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277

抑制剂 & 化合物

48

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T0049	Azlocillin sodium salt Sodium azlocillin,Azlocillin sodium,阿洛西林钠	Antibacterial; Antibiotic; Parasite	Microbiology/Virology
	Azlocillin sodium salt 是一种半合成青霉素，是内酰胺类广谱抗生素。它具有抗假单胞杆菌的活性，并对抗寄生虫Plasmodium falciparum 有效。
T28973	TIBI	Others	Others
	TIBI 是一种 ATP 竞争性 Rio1 抑制剂，作用方式和丰加霉素相似，可增强酶的热稳定性。
T2131	Articaine hydrochloride Ultracaine,盐酸阿替卡因,阿替卡因,Articaine HCl,Hoe-045	Sodium Channel	Membrane transporter/Ion channel
	Articaine hydrochloride (Hoe-045) 一种牙科局部麻醉剂。
T19672	Amtolmetin guacil MED 15,MED15,ST679,呱氨托美丁,ST-679,ST 679,MED-15	COX	Immunology/Inflammation; Neuroscience
	Amtolmetin guacil (ST-679) 抑制前列腺素合成和环氧合酶。 Amtolmetin guacil 具有与托美汀类似的 NSAID 特性，具有额外的镇痛、解热和胃保护特性。
T25702	Levovirin ICN 17261,L-Ribavirin,ICN-17261,ICN17261
	Levovirin is a monocyclic L-nucleosides with type 1 cytokine-inducing activity. Levovirin is the L-enantiomer of Ribavirin. Levovirin has similar immunomodulatory activity but does not have direct antiviral activity or hemolytic anemia.
T38311	(S)-3-Thienylglycine	Others	Others
	(S)-3-Thienylglycine 是一种噻吩衍生物，可用于研究与噻吩衍生物相似结构的遗传毒性。
T1333	Tolazamide 甲磺氮草脲,妥拉磺脲,U-17835	Potassium Channel	Membrane transporter/Ion channel
	Tolazamide (U-17835) 是一种磺脲类降糖药，用于研究 2 型糖尿病，其作用和用途与氯丙酰胺相似。
T0985	Oxacillin sodium salt 苯唑西林,Oxacillin sodium,Oxabel	Antibacterial; Antibiotic	Microbiology/Virology
	Oxacillin sodium salt (Oxabel) 是一种青霉素类的窄谱β-内酰胺抗生素，用于耐药葡萄球菌感染。
T5531	GSK-4716	Estrogen Receptor/ERR	Endocrinology/Hormones
	GSK-4716 是一种ERRβ/γ选择性激动剂。
T16742	Rhodamine 110 Rhodamine 110 chloride,RH110,罗丹明110	Others	Others
	Rhodamine 110 (RH110) 是灵敏的选择性底物，激发波长为 498 nm，发射波长为 521 nm，可用于测定溶液或活细胞内的蛋白酶。
T6584	MG 149 MG149,Tip60 HAT inhibitor	Apoptosis; Others; Epigenetic Reader Domain; Histone Acetyltransferase	Apoptosis; Chromatin/Epigenetic; Others
	MG 149 (Tip60 HAT inhibitor) 是一种Tip60抑制剂，IC50为 74 μM。它对 MOF 的抑制性较相似，IC50为 47 μM。
T6638	Retapamulin 瑞他莫林,SB-275833	ribosome; Antibacterial; Antibiotic	Microbiology/Virology
	Retapamulin (SB-275833) 是一种能结合金黄色葡萄球菌和大肠杆菌核糖体的局部抗生素，Kd 为3 nM。
T0274	Cinoxacin 西诺沙星,Compound 64716	Topoisomerase; Antibacterial; Antibiotic	DNA Damage/DNA Repair; Microbiology/Virology
	Cinoxacin (Compound 64716) 是一种喹诺酮类的合成抗生素, 与Oxolinic acid 和 Nalidixic acid 活性相似。
T0172	Maprotiline hydrochloride Maprotiline HCl,盐酸马普替林,Psymion,Deprilept,Ludiomil	5-HT Receptor; Adrenergic Receptor; AChR; Norepinephrine; Autophagy; Histamine Receptor	Autophagy; GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Maprotiline hydrochloride (Psymion) 是一种桥环四环类抗抑郁药，是去甲肾上腺素重吸收抑制剂。
T1054	Tolbutamide 甲苯磺丁脲,HLS 831	Potassium Channel; Autophagy	Autophagy; Membrane transporter/Ion channel
	Tolbutamide (HLS 831) 是一种磺脲类降糖药，作用和用途与氯丙酰胺相似。
T0741	Sulfamethazine Sulfadimerazine,磺胺二甲嘧啶,Sulfadimidine	Antibacterial; Antibiotic	Microbiology/Virology
	Sulfamethazine (Sulfadimidine) 是一种抗菌剂，可广泛用于研究和预防各种动物疾病。在中国和欧盟委员会中，动物产品中它的最大残留量为 100 µg/kg。
T14379	AZD5904	Glutathione Peroxidase	Metabolism
	AZD5904 是一种不可逆的人髓过氧化物酶选择性抑制剂，其IC50=140 nM，在小鼠和大鼠中也具有相似的效力。
TP1469	Lixisenatide acetate (320367-13-3 free base) Lixisenatide acetate	Glucagon Receptor	GPCR/G Protein
	Lixisenatide acetate 是一种胰高血糖素样肽 1 受体的激动剂，可用于研究 2 型糖尿病。
T4117	Zuclopenthixol 珠氯噻醇,cis-Clopenthixol,Cisordinol,(Z)-Clopenthixol	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Zuclopenthixol (cis-Clopenthixol) 是一种多巴胺 D1/D2受体的拮抗剂，是一种噻吨衍生物。
TP1457	BIO-11006 acetate salt (901117-03-1 free base) BIO-11006 acetate salt	Others	Others
	BIO-11006 acetate salt (901117-03-1 free base) 是一种多糖基化富含丙氨酸的 C 激酶底物 (MARCKS) 抑制剂，类似于 MANS 肽。
T7108	Omberacetam SGS-111,Noopept,GVS-111	Others; iGluR	Membrane transporter/Ion channel; Neuroscience; Others
	Omberacetam (Noopept) 是一种可作为膳食补充剂的合成二肽，有促智和提高认知作用。
T13587	BT18	Others	Others
	BT18 是一种功能类似于胶质细胞源神经营养因子的分子模拟物。它能够影响 GDNF 家族受体 GFRα1 和 RET 受体酪氨酸激酶 RetA 的功能。
T11044	Dihydromunduletone DHM	GPR	Endocrinology/Hormones; GPCR/G Protein
	Dihydromunduletone (DHM) 是一种粘附 G 蛋白偶联受体 (aGPCR）拮抗剂，可做一种化学探针，对具有相似拴系激动剂的 GPR56 和 GPR114/ADGRG5 有抑制作用。
TP1497L	Mast Cell Degranulating Peptide HR-2 acetate Mast Cell Degranulating Peptide HR-2 acetate(80388-04-1 free base)	Others	Others
	Mast Cell Degranulating Peptide HR-2 acetate(80388-04-1 free base) 来自大黄蜂 Vespa orientalis 的肥大细胞脱粒肽，其生物学效应类似于来自蜂毒的肥大细胞脱粒肽。
T0235	Modaline sulfate	MAO; Monoamine Oxidase	Metabolism; Neuroscience
	Modaline sulfate 是一种 MAO 抑制剂，用于研究抑郁症。
T6411	Biapenem CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627	Antibacterial; Antibiotic	Microbiology/Virology
	Biapenem (CLI 86815) 是不经肠道的广谱碳青霉烯抗生素。
T0280	Spiperone 螺哌隆,Spiroperidol,Spiropitan	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Spiperone (Spiropitan) 是多巴胺 D2、血清素5-HT1A 和血清素5-HT2A 拮抗剂。它是广泛使用的药理学工具。它具有研究神经系统疾病的潜力。
T0255	Clomipramine hydrochloride Clomipramine HCl,Anafranil,盐酸氯米帕明	Dopamine Receptor; 5-HT Receptor; Serotonin Transporter; Norepinephrine; GST	GPCR/G Protein; Neuroscience; oxidation-reduction
	Clomipramine hydrochloride (Anafranil) 是一种5-羟色胺转运体(Ki:0.14 nM)、去甲肾上腺素转运体(Ki:54 nM)和多巴胺转运体(Ki:3 nM)阻断剂。
T0766	Promazine hydrochloride Romtiazin hydrochloride,Sinophenin hydrochloride,盐酸丙嗪	Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR	GPCR/G Protein; Neuroscience
	Promazine hydrochloride (Romtiazin hydrochloride) 是一种抗精神病药，也是一种多巴胺受体 (D2) 拮抗剂，能够抑制多巴胺能神经传递。
T0514	Phenindione Rectadione,phenylindandione,苯茚二酮,Phenylindione
	Phenindione (Rectadione) 是一种茚满二酮，已被用作抗凝剂，可作为维生素 K 拮抗剂。它的作用类似于华法林，但由于其严重不良反应的发生率较高，现在很少使用。
T12854	SBI-797812	NAMPT	Metabolism
	SBI-797812 是在结构上类似于活性位点定向的 NAMPT 抑制剂的化合物，能够阻断这些抑制剂与 NAMPT 的结合。它将 NAMPT 反应平衡转向 NMN 形成，提高 NAMPT 对 ATP 的亲和力，稳定 His247 处的磷酸化 NAMPT，增加焦磷酸盐副产物的消耗，并通过 NAD+钝化反馈抑制。
T0305	Erythrosine B Erythrosine I,Erythrosin extra bluish,Erythrosin B,赤藓红B	Others	Others
	Erythrosine B (Erythrosine I) 是一种已被用于开发动物模型的新型光敏剂，在食品和纺织工业的人造染料中具有广泛的应用。
T15422	GSK-626616	DYRK	Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors
	GSK-626616 是一种口服具有活力的 DYRK3抑制剂 (IC50:0.7 nM)。它以相似的效力抑制 DYRK 家族的其他成员，可用于研究贫血。
T17103	TM-N1324	Others; GHSR	GPCR/G Protein; Others
	TM-N1324 是一种 GPR39 激动剂。 TM-N1324 在没有和存在 Zn2+ 的情况下分别以 280 nM 和 9 nM 的高效率和效力激活人 GPR39。 TM-N1324 对鼠 GPR39 表现出相似的效力，EC50 分别为 180 nM 和 5 nM。
T21335	Fluorogestone acetate Flurogestone Acetate Flugestone Acetate Fluorogesterone Acetate SC9880,氟孕酮醋酸酯	Others	Others
	Fluorogestone acetate (Flurogestone Acetate Flugestone Acetate Fluorogesterone Acetate SC9880) 显示出高效力且活性持续时间短，并且在生理上与孕酮相似。 FGA 的效力大约是黄体酮的 20-25 倍。
T10820L1	Ciraparantag acetate Ciraparantag acetate(1438492-26-2 Free base)	Others	Others
	Ciraparantag acetate 是一种抗凝逆转剂，是一种小分子，专门设计用于通过电荷-电荷相互作用与普通肝素和低分子量肝素非共价结合。它显示出与直接口服抗凝剂 (DOAC) 相似的结合特性。
T1634	Glibenclamide 格列本脲,Glyburide	Potassium Channel; Mitochondrial Metabolism; CFTR; P-gp; Autophagy	Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience
	Glibenclamide (Glyburide) 是一种具有口服活性的 ATP 敏感的 K+通道抑制剂，可研究糖尿病和肥胖。它抑制 P-糖蛋白，可直接结合并阻断 KATP 的 SUR1亚基并抑制囊性纤维化跨膜传导调节蛋白。它通过诱导膜离子通透性干扰线粒体生物能，可诱导自噬。
T0578	Erythrosin B Iodeosin,Tetraiodofluorescein,藻红B	Others	Others
	Erythrosin B (Iodeosin) 是一种四碘荧光素，在某些食物（樱桃、鱼）中用作红色色素，用作某些细胞类型的染色剂，以及用作牙菌斑的披露物。其分子结构与甲状腺素相似。
T12941	SN 2	TRP/TRPV Channel	Membrane transporter/Ion channel
	SN 2 是TRPML3离子通道的有效激活剂，EC50为 1.8 μM。它对登革热病毒 2 和寨卡病毒具有有效的抑制作用。
T1514	Norethindrone Norethisterone,炔诺酮	Estrogen/progestogen Receptor; Progesterone Receptor	Endocrinology/Hormones; Others
	Norethindrone (Norethisterone) 是孕激素，能够用于子宫内膜异位症、由激素水平异常引起的子宫出血和继发性闭经的研究。
T50089	2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine	Others	Others
	2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine 是一种吲哚胺类化合物，在结构上与血清素相似。它是5-HT2A 受体的选择性激动剂，在神经科学领域具有潜在的应用。
T77392	Pepinemab VX 15/2503	Others	Others
	Pepinemab(VX 15/2503) 是一种靶向信号素 4D 的 IgG4 人源化单克隆抗体。Pepinemab 具有抗癌活性，可阻断 SEMA4D 的活性，用于研究阿尔茨海默病类似的退行性疾病。
T4688	Pipequaline hydrochloride PK-8165 hydrochloride,盐酸哌夸林	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Pipequaline hydrochloride (PK-8165 hydrochloride) 是一种苯二氮卓受体部分激动剂，有抗焦虑作用。
T15830	M-110	Pim	Chromatin/Epigenetic; JAK/STAT signaling
	M-110 是一种高选择性的，ATP 竞争性的 PIM 激酶抑制剂，M-110 对 PIM-3 抑制作用较好，IC50=47 nM。M-110 抑制 PIM-1 和 PIM-2 的IC50 为 2.5 μM。M-110 抑制前列腺癌细胞的增殖，IC50 为 0.6-0.9 μM。
T13177	Taquidil
	Tocainide hydrochloride 是一种sodium channel 阻滞剂，它阻断神经膜中产生疼痛的病灶中的钠通道。Tocainide hydrochloride 是利多卡因 (lignocaine) 的一种伯胺类似物，可有效抑制各种情况下的室性心律失常。
T1312	Nafcillin sodium monohydrate CL 8491,萘夫西林钠,nafcillin sodium	Antibacterial; Antibiotic	Microbiology/Virology
	Nafcillin sodium monohydrate (CL 8491) 是一种抗生素，是可逆的β-lactamase 抑制剂。它用于治疗由耐青霉素的葡萄球菌菌株引起的感染。
T19450	N-desmethyl Enzalutamide 4-[3-[4-氰基-3-(三氟甲基)苯基]-5,5-二甲基-4-氧代-2-硫代-1-咪唑烷基]-2-氟苯甲酰胺,N-desmethyl MDV 3100	Androgen Receptor	Endocrinology/Hormones
	N-desmethyl Enzalutamide (N-desmethyl MDV 3100) 是一种 Enzalutamide 的主要活性代谢物，具有与 Enzalutamide 相似的一级和二级药效功效，并在与 Enzalutamide 大致相同的血浆浓度下循环。
TP1093	TAK-448 acetate TAK-448 acetate (1234319-68-6 Free base),MVT-602 acetate	Kisspeptin	GPCR/G Protein
	TAK-448 acetate (MVT-602 acetate) 是一种小分子 KISS1R 激动剂，是一种和 kisspeptin 类似的合成肽。TAK-448 acetate 具有抗肿瘤活性，抑制 VCaP 细胞增殖，可用于研究前列腺癌。
T21013	Clomipramine Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明	5-HT Receptor	GPCR/G Protein; Neuroscience
	Clomipramine (Clomicalm) 是一种三环类抗抑郁药，能够有效阻断 5-HT 再摄取 (IC50:1.5 nM) ，可用于研究强迫症 (OCD) 及抑郁症。
T0948	Adrenalone hydrochloride Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Adrenalone hydrochloride (Adrenalone HCl) 是一种多巴胺β氧化酶 (dopamine β oxidase) 抑制剂，结构与去甲肾上腺素转运蛋白 (NET) 配体相似，IC50=36.9 μM。它是一种肾上腺素能 (adrenergic) 激动剂，用作局部血管收缩剂和止血剂。

化合物

Azlocillin sodium salt

Cat.No: T0049

Synonym: Sodium azlocillin,Azlocillin sodium,阿洛西林钠

Target: Antibacterial, Antibiotic, Parasite

Cat.No: T28973

Target: Others

Articaine hydrochloride

Cat.No: T2131

Synonym: Ultracaine,盐酸阿替卡因,阿替卡因,Articaine HCl,Hoe-045

Target: Sodium Channel

Amtolmetin guacil

Cat.No: T19672

Synonym: MED 15,MED15,ST679,呱氨托美丁,ST-679,ST 679,MED-15

Target: COX

Cat.No: T25702

Synonym: ICN 17261,L-Ribavirin,ICN-17261,ICN17261

(S)-3-Thienylglycine

Cat.No: T38311

Target: Others

Cat.No: T1333

Synonym: 甲磺氮草脲,妥拉磺脲,U-17835

Target: Potassium Channel

Oxacillin sodium salt

Cat.No: T0985

Synonym: 苯唑西林,Oxacillin sodium,Oxabel

Target: Antibacterial, Antibiotic

Cat.No: T5531

Target: Estrogen Receptor/ERR

Cat.No: T16742

Synonym: Rhodamine 110 chloride,RH110,罗丹明110

Target: Others

Cat.No: T6584

Synonym: MG149,Tip60 HAT inhibitor

Target: Apoptosis, Others, Epigenetic Reader Domain, Histone Acetyltransferase

Cat.No: T6638

Synonym: 瑞他莫林,SB-275833

Target: ribosome, Antibacterial, Antibiotic

Cat.No: T0274

Synonym: 西诺沙星,Compound 64716

Target: Topoisomerase, Antibacterial, Antibiotic

Maprotiline hydrochloride

Cat.No: T0172

Synonym: Maprotiline HCl,盐酸马普替林,Psymion,Deprilept,Ludiomil

Target: 5-HT Receptor, Adrenergic Receptor, AChR, Norepinephrine, Autophagy, Histamine Receptor

Cat.No: T1054

Synonym: 甲苯磺丁脲,HLS 831

Target: Potassium Channel, Autophagy

Cat.No: T0741

Synonym: Sulfadimerazine,磺胺二甲嘧啶,Sulfadimidine

Target: Antibacterial, Antibiotic

Cat.No: T14379

Target: Glutathione Peroxidase

Lixisenatide acetate (320367-13-3 free base)

Cat.No: TP1469

Synonym: Lixisenatide acetate

Target: Glucagon Receptor

Cat.No: T4117

Synonym: 珠氯噻醇,cis-Clopenthixol,Cisordinol,(Z)-Clopenthixol

Target: Dopamine Receptor

BIO-11006 acetate salt (901117-03-1 free base)

Cat.No: TP1457

Synonym: BIO-11006 acetate salt

Target: Others

Cat.No: T7108

Synonym: SGS-111,Noopept,GVS-111

Target: Others, iGluR

Cat.No: T13587

Target: Others

Dihydromunduletone

Cat.No: T11044

Synonym: DHM

Target: GPR

Mast Cell Degranulating Peptide HR-2 acetate

Cat.No: TP1497L

Synonym: Mast Cell Degranulating Peptide HR-2 acetate(80388-04-1 free base)

Target: Others

Modaline sulfate

Cat.No: T0235

Target: MAO, Monoamine Oxidase

Cat.No: T6411

Synonym: CLI 86815,比阿培南,Biapenern,Omegacin,L 627,LJC 10627

Target: Antibacterial, Antibiotic

Cat.No: T0280

Synonym: 螺哌隆,Spiroperidol,Spiropitan

Target: Dopamine Receptor

Clomipramine hydrochloride

Cat.No: T0255

Synonym: Clomipramine HCl,Anafranil,盐酸氯米帕明

Target: Dopamine Receptor, 5-HT Receptor, Serotonin Transporter, Norepinephrine, GST

Promazine hydrochloride

Cat.No: T0766

Synonym: Romtiazin hydrochloride,Sinophenin hydrochloride,盐酸丙嗪

Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, AChR

Cat.No: T0514

Synonym: Rectadione,phenylindandione,苯茚二酮,Phenylindione

Cat.No: T12854

Target: NAMPT

Cat.No: T0305

Synonym: Erythrosine I,Erythrosin extra bluish,Erythrosin B,赤藓红B

Target: Others

Cat.No: T15422

Target: DYRK

Cat.No: T17103

Target: Others, GHSR

Fluorogestone acetate

Cat.No: T21335

Synonym: Flurogestone Acetate Flugestone Acetate Fluorogesterone Acetate SC9880,氟孕酮醋酸酯

Target: Others

Ciraparantag acetate

Cat.No: T10820L1

Synonym: Ciraparantag acetate(1438492-26-2 Free base)

Target: Others

Cat.No: T1634

Synonym: 格列本脲,Glyburide

Target: Potassium Channel, Mitochondrial Metabolism, CFTR, P-gp, Autophagy

Cat.No: T0578

Synonym: Iodeosin,Tetraiodofluorescein,藻红B

Target: Others

Cat.No: T12941

Target: TRP/TRPV Channel

Cat.No: T1514

Synonym: Norethisterone,炔诺酮

Target: Estrogen/progestogen Receptor, Progesterone Receptor

2-(5,7-dichloro-1H-indol-3-yl)ethan-1-amine

Cat.No: T50089

Target: Others

Cat.No: T77392

Synonym: VX 15/2503

Target: Others

Pipequaline hydrochloride

Cat.No: T4688

Synonym: PK-8165 hydrochloride,盐酸哌夸林

Target: GABA Receptor

Cat.No: T15830

Target: Pim

Cat.No: T13177

Nafcillin sodium monohydrate

Cat.No: T1312

Synonym: CL 8491,萘夫西林钠,nafcillin sodium

Target: Antibacterial, Antibiotic

N-desmethyl Enzalutamide

Cat.No: T19450

Synonym: 4-[3-[4-氰基-3-(三氟甲基)苯基]-5,5-二甲基-4-氧代-2-硫代-1-咪唑烷基]-2-氟苯甲酰胺,N-desmethyl MDV 3100

Target: Androgen Receptor

TAK-448 acetate

Cat.No: TP1093

Synonym: TAK-448 acetate (1234319-68-6 Free base),MVT-602 acetate

Target: Kisspeptin

Cat.No: T21013

Synonym: Chlorimipramine,Anafranil,Clomicalm,Anafranil (free base),Clomipramina,氯米帕明

Target: 5-HT Receptor

Adrenalone hydrochloride

Cat.No: T0948

Synonym: Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮

Target: Adrenergic Receptor

Cat. No.	Product Name	Target	Signaling Pathways
T21498	Phleomycin	DNA/RNA Synthesis; Antibacterial; Antibiotic	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
	Phleomycin 是在链霉菌中发现的，引起 DNA 切割的抗癌糖肽抗生素之一。它类似于博来霉素，它结合并插入 DNA 以破坏双螺旋的完整性。
T8034	Dimethyl Trisulfide	Others; Endogenous Metabolite	Metabolism; Others
	Dimethyl trisulfide 是存在于大蒜，洋葱，西兰花和类似植物中的有机三硫化物。它是一种氰化物解毒剂。
T0974	Novobiocin Sodium Albamycinsodium,新生霉素钠,Cathomycin,Albamycin	Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy	Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
	Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
T2S1840	Rebaudioside D 莱苞迪苷D,瑞鲍迪甙D	Others	Others
	Rebaudioside D 是一种苷类化合物，存在于甜菊叶中，可用作甜味剂。
T0004	Salicylamide 水杨酰胺,Salamide,2-Hydroxybenzamide	COX	Immunology/Inflammation; Neuroscience
	Salicylamide(2-Hydroxybenzamide) 是一种止痛剂和抗热解药剂，是一种微粒体 UDP-葡糖醛酸基转移酶抑制剂。
T0480	Doxofylline Doxophylline,多索茶碱	PDE; Adenosine Receptor	GPCR/G Protein; Metabolism; Neuroscience
	Doxofylline (Doxophylline) 是腺苷 A1 受体拮抗剂，且能抑制磷酸二酯酶 IV，用于治疗哮喘。
T5514	Epibrassinolide 24-Epibrassinolide,B1105,表油菜素内酯,BP55	Apoptosis	Apoptosis
	Epibrassinolide (BP55) 是一种广泛存在的植物生长激素，具有缓解植物重金属和农药胁迫潜力。它在各种癌细胞中是一种潜在的凋亡诱导剂。
T0581	Isomaltose D-Isomaltose,6-O-α-D-Glucopyranosyl-D-glucose,低聚异麦芽糖900	Others; Endogenous Metabolite	Metabolism; Others
	Isomaltose (D-Isomaltose) 是由两个葡萄糖组成的麦芽糖类似物，能够作为蔗糖的替代物，适合于糖尿病患者及有糖尿病倾向的人群。
T2S2109	Skimmianine beta-Fagarine,Skimmianin,茵芋碱,Chloroxylonine,Skimmiamine	Others	Others
	Skimmianine (Chloroxylonine) 是一种呋喹啉类生物碱，主要存在于芸香科，具有抗炎、抗痉挛和抗血小板聚集活性。它对多种癌细胞系具有细胞毒性和基因毒性。
T4S1869	12-Epinapelline 12-表欧乌头碱,12-表-欧乌头碱	Others	Others
	12-Epinapelline 是一种二萜生物碱，分离自Aconitum baikalense 中。它具有抗炎作用，能刺激成纤维细胞前体克隆的生长。
TJS0856	Dalbergin 黄檀素,6-Hydroxy-7-Methoxy-4-Phenylcoumarin	Others	Others
	Dalbergin (6-Hydroxy-7-Methoxy-4-Phenylcoumarin) 是一种 Dalbergia Sissoo Linn. knot wood 提取物的成分。它具有强大的抗氧化活性。
T2783	Methyl dihydrojasmonate Methyl Dihydrojasmonate,Kharismal,Hedione,二氢茉莉酮酸甲酯	Others	Others
	Methyl dihydrojasmonate (Kharismal) 是一种香料成分，具有茉莉花香气，常用于许多香料混合物中。
T1219	Sisomicin Sulfate 硫酸西索米星,Pathomycin,Extramycin,硫酸西索紫苏	Antibacterial; Antibiotic	Microbiology/Virology
	Sisomicin Sulfate (Pathomycin) 是由Micromonospora inyoensis 产生的一种广谱氨基糖苷类抗生素，对革兰氏阳性细菌有很大活性。
T4592	TOMATIDINE HYDROCHLORIDE Tomatidine,Tomatidine HCl,盐酸番茄碱	Others; NF-κB; JNK; Autophagy	Autophagy; MAPK; NF-κB; Others
	Tomatidine hydrochloride (Tomatidine HCl) 是一种甾体生物碱，可防止肌肉萎缩并促进肌肉生长。它通过阻断 NF-κB 和JNK 信号发挥抗炎作用，可激活哺乳动物细胞或秀丽隐杆线虫中的自噬。
TL0009	coniferin Coniferoside,松柏苷,Abietin	Others; Antifungal	Microbiology/Virology; Others
	Coniferin (Abietin) 是一种松柏醇中的葡萄糖苷。它抑制真菌生长和黑化反应，具有 ATP 依赖性转运活性并具有抗氧化作用。
T1284	Megestrol acetate SC10363,醋酸甲地孕酮,BDH1298	Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy	Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome
	Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性，可用于治疗厌食症和恶病质。
T21532	Anisodamine 6-Hydroxyhyoscyamine,6-beta-Hydroxyhyoscyamine	AChR	Neuroscience
	Anisodamine (6-beta-Hydroxyhyoscyamine) 是毒蕈碱和烟碱胆碱受体的拮抗剂，对毒蕈碱受体的亲和力与东莨菪碱和阿托品相似。 Anisodamine 改善休克状态下的微循环，可用于有机磷中毒的研究。
T4875	Palatinose hydrate 6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物	Others; Endogenous Metabolite	Metabolism; Others
	Palatinose hydrate (6-O-α-D-Glucopyranosyl-D-fructose, Isoma) 是内源性代谢产物的一种。
T4973	Paraxanthine 1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE	Endogenous Metabolite	Metabolism
	Paraxanthine (1,7-dimethylxanthine) 是一种 caffeine 的代谢物，能够刺激Ryanodine 受体通道来抑制多巴胺能细胞的死亡。
T0266	Quinidine hydrochloride monohydrate 奎宁树,奎尼丁盐酸盐一水合物,奎尼丁盐酸盐,Quinidine hydrochloride	Potassium Channel; Sodium Channel; Parasite	Membrane transporter/Ion channel; Microbiology/Virology
	Quinidine hydrochloride monohydrate 是一种抗心律失常剂，也是 K+通道 (K+channel) 的有效阻断剂，其IC50值为 19.9 μM。它是一种有效且选择性的细胞色素 P450db (cytochrome P450db) 抑制剂，也可用作疟疾的研究。
T2S1464	Thiocolchicoside 硫秋水仙苷;噻可撒可,Thiocolchicine 2-glucoside analog,硫秋水仙苷,Coltramyl	Others; GABA Receptor	Membrane transporter/Ion channel; Neuroscience; Others
	Thiocolchicoside (Thiocolchicine 2-glucoside analog) 是秋水仙碱的半合成硫衍生物，是竞争性 GABAA 受体拮抗剂和甘氨酸受体拮抗剂。它是肌肉松弛剂，具有抗炎作用，可用于缓解疼痛的研究。
T4S1422	Praeruptorin E 白花前胡素 E,白花前胡素E	Others; Calcium Channel	Membrane transporter/Ion channel; Metabolism; Others
	Praeruptorin E 是白花前胡中的一种主要成分，是钙拮抗剂，pD2′值为 5.2。
T3874	Diosgenin glucoside 延龄草苷,地索苷,Disogluside,Trillin	Apoptosis; Others; Autophagy	Apoptosis; Autophagy; Others
	Diosgenin glucoside (Trillin) 是一种来自蒺藜的皂苷元类天然产物，可通过调节自噬和减轻细胞凋亡来保护脊髓免受损伤。它通过调节小胶质细胞 M1 极化提供神经保护，和其他具有类似活性的合成糖苷可用于治疗高胆固醇血症和动脉粥样硬化。
T6S1653	Albiflorin Alibiflorin,芍药内酯苷	Reactive Oxygen Species	Immunology/Inflammation; Metabolism; NF-κB
	Albiflorin (Alibiflorin) 是一种牡丹根中的主要成分，是一种单萜糖苷。它具有神经保护、抗炎、抗氧化和缓解疼痛作用。
T4000	(±)-Equol Equol,(±)-雌马酚,(R,S)-Equol	Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Drug Metabolite	Endocrinology/Hormones; Metabolism
	(±)-Equol ((R,S)-Equol) 是 equol 的外消旋体。它对 ERα 和 ERβ 的 EC50s of 分别为 200 和 74 nM。Equol 是大豆异黄酮黄豆苷和大豆黄素的代谢产物。
T3339	Sophoridine 5-Epidihydrosophocarpine,槐定碱,Dihydro-5-episophocarpine	Apoptosis; Topoisomerase	Apoptosis; DNA Damage/DNA Repair
	Sophoridine (Dihydro-5-episophocarpine) 是一种从豆科植物槐豆斜生植物的叶子中分离出来的喹喔啉生物碱。它是胰腺癌的候选药物，诱导细胞凋亡。
T4716	Pyrrole-2-carboxylic acid 吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline	Endogenous Metabolite	Metabolism
	Pyrrole-2-carboxylic acid (Minaline) 是一种天然生物碱类，从海洋细菌Pelomonas puraquaesp. Nov 中分离得到。
TN2034	Paeoniflorigenone	Others; Caspase	Apoptosis; Others; Proteases/Proteasome
	Paeoniflorigenone is a depolarizing neuromuscular blocking agent, being similar to succinylcholine.
T13653	Dihydrocephalomannine	Others	Others
	Dihydrocephalomannine is similar to paclitaxel, showing reduced cytotoxicity and tubulin binding.
TN6542	Humic acid sodium salt
	Sodium salt of humic acid and sodium silicate have similar enhancement on kerosene contaminated soil washing with saponin.
T25204	Carbomycin B Magnamycin B
	Carbomycin B is an intermediate in the synthesis of Carbomycin. Carbomycin is a macrolite antibiotic complex produced by Stroptomyces halstedii, that is similar to Leucomycin and Erythromycin.
T22357	Lobeline sulfate 硫酸山梗菜碱,Lobelin sulphate	Others	Others
	Lobelin sulphate is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has a variety of therapeutic uses including in insomnia, and smoking cessation, peripheral vascular disorders, respiratory disor
T39148	FR179642 FR179642
	FR179642 is an essential intermediate compound utilized in the synthesis of Micafungin, an antifungal drug belonging to the echinocandin class. It serves as the cyclic peptide foundation for the structurally similar antifungal lipopeptide FR901379.
TN1366	Alcesefoliside	Others	Others
	Alcesefoliside has statistically significant cytoprotective activity similar to that of silymarin, tested at 60 ug/mL.
T1235L	Lincomycin U 10149,U10149,U-10149
	Lincomycin is a lincosamide antibiotic that comes from the actinomycete Streptomyces lincolnensis. Although similar in structure, antibacterial spectrum, and mechanism of action to macrolides, lincomycin is also effective against other organisms including
TN4299	Isoiridogermanal	Others	Others
	Isoiridogermanal shows similar cytotoxicity with IG(50) around 11 microM and 23 microM against MCF-7 and C32 cell lines, respectively.
T6601	Nanchangmycin Nanchangmycin A,南昌霉素	Antibacterial; Antibiotic	Microbiology/Virology
	Nanchangmycin (Nanchangmycin A) 由 Streptomyces nanchangensis 产生的一种聚醚抗生素，抑制革兰氏阳性菌。它也是一种广谱抗病毒药物，有抗 Zika 病毒作用。
TN2792	2-Oxopomolic acid
	2-Oxopomolic acid shows cytotoxic activity, it shows a significant decrease in intracellular melanin content in B16-F10 cells, and in culture media melanin. 2-Oxopomolic acid shows radical-scavenging activities similar to that of the reference antioxidant
T19268	D-Sedoheptulose 7-phosphate	Others	Others
	D-Sedoheptulose 7-phosphate is a common precursor of heptaic acid (group III) and hygromycin B (group IV) heptasaccharide. D-heptadecane 7-phosphate can be converted to NDP-heptose by similar biosynthetic pathways in these compounds.
T81814	Methyl Ganoderic acid B
	Methyl Ganoderic acid B, 一种从灵芝中分离得到的三萜类化合物，具有类似神经生长因子的神经元存活促进作用。
T38331	Commendamide
	Commendamide is a natural bacterial product that was discovered in a screen for commensal bacteria effector genes (Cbegs). Cbeg12 is a bacterial effector gene that encodes for its production. Commendamide is structurally similar to long-chain N-acyl-amides, which commonly signal, in mammals, through G protein-coupled receptors. Commendamide activates GPR132 (also known as G2A) with an EC50 value of 11.8 μM.
T73073	PTP1B-IN-21
	PTP1B-IN-21 是蛋白酪氨酸磷酸酶 1B (PTP1B) 的选择性抑制剂 (IC50=1.56 μM)，抑制力超出高度同源 T 细胞蛋白酪氨酸磷酸酶 (TCPTP；IC50>100 μM)，PTP1B 是抑制 2 型糖尿病的重要靶点。
T37911	cis-Resveratrol 顺式白藜芦醇,(Z)-Resveratrol
	Resveratrol is a potent phenolic antioxidant found in grapes, red wine, and various berries that also has antiproliferative and anti-inflammatory activity. cis-Resveratrol is the double bond isomer of trans-resveratrol, the more often studied and naturally abundant of the two resveratrol isomers. cis-Resveratrol exhibits antioxidant activity in the &#181M range similar to that observed with trans-resveratrol. It blocks production of reactive oxygen species (ROS) by inhibition of NAD(P)H oxidase ...
TN4053	FD-838	Antifection	Microbiology/Virology
	FD-838 shows good antileishmanial and moderate anticancer activities, it can moderately inhibit the growth of cultured P388 and HL-60 cell lines. FD-838 has anti-fungal activity, it can significantly inhibit the growth of two plant fungal pathogens Botryt
T39562	γ-Amanitin
	γ-Amanitin an ADC cytotoxin and isolated from the mushroom. γ-Amanitin inhibits RNA polymerase II and disrupts synthesis of mRNA. γ-Amanitin shows similar effects to α-Amanitin and β-Amanitin.
TN1875	Liriodenine 鹅掌揪碱	BCL; Caspase; p53	Apoptosis; Proteases/Proteasome
	Liriodenine is a potent inhibitor of topoisomerase II (EC 5.99.1.3) both in vivo and in vitro, it has antitumor, antibacterial and antifungal activities, it can suppress ventricular arrhythmias induced by myocardial ischaemia reperfusion, through inhibiti
T37219	N-Palmitoyl Glycine
	The acyl amides are a family of endogenous lipids that act as potent modulators of pain and inflammation. The best characterized members of this family are the arachidonoyl amides, which includes N-arachidonoyl ethanolamide (AEA; anandamide). N-palmitoyl glycine (PalGly) contains an 18-carbon saturated fatty acid that is amide-linked to glycine and is structurally similar to the phospholipid-derived N-acyl ethanolamines. Endogenously produced in rat skin and spinal cord, PalGly is present in 100...
TN5164	trans-Hinokiresinol	IL Receptor; TNF; NOS; LTR	Apoptosis; Immunology/Inflammation
	Hinokiresinol is a novel inhibitor of LTB4 binding to the human neutrophils, it has antiallergic effect, it inhibits IgE-induced mouse passive cutaneous anaphylaxis reaction. Hinokiresinol (trans-hinokiresinol) and nyasol (cis-hinokiresinol) are estrogen

天然产物

Cat.No: T21498

Target: DNA/RNA Synthesis, Antibacterial, Antibiotic

Dimethyl Trisulfide

Cat.No: T8034

Target: Others, Endogenous Metabolite

Novobiocin Sodium

Cat.No: T0974

Synonym: Albamycinsodium,新生霉素钠,Cathomycin,Albamycin

Target: Potassium Channel, DNA gyrase, Topoisomerase, Antibacterial, Antibiotic, ABC, Autophagy

Cat.No: T2S1840

Synonym: 莱苞迪苷D,瑞鲍迪甙D

Target: Others

Cat.No: T0004

Synonym: 水杨酰胺,Salamide,2-Hydroxybenzamide

Target: COX

Cat.No: T0480

Synonym: Doxophylline,多索茶碱

Target: PDE, Adenosine Receptor

Epibrassinolide

Cat.No: T5514

Synonym: 24-Epibrassinolide,B1105,表油菜素内酯,BP55

Target: Apoptosis

Cat.No: T0581

Synonym: D-Isomaltose,6-O-α-D-Glucopyranosyl-D-glucose,低聚异麦芽糖900

Target: Others, Endogenous Metabolite

Cat.No: T2S2109

Synonym: beta-Fagarine,Skimmianin,茵芋碱,Chloroxylonine,Skimmiamine

Target: Others

12-Epinapelline

Cat.No: T4S1869

Synonym: 12-表欧乌头碱,12-表-欧乌头碱

Target: Others

Cat.No: TJS0856

Synonym: 黄檀素,6-Hydroxy-7-Methoxy-4-Phenylcoumarin

Target: Others

Methyl dihydrojasmonate

Cat.No: T2783

Synonym: Methyl Dihydrojasmonate,Kharismal,Hedione,二氢茉莉酮酸甲酯

Target: Others

Sisomicin Sulfate

Cat.No: T1219

Synonym: 硫酸西索米星,Pathomycin,Extramycin,硫酸西索紫苏

Target: Antibacterial, Antibiotic

TOMATIDINE HYDROCHLORIDE

Cat.No: T4592

Synonym: Tomatidine,Tomatidine HCl,盐酸番茄碱

Target: Others, NF-κB, JNK, Autophagy

Cat.No: TL0009

Synonym: Coniferoside,松柏苷,Abietin

Target: Others, Antifungal

Megestrol acetate

Cat.No: T1284

Synonym: SC10363,醋酸甲地孕酮,BDH1298

Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, HIV Protease, Autophagy

Cat.No: T21532

Synonym: 6-Hydroxyhyoscyamine,6-beta-Hydroxyhyoscyamine

Target: AChR

Palatinose hydrate

Cat.No: T4875

Synonym: 6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物

Target: Others, Endogenous Metabolite

Cat.No: T4973

Synonym: 1,7-二甲基黄嘌呤,1,7-DIMETHYLXANTHINE

Target: Endogenous Metabolite

Quinidine hydrochloride monohydrate

Cat.No: T0266

Synonym: 奎宁树,奎尼丁盐酸盐一水合物,奎尼丁盐酸盐,Quinidine hydrochloride

Target: Potassium Channel, Sodium Channel, Parasite

Thiocolchicoside

Cat.No: T2S1464

Synonym: 硫秋水仙苷;噻可撒可,Thiocolchicine 2-glucoside analog,硫秋水仙苷,Coltramyl

Target: Others, GABA Receptor

Cat.No: T4S1422

Synonym: 白花前胡素 E,白花前胡素E

Target: Others, Calcium Channel

Diosgenin glucoside

Cat.No: T3874

Synonym: 延龄草苷,地索苷,Disogluside,Trillin

Target: Apoptosis, Others, Autophagy

Cat.No: T6S1653

Synonym: Alibiflorin,芍药内酯苷

Target: Reactive Oxygen Species

Cat.No: T4000

Synonym: Equol,(±)-雌马酚,(R,S)-Equol

Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Drug Metabolite

Cat.No: T3339

Synonym: 5-Epidihydrosophocarpine,槐定碱,Dihydro-5-episophocarpine

Target: Apoptosis, Topoisomerase

Pyrrole-2-carboxylic acid

Cat.No: T4716

Synonym: 吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline

Target: Endogenous Metabolite

Paeoniflorigenone

Cat.No: TN2034

Target: Others, Caspase

Dihydrocephalomannine

Cat.No: T13653

Target: Others

Humic acid sodium salt

Cat.No: TN6542

Cat.No: T25204

Synonym: Magnamycin B

Lobeline sulfate

Cat.No: T22357

Synonym: 硫酸山梗菜碱,Lobelin sulphate

Target: Others

Cat.No: T39148

Synonym: FR179642

Cat.No: TN1366

Target: Others

Cat.No: T1235L

Synonym: U 10149,U10149,U-10149

Isoiridogermanal

Cat.No: TN4299

Target: Others

Cat.No: T6601

Synonym: Nanchangmycin A,南昌霉素

Target: Antibacterial, Antibiotic

2-Oxopomolic acid

Cat.No: TN2792

D-Sedoheptulose 7-phosphate

Cat.No: T19268

Target: Others

Methyl Ganoderic acid B

Cat.No: T81814

Cat.No: T38331

Cat.No: T73073

cis-Resveratrol

Cat.No: T37911

Synonym: 顺式白藜芦醇,(Z)-Resveratrol

Cat.No: TN4053

Target: Antifection

Cat.No: T39562

Cat.No: TN1875

Synonym: 鹅掌揪碱

Target: BCL, Caspase, p53

N-Palmitoyl Glycine

Cat.No: T37219

trans-Hinokiresinol

Cat.No: TN5164

Target: IL Receptor, TNF, NOS, LTR

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