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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T10463L Bax inhibitor peptide V5 acetate

Bax inhibitor peptide V5 acetate(579492-81-2 free base)

Apoptosis Apoptosis
Bax inhibitor peptide V5 acetate (Bax inhibitor peptide V5 acetate(579492-81-2 free base)) 是一种 Bax 介导的细胞凋亡抑制剂,用于癌症治疗。
T10463 Bax inhibitor peptide V5

BIP-V5,BAX Inhibiting Peptide V5

BCL Apoptosis
Bax inhibitor peptide V5 (BIP-V5) is a Bax-mediated apoptosis inhibitor with anticancer activity.
T40379 Bax BH3 peptide (55-74), wild type

Bax BH3 peptide (55-74), wild type

Bax BH3 peptide (55-74), wild type is a 20-amino acid peptide (Bax 1) known for its ability to induce apoptosis in various cell line models.
T14499 Bax activator-1

BCL Apoptosis
Bax activator-1 (compound 106) is a Bax activator. It induces Bax-dependent tumor cell apoptosis[1].
TP2203 Bax inhibitor peptide, negative control

Others Others
The compound is a negative control peptide for the Bax inhibitor peptides V5 and P5.
T8649 TMBIM6 antagonist-1

BAX-inhibitor-1,1-(2-氨基苯基)-3-(3-硝基苯基)-2-丙烯-1-酮,BIA

mTOR PI3K/Akt/mTOR signaling
TMBIM6 antagonist-1 (BAX-inhibitor-1) 是有潜力的TMBIM6拮抗剂,能够抑制 TMBIM6 与 mTORC2 结合,抑制 mTORC2 活性,调节TMBIM6 释放 Ca2+。
T26737 Bamifylline Hydrochloride

BAX-2793Z,AC 3810,AC-3810,BAX2793Z,BAX 2793Z

Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.
T82918 BAX-IN-1

BAX-IN-1为潜在的Bcl-2相关x蛋白(BAX)选择性抑制剂。
T7538 Tetraethylammonium chloride

Potassium Channel Membrane transporter/Ion channel
Tetraethylammonium chloride 是非选择性钾通道阻滞剂。它是有机阳离子转运蛋白的良好底物,并具有抗肿瘤特性。
T5210 BAI1

Apoptosis; BCL Apoptosis
BAI1 是一种选择性凋亡因子BAX 变构抑制剂。它结合 BAX 并变构抑制其激活,具有潜力研究 BAX 依赖性细胞死亡介导的疾病。
T5104 BTSA1

Apoptosis; BCL Apoptosis
BTSA1 是一种有口服活性的 BAX 激活剂,IC50为 250 nM,EC50为 144 nM。它以高亲和力和特异性与 N 末端激活位点结合,并诱导 BAX 发生构象变化,从而导致BAX 介导的细胞凋亡。
T2099 ABT-737

Mitophagy; BCL; Autophagy Apoptosis; Autophagy
ABT737 是 BH3 模拟物,是Bcl-2、Bcl-xL 和Bcl-w 抑制剂,EC50分别为 30.3 nM、78.7 nM 和 197.8 nM。它诱导自噬,有研究急性髓系白血病的潜力。它还诱导 BCL-2/BAX 复合物的破坏和 BAK 依赖性。
T15771 Lobaplatin

D-19466,络铂

DNA Alkylation DNA Damage/DNA Repair
Lobaplatin (D-19466) 是一种铂 (II) 复合物的非对映混合物,是一种有前途的抗肿瘤化疗药物,在多种肿瘤类型的患者中具有活性。
T12412L PDK4-IN-1 hydrochloride

Apoptosis; PDK Apoptosis; PI3K/Akt/mTOR signaling
PDK4-IN-1 hydrochloride 是一种蒽醌衍生物,对丙酮酸脱氢酶激酶 4有抑制作用,IC50为 84 nM,具有口服活性。它抑制细胞转化和细胞增殖并诱导细胞凋亡。它具有抗过敏,抗糖尿病和抗癌作用。
T8978 DD1

3,3'-Diamino-4'-methoxyflavone,HUN85111

Proteasome Proteases/Proteasome; Ubiquitination
DD1 (HUN85111) 是一种蛋白酶体抑制剂,可诱导人髓系肿瘤选择性凋亡。
T4215 TCS-PIM-1-4a

5-[[3-(三氟甲基)苯基]亚甲基]-2,4-噻唑烷二酮,SMI-4a

Apoptosis; Pim Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling
TCS-PIM-1-4a (SMI-4a) 是一种泛-Pim 激酶抑制剂,可通过激活 AMPK 来阻断 mTORC1的活性。它可杀死多种髓样和淋巴样细胞系,IC50值为 0.8 μM 至 40 μM。
T23861 CAY10526

CAY-10526,BTH,CAY 10526

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
CAY10526 (BTH) 是 mPGES-1 的选择性抑制剂,可抑制 NF-κB 信号通路。
T0942 Quinacrine dihydrochloride

疟疾平,Mepacrine dihydrochloride,阿的平,SN-390,Quinacrine 2HCl

Apoptosis; Mitophagy; DNA; Phospholipase; Parasite; Autophagy; Histamine Receptor Apoptosis; Autophagy; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Quinacrine dihydrochloride (Mepacrine dihydrochloride) 是一种具有口服活性的抗疟剂,抑制 NF-κB 并激活 p53 信号转导,诱导肿瘤细胞发生凋亡,具有抗肿瘤和抗寄生虫活性。
T6583 MG-101

ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I

Cysteine Protease; Proteasome Proteases/Proteasome; Ubiquitination
MG-101 (Calpain inhibitor I) 是一种有效的半胱氨酸蛋白酶抑制剂,能够抑制钙蛋白酶I (Ki:190 pM),钙蛋白酶II (Ki:220 pM),组织蛋白酶B (Ki:150 pM)和组织蛋白酶L (Ki:500 pM)。
T15212 Emamectin Benzoate

MK-244,甲胺基阿维菌素苯甲酸盐

Apoptosis; Reactive Oxygen Species; GABA Receptor; Parasite Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
Emamectin Benzoate (MK-244) 是口服有效的神经系统毒物,其通过结合昆虫中的 GABA 受体发挥作用。它是阿维菌素的半合成衍生物之一,具有广谱的杀虫和杀螨活性。它诱导ROS 介导的 DNA 损伤和细胞凋亡。
T61373 Baxdrostat

Others Others
Baxdrostat 是一种醛固酮合成酶抑制剂。
T31668 Eribaxaban

PD 348292,PD0348292,PD-0348292,PD-348292,PD 0348292,PD348292

Factor Xa Metabolism
Eribaxaban (PD348292) 是一种可口服的 Xa 因子抑制剂,可用于预防和治疗静脉血栓栓塞。
T61372 (S)-Baxdrostat

(S)-Baxdrostat is an S-enantiomer of Baxdrostat, which functions as an inhibitor of aldosterone synthase [1].
T76822 Pagibaximab

Pagibaximab为一种嵌合IgG1抗体,针对金黄色葡萄球菌与表皮链球菌的表面脂肪酸成分具有特异性识别能力。其主要应用于预防葡萄球菌所引起的败血症。
T68632 Pibaxizine

Pibaxizine is diphenylmethyl piperazine derivatives. It is a histamine H1 receptor antagonist.
T2453 BAM7

BCL Apoptosis
BAM7 是一种促凋亡 Bax 的直接和特异性激活剂,IC50为 3.3 μM。
T83636L NSC 122393

3,4,5,6-Tetrabromofluorescein

NSC 122393 是一种荧光染料,抑制Bax和Bcl-X之间相互作用,可诱导Bcl-X过表达乳腺癌细胞的凋亡。
T14846 Bz 423

BZ48

Apoptosis; BCL Apoptosis
Bz 423 是一种有效的免疫调节剂,通过激活 Bax 和 Bak 来诱导线粒体外膜通透和细胞色素 c 释放来诱导细胞凋亡。Bz 423 在狼疮小鼠模型中显示出部分活性。
T21911 Rilmenidine hemifumarate

Rilmenidine (hemifumarate),S-3341 hemifumarate

Apoptosis; Imidazoline Receptor Apoptosis; Neuroscience
Rilmenidine hemifumarate (S-3341 hemifumarate) 是一种新型且具有口服活性和选择性 的 I1咪唑啉受体 (I1 imidazoline receptor) 和α2肾上腺素受体激动剂,可诱导自噬 ,调节白血病细胞增殖,刺激促凋亡蛋白 Bax,诱导人白血病 K562 细胞线粒体通路的紊乱和凋亡。
T22094 JGB1741

ILS-JGB-1741

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
JGB1741 (ILS-JGB-1741) 是一种有效的选择性 SIRT1 抑制剂,IC50 为 15 μM。 JGB1741 调节 Bax/Bcl2 比率、细胞色素 c 释放和 PARP 裂解并增加乙酰化 p53 水平,导致 p53 介导的细胞凋亡。 JGB1741可用于乳腺癌研究。
T61046 Anticancer agent 43

Apoptosis Apoptosis
Anticancer agent 43 是一种有效的抗癌剂,通过 caspase 3, PARP1,Bax 蛋白依赖性途径诱导癌细胞凋亡 (apoptosis)。Anticancer agent 43 能够诱导 DNA 损伤,可用于研究大鼠胶质母细胞瘤 。
T37518 Diphenyl disulfide

Phenyl disulfide

Apoptosis; BCL; Endogenous Metabolite Apoptosis; Metabolism
Diphenyl disulfide (Phenyl disulfide) 在乳腺癌细胞系中显示出抗癌活性。Diphenyl disulfide 通过Bax 蛋白水解活化和伴随的自噬来诱导并增强乳腺癌细胞的凋亡。Diphenyl disulfide 以剂量依赖性方式抑制细胞增殖和活力,并减少集落形成。Diphenyl disulfide 可用来治疗乳腺癌。
T6641 Rilmenidine Phosphate

Apoptosis; Adrenergic Receptor; Autophagy; Imidazoline Receptor Apoptosis; Autophagy; GPCR/G Protein; Neuroscience
Rilmenidine phosphate 是一种新型的抗高血压药物和口服活性选择性 I1 咪唑啉受体激动剂。它可调节白血病细胞增殖,刺激促凋亡蛋白 Bax,从而诱导人白血病 K562 细胞线粒体通路的紊乱和凋亡。它可通过减少交感神经过度活跃而发挥中枢作用,并通过抑制 Na+/H+反向转运而在肾脏中发挥作用。
T28117 MSN-50

MSN50,MSN 50

MSN-50, an inhibitor of Bax and Bak oligomerization, inhibits liposome permeabilization, prevents genotoxic cell death and promotes neuroprotection.
T60997 GL0388

GL0388 是一种Bax 激活剂,可导致 Bax 插入线粒体膜,从而诱导 Bax 介导的细胞凋亡。GL0388 在体内抑制乳腺癌异种移植的肿瘤生长,并且对多种癌细胞表现出抗增殖活性,IC50值为 0.299-1.57 μM。
T16155 MSN-125

Akt Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
MSN-125 effectively inhibits Bax/Bak-mediated apoptosis in HCT-116, BMK Cells, and primary cortical neurons protect primary neurons against glutamate excitotoxicity. MSN-125 is an effective Bax and Bak oligomerization inhibitor. MSN-125 prevents mitochond
T23925 CYD-2-11

CYD 2 11,CYD211

CYD-2-11 is an effective and selective Bax agonist. It acts by targeting the structural pocket proximal to S184 in the C-terminal region of Bax.
T8792 SMBA1

SMBA1 是一种 Bax 激活因子,是一种有效的 Bax 激动剂(Ki :43.3 nM),诱导恶性胶质瘤细胞周期阻滞和凋亡。SMBA1 有增强 Bax 表达的作用,显示出抗肿瘤活性。SMBA1 可用于研究癌症。
T24806 SMBA2

SMBA-2,NSC4436,NSC 4436,NSC-4436,SMBA 2

SMBA2 is a Bax activator. It acts by specifically targeting the binding pocket at S184.
T28411 Physapubenolide

NSC 368674,NSC368674,NSC-368674

Physapubenolide is natural cytotoxic withanolide antitumor agent. Physapubenolide induces apoptosis by decreasing mitochondrial membrane potential and elevating the Bax/Bcl-2 protein expression ratio.
T63530 Apoptotic agent-3

Apoptotic agent-3 利用潜在的线粒体介导的 Bcl-2/Bax 通路和激活 caspase-3 途径促进凋亡,表现出抗增殖作用,能够用于研究癌症。
T72570 Antitumor agent-83

Antitumor agent-83 是一种促凋亡蛋白 BAX 的激活剂,对肿瘤细胞有显著的抗增殖作用。Antitumor agent-83 通过诱导 BAX 的构象激活介导细胞凋亡 (Apoptosis),对 A549 细胞周期有抑制作用。Antitumor agent-83 具有良好的体外代谢稳定性和 CYP 谱。
T63188 Apoptotic agent-2

Apoptotic agent-2 能够使 Bcl-2 下调,并上调 Bax 和 caspase-3 诱导细胞凋亡 (apoptosis),表现出抗增殖作用,能够用于研究癌症。
T62814 Antitumor agent-77

Antitumor agent-77 对癌细胞的生长和迁移具有抑制作用,具有抗癌作用。Antitumor agent-77 能够抑制 GPx-4 和提高 COX2 引发铁下垂。Antitumor agent-77 可以激活肿瘤细胞固有凋亡通路 (Bax-Bcl-2-caspase-3),阻碍肿瘤细胞上皮间质转化 (EMT) 过程。
T76033 Humanin

Humanin 是一种 24 个氨基酸组成的抗凋亡肽,是Bax 抑制剂。Humanin 可以阻止Bax 从细胞质向线粒体的转运,阻断Bax 由活性构象向活性构象的转变。Humanin 是一种线粒体相关肽,具有对抗 AD 相关神经毒性的神经保护作用。Humanin 还可以改善动物的整体胰岛素敏感性。Humanin 与衰老有关。HNG,是 Humanin 的 14号位置的丝氨酸被甘氨酸取代的类似物。
T26817 Bim-BLK-A

Bim Blocker A,Compound A,Bim BLK A,BimBLKA

Bim-BLK-A efficiently blocks Bim-induced apoptosis after Bax is activated on the mitochondria. The cellular target of Bim-BLK-A was identified to be the succinate dehydrogenase subunit B (SDHB) protein of complex II of the mitochondrial electron transfer
T76073 BH3 hydrochloride

BH3 hydrochloride是一种能够穿透血脑屏障的多肽,其机制是通过直接激活促凋亡蛋白Bax/Bak或中和抗凋亡Bcl-2家族蛋白(Bcl-2、Bcl-XL、Bcl-w、mcl1和A-1),从而诱导细胞凋亡。这一作用是通过与BH3结构域的结合实现的。
T61385 IDO1/TDO-IN-1

IDO1/TDO-IN-1 (30) is a highly effective inhibitor that targets both IDO1 and TDO enzymes with uncompetitive (Ki = 0.23 μM) and competitive (Ki = 0.73 μM) mechanisms, respectively. This compound, IDO1/TDO-IN-1 (30), exhibits a significant capacity to induce cell apoptosis via the potential mitochondria-mediated Bcl-2/Bax pathway [1].
T30807 CG0009

CG-0009,CG 0009

CG0009 is a potent and highly selective glycogen synthase kinase 3 (GSK3) inhibitor that inhibitions proliferation, induces apoptosis, and activates the p53-Bax pathway in breast cancer cells through cyclin D1 depletion. CG0009 inhibit breast cancer cell
T62044 Anticancer agent 71

Anticancer agent 71 (Compound 4b) 是有效的抗癌剂。Anticancer agent 71 将细胞周期阻滞在 G2/M 期。Anticancer agent 71通过上调 Bax、Ikb-α 和切割 PARP 并下调 Bcl-2 表达水平诱导细胞凋亡。

化合物

Bax inhibitor peptide V5 acetate
Cat.No: T10463L
Synonym: Bax inhibitor peptide V5 acetate(579492-81-2 free base)
Target: Apoptosis
Bax inhibitor peptide V5
Cat.No: T10463
Synonym: BIP-V5,BAX Inhibiting Peptide V5
Target: BCL
Bax BH3 peptide (55-74), wild type
Cat.No: T40379
Synonym: Bax BH3 peptide (55-74), wild type
Target:
Bax activator-1
Cat.No: T14499
Synonym:
Target: BCL
Bax inhibitor peptide, negative control
Cat.No: TP2203
Synonym:
Target: Others
TMBIM6 antagonist-1
Cat.No: T8649
Synonym: BAX-inhibitor-1,1-(2-氨基苯基)-3-(3-硝基苯基)-2-丙烯-1-酮,BIA
Target: mTOR
Bamifylline Hydrochloride
Cat.No: T26737
Synonym: BAX-2793Z,AC 3810,AC-3810,BAX2793Z,BAX 2793Z
Target:
BAX-IN-1
Cat.No: T82918
Synonym:
Target:
Tetraethylammonium chloride
Cat.No: T7538
Synonym:
Target: Potassium Channel
BAI1
Cat.No: T5210
Synonym:
Target: Apoptosis, BCL
BTSA1
Cat.No: T5104
Synonym:
Target: Apoptosis, BCL
ABT-737
Cat.No: T2099
Synonym:
Target: Mitophagy, BCL, Autophagy
Lobaplatin
Cat.No: T15771
Synonym: D-19466,络铂
Target: DNA Alkylation
PDK4-IN-1 hydrochloride
Cat.No: T12412L
Synonym:
Target: Apoptosis, PDK
DD1
Cat.No: T8978
Synonym: 3,3'-Diamino-4'-methoxyflavone,HUN85111
Target: Proteasome
TCS-PIM-1-4a
Cat.No: T4215
Synonym: 5-[[3-(三氟甲基)苯基]亚甲基]-2,4-噻唑烷二酮,SMI-4a
Target: Apoptosis, Pim
CAY10526
Cat.No: T23861
Synonym: CAY-10526,BTH,CAY 10526
Target: Prostaglandin Receptor
Quinacrine dihydrochloride
Cat.No: T0942
Synonym: 疟疾平,Mepacrine dihydrochloride,阿的平,SN-390,Quinacrine 2HCl
Target: Apoptosis, Mitophagy, DNA, Phospholipase, Parasite, Autophagy, Histamine Receptor
MG-101
Cat.No: T6583
Synonym: ALLN,Ac-LLnL-CHO,Calpain inhibitor I,Calpain inhibitor-1,MG101,钙蛋白酶抑制剂I
Target: Cysteine Protease, Proteasome
Emamectin Benzoate
Cat.No: T15212
Synonym: MK-244,甲胺基阿维菌素苯甲酸盐
Target: Apoptosis, Reactive Oxygen Species, GABA Receptor, Parasite
Baxdrostat
Cat.No: T61373
Synonym:
Target: Others
Eribaxaban
Cat.No: T31668
Synonym: PD 348292,PD0348292,PD-0348292,PD-348292,PD 0348292,PD348292
Target: Factor Xa
(S)-Baxdrostat
Cat.No: T61372
Synonym:
Target:
Pagibaximab
Cat.No: T76822
Synonym:
Target:
Pibaxizine
Cat.No: T68632
Synonym:
Target:
BAM7
Cat.No: T2453
Synonym:
Target: BCL
NSC 122393
Cat.No: T83636L
Synonym: 3,4,5,6-Tetrabromofluorescein
Target:
Bz 423
Cat.No: T14846
Synonym: BZ48
Target: Apoptosis, BCL
Rilmenidine hemifumarate
Cat.No: T21911
Synonym: Rilmenidine (hemifumarate),S-3341 hemifumarate
Target: Apoptosis, Imidazoline Receptor
JGB1741
Cat.No: T22094
Synonym: ILS-JGB-1741
Target: Sirtuin
Anticancer agent 43
Cat.No: T61046
Synonym:
Target: Apoptosis
Diphenyl disulfide
Cat.No: T37518
Synonym: Phenyl disulfide
Target: Apoptosis, BCL, Endogenous Metabolite
Rilmenidine Phosphate
Cat.No: T6641
Synonym:
Target: Apoptosis, Adrenergic Receptor, Autophagy, Imidazoline Receptor
MSN-50
Cat.No: T28117
Synonym: MSN50,MSN 50
Target:
GL0388
Cat.No: T60997
Synonym:
Target:
MSN-125
Cat.No: T16155
Synonym:
Target: Akt
CYD-2-11
Cat.No: T23925
Synonym: CYD 2 11,CYD211
Target:
SMBA1
Cat.No: T8792
Synonym:
Target:
SMBA2
Cat.No: T24806
Synonym: SMBA-2,NSC4436,NSC 4436,NSC-4436,SMBA 2
Target:
Physapubenolide
Cat.No: T28411
Synonym: NSC 368674,NSC368674,NSC-368674
Target:
Apoptotic agent-3
Cat.No: T63530
Synonym:
Target:
Antitumor agent-83
Cat.No: T72570
Synonym:
Target:
Apoptotic agent-2
Cat.No: T63188
Synonym:
Target:
Antitumor agent-77
Cat.No: T62814
Synonym:
Target:
Humanin
Cat.No: T76033
Synonym:
Target:
Bim-BLK-A
Cat.No: T26817
Synonym: Bim Blocker A,Compound A,Bim BLK A,BimBLKA
Target:
BH3 hydrochloride
Cat.No: T76073
Synonym:
Target:
IDO1/TDO-IN-1
Cat.No: T61385
Synonym:
Target:
CG0009
Cat.No: T30807
Synonym: CG-0009,CG 0009
Target:
Anticancer agent 71
Cat.No: T62044
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2S0500 Ilexsaponin A

毛冬青皂苷A,毛冬青皂苷甲,Ilexsaponin A1

Others Others
Ilexsaponin A (Ilexsaponin A1)1 是分离自冬凌草的根中,利用抗凋亡途径减轻缺血再灌注引起的心肌损伤。它能够减少心肌梗塞的大小,减少 LDH,AST 和 CK-MB 的血清水平,促进细胞活力并抑制缺氧/复氧心肌细胞的凋亡。
TN1195 17-Hydroxy sprengerinin C

17-羟基麦冬皂苷C

BCL; Others; Caspase Apoptosis; Others; Proteases/Proteasome
17-Hydroxy sprengerinin C 是从黄精的根茎中分离得到的一种糖苷化合物,具有更强的抗癌活性。17-Hydroxy sprengerinin C 降低 Blc-2 和 pro-caspase3 的表达并增加 Bax 的产生。
T1079 Metronidazole

Flagyl,Metronidazol,甲硝唑,Anagiardil

Apoptosis; NADPH; Hydrogenase; Antibacterial; Antibiotic; Parasite; Antifection Apoptosis; Metabolism; Microbiology/Virology
Metronidazole (Metronidazol) 是一种合成的硝基咪唑衍生物,具有抗原生动物和抗菌活性。
T2764 (S)-10-Hydroxycamptothecin

10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT

Apoptosis; Topoisomerase Apoptosis; DNA Damage/DNA Repair
(S)-10-Hydroxycamptothecin (10-HCPT) 是一种从喜树中分离的 DNA 拓扑异构酶 I 抑制剂。它显著诱导细胞凋亡,可研究肝癌、胃癌、结肠癌和白血病。
T3322 trans-Chalcone

Chalcone,反-查耳酮,查尔酮,Cinnamophenone,Chalkone

Apoptosis; Others; Antifungal; Fatty Acid Synthase Apoptosis; Metabolism; Microbiology/Virology; Others
trans-Chalcone (Chalkone) 是从 Aronia melanocarpa 果皮中分离出来的一种天然产物,是类黄酮前体的双酚核心结构。它是脂肪酸合酶和 α-淀粉酶的抑制剂,具有抗真菌和抗癌活性。
TN1349 9-Hydroxycalabaxanthone

Antifection Microbiology/Virology
9-Hydroxycalabaxanthone exhibits cytotoxicity against the HT-29 cell line with ED50 values of 9.1 microM. The combination of 9-hydroxycalabaxanthone with α±-mangostin shows the synergistic antimalarial interaction in both clones.
T9503 PHYTOSPHINGOSINE

Apoptosis Apoptosis
Phytosphingosine 是具有抗癌作用的一种磷脂。在癌细胞中,它通过 caspase 8 的激活和 Bax 转位诱导细胞凋亡。
T5715 (E)-Flavokawain A

(E)-1-(2-羟基-4,6-二甲氧基苯基)-3-(4-甲氧基苯基)-2-丙烯-1-酮,FLAVOKAVAIN A(P),卡瓦胡椒素A

Apoptosis; P450 Apoptosis; Metabolism
(E)-Flavokawain A 是一种来自卡瓦提取物的新型查尔酮,通过参与 Bax 蛋白依赖性和线粒体依赖性凋亡途径诱导膀胱癌细胞凋亡,并抑制小鼠肿瘤生长,具有抗癌作用。
T6S1529 Cynarin

Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1R,​3R,​4S,​5R)​-,Cynarine,1,5-Dicaffeoylquinic acid,洋蓟素,金银花

Antioxidant; Antiviral; Influenza Virus; Reactive Oxygen Species Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; oxidation-reduction
Cynarin (1,5-Dicaffeoylquinic acid) 是一种抗窒息剂,具有抗氧化、抗组胺和抗病毒等多种生物活性。
T3902 Atractylenolide III

白术内酯 III,ICodonolactone,8β-Hydroxyasterolide

Apoptosis Apoptosis
Atractylenolide III (ICodonolactone) 是白术根茎主要成分,通过诱导细胞色素 c 的释放、上调 Bax 的表达和易位凋亡诱导因子,是治疗人肺癌的潜力。
T5679 (E)-Ferulic acid

trans-Ferulic acid,反式阿魏酸,(E)-Coniferic acid

BCL; Ferroptosis; Wnt/beta-catenin; Endogenous Metabolite Apoptosis; Cytoskeletal Signaling; Metabolism; Stem Cells
(E)-Ferulic acid ((E)-Coniferic acid) 是阿魏酸的异构体,阿魏酸是在植物细胞壁中丰富存在的芳香族天然产物。 它引起 β-catenin 的磷酸化,导致其蛋白酶体降解,增加促凋亡因子 Bax 的表达,降低促生存因子的表达。它在人肺癌细胞系 H1299 中发挥抗增殖和抗迁移作用。
T7027 EURYCOMANONE

东革阿里提取物,Pasakbumin A

Others Others
Eurycomanone (Pasakbumin A) 能够抑制雌激素生成过程中磷酸二酯酶和芳香酶的活性,促进精子生成。它对 HepG2 细胞具有细胞毒性,能够上调 p53 和 Bax 以及下调 Bcl-2 ,诱导细胞凋亡。它具有抗癌活性,在浓度范围内以剂量依赖性方式抑制 A549 肺癌细胞增殖 从 5 到 20 微克/毫升。
TN1393 (-)-Anonaine

番荔枝碱

Apoptosis; Antioxidant; Parasite; Antifungal Apoptosis; Microbiology/Virology; oxidation-reduction
(-)-Anonaine 可从木兰科和安妮科的几个物种中提取出来,具有抗疟、抗菌、抗真菌、抗氧化、抗癌、抗抑郁和血管舒张的活性。(-)-Anonaine 通过 Bax 和 caspase 依赖性途径诱导人类宫颈癌(HeLa)细胞的凋亡,诱导 DNA 损伤并抑制人类肺癌 h1299细胞的生长和迁移。
T5S2083 Puerarin 6''-O-Xyloside

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Puerarin 6''-O-Xyloside 是从葛根中分离得到的一种天然产物,可诱导线粒体介导的细胞凋亡通路,有抗炎和抗癌活性。
T2795 Amygdalin

苦杏仁苷,Laetrile

Others Others
Amygdalin (Laetrile) 是一种植物葡萄糖苷,分离自蔷薇果实的果核中,如杏,桃,杏仁,樱桃和李子。
T13818 Phytohemagglutinin

PHA-M,植物血球凝集素,PHA,植物血凝素

Apoptosis Apoptosis
Phytohemagglutinin (PHA-M) 是一种普通豆菜豆的主要种子凝集素,聚集在子叶的薄壁细胞中。它是一种 T 细胞激活剂,能够刺激人单核白细胞,可诱导 ChAT mRNA 表达,增强 ACh 合成。
T2909 Fraxetin

7,8-dihydroxy-6-methoxy coumarin,秦皮素,弗拉西汀

Apoptosis; Others Apoptosis; Others
Fraxetin (7,8-dihydroxy-6-methoxy coumarin) 是从秦皮中分离出来的一种天然产物,可诱导细胞凋亡,具有抗肿瘤、抗氧化作用和抗炎作用。
T6S1653 Albiflorin

Alibiflorin,芍药内酯苷

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Albiflorin (Alibiflorin) 是一种牡丹根中的主要成分,是一种单萜糖苷。它具有神经保护、抗炎、抗氧化和缓解疼痛作用。
T5S2358 Dehydrocorydaline

Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline (13-Methylpalmatine) 是一种生物碱。它调节Bax,Bcl-2蛋白表达,激活caspase-7,caspase-8,并使PARP 失活。它能增强p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
TN2103 PROCYANIDIN C1

原花青素 C1,原花青素C1

Apoptosis Apoptosis
Procyanidin C1 是一种天然多酚,可造成 DNA 损伤,细胞周期停滞,诱导凋亡。它降低癌细胞中 Bcl-2 的蛋白水平,增强 BAX,caspase 3 和 9 的表达。
T3S2344 β,β-Dimethylacrylshikonin

β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin

ERK; HIF/HIF Prolyl-Hydroxylase Chromatin/Epigenetic; MAPK; Metabolism
β,β-Dimethylacrylshikonin (Dimethylacrylshikonin) 是一种萘醌衍生物,从 Arnebia nobilis 中提取得到。它利用 PI3K 通路诱导 eNOS、VEGF 和 HIF-1α 的表达,促进血管生成,具有抗肿瘤活性。
T3864 Erianin

BCL; Antibacterial Apoptosis; Microbiology/Virology
Erianin 能抑制吲哚胺-2,3-双加氧酶诱导的肿瘤血管生成,可用作退烧药和止疼剂。
T2860 Vanillyl Alcohol

4-Hydroxy-3-methoxybenzenemethanol,3-Methoxy-4-hydroxybenzyl alcohol,4-Hydroxy-3-methoxybenzyl alcohol,香兰醇,Vanillin alcohol,Vanillic alcohol

Apoptosis; Others Apoptosis; Others
Vanillyl Alcohol (3-Methoxy-4-hydroxybenzyl alcohol) 是一种酚类醇,具有抗血管生成、抗惊厥、抗炎、抗氧化、神经保护和抗伤害活性。它由香兰素衍生而来,在食品和饮料中用作调味剂。
T3895 Polyphyllin I

重楼皂苷I,重楼皂甙

Apoptosis; Akt; JNK; PDK; mTOR; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
Polyphyllin I 是从七叶一枝花中提取的生物活性成分,具有很强的抗肿瘤活性。它是 JNK 信号通路的激活剂,也是 PDK1/Akt/mTOR 信号传导的抑制剂。它诱导自噬,G2/M 期阻滞和细胞凋亡。
T6917 Oleuropein

洋橄榄苦甙,橄榄苦苷

Apoptosis; Aromatase; ROS; PPAR Apoptosis; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Oleuropein 在橄榄叶和油中发现的天然产物,通过 p53 依赖性途径以及 Bax 和 Bcl2基因的调控来诱导乳腺癌细胞凋亡,还抑制芳香化酶。它可通过直接抑制 PPARγ转录活性来发挥抗氧化,抗炎和抗动脉粥样硬化作用。
T10990 Dehydrocorydaline chloride

盐酸脱氢紫堇碱,13-Methylpalmatine chloride

BCL; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Proteases/Proteasome
Dehydrocorydaline chloride (13-Methylpalmatine chloride) 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达;激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌等功效。它具有强大的抗疟疾作用,并具低细胞毒性。
T3729 Ethyl gallate

Nipagallin A,Phyllemblin,gallic acid ethyl ester,没食子酸乙酯

MMP; NF-κB; Akt; Antibacterial Cytoskeletal Signaling; Microbiology/Virology; NF-κB; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Ethyl gallate (gallic acid ethyl ester) 是一种非类黄酮酚过氧化氢清除剂。
T2698 Asperosaponin VI

Akebia saponin D,Asperosaponin Ⅵ,川续断皂苷 VI

Apoptosis; Others; Caspase Apoptosis; Others; Proteases/Proteasome
Asperosaponin VI (Akebia saponin D) 是一种来自续断壁的皂苷组分。它通过增加 Bcl-2/Bax 比值,降低活性 caspase-3 表达,以及增强 p-Akt 和 p-CREB,从而抑制缺氧诱导的心肌细胞凋亡。它通过 BMP-2/p38 和 ERK1/2 信号途径诱导成骨细胞分化。
T6S0052 Chelerythrine

Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine (Broussonpapyrine) 是一种天然生物碱,为有效、选择性的 Ca2+/磷脂依赖性PKC 拮抗剂,IC50值为 0.7 μM。它具有抗肿瘤、抗糖尿病、抗炎的活性。它抑制BclXL-Bak BH3肽结合,IC50为 1.5 μM,并从 BclXL 取代了 Bax。它诱导细胞凋亡和自噬。
T2S2362 Dehydrocorydaline nitrate

去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱

BCL; Others; PARP; p38 MAPK; Caspase; Parasite; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; DNA Damage/DNA Repair; MAPK; Microbiology/Virology; Others; Proteases/Proteasome
Dehydrocorydaline nitrate 是生物碱。Dehydrocorydaline 调节 Bax,Bcl-2蛋白表达,激活 caspase-7,caspase-8,并使 PARP 失活。它能增强 p38 MAPK 活化,具有抗炎、抗癌、抗疟疾等功效。
T5S0661 Koumine

Others Others
Koumine 是一种从钩吻中得到的生物碱,具有高效抗肿瘤活性,在肿瘤细胞中能够提高 Bax/Bcl-2 的蛋白比例和 caspase-3 的表达。在类风湿性关节炎动物模型中,它能够预防关节炎的发展。它具有抗焦虑、抗应激、抗银屑病作用,也可用于缓解疼痛的研究。
T3S0737 Flavokawain A

2'-羟基-4,4',6'-三甲氧基查耳酮,Flavokavain A

Apoptosis; p38 MAPK Apoptosis; MAPK
Flavokawain A (Flavokavain A) 是 kava 提取物中的查耳酮,是一种抗癌试剂,具有抗肿瘤活性。它通过 Bax 蛋白依赖和线粒体依赖的凋亡途径诱导细胞凋亡,有潜力用于膀胱癌的相关研究。
T3824 Jaceosidin

Apoptosis; BCL; COX; UGT Apoptosis; Immunology/Inflammation; Metabolism; Neuroscience
Jaceosidin 是从毛莲蒿中得到的一种黄酮类天然产物,可激活Bax,下调 Mcl-1 和 c-FLIP 的表达,诱导癌细胞凋亡。它能够降低炎性因子水平,激活 NF-κB,抑制COX-2的表达,具有抗癌和抗炎作用。
TN3653 Cimidahurinine

BCL; ROS Apoptosis; Immunology/Inflammation
Cimidahurinine can attenuate Doxorubicin (DOX)-induced cardiotoxicity in a dose-dependent manner with EC50 values of 45.79 uM; it protects against cardiotoxicity by decreasing reactive oxygen species (ROS) accumulation and downregulating apoptosis-related Bax/Bcl-2 proteins.
TN6394 Alisol B acetate

Alisol B acetate can induce Bax nuclear translocation and apoptosis in human hormone-resistant prostate cancer PC-3 cells, the Bax activation and translocation from the cytosol to nucleus might be a crucial response to the apoptotic effect. Alisol B aceta
TN1093 Ginsenoside F4

人参皂苷F4

MMP; IL Receptor; BCL Apoptosis; Immunology/Inflammation; Proteases/Proteasome
Ginsenoside F4 has inhibitory effect on human lymphocytoma JK cell by inducing its apoptosis, the mechanism is related to the mitochondrial dysfunction and the increase of Bax expression and decrease of Bcl-2 expression.
TMA1743 Ergosterol peroxide

ERK; VEGFR; p38 MAPK; Wnt/beta-catenin; Akt; JAK; CDK; JNK; STAT; Antifection Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling; Stem Cells; Tyrosine Kinase/Adaptors
Ergosterol peroxide is an inhibitor of osteoclast differentiation, which has antiviral, trypanocidal, antitumor, and antiangiogenic actions, it can stimulate Foxo3a activity by inhibiting pAKT and c-Myc and activating pro-apoptotic protein Puma and Bax to
T40940 7,3′,5′-Trihydroxyflavanone

7,3′,5′-Trihydroxyflavanone, a flavanoid derivative, promotes apoptotic cell death in MCF-7 cells by augmenting Bax expression. Additionally, this compound demonstrates antioxidant properties.
TN1139 Dehydrocavidine

Dehydrocorydaline,岩黄连碱

BCL; PARP Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair
Dehydrocavidine (Dehydrocorydaline) 具有抗肿瘤活性,它通过诱导调节 Bax/Bcl-2 介导的细胞凋亡、激活半胱天冬酶以及切割 PARP 来抑制 MCF-7 细胞增殖。
TN2308 Wilfortrine

BCL Apoptosis
Wilfortrine can induce liver cancer cell HepG2 apoptosis, but with no effect on the cell cycle, mainly by promoting Bax expression and inhibiting anti-apoptotic protein Bcl-2 expression.
TN6419 Chamaejasmine

Chamaejasmine could be a candidate drug for osteosarcoma and breast cancer chemoprevention, induces apoptosis in MG63 and HEp-2 cells by Akt inactivation and dephosphorylation of BAD. It inhibits Bcl-2 expression and induces Bax expression to desintegrate
T75485 Dehydrobruceine B

Dehydrobruceine B 是一种苦木素,可从鸦胆子 (Brucea javanica) 中分离得到。Dehydrobruceine B 与 Cisplatin 通过线粒体途径,协同诱导细胞凋亡 (apoptosis)。Dehydrobruceine B 还增加凋亡诱导因子 (AIF) 和 Bax 表达,抑制 Keap1-Nrf2。
TN5201 Uncarinic acid E

BCL; MEK; Caspase; PI3K; Antifection; p53 Apoptosis; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Uncarinic acid E has anti-cancer activity, it induces apoptosis in HepG2 cells via accumulation of p53, alters the Bax/Bcl-2 ratio, and activates caspases, resulting in cytochrome c release from the mitochondria. A mixture of uncarinic acid E and 27-O-p-(
TN2257 Tanshinone IIB

丹参酮ⅡB

BCL; Caspase; P-gp Apoptosis; Membrane transporter/Ion channel; Neuroscience; Proteases/Proteasome
Co-treatment with Tanshinone IIB (TSB) significantly inhibits the DNA laddering, cytotoxicity and apoptosis of rat cortical neurons induced by staurosporine in a concentration-dependent manner; TSB also suppresses the elevated Bax protein and decreased bc
T66078 Cardamonin

Cardamonin, a chalcone extracted from cardamom spice with anti-inflammatory and anti-tumor activities. Cardamonin decreased viability of NPC(Nasopharyngeal carcinoma ) cells in a concentration-dependent manner. The IC50 values were 16.22 μM(CNE-1), 14.34 μM (CNE-2), 16.50 μM (HONE-1), and 68.12 μM (SUNE-1). Moreover, the expression level of the proapoptotic effector protein Bax and Bid was also markedly increased after treatment with cardamonin(15μM) in CNE-2 cells.In vivo, cardamonin (25 mg/kg ...
T73403 Aviculin

Aviculin 是一种木聚糖苷,是一种有效的抗癌剂 (anticanceragent)。Aviculin 可降低 MCF-7 细胞代谢活性到 50% 以下,IC50为 75.47 μM。Aviculin 通过内在凋亡途径诱导乳腺癌细胞凋亡 (apoptosis)。Aviculin 增加了 caspase-9、caspase-7和 PARP 的表达。Aviculin 使 Bax/Bcl-2 的比值升高。
TN4999 Serratenediol

BCL; PARP; Caspase Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Proteases/Proteasome
Serratenediol demonstrates strong inhibitory effects on the Epstein-Barr virus early antigen (EBV-EA) activation without showing any cytotoxicity, its effects being stronger than that of a representative control, oleanolic acid. Serratenediol can promote
TN1094 Ginsenoside Rg6

人参皂苷Rg6,人参皂苷 Rg6

Apoptosis; NF-κB Apoptosis; NF-κB
Ginsenoside Rg6 抑制人淋巴瘤 JK 细胞增殖并诱导其凋亡,在 HepG2 细胞中抑制 TNF-α 诱导的 NF-κB 转录活性,IC50为 29.34 μM。

天然产物

Ilexsaponin A
Cat.No: T2S0500
Synonym: 毛冬青皂苷A,毛冬青皂苷甲,Ilexsaponin A1
Target: Others
17-Hydroxy sprengerinin C
Cat.No: TN1195
Synonym: 17-羟基麦冬皂苷C
Target: BCL, Others, Caspase
Metronidazole
Cat.No: T1079
Synonym: Flagyl,Metronidazol,甲硝唑,Anagiardil
Target: Apoptosis, NADPH, Hydrogenase, Antibacterial, Antibiotic, Parasite, Antifection
(S)-10-Hydroxycamptothecin
Cat.No: T2764
Synonym: 10-羟喜树碱,10-羟基喜树碱,10-Hydroxycamptothecin,10-HCPT
Target: Apoptosis, Topoisomerase
trans-Chalcone
Cat.No: T3322
Synonym: Chalcone,反-查耳酮,查尔酮,Cinnamophenone,Chalkone
Target: Apoptosis, Others, Antifungal, Fatty Acid Synthase
9-Hydroxycalabaxanthone
Cat.No: TN1349
Synonym:
Target: Antifection
PHYTOSPHINGOSINE
Cat.No: T9503
Synonym:
Target: Apoptosis
(E)-Flavokawain A
Cat.No: T5715
Synonym: (E)-1-(2-羟基-4,6-二甲氧基苯基)-3-(4-甲氧基苯基)-2-丙烯-1-酮,FLAVOKAVAIN A(P),卡瓦胡椒素A
Target: Apoptosis, P450
Cynarin
Cat.No: T6S1529
Synonym: Cyclohexanecarboxyli​c acid, 1,​3-​bis[[3-​(3,​4-​dihydroxyphenyl)​-​1-​oxo-​2-​propen-​1-​yl]​oxy]​-​4,​5-​dihydroxy-​, (1R,​3R,​4S,​5R)​-,Cynarine,1,5-Dicaffeoylquinic acid,洋蓟素,金银花
Target: Antioxidant, Antiviral, Influenza Virus, Reactive Oxygen Species
Atractylenolide III
Cat.No: T3902
Synonym: 白术内酯 III,ICodonolactone,8β-Hydroxyasterolide
Target: Apoptosis
(E)-Ferulic acid
Cat.No: T5679
Synonym: trans-Ferulic acid,反式阿魏酸,(E)-Coniferic acid
Target: BCL, Ferroptosis, Wnt/beta-catenin, Endogenous Metabolite
EURYCOMANONE
Cat.No: T7027
Synonym: 东革阿里提取物,Pasakbumin A
Target: Others
(-)-Anonaine
Cat.No: TN1393
Synonym: 番荔枝碱
Target: Apoptosis, Antioxidant, Parasite, Antifungal
Puerarin 6''-O-Xyloside
Cat.No: T5S2083
Synonym:
Target: Apoptosis, Caspase
Amygdalin
Cat.No: T2795
Synonym: 苦杏仁苷,Laetrile
Target: Others
Phytohemagglutinin
Cat.No: T13818
Synonym: PHA-M,植物血球凝集素,PHA,植物血凝素
Target: Apoptosis
Fraxetin
Cat.No: T2909
Synonym: 7,8-dihydroxy-6-methoxy coumarin,秦皮素,弗拉西汀
Target: Apoptosis, Others
Albiflorin
Cat.No: T6S1653
Synonym: Alibiflorin,芍药内酯苷
Target: Reactive Oxygen Species
Dehydrocorydaline
Cat.No: T5S2358
Synonym: Dehydrocorydalin,脱氢紫堇碱,13-Methylpalmatine
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
PROCYANIDIN C1
Cat.No: TN2103
Synonym: 原花青素 C1,原花青素C1
Target: Apoptosis
β,β-Dimethylacrylshikonin
Cat.No: T3S2344
Synonym: β,β-二甲基丙烯酰紫草素,Dimethylacrylshikonin,β, β-Dimethylacrylshikonin
Target: ERK, HIF/HIF Prolyl-Hydroxylase
Erianin
Cat.No: T3864
Synonym:
Target: BCL, Antibacterial
Vanillyl Alcohol
Cat.No: T2860
Synonym: 4-Hydroxy-3-methoxybenzenemethanol,3-Methoxy-4-hydroxybenzyl alcohol,4-Hydroxy-3-methoxybenzyl alcohol,香兰醇,Vanillin alcohol,Vanillic alcohol
Target: Apoptosis, Others
Polyphyllin I
Cat.No: T3895
Synonym: 重楼皂苷I,重楼皂甙
Target: Apoptosis, Akt, JNK, PDK, mTOR, Autophagy
Oleuropein
Cat.No: T6917
Synonym: 洋橄榄苦甙,橄榄苦苷
Target: Apoptosis, Aromatase, ROS, PPAR
Dehydrocorydaline chloride
Cat.No: T10990
Synonym: 盐酸脱氢紫堇碱,13-Methylpalmatine chloride
Target: BCL, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Ethyl gallate
Cat.No: T3729
Synonym: Nipagallin A,Phyllemblin,gallic acid ethyl ester,没食子酸乙酯
Target: MMP, NF-κB, Akt, Antibacterial
Asperosaponin VI
Cat.No: T2698
Synonym: Akebia saponin D,Asperosaponin Ⅵ,川续断皂苷 VI
Target: Apoptosis, Others, Caspase
Chelerythrine
Cat.No: T6S0052
Synonym: Toddalin,Broussonpapyrine,白屈菜红碱,Cheleritrine
Target: Apoptosis, BCL, PKC, Autophagy
Dehydrocorydaline nitrate
Cat.No: T2S2362
Synonym: 去氢延胡索甲素硝酸盐,硝酸脱氢紫堇碱
Target: BCL, Others, PARP, p38 MAPK, Caspase, Parasite, Autophagy
Koumine
Cat.No: T5S0661
Synonym:
Target: Others
Flavokawain A
Cat.No: T3S0737
Synonym: 2'-羟基-4,4',6'-三甲氧基查耳酮,Flavokavain A
Target: Apoptosis, p38 MAPK
Jaceosidin
Cat.No: T3824
Synonym:
Target: Apoptosis, BCL, COX, UGT
Cimidahurinine
Cat.No: TN3653
Synonym:
Target: BCL, ROS
Alisol B acetate
Cat.No: TN6394
Synonym:
Target:
Ginsenoside F4
Cat.No: TN1093
Synonym: 人参皂苷F4
Target: MMP, IL Receptor, BCL
Ergosterol peroxide
Cat.No: TMA1743
Synonym:
Target: ERK, VEGFR, p38 MAPK, Wnt/beta-catenin, Akt, JAK, CDK, JNK, STAT, Antifection
7,3′,5′-Trihydroxyflavanone
Cat.No: T40940
Synonym:
Target:
Dehydrocavidine
Cat.No: TN1139
Synonym: Dehydrocorydaline,岩黄连碱
Target: BCL, PARP
Wilfortrine
Cat.No: TN2308
Synonym:
Target: BCL
Chamaejasmine
Cat.No: TN6419
Synonym:
Target:
Dehydrobruceine B
Cat.No: T75485
Synonym:
Target:
Uncarinic acid E
Cat.No: TN5201
Synonym:
Target: BCL, MEK, Caspase, PI3K, Antifection, p53
Tanshinone IIB
Cat.No: TN2257
Synonym: 丹参酮ⅡB
Target: BCL, Caspase, P-gp
Cardamonin
Cat.No: T66078
Synonym:
Target:
Aviculin
Cat.No: T73403
Synonym:
Target:
Serratenediol
Cat.No: TN4999
Synonym:
Target: BCL, PARP, Caspase
Ginsenoside Rg6
Cat.No: TN1094
Synonym: 人参皂苷Rg6,人参皂苷 Rg6
Target: Apoptosis, NF-κB
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