR Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
Cholesterol myristate (Cholesteryl myristate) 是粗吻海龙中的一种类固醇,可与多种离子通道结合,例如nAChR、GABAA 受体和内向整流钾离子通道。
T8713 1-Oleoyl-sn-glycero-3-phosphocholine

Others Others
1-Oleoyl-sn-glycero-3-phosphocholine 是分析溶血卵磷脂的参考。
T19161 7α-Hydroxycholesterol

Others Others
7α-Hydroxycholesterol 是一种由酶促氧化和非酶促氧化形成的胆固醇氧化物,可用作脂质过氧化的生物标志物。
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天然产物

Cholesteryl linoleate
Cat.No: T5214
Synonym: CE(18:2(9Z,12Z)),Cholesterol Linoleate,Linoleic Acid cholesteryl ester,胆甾烯基亚油酸酯
Target: Others, Endogenous Metabolite
Hyodeoxycholic acid
Cat.No: T2968
Synonym: NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA
Target: FXR, Endogenous Metabolite, GPCR19
Choline bitartrate
Cat.No: T6805
Synonym: 2,3,4-trihydroxy-4-oxobutanoate,2-hydroxyethyl(trimethyl)azanium,酒石酸氢胆碱
Target: Others, AChR
25-Hydroxycholesterol
Cat.No: T4717
Synonym: 25-羟基胆固醇,25-羟基胆甾醇
Target: Others, Endogenous Metabolite, HMG-CoA Reductase
3-​Oxocholic acid
Cat.No: T19124
Synonym: 3-Ketocholic acid
Target: Endogenous Metabolite
Acetylcholine iodide
Cat.No: T6751
Synonym: Acetylcolina
Target: Others
Cholestenone
Cat.No: T5240
Synonym: 胆甾烯酮,4-胆甾烯-3-酮,(+)-4-Cholesten-3-one
Target: Others, Endogenous Metabolite
Taurodeoxycholate sodium salt
Cat.No: TN2349
Synonym: Sodium taurodeoxylate,牛磺脱氧胆酸钠
Target: Endogenous Metabolite
Taurodeoxycholic acid sodium hydrate
Cat.No: TJA2398
Synonym: Sodium taurodeoxycholate monohydrate,Taurodeoxychloic Acid sodium hydrate,Taurohyodeoxycholic acid sodium salt,牛磺猪去氧胆酸
Target: Apoptosis, Caspase
3-Methylcatechol
Cat.No: T3742
Synonym: 3-甲基苯邻二酚,3-Methylpyrocatechol,2,3-Toluenediol,3-甲基邻苯二酚,2,3-dihydroxytoluene
Target: Others
Lipoteichoic acid
Cat.No: T40646
Synonym:
Target: Complement System
Taurochenodeoxycholic acid sodium
Cat.No: TN2215
Synonym: 牛磺鹅去氧胆酸钠盐,Sodium taurochenodeoxycholate,牛磺鹅去氧胆酸钠
Target: Apoptosis, Endogenous Metabolite
5α-Cholestan-3β-ol
Cat.No: T2962
Synonym: Dihydrocholesterol,Zymostanol,5α-Cholestanol,5alpha-Cholestanol,NSC 18188,Beta-Cholestanol,二氢胆甾醇
Target: Others, Endogenous Metabolite
3b-Hydroxy-5-cholenoic acid
Cat.No: T7628
Synonym:
Target: Endogenous Metabolite
Cichoriin
Cat.No: TN3651
Synonym:
Target: Others
Phosphorylcholine chloride calcium salt tetrahydrate
Cat.No: T4713
Synonym: Phosphocholine chloride calcium salt tet,胆碱磷酸氯化钙四水,CalciuM Phosphorylcholine Tetrahydrate
Target: Others, Endogenous Metabolite
1,2-Distearoyl-sn-glycero-3-phosphorylcholine
Cat.No: T9510
Synonym: DSPC,L-ALPHA-PHOSPHATIDYLCHOLINE, DISTEAROYL,1,2-Distearoyl-sn-glycero-3-PC,二硬脂酰磷脂酰胆碱
Target: Others
Cinchonidine
Cat.No: T1317
Synonym: 奎宁树,α-Quinidine,辛可尼丁,L-Cinchonidine
Target: 5-HT Receptor, Serotonin Transporter, Parasite
Deoxycholic acid sodium salt
Cat.No: T5077
Synonym: 脱氧胆酸钠,Sodium deoxycholate,Sodium Desoxycholate
Target: Endogenous Metabolite, GPCR19
Taurolithocholic acid sodium salt
Cat.No: T4727
Synonym: 牛磺石胆酸钠,Sodium taurolithocholate
Target: Others, Calcium Channel
27-Hydroxycholesterol
Cat.No: TQ0274
Synonym: 27-羟基胆固醇,5,25R-胆甾烯-3BETA,26-二醇,25(R)-27-hydroxy Cholesterol
Target: Estrogen/progestogen Receptor, Liver X Receptor
4-methoxylonchocarpin
Cat.No: TN7235
Synonym:
Target: TNF, NF-κB
Allocholic acid
Cat.No: T19189
Synonym:
Target: Others
Lapachol
Cat.No: T4136
Synonym: Bethabarra wood,CI75490,黄钟花醌,Greenhartin,Tecomin
Target: Others, Influenza Virus, Antibacterial, Parasite, Antifungal
Taurohyodeoxycholic acid sodium salt
Cat.No: T8092
Synonym: Sodium taurohyodeoxycholate hydrate
Target: Caspase
1-Palmitoyl-sn-glycero-3-phosphocholine
Cat.No: T8712
Synonym: 1-十六酰-SN-丙三醇-磷酸胆碱,1-Hexadecanoyl-sn-glycero-3-phosphocholine
Target: Others
Glycocholic acid hydrate
Cat.No: T5072
Synonym:
Target: Others, Endogenous Metabolite
Rhynchophylline
Cat.No: T6S0659
Synonym: 钩藤碱,Rhynchophyllin,Rhyncophylline,Mitrinermine,Mitrinermin
Target: Calcium Channel, NF-κB
4-Hydroxylonchocarpin
Cat.No: T2S0142
Synonym: 异补骨脂色烯查耳酮,Isobavachromene
Target: Others
GLYCODEOXYCHOLIC ACID
Cat.No: T5352
Synonym:
Target: Others, Endogenous Metabolite
Glycolithocholic acid
Cat.No: T31964
Synonym: Lithocholic acid glycine conjugate,甘氨石胆酸,Lithocholylglycine
Target: Others
Taurodeoxycholic acid
Cat.No: T75319
Synonym: Taurodeoxychloic acid
Target: Apoptosis, Calcium Channel, Caspase
20(S)-Hydroxycholesterol
Cat.No: T10085
Synonym: 20α-Hydroxycholesterol
Target: Smo
3α,12β-Dihydroxycholanoic acid
Cat.No: T13505
Synonym:
Target: Others
Hyocholic acid
Cat.No: TN7024
Synonym:
Target:
Methyl Cholate
Cat.No: T2744
Synonym: 胆酸甲酯,Cholic acid methyl ester
Target: Others
Deoxycholic acid
Cat.No: T2965
Synonym: Cholorebic,去氧胆酸,脱氧胆酸,Deoxycholate,Desoxycholic acid,Cholanoic Acid,Cholerebic
Target: Endogenous Metabolite, GPCR19
Cholesterol
Cat.No: T0760
Synonym: Cholesterin,Cholesteryl alcohol,胆固醇
Target: Estrogen Receptor/ERR, MRP, Endogenous Metabolite, ROR
Cholic Acid
Cat.No: T2963
Synonym: Cholanic acid,胆汁酸,Cholate,Colalin
Target: Endogenous Metabolite
1-Stearoyl-sn-glycero-3-phosphocholine
Cat.No: T8714
Synonym: 1-硬脂酰-SN-甘油-3-磷酰胆碱,1-stearoyl-lysophosphatidylcholine,L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY
Target: Others
Isodeoxycholic Acid
Cat.No: T36585
Synonym: isoDCA
Target: Chloride channel, Antibacterial
(-)-Fenchone
Cat.No: TN1641
Synonym:
Target: Others, Antioxidant, Antifungal
Taurocholic acid sodium salt hydrate
Cat.No: T1138
Synonym: 牛胆酸钠,牛磺胆酸钠水合物,Sodium taurocholate hydrate,Taurocholic Acid sodium hydrate
Target: Others, Potassium Channel, Endogenous Metabolite
4-Allylcatechol
Cat.No: TN1274
Synonym: 2-羟基胡椒酚,4-Allylpyrocatechol,Hydroxychavicol
Target: Others
24-Hydroxycholesterol
Cat.No: T10086
Synonym: Cholest-5-ene-3beta,24-diol
Target: Liver X Receptor, NMDAR
Choline chloride
Cat.No: T1039
Synonym: Biocolina,Biocoline,Hepacholine,氯化胆碱
Target: AChR
Chondroitine sulfate
Cat.No: T22293
Synonym: Chondroitine sulfate (From cattle)
Target: Others
Cholesterol myristate
Cat.No: T8040
Synonym: 胆甾烯基豆蔻酸酯,Cholesteryl myristate,胆固醇肉豆蔻酸,Cholesteryl tetradecanoate
Target: Others, Potassium Channel, GABA Receptor, Endogenous Metabolite, AChR
1-Oleoyl-sn-glycero-3-phosphocholine
Cat.No: T8713
Synonym:
Target: Others
7α-Hydroxycholesterol
Cat.No: T19161
Synonym:
Target: Others
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