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492

抑制剂 & 化合物

174

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Cat. No. Product Name Target Signaling Pathways
T40284 B-Raf IN 2

Raf MAPK
B-Raf IN 2, compound Ia, is a highly effective and specific inhibitor of BRAF. It exhibits significant potential for cancer research.
T9560 MAO-B-IN-2

MAO-B-IN-2 是一种选择性和竞争性的MAO-BBChE 抑制剂,其IC50值分别为 0.51 和 7.00 μM。MAO-B-IN-2 通过良好的 ROS 清除特性减轻 H2O2 诱导的细胞损伤。
T60001 Benzamide, 3-methoxy-N-(3-thiazolo[5,4-b]pyridin-2-ylphenyl)

3-methoxy-N-(3-(thiazolo[5,4-b]pyridin-2-yl)phenyl)benzamide

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
Benzamide, 3-methoxy-N-(3-thiazolo[5,4-b]pyridin-2-ylphenyl) (3-methoxy-N-(3-(thiazolo[5,4-b]pyridin-2-yl)phenyl)benzamide) 是一种 sirtuin 调节剂,可用于延长细胞寿命,治疗和/或预防多种 疾病和障碍包括糖尿病、心血管疾病、凝血障碍、炎症、癌症等。
T63898 Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-

PPAR DNA Damage/DNA Repair; Metabolism
Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-是一种PPARα/γ双激动剂,EC50 分别为 0.358μM 和1.21μM。Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-是Aleglitazar 的R 型异构体。
T50009L sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate

Others Others
sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate 是一种有机硫化合物。它已被用作研究含硫化合物对酶活性和代谢途径的影响的模型化合物,也被用于研究含硫化合物对细菌生长和基因表达调控的影响。
T22595 B2

Linazolamide intermediate B impurity 2,CPNQ,5-[4-(4-Chlorobenzoyl)-1-piperazinyl]-8-nitroquinoline,奥司他韦杂质B(2-叠氮杂合物)

Others; Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
B2 (Linazolamide intermediate B impurity 2) 促进亨廷顿病和帕金森病细胞模型中的包涵体形成。
T9752 3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile

Androgen Receptor Endocrinology/Hormones
3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile 是一种雄激素受体调节剂。
T5103 AKOS B018304

(5E)-5-(2-硝基苯亚甲基)-2-硫代-四氢噻唑-4-酮

Others Others
AKOS B018304 是芳基衍生物,能够在para 位置进行极性替换。
T9315 2H-​Imidazo[4,​5-​b]​pyrazin-​2-​one, 1,​3-​dihydro-​6-​[6-​(1-​hydroxy-​1-​methylethyl)​-​3-​pyridinyl]​-​1-​[(tetrahydro-​2H-​pyran-​4-​yl)​methyl]​-

Others Others
2H-Imidazo[4,5-b]pyrazin-2-one, 1,3-dihydro-6-[6-(1-hydroxy-1-​methylethyl)-3-pyridinyl]-1-[(tetrahydro-2H-pyran-4-yl)methyl]- 是有效的mTOR 抑制剂,对于mTOR 和PI3Kα的IC50分别为0.176 μM 和 >30 μM。
T10707 CCK-B Receptor Antagonist 2

Others Others
CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin/CCK-B (IC50: 0.43 nM). It also inhibits gastrin/CCK-A activity (IC50: 1.82 μM).
T41094 Wnt/β-catenin agonist 2

GSK-3; Wnt/beta-catenin Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Stem Cells
Wnt/β-catenin agonist 2激活 Wnt/β-catenin 信号传导,是一种有效的 Wnt 激动剂。 Wnt/β-catenin agonist 2可用于与信号转导相关的疾病研究,与癌症侵袭转移密切相关。
T0660 Beta-Tetralone

2-Tetralone,beta-四氢萘酮

P450 Metabolism
Beta-Tetralone (2-Tetralone) 是 tetralin 的酮衍生物。
T9871 Dazonone

Imidazo[2,1-b]quinazolin-2(3H)-one, 6-chloro-1,5-dihydro-3-methyl-

PDE Metabolism
Dazonone (Imidazo[2,1-b]quinazolin-2(3H)-one, 6-chloro-1,5-dihydro-3-methyl-) 是一种特异性的 PDE III 抑制剂。
T9999 Sirtuin modulator 2

N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide

Others; Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
Sirtuin modulator 2 (N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide) 具有抗糖尿病、抗炎和抗肿瘤活性。
T12110 MRZ 2-514

8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one

NMDAR Neuroscience
MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) 是 NMDA receptor(glycineB) 的拮抗剂,Ki=33 μM。
T9659 LCB 03-0110

3-(2-(3-(Morpholinomethyl)phenyl)thieno[3,2-b]pyridin-7-ylamino)phenol

Discoidin Domain Receptor (DDR) Tyrosine Kinase/Adaptors
LCB 03-0110 (3-(2-(3-(Morpholinomethyl)phenyl)thieno[3,2-b]pyridin-7-ylamino)phenol) 是一种盘状结构域受体家族酪氨酸激酶的强效抑制剂,可强烈抑制多种酪氨酸激酶,包括 c-Src 家族、脾酪氨酸激酶、布鲁顿酪氨酸激酶和血管内皮生长因子受体 2,它们对免疫很重要细胞信号传导和炎症反应。
T9734 InhA-IN-2

CDK Cell Cycle/Checkpoint
InhA-IN-2直接抑制 InhA,不需要过氧化氢酶过氧化物酶 KatG 的激活。
T8430 Senexin B

4-[[2-[6-[(4-甲基-1-哌嗪基)羰基]-2-萘基]乙基]氨基]-6-喹唑啉甲腈

CDK Cell Cycle/Checkpoint
Senexin B 是一种有效的选择性 CDK8/19 抑制剂(CDK8 和 CDK19,Kd 分别为 140 nM 和 80 nM)。
T9017 HPK1-IN-2

Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2,HPK1-IN-2

Others; FLT; Src Angiogenesis; Others; Tyrosine Kinase/Adaptors
HPK1-IN-2 (Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2) 是一种有效且具有口服活性的造血祖细胞激酶-1 抑制剂(HPK1;IC50<0.05 µM)。它还抑制 Lck (0.05 µM<IC50<0.5 µM) 和 Flt3 (IC50<0.05 µM) 激酶活性,具有抗肿瘤活性。
T3346 AKT inhibitor VIII

AKTi-1/2

Apoptosis; Akt Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
AKT inhibitor VIII (AKTi-1/2) 是一种细胞渗透的喹喔啉化合物,可逆的选择性抑制Akt1、Akt2和Akt3的活性,IC50值分别为 58 nM、210 nM 和 2119 nM。
T27119L (Rac)-Daglutril

SLV 306 acetic acid,2-((3S)-3-(1-(2-(ethoxycarbonyl)-4-phenylbutyl)cyclopentane-1-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)acetic acid

Others Others
(Rac)-Daglutril (SLV 306 acetic acid) 是 Daglutril 的消旋体。Daglutril 是一种口服活性的混合中性内肽酶/内皮素转化酶抑制剂,正在开发用于治疗原发性高血压和充血性心力衰竭。
T15559 TBK1/IKKε-IN-2

B/IKK NF-κB
TBK1/IKKε-IN-2 是双重TBK1和IKKε抑制剂。
T50083 12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide

Others Others
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide 可用作分子结构单元,用于多种化合物的合成。
T10237 ACHP Hydrochloride

IKK-2 Inhibitor VIII

B/IKK NF-κB
ACHP Hydrochloride (IKK-2 Inhibitor VIII) 是选择性的IKK-β抑制剂 (IC50=5.8 nM)。
TNU0159 FMAU

2'-Deoxy-2'-fluoro-5-methyl-beta-D-arabinouridine

Apoptosis Apoptosis
FMAU (2'-Deoxy-2'-fluoro-5-methyl-beta-D-arabinouridine) is a thymine nucleoside analog with insertional activity on replicating DNA.FMAU can be used to label cells and track DNA synthesis.
T19206 β-Lactamase-IN-1

4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one,beta-lactamase-IN-1

Antibacterial Microbiology/Virology
β-Lactamase-IN-1 (4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one) 是一种 β-Lactamase 抑制剂,针对淋病奈瑟菌的感染。
T9696 β-catenin-IN-2

Wnt/beta-catenin Cytoskeletal Signaling; Stem Cells
β-catenin-IN-2 是有效的β-catenin 抑制剂。β-catenin-IN-2在结直肠癌中有研究的价值。
T19497 ONPG

2-硝基苯-beta-D-半乳糖苷,2-Nitrophenyl β-D-galactopyranoside

Others Others
ONPG (2-Nitrophenyl β-D-galactopyranoside) 是用作比色和分光光度计底物,可用作 β-半乳糖苷酶活性的检测。
T50093 MASM7

Others Others
MASM7 又称MASM7,是一种用作分子结构单元的化合物。它是一种线粒体融合蛋白激活剂,可以通过线粒体融合蛋白实现线粒体融合。
T28257L (-)-OPC-51803

AChR Neuroscience
(-)-OPC-51803 是一种抗利尿激素 V2受体激动剂,可用于夜尿症和尿失禁的治疗。
T39924 NF-κΒ activator 2

NF-κB NF-κB
NF-κΒ activator 2 是口服有效的 NF-ҡB 激活剂,EC50为 1.58 μM。它通过增加 NF-κB 的表达和激活来诱导 SOD2。它具有用于研究肌萎缩性侧索硬化症的价值。
T21620 Adenosine receptor antagonist 4

Adenosine Receptor GPCR/G Protein; Neuroscience
Adenosine receptor antagonist 4 是一种腺苷受体拮抗剂。
T35427 β-Lactamase-IN-2

Antibacterial Microbiology/Virology
β-Lactamase-IN-2 是 β-内酰胺酶的有效抑制剂。β-Lactamase-IN-2显示出抗菌活性。
T21000 PiB

2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇,Pittsburgh Compound-B,6-OH-BTA-1

Others Others
PiB (Pittsburgh Compound-B) 是分析 11C-PiB 的标准品。 11C-PiB 是一种用于阿尔茨海默病诊断的 β-淀粉样蛋白 PET 成像示踪剂。
T7433 2-Phenylethylamine hydrochloride

&beta,-Phenylethylamine hydrochloride,2-苯乙胺盐酸盐,benzeneethanamine hydrochloride,&beta,-aminoethylbenzene hydrochloride

Others Others
2-Phenylethylamine hydrochloride (benzeneethanamine hydrochloride) 是神经调节剂或神经递质。
T8749 CS-B1628

2-(6-溴-5-甲基-2,4-二氧代-1,4-二氢噻吩并[2,3-D]嘧啶-3(2H) - 基)-,tert-Butyl 2-(6-bromo-5-methyl-2,4-dioxo-1,4-dihydrothieno[2,3-d]pyrimidin-3(2H)-yl)-2-methylpropanoate,ACN-053859

Others Others
CS-B1628 (tert-Butyl 2-(6-bromo-5-methyl-2,4-dioxo-1,4-dihydrothieno[2,3-d]pyrimidin-3(2H)-yl)-2-methylpropanoate) 可用于合成嘧啶衍生物,具有成为各种有机化合物(包括药物和农用化学品)起始材料的潜在用途。
TP1730L β-catenin peptide acetate(265669-37-2 free base)

Others Others
β-catenin peptide acetate(265669-37-2 free base) 是一种由 Kb 呈递的天然存在的自身肽,可非常有效地介导 OT-I 胸腺细胞的阳性选择。
TP2359 FMOC-DL-7-AZATRYPTOPHAN

2-({[(9H-fluoren-9-yl)methoxy]carbonyl}amino)-3-{1H-pyrrolo[2,3-b]pyridin-3-yl}propanoic acid

Others Others
FMOC-DL-7-AZATRYPTOPHAN (2-({[(9H-fluoren-9-yl)methoxy]carbonyl}amino)-3-{1H-pyrrolo[2,3-b]pyridin-3-yl}propanoic acid) 是肽。
T14909 CCX140

3-三氟甲基-4-氯-N-[2-[7H-吡咯并[2,3-D]嘧啶-4-羰基]-5-甲基-3-吡啶基]苯磺酰胺,CCX140-B

CCR Immunology/Inflammation; Microbiology/Virology
CCX140 (CCX140-B) 是 CCR2 的拮抗剂。
T2234 TCS JNK 5a

N-(3-氰基-4,5,6,7-四氢苯并[b]噻吩-2-基)-1-萘甲酰胺,SC202671,SC 202671,N-(3-Cyano-4,5,6,7-tetrahydrobenzo[b]thienyl-2-yl)-1-naphthalenecarboxamide,JNK Inhibitor IX,SC-202671

Apoptosis; JNK Apoptosis; MAPK
TCS JNK 5a (SC202671) 是一种 JNK2和 JNK3的有效抑制剂,pIC50分别为 6.5和 6.7。
T20889 AalphaC

2-Amino-alpha-carboline,Aalpha C,2-氨基-9H-吡啶[2,3-b]吲哚,Aalpha-C

Others Others
AalphaC (2-Amino-alpha-carboline) 是一种潜在的致癌物质。
T9320 YK-3-237

B-[2-Methoxy-5-[(1E)-3-oxo-3-(3,4,5-trimethoxyphenyl)-1-propen-1-yl]phenyl]boronic acid

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
YK-3-237 (B-[2-Methoxy-5-[(1E)-3-oxo-3-(3,4,5-trimethoxyphenyl)-1-propen-1-yl]phenyl]boronic acid) 是 SIRT1 激活剂,靶向突变体 p53。它抑制三阴性乳腺癌细胞的增殖。
T7546 Bethoxazin

3-苯并[b]噻吩-2-基-5,6-二氢-1,4,2-噻嗪 4-氧化物

Antibacterial Microbiology/Virology
Bethoxazin 是一种新型广谱工业杀菌剂。
T8326 BMS-2

1-(4-氟苯基)-N-[3-氟-4-(1H-吡咯并[2,3-B]吡啶-4-基氧基)苯基]-1,2-二氢-2-氧代-3-吡啶甲酰胺

VEGFR; FLT; c-Met/HGFR Angiogenesis; Tyrosine Kinase/Adaptors
BMS-2 是 Met/Flt-3/VEGFR2 酪氨酸激酶抑制剂。
T6746 6-Thio-2'-Deoxyguanosine

6-Thio-dG,β-TGdR

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
6-Thio-2'-Deoxyguanosine (β-TGdR) 是一种核苷类似物和端粒酶底物,可以通过端粒酶掺入重新合成的端粒中。
T3467 Miransertib

ARQ-092,AKT inhibitor 2

Akt; Parasite Cytoskeletal Signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling
Miransertib (ARQ-092) 是一种具有口服活性的,选择性和变构性Akt 抑制剂。它有效抑制利什曼原虫,还是 AKT1-E17K 突变蛋白抑制剂,可研究PI3K/AKT 驱动的肿瘤和 Proteus 综合征。
T21667 FAUC-365

FAUC-365 Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro- phenyl)-piperazin-1-yl]-butyl}-amide,FAUC-365 Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro- phenyl)-piperazin-1-yl]-butyl}-amide

Dopamine Receptor GPCR/G Protein; Neuroscience
FAUC-365 是一种高度选择性的多巴胺D3受体拮抗剂,能够作用于 D3 受体(Ki:0.5 nM)、D4.4 受体(Ki:340 nM)、D2short 受体(Ki:2600 nM)和 D2Long 受体(Ki:3600 nM)。它可用于研究帕金森病、精神分裂症等疾病。
T8917 PAR-2-IN-1

IUN76750,8-(叔丁基)-6-氯咪唑并[1,2-B]吡啶-2-羧酸甲酯

Protease-activated Receptor GPCR/G Protein
PAR-2-IN-1 (IUN76750) 是一种 PAR-​2 信号通路抑制剂,具有抗炎和抗癌作用。
T9040 Aurora kinase inhibitor-2

IUN-70219,Aurora Kinase Inhibitor II

Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic
Aurora kinase inhibitor-2 (IUN-70219) 是一种可渗透细胞的苯胺喹唑啉,可抑制极光激酶的活性,对Aurora A 和Aurora B 的IC50分别为 390 nM 和 240 nM。
T6065 Triciribine

VD-0002,Tricyclic nucleoside,NSC 154020,曲西立滨,API-2,TCN

Akt; HIV Protease; DNA/RNA Synthesis Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Microbiology/Virology; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Triciribine (NSC-154020) 是一种 DNA 合成抑制剂,也抑制 Akt 和 HIV-1/2,IC50分别为 130 nM 和 0.02-0.46 μM。

化合物

B-Raf IN 2
Cat.No: T40284
Synonym:
Target: Raf
MAO-B-IN-2
Cat.No: T9560
Synonym:
Target:
Benzamide, 3-methoxy-N-(3-thiazolo[5,4-b]pyridin-2-ylphenyl)
Cat.No: T60001
Synonym: 3-methoxy-N-(3-(thiazolo[5,4-b]pyridin-2-yl)phenyl)benzamide
Target: Sirtuin
Benzo[b]thiophene-7-propanoic acid, α-methoxy-4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]-, (αR)-
Cat.No: T63898
Synonym:
Target: PPAR
sodium 3-amino-4,6-dimethylthieno[2,3-b]pyridine-2-carboxylate
Cat.No: T50009L
Synonym:
Target: Others
B2
Cat.No: T22595
Synonym: Linazolamide intermediate B impurity 2,CPNQ,5-[4-(4-Chlorobenzoyl)-1-piperazinyl]-8-nitroquinoline,奥司他韦杂质B(2-叠氮杂合物)
Target: Others, Sirtuin
3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
Cat.No: T9752
Synonym:
Target: Androgen Receptor
AKOS B018304
Cat.No: T5103
Synonym: (5E)-5-(2-硝基苯亚甲基)-2-硫代-四氢噻唑-4-酮
Target: Others
2H-​Imidazo[4,​5-​b]​pyrazin-​2-​one, 1,​3-​dihydro-​6-​[6-​(1-​hydroxy-​1-​methylethyl)​-​3-​pyridinyl]​-​1-​[(tetrahydro-​2H-​pyran-​4-​yl)​methyl]​-
Cat.No: T9315
Synonym:
Target: Others
CCK-B Receptor Antagonist 2
Cat.No: T10707
Synonym:
Target: Others
Wnt/β-catenin agonist 2
Cat.No: T41094
Synonym:
Target: GSK-3, Wnt/beta-catenin
Beta-Tetralone
Cat.No: T0660
Synonym: 2-Tetralone,beta-四氢萘酮
Target: P450
Dazonone
Cat.No: T9871
Synonym: Imidazo[2,1-b]quinazolin-2(3H)-one, 6-chloro-1,5-dihydro-3-methyl-
Target: PDE
Sirtuin modulator 2
Cat.No: T9999
Synonym: N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide
Target: Others, Sirtuin
MRZ 2-514
Cat.No: T12110
Synonym: 8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one
Target: NMDAR
LCB 03-0110
Cat.No: T9659
Synonym: 3-(2-(3-(Morpholinomethyl)phenyl)thieno[3,2-b]pyridin-7-ylamino)phenol
Target: Discoidin Domain Receptor (DDR)
InhA-IN-2
Cat.No: T9734
Synonym:
Target: CDK
Senexin B
Cat.No: T8430
Synonym: 4-[[2-[6-[(4-甲基-1-哌嗪基)羰基]-2-萘基]乙基]氨基]-6-喹唑啉甲腈
Target: CDK
HPK1-IN-2
Cat.No: T9017
Synonym: Thieno[2,3-b]pyridin-6(7H)-one, 4-amino-5-[6-(4-methyl-1-piperazinyl)-1H-benzimidazol-2-yl]-HPK1-IN-2,HPK1-IN-2
Target: Others, FLT, Src
AKT inhibitor VIII
Cat.No: T3346
Synonym: AKTi-1/2
Target: Apoptosis, Akt
(Rac)-Daglutril
Cat.No: T27119L
Synonym: SLV 306 acetic acid,2-((3S)-3-(1-(2-(ethoxycarbonyl)-4-phenylbutyl)cyclopentane-1-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)acetic acid
Target: Others
TBK1/IKKε-IN-2
Cat.No: T15559
Synonym:
Target: B/IKK
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide
Cat.No: T50083
Synonym:
Target: Others
ACHP Hydrochloride
Cat.No: T10237
Synonym: IKK-2 Inhibitor VIII
Target: B/IKK
FMAU
Cat.No: TNU0159
Synonym: 2'-Deoxy-2'-fluoro-5-methyl-beta-D-arabinouridine
Target: Apoptosis
β-Lactamase-IN-1
Cat.No: T19206
Synonym: 4-(1,3-dihydroxypropan-2-yl)-6-methoxypyrido[2,3-b]pyrazin-3-one,beta-lactamase-IN-1
Target: Antibacterial
β-catenin-IN-2
Cat.No: T9696
Synonym:
Target: Wnt/beta-catenin
ONPG
Cat.No: T19497
Synonym: 2-硝基苯-beta-D-半乳糖苷,2-Nitrophenyl β-D-galactopyranoside
Target: Others
MASM7
Cat.No: T50093
Synonym:
Target: Others
(-)-OPC-51803
Cat.No: T28257L
Synonym:
Target: AChR
NF-κΒ activator 2
Cat.No: T39924
Synonym:
Target: NF-κB
Adenosine receptor antagonist 4
Cat.No: T21620
Synonym:
Target: Adenosine Receptor
β-Lactamase-IN-2
Cat.No: T35427
Synonym:
Target: Antibacterial
PiB
Cat.No: T21000
Synonym: 2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇,Pittsburgh Compound-B,6-OH-BTA-1
Target: Others
2-Phenylethylamine hydrochloride
Cat.No: T7433
Synonym: &beta,-Phenylethylamine hydrochloride,2-苯乙胺盐酸盐,benzeneethanamine hydrochloride,&beta,-aminoethylbenzene hydrochloride
Target: Others
CS-B1628
Cat.No: T8749
Synonym: 2-(6-溴-5-甲基-2,4-二氧代-1,4-二氢噻吩并[2,3-D]嘧啶-3(2H) - 基)-,tert-Butyl 2-(6-bromo-5-methyl-2,4-dioxo-1,4-dihydrothieno[2,3-d]pyrimidin-3(2H)-yl)-2-methylpropanoate,ACN-053859
Target: Others
β-catenin peptide acetate(265669-37-2 free base)
Cat.No: TP1730L
Synonym:
Target: Others
FMOC-DL-7-AZATRYPTOPHAN
Cat.No: TP2359
Synonym: 2-({[(9H-fluoren-9-yl)methoxy]carbonyl}amino)-3-{1H-pyrrolo[2,3-b]pyridin-3-yl}propanoic acid
Target: Others
CCX140
Cat.No: T14909
Synonym: 3-三氟甲基-4-氯-N-[2-[7H-吡咯并[2,3-D]嘧啶-4-羰基]-5-甲基-3-吡啶基]苯磺酰胺,CCX140-B
Target: CCR
TCS JNK 5a
Cat.No: T2234
Synonym: N-(3-氰基-4,5,6,7-四氢苯并[b]噻吩-2-基)-1-萘甲酰胺,SC202671,SC 202671,N-(3-Cyano-4,5,6,7-tetrahydrobenzo[b]thienyl-2-yl)-1-naphthalenecarboxamide,JNK Inhibitor IX,SC-202671
Target: Apoptosis, JNK
AalphaC
Cat.No: T20889
Synonym: 2-Amino-alpha-carboline,Aalpha C,2-氨基-9H-吡啶[2,3-b]吲哚,Aalpha-C
Target: Others
YK-3-237
Cat.No: T9320
Synonym: B-[2-Methoxy-5-[(1E)-3-oxo-3-(3,4,5-trimethoxyphenyl)-1-propen-1-yl]phenyl]boronic acid
Target: Sirtuin
Bethoxazin
Cat.No: T7546
Synonym: 3-苯并[b]噻吩-2-基-5,6-二氢-1,4,2-噻嗪 4-氧化物
Target: Antibacterial
BMS-2
Cat.No: T8326
Synonym: 1-(4-氟苯基)-N-[3-氟-4-(1H-吡咯并[2,3-B]吡啶-4-基氧基)苯基]-1,2-二氢-2-氧代-3-吡啶甲酰胺
Target: VEGFR, FLT, c-Met/HGFR
6-Thio-2'-Deoxyguanosine
Cat.No: T6746
Synonym: 6-Thio-dG,β-TGdR
Target: Others, DNA/RNA Synthesis
Miransertib
Cat.No: T3467
Synonym: ARQ-092,AKT inhibitor 2
Target: Akt, Parasite
FAUC-365
Cat.No: T21667
Synonym: FAUC-365 Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro- phenyl)-piperazin-1-yl]-butyl}-amide,FAUC-365 Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro- phenyl)-piperazin-1-yl]-butyl}-amide
Target: Dopamine Receptor
PAR-2-IN-1
Cat.No: T8917
Synonym: IUN76750,8-(叔丁基)-6-氯咪唑并[1,2-B]吡啶-2-羧酸甲酯
Target: Protease-activated Receptor
Aurora kinase inhibitor-2
Cat.No: T9040
Synonym: IUN-70219,Aurora Kinase Inhibitor II
Target: Aurora Kinase
Triciribine
Cat.No: T6065
Synonym: VD-0002,Tricyclic nucleoside,NSC 154020,曲西立滨,API-2,TCN
Target: Akt, HIV Protease, DNA/RNA Synthesis
Cat. No. Product Name Target Signaling Pathways
T6S0735 Flavokawain B

黄卡瓦胡椒素B,Flavokavain B,Flavokawin B,2'-Hydroxy-4',6'-Dimethoxychalcone

Apoptosis; Others Apoptosis; Others
Flavokawain B (Flavokavain B) 是从卡瓦醉椒的根提取物中,分离出的查尔酮。它是一种凋亡诱导剂,可抑制各种癌细胞株生长。它以极低的无毒浓度抑制人脑内皮细胞的迁移和血管形成,具有抗血管生成活性。
T6S1367 Procyanidin B2

原花青素 B2,Proanthocyanidin B2

Reactive Oxygen Species; NOD Immunology/Inflammation; Metabolism; NF-κB
Procyanidin B2 (Proanthocyanidin B2) 是天然黄酮类物质,具有抗肿瘤,抗氧化等活性。
TN5569 2-Deacetoxytaxinine B

2-Deacetoxytaxinine B is a strongly inhibitor against U46619-induced aggregation, it shows strong inhibitory effects against arachidonic acid (AA)-induced aggregation.
T3780 Oroxin B

Hypocretin-2,木蝴蝶苷B

Apoptosis; PTEN; Antioxidant; PI3K; Autophagy Apoptosis; Autophagy; oxidation-reduction; PI3K/Akt/mTOR signaling
Oroxin B (Hypocretin-2) 是从传统中草药木蝴蝶中分离出来的黄酮类天然产物,在恶性淋巴瘤细胞中诱导肿瘤抑制性 ER 应激。它通过上调 PTEN,下调 COX-2,VEGF,PI3K 和 p-AKT,对肝癌细胞具有明显的抑制作用,诱导细胞早期凋亡。
TN1530 Cowaxanthone B

β-倒捻子素类似物2

Antioxidant; Parasite Microbiology/Virology; oxidation-reduction
Cowaxanthone B 是从小叶藤黄果实中分离出的新的四氧氧杂蒽酮。Cowaxanthone B 具有潜在的抗菌活性。
TN4857 (+)-Puerol B 2''-O-glucoside

Others Others
(+)-Puerol B 2''-O-glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4857,CAS号为 868409-19-2
T5713 2"-O-beta-L-galactopyranosylorientin

荭草素-2"-0-B-L半乳糖苷,荭草素-2"-O-BETA-L-半乳糖苷,2''-O-β-L-Galorientin

Others Others
2"-O-beta-L-galactopyranosylorientin (2''-O-β-L-Galorientin) 提取自Trollius ledebouri 的花朵。它是多药耐药蛋白2 (MRP2) 的底物,能够被动扩散,并涉及转运蛋白介导的外排作用。
T3344 Ciwujianoside B

yemuoside YM,刺五加皂苷 B,acanthopanax senticosides B,刺五加皂甙 B,Ciwujianoside-B

BCL; Others Apoptosis; Others
Ciwujianoside B (acanthopanax senticosides B) 是刺五加的主要成分,能缓解疲劳,增强记忆力,提高人的认知能力。
T20587 2-Acetonaphthone

2-萘乙酮,beta-Acetylnaphthalene,beta-Acetonaphthalene,2Acetylnaphthalene,2-Acetylnaphthalene,2 Acetylnaphthalene,beta-Naphthyl methyl ketone

Endogenous Metabolite Metabolism
2-Acetonaphthone (beta-Naphthyl methyl ketone) 是内源性代谢产物的一种。
T3810 Saikosaponin B2

柴胡皂苷 B2,柴胡皂甙 B2

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
Saikosaponin B2 是从柴胡根中分离得到的一种活性成分,可抑制 HCV 病毒感染的侵入,有抗癌作用。
T2964 2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside

芪多酚,2,3,4',5-Tetrahydroxystilbene 2-O-D-glucoside,2,3,5,4'-Tetrahydroxystilbene-2-O-b-D-glucopyranoside,Astragalus polyphenols

Others Others
2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside (Astragalus polyphenols) 是分离自蓼属植物物种的根中,对5-HETE、HHT、thromboxane B2的形成具有抑制作用。
TN1534 Cucurbitacin B 2-O-beta-D-glucoside

Others Others
Cucurbitacin B 2-o-α²-D-glucoside has anticancer activity.
T3779 Crocin II

Crocin 2,西红花苷II,Crocetin gentiobiosylglucosyl ester,藏红花,Tricrocin,Crocin B

Caspase; COX; NO Synthase Apoptosis; Immunology/Inflammation; Neuroscience; Proteases/Proteasome
Crocin II (Crocetin gentiobiosylglucosyl ester) 是从栀子果实中分离出来的一种天然产物,具有抗氧化、抗癌和抗抑郁活性。它抑制 iNOS 和 COX-2的蛋白质和 m-RNA 的表达,还抑制NO 产生,IC50值为 31.1 μM。
TN1921 Meloside A

异牡荆素-2''-O-葡萄糖苷,Isovitexin 2''-O-glucoside,Isovitexin 2''-O-β-D-glucoside

Others Others
Meloside A (Isovitexin 2''-O-β-D-glucoside) 是一种从大麦中提取的苯丙烷类天然产物。 Meloside A 对过量的 UV-B 辐射具有抗氧化和保护作用,并与对病原体的抵抗力有关。
TN1470 Cassiaside B2

决明子苷B2

Phosphatase; MAO; 5-HT Receptor GPCR/G Protein; Metabolism; Neuroscience
Cassiaside B2 是蛋白酪氨酸磷酸酶1B (PTP1B) 和人单胺氧化酶A (hMAO-A) 的抑制剂。Cassiaside B2是 5-HT2C 受体的激动剂, 具有抗过敏活性。Cassiaside B2 是萘吡喃酮参比提取物(NRE)的有效成分之一。
T3122 Fangchinoline

Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline

Apoptosis; FAK; HIV Protease; Autophagy Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Fangchinoline (Tetrandrine B) 是从Stephaniatetrandra 中分离出来的,一种具有广泛生物学活性的天然产物。它是新型HIV-1抑制剂,通过损害 gp160 蛋白水解过程来抑制 HIV-1 复制。它靶向Focal adhesion kinase (FAK)并抑制肿瘤细胞中 FAK 介导的的信号传导途径。
TN2139 Regaloside B

鸦胆子苦醇,王百合苷 B

NOS; COX; NO Synthase Immunology/Inflammation; Neuroscience
Regaloside B 是从麝香百合中分离出来的一种苯丙烷,可抑制iNOS 和COX-2的表达,具有抗炎活性。
T0937 Riboflavin

Vitamin B2,维生素B2,E101

Endogenous Metabolite Metabolism
Riboflavin (E101),一种人内源性代谢物, 是极易吸收的微量营养素。
T2769 3-Aminopropionitrile fumarate (2:1)

Di-β-aminopropionitrile fumarate,3-Aminopropionitrile fumarate,3-氨基丙腈,β-Aminopropionitrile fumarate,3-Aminopropionitrile fumarate 2:1,Beta-Aminopropionitrile fumarate,β-Ammoniumpropionitrile hemifumarate

Others Others
3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) 是一种能抑制胶原蛋白(collagen)交联的山黧豆素。
TN1259 Complanatoside B

3-O-Β-D-芹糖(1-2)-Β-D-葡萄糖-鼠李柠檬素4'-O-Β-D-葡萄糖苷,沙苑子苷B

Others Others
Complanatoside B 是一种黄酮类天然产物,具有抗炎作用。
T6S1917 Schisandrol B

Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B

P450; Reactive Oxygen Species; Autophagy Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Schisandrol B (Besigomsin) 是华中五味子的主要活性成分,具有保肝、抗炎、抗糖尿病和抗氧化的作用。它抑制活性氧的产生,也抑制 P-糖蛋白和CYP3A 的活性。
T4956 Tetrahydroxystilbene-2-O-β-D-glucoside

tetrahydroxyl diphenylethylene-2-o-gluco,何首乌苷,EH-201

Others Others
Tetrahydroxystilbene-2-O-β-D-glucoside (EH-201) 是一种低分子量的促红细胞生成素诱导剂。
TN1433 Batatasin III

FAK; Others; Akt Angiogenesis; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Batatasin III 通过抑制上皮间质转化和 FAK-AKT 信号来抑制癌症迁移和侵袭,并具有抗癌活性。 Batatasin III 对整株生长有长期抑制作用,显示出抑制萌发活性。
TN7028 Eurycomanol 2-O-β-D-glucopyranoside

Others Others
Eurycomanol 2-O-β-D-glucopyranoside是一种天然化合物,属于二萜类,提取于东革阿里。
T5704 Entadamide-A-β-D-glucopyranoside

(E)-N-[2-(β-D-Glucopyranosyloxy)ethyl]-,榼藤子酰胺A-Β-D-吡喃葡萄糖苷,榼藤子酰胺A-β-D-吡喃葡萄糖

Others Others
Entadamide-A-β-D-glucopyranoside ((E)-N-[2-(β-D-Glucopyranosyloxy)ethyl]-) 是一种菜豆虫种子的主要成分,具有抗补体作用。
T0627 β-Alanine

beta-Alanine,beta-氨基丙酸,3-Aminopropanoic acid,2-Carboxyethylamine,β-丙氨酸

GABA Receptor; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Neuroscience
β-Alanine (3-Aminopropanoic acid) 是一种天然存在的β-氨基酸,在体内由二氢尿嘧啶和肌肽降解形成,它作为神经递质可激活甘氨酸和GABA受体。
T4024 Norharmane

2-Azacarbazole,2,9-Diazafluorene,β-Carboline,去甲哈尔满

DNA; Endogenous Metabolite; Monoamine Oxidase DNA Damage/DNA Repair; Metabolism; Neuroscience
Norharmane (β-Carboline) 是一种有效的选择性单胺氧化酶 A (MAO-A) 抑制剂,Ki=3.34 μM。
TN6909 Polyporusterone B

猪苓酮B,(1R,2R,4S,5R,7R,11R,14S,15R)-14-[(2R,3R)-2,3-dihydroxy-6-methyl-5-methylideneheptan-2-yl]-4,5,11-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,?.011,1?]heptadec-9-en-8-one

Others Others
Polyporusterone B ((1R,2R,4S,5R,7R,11R,14S,15R)-14-[(2R,3R)-2,3-dihydroxy-6-methyl-5-methylideneheptan-2-yl]-4,5,11-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,?.011,1?]heptadec-9-en-8-one) 是一种三萜羧酸,从Polyporus umbellatusFries 中分离得到。它对自由基诱导的红细胞裂解 (溶血) 具有抑制作用。
T2932 Ginsenoside Rh1

Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1

IL Receptor; TNF; Endogenous Metabolite; PPAR; Interleukin Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism
Ginsenoside Rh1 (Sanchinoside B2) 是人参的一种主要成分,具有抗炎作用,抑制PPAR-γ,TNF-α,IL-6和IL-1β的表达。
TP2167 β-CGRP, human acetate

β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate

CGRP Receptor GPCR/G Protein; Neuroscience
β-CGRP, human acetate 是降钙素肽之一,通过受体活性修饰蛋白 (RAMP) 和降钙素受体样受体 (CRLR) 的复合物发挥作用(对于 CRLR/RAMP1 和 CRLR,IC50:1 nM 和 300 nM /RAMP2 在单元格中)。
T6460 Cysteamine hydrochloride

2-Mercaptoethylamine Hydrochloride,β-Mercaptoethylamine Hydrochloride,半胱胺盐酸盐,Thioethanolamine Hydrochloride,2-Aminoethanethiol Hydrochloride,Cysteamine HCl,Bekaptan

Apoptosis; Others; Reactive Oxygen Species; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB; Others
Cysteamine hydrochloride (Thioethanolamine Hydrochloride) 是一种可口服的,用于肾病型胱胺酸症的小分子药物,也可作为抗氧化剂。
TN1489 3'-Methoxyapiin

Graveobioside B,3'-Methoxy apiin,Chrysoeriol 7-apiosylglucoside,3'-甲氧基芹菜苷

Others Others
3'-Methoxyapiin (Graveobioside B) 是一种来自 Eminium spiculatum 植物的类黄酮。
T2872 Ginsenoside Re

人参皂苷 Re,Ginsenoside B2,Panaxoside Re,Chikusetsusaponin Ivc,Sanchinoside Re,人参皂苷Re

Beta Amyloid; NF-κB; Endogenous Metabolite; JNK MAPK; Metabolism; Neuroscience; NF-κB
Ginsenoside Re (Ginsenoside B2) 是一种人参提取物,可降低 β-淀粉样蛋白 (Aβ),还通过抑制 JNK 和 NF-κB 发挥抗炎作用。
TN3500 beta-Amyrone

β-Amyron,β-香树脂酮

COX; AChR; PPAR; Antifection DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
beta-Amyrone (β-Amyron) 对基孔肯雅病毒复制具有抗真菌活性,EC50 为 86 uM。 beta-Amyrone 通过抑制 COX-2 的表达而具有抗炎活性。 beta-Amyrone 表现出抗α-葡萄糖苷酶抑制活性和中等 AChE 活性。 β-Amyrone 可用于炎症、感染和肥胖等疾病的研究。
TN6719 Kaempferol-3-O-β-D-glucosyl(1-2)rhamnoside

Others Others
Kaempferol-3-O-β-D-glucosyl(1-2)rhamnoside 是一种从阿拉伯茉莉中分离出来的天然产物。
T5246 Trans-​2-​butene-​1,​4-​dicarboxylic acid

trans-2-Butene-1,4-dicarboxylic Acid,3-Hexenedioic Acid,trans-3-Hexenedioic Acid,β-Hydromuconic Acid,反式-2-丁烯-1,4-二甲酸

Others; Endogenous Metabolite Metabolism; Others
Trans-​2-​butene-​1,​4-​dicarboxylic acid (3-Hexenedioic Acid) 是内源性代谢产物的一种。
TN6734 Quercetin-3-O-D-glucosyl]-(1-2)-L-rhamnoside

Quercetin 3-O-beta-D-glucosyl-(1->2)-rhamnoside,槲皮素-3-O-葡萄糖基-(1-2)-L-鼠李糖苷,槲皮素 3-O-葡萄糖基 (1→2)鼠李糖苷

Others Others
Quercetin-3-O-D-glucosyl]-(1-2)-L-rhamnoside (Quercetin 3-O-beta-D-glucosyl-(1->2)-rhamnoside) 是 Shuxuenin 中的一种主要抗氧化剂。
T5621 β-Phellandrene

beta-Phellandrene,3-异丙基-6-亚甲基-1-环己烯,p-mentha-1(7),2-diene,(±)-beta-水芹烯

Others Others
β-Phellandrene (p-mentha-1(7),2-diene) 是由加拿大香脂油分馏取得,可用作精油添加剂。
TN4537 Methyl 8-hydroxy-3-(2-methoxy-2-oxoethyl)-6-methyl-9-oxo-9H-furo[3,4-b]chromene-1-carboxylate

Others Others
Methyl 8-hydroxy-3-(2-methoxy-2-oxoethyl)-6-methyl-9-oxo-9H-furo[3,4-b]chromene-1-carboxylate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4537,CAS号为 96287-41-1。
T1048 Estradiol

雌二醇,E2,17β-Estradiol,17β-Oestradiol,β-Estradiol

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Estradiol (E2) 是一种天然的类固醇性激素,对于女性生育能力和第二性征的维持至关重要。Estradiol 通过雌激素受体 β (ERβ) 上调 IL-6 表达。
T4887 3-Amino-2-methylpropanoic acid

DL-3-AMINOISOBUTYRIC ACID,3-氨基异丁酸,α-Methyl-β-alanine

Endogenous Metabolite Metabolism
3-Amino-2-methylpropanoic acid (α-Methyl-β-alanine) 是 N-carbamyl-beta-aminoisobutyric acid 经 enzyme Beta-ureidopropionase (EC 3.5.1.6)转化后的产物,是嘧啶降解的最后一步。-尿嘧啶丙酸酶缺乏症是一种与神经异常相关的嘧啶降解的先天性错误。
T6185 Gambogic Acid

藤黄酸,Beta-Guttiferrin,藤黄酸 A,Guttatic Acid,Guttic Acid

BCL; Autophagy Apoptosis; Autophagy
Gambogic Acid (Guttic Acid) 是来自藤黄树的一种藤黄树脂,抑制 Bcl-XL、Bcl-2Bcl-W、Bcl-BBfl-1和 Mcl-1,IC50分别为 1.47 μM、1.21 μM、2.02 μM、0.66 μM、1.06 μM 和 0.79 μM。
T5S0483 (-)-Syringaresnol-4-O-β-D-apiofuranosyl-(1→2)-β-D-glucopyranoside

(-)-丁香树脂酚-4-O-beta-D-呋喃芹糖基-(1→2)-beta-D-吡喃葡萄糖苷,(-)-Syringaresnol-4-O-beta-D-apiofuranos

Others Others
(-)-Syringaresnol-4-O-β-D-apiofuranosyl-(1→2)-β-D-glucopyranoside ((-)-Syringaresnol-4-O-beta-D-apiofuranos) 是从Albizzia myriophylla 的树皮部分分离得到。
TN6287 Apigenin 7-O-(2'',6''-di-O-E-p-coumaroyl)glucoside

Anisofolin B

Apigenin 7-O-(2'',6''-di-O-E-p-coumaroyl)glucoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6287,CAS号为 1448779-19-8。
TN2768 2 beta-Hydroxykolavelool

Others Others
2 beta-Hydroxykolavelool is a natural product from Sagittaria trifolia.
TN6176 Platachromone B

5,7,4'-Trihydroxy-8-isoprenyl-2-styrylchromone

Platachromone B 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6176,CAS号为 1606149-63-6。
TN2117 Pulsatilloside E

3-O-B-D-葡萄糖( 1→4)-[ A -L-鼠李糖(1→2)]- A-L-阿拉伯糖 23-羟基羽扇豆20(29)-烯-28–酸- 28-O-鼠李糖(1→4)葡萄糖(1→6)葡萄糖苷,Pulchinenoside E,白头翁皂苷E

Others Others
Pulsatilloside E (Pulchinenoside E) 是一种从毛茛科白头翁Pulsatilla chinensis (Ranunculaceae)的根中分离出来的天然产物。
TN3083 Artoindonesianin B-1

5-(6-Hydroxybenzofuran-2-yl)-2-(3-methylbut-1-enyl)benzene-1,3-diol

Others Others
Artoindonesianin B-1 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN3083,CAS号为 936006-11-0。
T1080 2-Aminoethanethiol

2-Mercaptoethylamine,巯基乙胺,β-Mercaptoethylamine,β-MEA,Cysteamine

Apoptosis; Others; Reactive Oxygen Species; Cysteine Protease; Somatostatin; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; GPCR/G Protein; Immunology/Inflammation; Metabolism; NF-κB; Others; Proteases/Proteasome
2-Aminoethanethiol (Cysteamine) 是一种胱氨酸消耗剂。半胱胺的作用机制是胱氨酸二硫化物还原。
T19359 Hydrolyzed Fumonisin B2

Others Others
Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.
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天然产物

Flavokawain B
Cat.No: T6S0735
Synonym: 黄卡瓦胡椒素B,Flavokavain B,Flavokawin B,2'-Hydroxy-4',6'-Dimethoxychalcone
Target: Apoptosis, Others
Procyanidin B2
Cat.No: T6S1367
Synonym: 原花青素 B2,Proanthocyanidin B2
Target: Reactive Oxygen Species, NOD
2-Deacetoxytaxinine B
Cat.No: TN5569
Synonym:
Target:
Oroxin B
Cat.No: T3780
Synonym: Hypocretin-2,木蝴蝶苷B
Target: Apoptosis, PTEN, Antioxidant, PI3K, Autophagy
Cowaxanthone B
Cat.No: TN1530
Synonym: β-倒捻子素类似物2
Target: Antioxidant, Parasite
(+)-Puerol B 2''-O-glucoside
Cat.No: TN4857
Synonym:
Target: Others
2"-O-beta-L-galactopyranosylorientin
Cat.No: T5713
Synonym: 荭草素-2"-0-B-L半乳糖苷,荭草素-2"-O-BETA-L-半乳糖苷,2''-O-β-L-Galorientin
Target: Others
Ciwujianoside B
Cat.No: T3344
Synonym: yemuoside YM,刺五加皂苷 B,acanthopanax senticosides B,刺五加皂甙 B,Ciwujianoside-B
Target: BCL, Others
2-Acetonaphthone
Cat.No: T20587
Synonym: 2-萘乙酮,beta-Acetylnaphthalene,beta-Acetonaphthalene,2Acetylnaphthalene,2-Acetylnaphthalene,2 Acetylnaphthalene,beta-Naphthyl methyl ketone
Target: Endogenous Metabolite
Saikosaponin B2
Cat.No: T3810
Synonym: 柴胡皂苷 B2,柴胡皂甙 B2
Target: Others, HCV Protease
2,3,5,4'-Tetrahydroxystilbene 2-O-β-D-glucoside
Cat.No: T2964
Synonym: 芪多酚,2,3,4',5-Tetrahydroxystilbene 2-O-D-glucoside,2,3,5,4'-Tetrahydroxystilbene-2-O-b-D-glucopyranoside,Astragalus polyphenols
Target: Others
Cucurbitacin B 2-O-beta-D-glucoside
Cat.No: TN1534
Synonym:
Target: Others
Crocin II
Cat.No: T3779
Synonym: Crocin 2,西红花苷II,Crocetin gentiobiosylglucosyl ester,藏红花,Tricrocin,Crocin B
Target: Caspase, COX, NO Synthase
Meloside A
Cat.No: TN1921
Synonym: 异牡荆素-2''-O-葡萄糖苷,Isovitexin 2''-O-glucoside,Isovitexin 2''-O-β-D-glucoside
Target: Others
Cassiaside B2
Cat.No: TN1470
Synonym: 决明子苷B2
Target: Phosphatase, MAO, 5-HT Receptor
Fangchinoline
Cat.No: T3122
Synonym: Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline
Target: Apoptosis, FAK, HIV Protease, Autophagy
Regaloside B
Cat.No: TN2139
Synonym: 鸦胆子苦醇,王百合苷 B
Target: NOS, COX, NO Synthase
Riboflavin
Cat.No: T0937
Synonym: Vitamin B2,维生素B2,E101
Target: Endogenous Metabolite
3-Aminopropionitrile fumarate (2:1)
Cat.No: T2769
Synonym: Di-β-aminopropionitrile fumarate,3-Aminopropionitrile fumarate,3-氨基丙腈,β-Aminopropionitrile fumarate,3-Aminopropionitrile fumarate 2:1,Beta-Aminopropionitrile fumarate,β-Ammoniumpropionitrile hemifumarate
Target: Others
Complanatoside B
Cat.No: TN1259
Synonym: 3-O-Β-D-芹糖(1-2)-Β-D-葡萄糖-鼠李柠檬素4'-O-Β-D-葡萄糖苷,沙苑子苷B
Target: Others
Schisandrol B
Cat.No: T6S1917
Synonym: Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B
Target: P450, Reactive Oxygen Species, Autophagy
Tetrahydroxystilbene-2-O-β-D-glucoside
Cat.No: T4956
Synonym: tetrahydroxyl diphenylethylene-2-o-gluco,何首乌苷,EH-201
Target: Others
Batatasin III
Cat.No: TN1433
Synonym:
Target: FAK, Others, Akt
Eurycomanol 2-O-β-D-glucopyranoside
Cat.No: TN7028
Synonym:
Target: Others
Entadamide-A-β-D-glucopyranoside
Cat.No: T5704
Synonym: (E)-N-[2-(β-D-Glucopyranosyloxy)ethyl]-,榼藤子酰胺A-Β-D-吡喃葡萄糖苷,榼藤子酰胺A-β-D-吡喃葡萄糖
Target: Others
β-Alanine
Cat.No: T0627
Synonym: beta-Alanine,beta-氨基丙酸,3-Aminopropanoic acid,2-Carboxyethylamine,β-丙氨酸
Target: GABA Receptor, Endogenous Metabolite
Norharmane
Cat.No: T4024
Synonym: 2-Azacarbazole,2,9-Diazafluorene,β-Carboline,去甲哈尔满
Target: DNA, Endogenous Metabolite, Monoamine Oxidase
Polyporusterone B
Cat.No: TN6909
Synonym: 猪苓酮B,(1R,2R,4S,5R,7R,11R,14S,15R)-14-[(2R,3R)-2,3-dihydroxy-6-methyl-5-methylideneheptan-2-yl]-4,5,11-trihydroxy-2,15-dimethyltetracyclo[8.7.0.02,?.011,1?]heptadec-9-en-8-one
Target: Others
Ginsenoside Rh1
Cat.No: T2932
Synonym: Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1
Target: IL Receptor, TNF, Endogenous Metabolite, PPAR, Interleukin
β-CGRP, human acetate
Cat.No: TP2167
Synonym: β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate
Target: CGRP Receptor
Cysteamine hydrochloride
Cat.No: T6460
Synonym: 2-Mercaptoethylamine Hydrochloride,β-Mercaptoethylamine Hydrochloride,半胱胺盐酸盐,Thioethanolamine Hydrochloride,2-Aminoethanethiol Hydrochloride,Cysteamine HCl,Bekaptan
Target: Apoptosis, Others, Reactive Oxygen Species, Endogenous Metabolite, Autophagy
3'-Methoxyapiin
Cat.No: TN1489
Synonym: Graveobioside B,3'-Methoxy apiin,Chrysoeriol 7-apiosylglucoside,3'-甲氧基芹菜苷
Target: Others
Ginsenoside Re
Cat.No: T2872
Synonym: 人参皂苷 Re,Ginsenoside B2,Panaxoside Re,Chikusetsusaponin Ivc,Sanchinoside Re,人参皂苷Re
Target: Beta Amyloid, NF-κB, Endogenous Metabolite, JNK
beta-Amyrone
Cat.No: TN3500
Synonym: β-Amyron,β-香树脂酮
Target: COX, AChR, PPAR, Antifection
Kaempferol-3-O-β-D-glucosyl(1-2)rhamnoside
Cat.No: TN6719
Synonym:
Target: Others
Trans-​2-​butene-​1,​4-​dicarboxylic acid
Cat.No: T5246
Synonym: trans-2-Butene-1,4-dicarboxylic Acid,3-Hexenedioic Acid,trans-3-Hexenedioic Acid,β-Hydromuconic Acid,反式-2-丁烯-1,4-二甲酸
Target: Others, Endogenous Metabolite
Quercetin-3-O-D-glucosyl]-(1-2)-L-rhamnoside
Cat.No: TN6734
Synonym: Quercetin 3-O-beta-D-glucosyl-(1->2)-rhamnoside,槲皮素-3-O-葡萄糖基-(1-2)-L-鼠李糖苷,槲皮素 3-O-葡萄糖基 (1→2)鼠李糖苷
Target: Others
β-Phellandrene
Cat.No: T5621
Synonym: beta-Phellandrene,3-异丙基-6-亚甲基-1-环己烯,p-mentha-1(7),2-diene,(±)-beta-水芹烯
Target: Others
Methyl 8-hydroxy-3-(2-methoxy-2-oxoethyl)-6-methyl-9-oxo-9H-furo[3,4-b]chromene-1-carboxylate
Cat.No: TN4537
Synonym:
Target: Others
Estradiol
Cat.No: T1048
Synonym: 雌二醇,E2,17β-Estradiol,17β-Oestradiol,β-Estradiol
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
3-Amino-2-methylpropanoic acid
Cat.No: T4887
Synonym: DL-3-AMINOISOBUTYRIC ACID,3-氨基异丁酸,α-Methyl-β-alanine
Target: Endogenous Metabolite
Gambogic Acid
Cat.No: T6185
Synonym: 藤黄酸,Beta-Guttiferrin,藤黄酸 A,Guttatic Acid,Guttic Acid
Target: BCL, Autophagy
(-)-Syringaresnol-4-O-β-D-apiofuranosyl-(1→2)-β-D-glucopyranoside
Cat.No: T5S0483
Synonym: (-)-丁香树脂酚-4-O-beta-D-呋喃芹糖基-(1→2)-beta-D-吡喃葡萄糖苷,(-)-Syringaresnol-4-O-beta-D-apiofuranos
Target: Others
Apigenin 7-O-(2'',6''-di-O-E-p-coumaroyl)glucoside
Cat.No: TN6287
Synonym: Anisofolin B
Target:
2 beta-Hydroxykolavelool
Cat.No: TN2768
Synonym:
Target: Others
Platachromone B
Cat.No: TN6176
Synonym: 5,7,4'-Trihydroxy-8-isoprenyl-2-styrylchromone
Target:
Pulsatilloside E
Cat.No: TN2117
Synonym: 3-O-B-D-葡萄糖( 1→4)-[ A -L-鼠李糖(1→2)]- A-L-阿拉伯糖 23-羟基羽扇豆20(29)-烯-28–酸- 28-O-鼠李糖(1→4)葡萄糖(1→6)葡萄糖苷,Pulchinenoside E,白头翁皂苷E
Target: Others
Artoindonesianin B-1
Cat.No: TN3083
Synonym: 5-(6-Hydroxybenzofuran-2-yl)-2-(3-methylbut-1-enyl)benzene-1,3-diol
Target: Others
2-Aminoethanethiol
Cat.No: T1080
Synonym: 2-Mercaptoethylamine,巯基乙胺,β-Mercaptoethylamine,β-MEA,Cysteamine
Target: Apoptosis, Others, Reactive Oxygen Species, Cysteine Protease, Somatostatin, Endogenous Metabolite, Autophagy
Hydrolyzed Fumonisin B2
Cat.No: T19359
Synonym:
Target: Others
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