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61

抑制剂 & 化合物

61

天然产物

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Cat. No. Product Name Target Signaling Pathways
T7969 Dipyrithione

Others Others
Dipyrithione 似乎具有新的细胞毒性和强大的广谱抗肿瘤活性。
T11888 LtaS-IN-1

Others; Antibacterial Microbiology/Virology; Others
LtaS-IN-1 是多药耐药粪肠球菌中脂磷壁酸合成的有效抑制剂,可改变细胞壁形态。 LtaS-IN-1 对抗肠球菌属 28 菌株,MIC 值从 0.5 μg/mL 到 64 μg/mL 不等。 LtaS-IN-1 抑制菌株 E1630 和 E1590,MIC 值为 0.5 μg/mL。
T35427 β-Lactamase-IN-2

Antibacterial Microbiology/Virology
β-Lactamase-IN-2 是 β-内酰胺酶的有效抑制剂。β-Lactamase-IN-2显示出抗菌活性。
T38240 2,6-Dichlorodiphenylamine

Antibacterial Microbiology/Virology
2,6-Dichlorodiphenylamine 是双氯芬酸钠的一种结构类似物,显示出抗白色念珠菌活性。2,6-Dichlorodiphenylamine 是非选择性抗炎剂,为COX 的抑制剂,在 CHO 细胞中,对人 COX-1 和 COX-2 的IC50分别为 4 和 1.3 nM。
T0767 Sulfapyridine

磺胺吡啶,Sulfidine,Sulfidin,2-Sulfapyridine

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Sulfapyridine (2-Sulfapyridine) 是一种磺酰胺类抗生素,是 Sulfasalazine 的代谢产物。它抑制重组 P. carinii 二氢蝶呤合成酶,IC50为 0.18 μM。它具有抗菌,抗炎和抗风湿作用。
T38359 Dup-721

Antibacterial Microbiology/Virology
DuP-721 是广谱的口服有效的抗菌剂,可以抑制多种临床敏感和耐药细菌,特别是结核杆菌M. tuberculosis。
T8694 ML406

Antibacterial; Antibiotic Microbiology/Virology
ML406 是一种小分子探针,通过抑制M.tuberculosisBioA(DAPA 合酶) 显示出抗结核活性,IC50为 30 nM。
T6439 Cetylpyridinium Chloride

西吡氯铵,Cetamium,Pristacin,Hexadecylpyridinium Chloride

Others; HBV; Antibacterial Microbiology/Virology; Others
Cetylpyridinium Chloride (Hexadecylpyridinium Chloride) 是阳离子季铵,是一种广谱抗菌剂。它有效抑制 HBV 衣壳装配,IC50为 2.5 μM。它被用于杀虫剂和各种漱口水以及其他个人护理产品中。
T1647 Ronidazole

洛硝哒唑,Ronidazol,罗硝唑,Ridzol

Antibacterial; Antibiotic; Parasite Microbiology/Virology
Ronidazole (Ronidazol) 是一种口服有效的抗原虫和抗菌试剂。它在猫模型中对胎儿三毛滴虫有效,还可研究组织口癣和猪痢疾。
T0456 Cinchophen

2-苯基-4-喹啉羧酸,辛可芬,Cinconal

COX Immunology/Inflammation; Neuroscience
Cinchophen (Cinconal) 是口服具有活性的非甾体抗炎试剂,具有抗菌活性。它可用于研究关节炎和某些肝脏疾病。
T8390 Cefazolin

头孢唑林,头孢唑啉

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazolin 是一种头孢类抗生素, 用于多种细菌感染的研究。
T1454 Acyclovir

Aciclovir,Acycloguanosine,阿昔洛韦

Apoptosis; DNA/RNA Synthesis; Antibacterial; Antibiotic; HSV Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Acyclovir (Aciclovir) 是鸟嘌呤类似物和具有口服活性的抗病毒剂。它对HSV-1(IC50为 0.85 μM),HSV-2(IC50为 0.86 μM) 和水痘带状疱疹病毒有活性。
T2692 A40926

Dalbavancin Impurity,达巴霉素杂质

Antibacterial Microbiology/Virology
A40926 (Dalbavancin Impurity) 是Dalbavancin 的前体,是一种糖肽抗生素。它抑制革兰氏阳性细菌,对淋病奈瑟氏球菌非常有效。
T0314 Hexylresorcinol

己雷锁辛,4-己基间苯二酚,4-Hexylresorcinol

Apoptosis; Tyrosinase; Antibacterial; Parasite Apoptosis; Microbiology/Virology; Proteases/Proteasome
Hexylresorcinol (4-Hexylresorcinol) 是在植物中发现的一种天然产物,具有抗菌、驱虫、防腐和抗肿瘤活性。它是一种可逆、非竞争性的 α-葡萄糖苷酶抑制剂,有抗 DNA 氧化损伤的保护作用。它可诱导鳞癌细胞凋亡。
T1640 Ciprofloxacin

Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ciprofloxacin (Bay-09867) 是一种有高抗菌活性的氟喹诺酮类抗生素。
T0250 Ciprofloxacin monohydrochloride

Bay-09867 (hydrochloride),Ciprofloxacin HCl,盐酸环丙沙星,环丙沙星盐酸盐,Ciprofloxacin hydrochloride

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Ciprofloxacin monohydrochloride (Bay-09867 hydrochloride) 是一种高抗菌活性的氟喹诺酮类抗生素。
T0341 Dimethyl sulfoxide

Methyl Sulfoxide,DMSO,二甲基亚砜

Others; Antibacterial Microbiology/Virology; Others
Dimethyl sulfoxide (DMSO) 是一种常用的溶剂,可溶解极性和非极性化合物。Dimethyl sulfoxide 已被广泛用于生物实验中化合物的母液配制。Dimethyl sulfoxide 具有抑菌活性。
T0953 Cefazolin sodium

Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin

Others; Antibacterial; Antibiotic Microbiology/Virology; Others
Cefazolin sodium (cephazolin sodium) salt 是一种头孢类抗生素, 可研究多种细菌感染。
T1140 Doxycycline hydrochloride

Doxylin,盐酸多西环素,Vibramycin,Hyclate

MMP; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hydrochloride (Hyclate) 是一种四环素抗生素,是口服有效的广谱金属蛋白酶抑制剂,具有抗菌活性。
T16465 Penicillin G benzathine

Benzathine benzylpenicillin,Benzathine penicilline G

Antibacterial Microbiology/Virology
Penicillin G benzathine 具有抗细菌感染活性,可用于研究早期梅毒。
T50057 N-(4-bromo-2-chlorophenyl)-5-chloro-2-hydroxybenzamide

Others Others
N-(4-bromo-2-chlorophenyl)-5-chloro-2-hydroxybenzamide 是一种苯甲酰胺类化合物,具有抗肿瘤、抗炎、抗细菌和抗真菌的活性。
T1427 2-(Phosphonooxy)benzoic acid

磷柳酸,Fosfosal,2-phosphonoxy benzoic acid,Salicyl phosphate,Disdolen

COX Immunology/Inflammation; Neuroscience
2-(Phosphonooxy)benzoic acid (Fosfosal) 是一种非乙酰化的水杨酸衍生物,对炎性疾病以及止痛具有潜在的研究价值。
TP1745L Ceratotoxin A acetate

Ceratotoxin A acetate(150671-04-8 Free base)

Antibacterial Microbiology/Virology
Ceratotoxin A acetate 是从副腺分泌液中分离出来的,具有抗菌作用。
T2353 BRD7116

BRD7716

DNA gyrase; Antibacterial DNA Damage/DNA Repair; Microbiology/Virology
BRD7116 与细菌 DNA 促旋酶竞争性结合, 作用于LSCe 细胞,EC50值为200 nM。它具有细胞非自主抗白血病活性。
T8138 Phenazine methylsulfate

5-甲基吩嗪硫酸甲酯,Phenazine methosulfate

Apoptosis; Antibacterial; Antibiotic Apoptosis; Microbiology/Virology
Phenazine methylsulfate 是一种自由基产生剂。 它已被用作细胞活力测定中的电子转移反应物。 它在还原剂 NADPH 存在下诱导 ssDNA 断裂形成。它在碱性彗星试验和细胞凋亡中诱导氧化性 DNA 损伤。
T50075 3,5-dimethyl-4-phenyl-1,2-oxazole

Others Others
3,5-dimethyl-4-phenyl-1,2-oxazole 是一种用作分子结构单元的杂环化合物,具有抗炎、抗肿瘤、抗细菌和抗真菌活性,以及调节免疫系统的能力。
T4202 Delamanid

迪拉马尼,德拉马尼,OPC-67683

Anti-infection; Antibacterial; Antibiotic Microbiology/Virology
Delamanid (OPC-67683) 是一种新的分枝杆菌细胞壁合成抑制剂,可用于耐多药结核病。
T25214 CCR-11

CCR11,CCR 11

Antibiotic Microbiology/Virology
CCR-11 是一种具有抗菌活性的绕丹宁衍生物。 CCR-11 可以抑制 B. subtilis细胞和 HeLa 细胞增殖。 CCR-11 通过抑制 FtsZ 的组装和 GTPase 活性来抑制细菌增殖和细菌胞质分裂。 CCR-11 具有潜在的抗肿瘤活性,可用于研究乳腺癌和小儿骨髓增生异常。
T13041 Surfactin

HSV Microbiology/Virology
Surfactin 是一种有效的环状脂肽生物表面活性剂,可介导单价和二价阳离子(如钙)穿过脂质双层膜的通量,具有抗菌、抗真菌、抗支原体和溶血作用。
T64750 Deoxyribonuclease I

DNase I

Others Others
Deoxyribonuclease I (DNase I) 是提纯蛋白质常用的一种酶,具有潜在的抗炎和抗癌活性,可用于研究细菌感染和真菌感染。
T77608 1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl-

Antifungal Microbiology/Virology
1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl- 可作为一种广谱抗菌剂,对黑曲霉枯草芽孢杆菌、白假丝酵母、大肠杆菌和金黄色葡萄球菌有抑制作用。1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl- 在体外实验中显示出抗炎活性,可用于治疗细菌感染。
T20159 Bilanafos

Herby,Bialaphos,Antibiotic SF 1293

Bilanafos is an agent of Anti-Bacterial.
T24761 Satranidazole

GO 10213,C 10213 Go

Satranidazole is an anti-bacterial. It is used to treat periodontitis.
T10750 Cecropin A TFA (80451-04-3 free base)

Cecropin A TFA

Others Others
Cecropin A TFA is an antimicrobial polypeptide isolated from Hyalaphora cecropia pupae with anti-inflammatory, anti-bacterial, and anti-cancer activity.
T63632 Anti-MRSA agent 3

Anti-MRSA agent 3 能够明显的抑制耐甲氧西林金黄色葡萄球菌 (MRSA) 的活性 (MIC: 0.098 μg/ml),并且对正常细胞毒性较低。Anti-MRSA agent 3 对细菌基因组 DNA 具有较高的结合亲和力,对细菌细胞壁和细胞膜具有较强的破坏能力。
T62383 Anti-MRSA agent 2

Anti-MRSA agent 2 (compound 14) 能够较好的抑制耐甲氧西林金黄色葡萄球菌 (MRSA) (MIC: 0.098 μg/ml),对正常细胞的毒性相对较低。Anti-MRSA agent 2 能够较强的破坏细菌膜,并具有较好的与细菌基因组DNA 结合的能力。
T61484 LasR-IN-1

LasR-IN-1 (compound 9g) is a highly effective inhibitor of LasR, exhibiting strong potency against E. coli. It also demonstrates significant anti-bacterial properties, displaying a minimum inhibitory concentration (MIC) of 28.13 μM against P. aeruginosa [1].
T82788 Calpurbatug

Calpurbatug是一种免疫球蛋白G1抗体,具有针对DNABII家族抗菌DNA结合蛋白和TRL1068γ1链的人单克隆抗体活性。
T74776 Antibacterial agent 139

Antibacterial agent 139 对革兰氏阳性菌具有抗菌活性。Antibacterial agent 139 具有抗 MRSA、抗 VISA 和抗 LRSE 活性。Antibacterial agent 139 去极化细菌细胞膜。
T74657 Balhimycin

Balhimycin为一种源自Amycolatopsis sp.发酵产物的糖肽类抗生素,其展现出针对葡萄球菌和厌氧菌的显著抗菌效果。
T76321 Brain Derived Basic Fibroblast Growth Factor (1-24)

Brain Derived BasicFibroblast Growth Factor(1-24) (FGF basic 1-24) 是一种合成肽,表现出抗细菌和抗HBV 的活性。Brain Derived BasicFibroblast Growth Factor(1-24) 可用于感染性疾病和免疫性疾病的研究。
T62577 Anti-MRSA agent 5

Anti-MRSA agent 是一种 MRSA 的有效拮抗剂 (MIC50: 0.38 μg/mL),hERG 活性较低 (IC50: 40 μM)。Anti-MRSA agent 对哺乳动物细胞的毒性也很低,几乎不可能获得细菌的耐药性。
T61937 DNA Gyrase-IN-3

DNA Gyrase-IN-3 (Compound 28) 是细菌DNA 旋转酶 B (bacterial DNA gyrase B) 抑制剂。DNA Gyrase-IN-3抑制大肠杆菌DNA 旋转酶的 IC50为5.41-15.64 μM。DNA Gyrase-IN-3显示出抗结核和抗菌活性。
T79778 Anti-MRSA agent 8

Anti-MRSA agent 8(Compound 7g)为DAPG衍生物,展现出显著的抗菌活性,主要通过作用于细菌细胞膜以发挥效能。此化合物可应用于耐甲氧西林Staphylococcus aureus(MRSA)的研究领域。
T75300 Cefazolin sodium pentahydrate

Cefazolin sodium pentahydrate 是一代头孢菌素类抗生素,可用于多种细菌感染的研究。Cefazolin sodium pentahydrate 具有抗炎作用,可以减轻术后认知功能障碍 (POCD)。
T0366L Cefadroxil (hydrate)

Cefadroxil is a first generation aminocephalosporin with good patient compliance, a long-acting therapeutic effect, high solubility and relatively broad spectrum of anti-bacterial activity. Cefadroxil is also a substrate of the intestinal peptide transporter PepT1, which is primarily responsible for the drug's uptake across the apical membrane of small intestine.
T75014 Antiproliferative agent-18

Antiproliferative agent-18 (Compound 5k) 为具抗增殖、中度抗细菌 (anti-bacterial) 及抗真菌 (anti-fungi) 活性的化合物。
T63588 Antibacterial agent 89

Antibacterial agent 89 是强效的抗菌剂,能够干扰细菌转录的过程,表现出抗梭菌效果。Antibacterial agent 89 能够抑制细胞毒素的释放和 β'CH-σ 相互作用。
T80390 HG4

HG4为快速作用的抗菌多肽,具有抗生物膜和抗炎活性。特别是针对MRSA菌株(MIC: 32-64 μg/mL),它对革兰氏阳性病原体表现出显著活性。此外,HG4能够与细菌脂质结合,并能减少S. aureus MRSA USA300细菌的ATP浓度。
T63370 FtsZ-IN-2

FtsZ-IN-2 是细菌细胞分裂蛋白 FtsZ 抑制剂,对 GTPase 的活性具有抑制作用。FtsZ-IN-2 表现出抗葡萄球菌作用,对 MSSA 和 MRSA 的MIC 值均为 2 μg/ml。

化合物

Dipyrithione
Cat.No: T7969
Synonym:
Target: Others
LtaS-IN-1
Cat.No: T11888
Synonym:
Target: Others, Antibacterial
β-Lactamase-IN-2
Cat.No: T35427
Synonym:
Target: Antibacterial
2,6-Dichlorodiphenylamine
Cat.No: T38240
Synonym:
Target: Antibacterial
Sulfapyridine
Cat.No: T0767
Synonym: 磺胺吡啶,Sulfidine,Sulfidin,2-Sulfapyridine
Target: Antibacterial, Antibiotic, Autophagy
Dup-721
Cat.No: T38359
Synonym:
Target: Antibacterial
ML406
Cat.No: T8694
Synonym:
Target: Antibacterial, Antibiotic
Cetylpyridinium Chloride
Cat.No: T6439
Synonym: 西吡氯铵,Cetamium,Pristacin,Hexadecylpyridinium Chloride
Target: Others, HBV, Antibacterial
Ronidazole
Cat.No: T1647
Synonym: 洛硝哒唑,Ronidazol,罗硝唑,Ridzol
Target: Antibacterial, Antibiotic, Parasite
Cinchophen
Cat.No: T0456
Synonym: 2-苯基-4-喹啉羧酸,辛可芬,Cinconal
Target: COX
Cefazolin
Cat.No: T8390
Synonym: 头孢唑林,头孢唑啉
Target: Others, Antibacterial, Antibiotic
Acyclovir
Cat.No: T1454
Synonym: Aciclovir,Acycloguanosine,阿昔洛韦
Target: Apoptosis, DNA/RNA Synthesis, Antibacterial, Antibiotic, HSV
A40926
Cat.No: T2692
Synonym: Dalbavancin Impurity,达巴霉素杂质
Target: Antibacterial
Hexylresorcinol
Cat.No: T0314
Synonym: 己雷锁辛,4-己基间苯二酚,4-Hexylresorcinol
Target: Apoptosis, Tyrosinase, Antibacterial, Parasite
Ciprofloxacin
Cat.No: T1640
Synonym: Ciproxan,环丙沙星,Ciprobay,Bay o 9867,Bay-09867
Target: Topoisomerase, Antibacterial, Antibiotic
Ciprofloxacin monohydrochloride
Cat.No: T0250
Synonym: Bay-09867 (hydrochloride),Ciprofloxacin HCl,盐酸环丙沙星,环丙沙星盐酸盐,Ciprofloxacin hydrochloride
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Dimethyl sulfoxide
Cat.No: T0341
Synonym: Methyl Sulfoxide,DMSO,二甲基亚砜
Target: Others, Antibacterial
Cefazolin sodium
Cat.No: T0953
Synonym: Ancef,头孢唑啉钠,头孢唑林钠,Cefazolin sodium salt,Sodium cephazolin,cephazolin sodium,cefazoline sodium,Sodium cefazolin
Target: Others, Antibacterial, Antibiotic
Doxycycline hydrochloride
Cat.No: T1140
Synonym: Doxylin,盐酸多西环素,Vibramycin,Hyclate
Target: MMP, Antibacterial, Antibiotic
Penicillin G benzathine
Cat.No: T16465
Synonym: Benzathine benzylpenicillin,Benzathine penicilline G
Target: Antibacterial
N-(4-bromo-2-chlorophenyl)-5-chloro-2-hydroxybenzamide
Cat.No: T50057
Synonym:
Target: Others
2-(Phosphonooxy)benzoic acid
Cat.No: T1427
Synonym: 磷柳酸,Fosfosal,2-phosphonoxy benzoic acid,Salicyl phosphate,Disdolen
Target: COX
Ceratotoxin A acetate
Cat.No: TP1745L
Synonym: Ceratotoxin A acetate(150671-04-8 Free base)
Target: Antibacterial
BRD7116
Cat.No: T2353
Synonym: BRD7716
Target: DNA gyrase, Antibacterial
Phenazine methylsulfate
Cat.No: T8138
Synonym: 5-甲基吩嗪硫酸甲酯,Phenazine methosulfate
Target: Apoptosis, Antibacterial, Antibiotic
3,5-dimethyl-4-phenyl-1,2-oxazole
Cat.No: T50075
Synonym:
Target: Others
Delamanid
Cat.No: T4202
Synonym: 迪拉马尼,德拉马尼,OPC-67683
Target: Anti-infection, Antibacterial, Antibiotic
CCR-11
Cat.No: T25214
Synonym: CCR11,CCR 11
Target: Antibiotic
Surfactin
Cat.No: T13041
Synonym:
Target: HSV
Deoxyribonuclease I
Cat.No: T64750
Synonym: DNase I
Target: Others
1H-Indole, 3,3'-(2-thienylmethylene)bis[2-methyl-
Cat.No: T77608
Synonym:
Target: Antifungal
Bilanafos
Cat.No: T20159
Synonym: Herby,Bialaphos,Antibiotic SF 1293
Target:
Satranidazole
Cat.No: T24761
Synonym: GO 10213,C 10213 Go
Target:
Cecropin A TFA (80451-04-3 free base)
Cat.No: T10750
Synonym: Cecropin A TFA
Target: Others
Anti-MRSA agent 3
Cat.No: T63632
Synonym:
Target:
Anti-MRSA agent 2
Cat.No: T62383
Synonym:
Target:
LasR-IN-1
Cat.No: T61484
Synonym:
Target:
Calpurbatug
Cat.No: T82788
Synonym:
Target:
Antibacterial agent 139
Cat.No: T74776
Synonym:
Target:
Balhimycin
Cat.No: T74657
Synonym:
Target:
Brain Derived Basic Fibroblast Growth Factor (1-24)
Cat.No: T76321
Synonym:
Target:
Anti-MRSA agent 5
Cat.No: T62577
Synonym:
Target:
DNA Gyrase-IN-3
Cat.No: T61937
Synonym:
Target:
Anti-MRSA agent 8
Cat.No: T79778
Synonym:
Target:
Cefazolin sodium pentahydrate
Cat.No: T75300
Synonym:
Target:
Cefadroxil (hydrate)
Cat.No: T0366L
Synonym:
Target:
Antiproliferative agent-18
Cat.No: T75014
Synonym:
Target:
Antibacterial agent 89
Cat.No: T63588
Synonym:
Target:
HG4
Cat.No: T80390
Synonym:
Target:
FtsZ-IN-2
Cat.No: T63370
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T2982 Xanthone

Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide

Apoptosis; Others; Influenza Virus; Antibacterial; Antifungal Apoptosis; Microbiology/Virology; Others
Xanthone (Xanthenone) 是一种从山竹果中分离得到的天然产物,具有抗炎,抗氧化,抗肿瘤,抗过敏,抗细菌,抗真菌和抗病毒活性。在癌变的不同阶段可控制细胞分裂和生长,凋亡,炎症和转移。
T8249 Hexahydrofarnesyl acetone

植酮,Phytone

Others; Antibacterial Microbiology/Virology; Others
Hexahydrofarnesyl acetone (Phytone) 是从Launaea mucronata 中分离得到的倍半萜,具有抗菌和抗炎活性,可研究缓解疼痛。
TN2085 Piperlonguminine

Anti-infection; Antibacterial; Antifungal Microbiology/Virology
Piperlonguminine 是一种从 Piper 中分离出的生物碱酰胺。它具有多种生物活性,如神经保护、抗炎、抗肿瘤、抗血小板、抗黑素生成、抗真菌和抗菌活性。
TN3690 Comanthoside B

Comanthosid B

Antibacterial Microbiology/Virology
Comanthoside B (Comanthosid B) 是一种黄酮类苷,分离自芦花属植物,具有抗菌、抗炎活性。
TN1686 Ginsenoside Rg4

人参皂苷 RG4

Antibacterial Microbiology/Virology
Ginsenoside Rg4 是分离自Panax ginsengC. A. Meyer 叶子中的一种人参三醇型人参皂苷。人参三醇型人参皂苷具有多种生物活性,包括防腐,抗糖尿病,伤口愈合,免疫刺激和抗氧化活性等。
TN1772 Isoastilbin

Anti-infection; Tyrosinase; Antibacterial Microbiology/Virology; Proteases/Proteasome
Isoastilbin 是Rhizoma Smilacis glabrae 和Astragalus membranaceus 中的二氢黄酮醇糖苷。它抑制酪氨酸酶活性,还抑制葡萄糖基转移酶,IC50值为 54.3 μg/mL。它具有神经保护、抗氧化、抗微生物和抗凋亡活性,可研究阿尔茨海默氏病。
TN1990 Norathyriol

芒果苷元

Akt; DNA/RNA Synthesis; AMPK; PPAR Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Metabolism; PI3K/Akt/mTOR signaling
Norathyriol 是来自芒果的芒果苷代谢物,具有抗氧化、抗癌、抗菌和抗炎活性。它以非竞争性方式抑制 α-葡萄糖苷酶,IC50为 3.12 μM。它还抑制PPARα、PPARβ和PPARγ,IC50分别为 92.8、102.4 和 153.5 µM。
T3843 Pinosylvin

银松素,3,5-stilbenediol,5-Styrylresorcinol

Apoptosis; Others; Antibacterial; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Others
Pinosylvin (5-Styrylresorcinol) 是从Pinus spp 的心材中分离出来的一种白藜芦醇类似物,可诱导白血病细胞凋亡和自噬。它是一种感染前的类苯乙烯类毒素,具有抗菌活性。
T13229 Tunicamycin

Influenza Virus; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Tunicamycin 是一种抗生素的混合物,通过阻断 GlcNAc 磷酸转移酶 (GPT),抑制 N-连接糖基化。Tunicamycin 具有抗肿瘤活性,还具有抗细菌、抗真菌和抗病毒活性。
T3254 PHYTOL

植醇,trans-Phytol,(E)-Phytol

Antibacterial; PPAR; Parasite DNA Damage/DNA Repair; Metabolism; Microbiology/Virology
PHYTOL (trans-Phytol) 是一种从叶绿素中提取的二萜醇,广泛应用于食品添加剂和医药领域,具有很好的抗血吸虫特性。它具有抗伤害、抗氧化、抗炎、抗过敏等作用。它对结核分枝杆菌和金黄色葡萄球菌具有抗菌活性。
T3399 Psoralidin

Others; Estrogen/progestogen Receptor; Reactive Oxygen Species; Lipoxygenase; Gamma-secretase; Akt; COX; Antibacterial Cytoskeletal Signaling; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB; Others; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Psoralidin 是COX-2和5-LOX 的抑制剂,有抗癌,抗菌和抗炎作用。它显著下调NOTCH1信号传导,还极大地诱导活化氧产生。
T2S0961 Chalcone

benzylideneacetophenone,phenyl styryl ketone,Cinnamophenone,benzalacetophenone,β-phenylacrylophenone,查耳酮

EGFR; Antibacterial Angiogenesis; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Chalcone (Cinnamophenone) 是从甘草中分离得到的一种芳香酮,可合成查耳酮衍生物。它具有多种生物和药理的活性,如抗炎、抗菌、抗癌、抗氧化、抗寄生虫等活性。
T3739 2,6-Dimethoxyquinone

2,6-Dimethoxy-1,4-benzoquinone,2,6-Dimethoxy-p-benzoquinone,2,6-Dimethoxybenzoquinone,2,6-二甲氧基-1,4-苯醌

Others Others
2,6-Dimethoxyquinone (2,6-Dimethoxy-p-benzoquinone) 是一种植物中提取吸脂诱导因子。它具有抗脂肪、抗癌、抗菌、抗疟疾和抗炎的作用。
T3907 Tenuigenin

Senegenin,Senegin,远志皂苷元

NF-κB; Caspase; Antibacterial Apoptosis; Microbiology/Virology; NF-κB; Proteases/Proteasome
Tenuigenin (Senegenin) 是从中草药远志根中分离出来的主要活性成分,用于中药,具有抗氧化和抗炎活性。它抑制 NF-κB 活化,预防金黄色葡萄球菌诱导的肺炎。
T0974 Novobiocin Sodium

Albamycinsodium,新生霉素钠,Cathomycin,Albamycin

Potassium Channel; DNA gyrase; Topoisomerase; Antibacterial; Antibiotic; ABC; Autophagy Autophagy; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology
Novobiocin Sodium (Albamycinsodium) 是源自 Streptomyces niveus 的抗生素。 它的化学结构类似于香豆素。Novobiocin 与 DNA 促旋酶结合并阻断三磷酸腺苷活性。
TN1926 Methyl caffeate

Methyl caffeate acid,金银花,咖啡酸甲酯

Others; Antibacterial Microbiology/Virology; Others
Methyl caffeate (Methyl caffeate acid) acid 是一种抗微生物剂,有抗菌和抗分枝杆菌活性。它还抑制 α-葡萄糖苷酶,有氧化应激抑制活性,抗血小板活性,子宫颈癌的抗增殖活性以及肺和白细胞的抗癌活性。
T3416 Aucubin

Aucuboside,桃叶珊瑚苷,Rhinanthin

IL Receptor; NF-κB; Antibacterial Immunology/Inflammation; Microbiology/Virology; NF-κB
Aucubin (Rhinanthin) 是一种可从许多传统的草药中提取的环烯醚萜苷,有许多生物学活性。
TN4893 Rapanone

拉帕酮,2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione,酸藤子醌

Apoptosis; Phospholipase; Antibacterial; Parasite Apoptosis; Metabolism; Microbiology/Virology
Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) 是一种具有广泛生物活性的天然苯醌,如抗肿瘤、抗氧化、抗炎、抗菌和抗寄生虫活性。它还是选择性人滑膜 PLA2抑制剂,IC50值为 2.6 μM。
T26288 Clovamide

trans-Clovamide,N-trans-Caffeoy-L-dopa

Apoptosis; Influenza Virus; ROS; Antibacterial Apoptosis; Immunology/Inflammation; Microbiology/Virology
Clovamide (trans-Clovamide) 是一种天然存在的咖啡酰结合物,具有抗菌、抗炎、抗氧化和神经保护作用。它是一种极好的活性氧和氧自由基清除剂。
T1687 Doxycycline

Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素

MMP; ribosome; Antibacterial; Antibiotic; Parasite Microbiology/Virology; Proteases/Proteasome
Doxycycline (Doxiciclina) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline 具有抗菌活性和抗肿瘤活性。
T0132 Etoposide

VP-16,依托泊苷,依托泊甙,VP-16-213

Apoptosis; Mitophagy; Topoisomerase; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Microbiology/Virology
Etoposide (VP-16-213) 是一种拓扑异构酶 II 的抑制剂,通过与拓扑异构酶 II 和 DNA 形成复合物来抑制 DNA 合成 (IC50=60.3 μM)。Etoposide 具有抗肿瘤活性,可以诱导细胞凋亡、自噬。
T4S1173 Agrimol B

仙鹤草酚B,仙鹤草酚 B

Sirtuin; PPAR Chromatin/Epigenetic; DNA Damage/DNA Repair; Metabolism
Agrimol B 是从仙鹤草中分离得到的一种多酚衍生物,可抑制脂肪形成,降低PPARγ的表达,诱导SIRT1易位和表达。
T3324 Lycorine

Galanthidine,Narcissine,石蒜碱,Amarylline,Belamarine,Licorine,番石榴碱

Apoptosis; Virus Protease; Antibacterial; AChR; Fatty Acid Synthase Apoptosis; Metabolism; Microbiology/Virology; Neuroscience
Lycorine (Narcissine) 是从金眼科植物科中提取的一种天然生物碱。它是一种具有口服活性的SCAP 抑制剂,Kd 值 15.24 nM。它也是黑色素瘤血管生成抑制剂,有用于前列腺癌和代谢疾病的研究潜力。
T1687L Doxycycline (hyclate)

Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate

MMP; ribosome; Antibacterial; Antibiotic Microbiology/Virology; Proteases/Proteasome
Doxycycline hyclate (WC2031) 属于四环素类抗生素,是一种广谱的金属蛋白酶 (MMP) 抑制剂,具有口服活性。Doxycycline hyclate 具有抗菌活性和抗肿瘤活性。
T3417 Amentoflavone

Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin

Apoptosis; P450; Phospholipase; Reactive Oxygen Species; Opioid Receptor; COX; Antibacterial; RSV; Antifungal Apoptosis; Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; NF-κB
Amentoflavone (3',8''-Biapigenin) 是一种具有很多生物活性的双黄酮类天然产物,有抗炎、抗氧化和神经保护等作用。
T21344 1-Deoxynojirimycin hydrochloride

Moranoline,去氧野艽霉素盐酸盐,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin

PI3K; Antibacterial; Antibiotic; Glucosidase Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
1-Deoxynojirimycin hydrochloride (Moranoline) 是一种口服有效的 α-葡萄糖苷酶抑制剂,具有降血糖、减肥和抗病毒的作用,可抑制餐后血糖,预防糖尿病。
TN6732 Oenothein B

Apoptosis; HCV Protease; Antibacterial; Antifungal Apoptosis; Microbiology/Virology; Proteases/Proteasome
Oenothein B 是一种聚(ADP-核糖)糖水解酶的特异性抑制剂。 Oenothein B 具有抗氧化、抗炎、抗真菌、抗 HCV 和抗肿瘤特性。
T11589 Hydroxycitric acid tripotassium hydrate

柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate

ATP Citrate Lyase; HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Chromatin/Epigenetic; Metabolism
Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) 是一种藤黄果的主要活性成分,也是一种柠檬酸的衍生物。它可竞争性抑制柠檬酸裂解酶 (ATP citrate lyase) ,并具有减肥作用。它有效抑制结石形成,并抑制HIF,具有抗氧化,抗炎和抗肿瘤活性。
T8130 Ciprofloxacin hydrochloride monohydrate

Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan

Antibacterial; Antibiotic Microbiology/Virology
Ciprofloxacin hydrochloride monohydrate (Bay-09867 hydrochloride monohydrate) 是一种具有高效抗菌活性的氟喹诺酮类抗生素。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
T1511 Daunorubicin hydrochloride

Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin

Apoptosis; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Daunorubicin hydrochloride (Rubidomycin hydrochloride) 是一种蒽环类氨基糖苷类抗肿瘤药物,可抑制 DNA 复制和修复以及 RNA 和蛋白质合成。
T3376 Cynaroside

朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside

Others; Influenza Virus; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Cynaroside (Luteolin 7-O-Glucoside) 是一个抗氧化类黄酮。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 32 nM。
T8020 Benzoyleneurea

亚苯甲酰基脲,2,4-喹唑啉二酮

Antibacterial Microbiology/Virology
Benzoyleneurea 拥有抗菌活性,常被用作合成新型 PGGTase-I 的抑制剂。
T5787 Macranthoside B

金银花,灰毡毛忍冬次皂苷乙

Antibacterial Microbiology/Virology
Macranthoside B 是一种从金银花中分离出来的天然产物,具有抗菌活性。
TN2316 Xanthyletin

花椒树皮素甲,美洲花椒素

MMP; ERK; Antifungal MAPK; Microbiology/Virology; Proteases/Proteasome
Xanthyletin 是从 Citrus 中得到的香豆素类化合物,具有抗炎、抗肿瘤和抗菌活性,还抑制切叶蚁培育的共生真菌。
T1313 Nitrofurantoin

Furadantine,呋喃妥因,Macrodantin,Furadonine

Antibacterial; Antibiotic Microbiology/Virology
Nitrofurantoin (Furadantine) 是一种具有口服活性的广谱内酰胺酶抗菌剂。它是一种抗生素,可研究尿路感染。
T4S1519 Pseudoginsenoside RT5

拟人参皂苷RT5

Others Others
Pseudoginsenoside RT5 分离于 Panax quinquefolium 中。它通过促进神经生长和提高认知能力,具有抗癫痫、抗抑郁活性,还具有抗菌、抗肿瘤、抗疟疾等活性。
T2S0765 Epibetulinic acid

NO Synthase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Epibetulinic acid 对细菌内毒素刺激的小鼠巨噬细胞 (RAW 264.7) 中 NO 和前列腺素 E(2) 的产生具有有效的抑制作用,IC50分别为 0.7 和 0.6 μM,具有抗炎活性。
T2790 Oridonin

NSC-250682,Rubescenin,冬凌草甲素,Isodonol,Rubescensin A

Akt; Antibacterial Cytoskeletal Signaling; Microbiology/Virology; PI3K/Akt/mTOR signaling
Oridonin (NSC-250682) 是从Rabdosia rubescens 中得到的二萜,是一种AKT 抑制剂,对 AKT1 和 AKT2 的IC50值分别为 8.4 和 8.9 μM,具有抗菌、抗炎、抗肿瘤等功效。
T3400 Bakuchiol

p38 MAPK; DNA/RNA Synthesis; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; MAPK
Bakuchiol 是一种从补骨脂种子中提取的植物雌激素,具有抗肿瘤和抗蠕虫特性,以及细胞毒活性和抗菌活性。
TN3033 4'-Hydroxy-2,4-dimethoxychalcone

Antibacterial; Parasite; Antifungal Microbiology/Virology
4'-Hydroxy-2,4-dimethoxychalcone 是红色龙血天竺葵草药树脂中的天然查尔酮衍生物。4'-Hydroxy-2,4-dimethoxychalcone 具有广泛的生物学活性,包括抗疟疾,抗细菌,抗真菌和抗原生动物活性。
T3811 Ginsenoside C-K

20(S)-人参皂苷 C-K,Ginsenoside compound K,Ginsenoside K,人参皂苷 C-K

P450; cell cycle arrest; COX; NO Synthase Cell Cycle/Checkpoint; Immunology/Inflammation; Metabolism; Neuroscience
Ginsenoside C-K (Ginsenoside K) 是 Ginsenoside Rb1 的细菌代谢物,可通过抑制诱生型一氧化氮合酶和COX-2来发挥抗炎作用。它在人肝微粒体中抑制CYP2C9和CYP2A6活性,IC50分别为 32.0±3.6 和 63.6±4.2 μM。
TN1622 Ermanin

堪非醇3,4'-二-O-甲醚

NOS; Influenza Virus; COX; HIV Protease; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ermanin 是一种从 Tanacetum microphyllum 中分离出来的类黄酮。Ermanin抑制血小板聚集,具有抗结核和抗病毒/细菌特性。Ermanin 可抑制 iNOS 和 COX-2 的表达,从而具有抗炎活性。Ermanin 可能具有抗 HIV-1 活性。Ermanin 在较低浓度下可有效地抑制 Dione juno 幼虫。
T2768 Saikosaponin A

柴胡皂苷A,柴胡皂苷 A

NF-κB; Antibacterial; Liver X Receptor Metabolism; Microbiology/Virology; NF-κB
Saikosaponin A 是银柴胡中的主要活性成分,有抗炎活性,可上调 LXRα的表达。
T4115 Auraptene

橙皮油内酯,7-geranyloxycoumarin,橙皮油素

MMP; BACE Neuroscience; Proteases/Proteasome
Auraptene 是一种丰富的天然香叶氧基香豆素。它能够抑制基质金属蛋白酶 2 以及关键炎症因子,包括 IL-6,IL-8 和趋化因子 (C-C 基序) 配体-5 (CCL5)的分泌。
T7028 Licochalcone C

LICOCHALCONEC,甘草查尔酮C

Phosphatase; Antioxidant; Glucosidase Metabolism; oxidation-reduction
Licochalcone C (LICOCHALCONEC) 能够抑制 α-葡萄糖苷酶,其对 α-葡萄糖苷酶的 IC50 <100 nM,对蛋白酪氨酸磷酸酶 1B 的 IC50=92.43 μM 。
T4S0867 Pogostone

DHELWANGIN,广藿香酮

Apoptosis; Antibacterial; Autophagy Apoptosis; Autophagy; Microbiology/Virology
Pogostone (DHELWANGIN) 是从薄荷中分离出,对革兰氏阴性菌、革兰氏阳性菌、大肠埃希菌等具有强效抗菌、抗真菌活性。它诱导细胞凋亡和自噬。
T2S2264 Linalool

Linalol,(±)-Linalool,Phantol,沉香醇

Apoptosis; IL Receptor; TNF; Endogenous Metabolite; iGluR Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Linalool (Linalol) 是存在芫荽等植物中的单萜类天然产物,是竞争性NMDA 受体拮抗剂,具有抗肿瘤和抗心脏毒性的作用。它通过激活 Nrf2 诱导抗氧化防御和通过抑制 NF-κB 减少炎症反应来保护其免受 LPS/GalN 诱导的肝损伤,具有镇痛、抗菌和抗炎的特性。
TN4478 Macrocarpal H

Antifection Microbiology/Virology
Macrocarpal H has anti-glucosyltransferase, and anti-bacterial activities.
TN4479 Macrocarpal I

Antifection Microbiology/Virology
Macrocarpal I has anti-glucosyltransferase, and anti-bacterial activities.
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天然产物

Xanthone
Cat.No: T2982
Synonym: Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide
Target: Apoptosis, Others, Influenza Virus, Antibacterial, Antifungal
Hexahydrofarnesyl acetone
Cat.No: T8249
Synonym: 植酮,Phytone
Target: Others, Antibacterial
Piperlonguminine
Cat.No: TN2085
Synonym:
Target: Anti-infection, Antibacterial, Antifungal
Comanthoside B
Cat.No: TN3690
Synonym: Comanthosid B
Target: Antibacterial
Ginsenoside Rg4
Cat.No: TN1686
Synonym: 人参皂苷 RG4
Target: Antibacterial
Isoastilbin
Cat.No: TN1772
Synonym:
Target: Anti-infection, Tyrosinase, Antibacterial
Norathyriol
Cat.No: TN1990
Synonym: 芒果苷元
Target: Akt, DNA/RNA Synthesis, AMPK, PPAR
Pinosylvin
Cat.No: T3843
Synonym: 银松素,3,5-stilbenediol,5-Styrylresorcinol
Target: Apoptosis, Others, Antibacterial, Autophagy
Tunicamycin
Cat.No: T13229
Synonym:
Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal
PHYTOL
Cat.No: T3254
Synonym: 植醇,trans-Phytol,(E)-Phytol
Target: Antibacterial, PPAR, Parasite
Psoralidin
Cat.No: T3399
Synonym:
Target: Others, Estrogen/progestogen Receptor, Reactive Oxygen Species, Lipoxygenase, Gamma-secretase, Akt, COX, Antibacterial
Chalcone
Cat.No: T2S0961
Synonym: benzylideneacetophenone,phenyl styryl ketone,Cinnamophenone,benzalacetophenone,β-phenylacrylophenone,查耳酮
Target: EGFR, Antibacterial
2,6-Dimethoxyquinone
Cat.No: T3739
Synonym: 2,6-Dimethoxy-1,4-benzoquinone,2,6-Dimethoxy-p-benzoquinone,2,6-Dimethoxybenzoquinone,2,6-二甲氧基-1,4-苯醌
Target: Others
Tenuigenin
Cat.No: T3907
Synonym: Senegenin,Senegin,远志皂苷元
Target: NF-κB, Caspase, Antibacterial
Novobiocin Sodium
Cat.No: T0974
Synonym: Albamycinsodium,新生霉素钠,Cathomycin,Albamycin
Target: Potassium Channel, DNA gyrase, Topoisomerase, Antibacterial, Antibiotic, ABC, Autophagy
Methyl caffeate
Cat.No: TN1926
Synonym: Methyl caffeate acid,金银花,咖啡酸甲酯
Target: Others, Antibacterial
Aucubin
Cat.No: T3416
Synonym: Aucuboside,桃叶珊瑚苷,Rhinanthin
Target: IL Receptor, NF-κB, Antibacterial
Rapanone
Cat.No: TN4893
Synonym: 拉帕酮,2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone,2,5-Dihydroxy-3-tridecylcyclohexa-2,5-diene-1,4-dione,酸藤子醌
Target: Apoptosis, Phospholipase, Antibacterial, Parasite
Clovamide
Cat.No: T26288
Synonym: trans-Clovamide,N-trans-Caffeoy-L-dopa
Target: Apoptosis, Influenza Virus, ROS, Antibacterial
Doxycycline
Cat.No: T1687
Synonym: Vibramycin,多西环素,Doxiciclina,Doxytetracycline,Doxycyclinum,强力霉素
Target: MMP, ribosome, Antibacterial, Antibiotic, Parasite
Etoposide
Cat.No: T0132
Synonym: VP-16,依托泊苷,依托泊甙,VP-16-213
Target: Apoptosis, Mitophagy, Topoisomerase, Antibacterial, Antibiotic, Autophagy
Agrimol B
Cat.No: T4S1173
Synonym: 仙鹤草酚B,仙鹤草酚 B
Target: Sirtuin, PPAR
Lycorine
Cat.No: T3324
Synonym: Galanthidine,Narcissine,石蒜碱,Amarylline,Belamarine,Licorine,番石榴碱
Target: Apoptosis, Virus Protease, Antibacterial, AChR, Fatty Acid Synthase
Doxycycline (hyclate)
Cat.No: T1687L
Synonym: Doxycycline hydrochloride hemiethanolate hemihydrate,盐酸强力霉素,WC2031,Doxycycline hyclate
Target: MMP, ribosome, Antibacterial, Antibiotic
Amentoflavone
Cat.No: T3417
Synonym: Didemethyl-ginkgetin,穗花杉双黄酮,Amenthoflavone,3',8''-Biapigenin
Target: Apoptosis, P450, Phospholipase, Reactive Oxygen Species, Opioid Receptor, COX, Antibacterial, RSV, Antifungal
1-Deoxynojirimycin hydrochloride
Cat.No: T21344
Synonym: Moranoline,去氧野艽霉素盐酸盐,AT2220,Duvoglustat hydrochloride,1-Deoxynojirimycin,DNJ,deoxynojirimycin
Target: PI3K, Antibacterial, Antibiotic, Glucosidase
Oenothein B
Cat.No: TN6732
Synonym:
Target: Apoptosis, HCV Protease, Antibacterial, Antifungal
Hydroxycitric acid tripotassium hydrate
Cat.No: T11589
Synonym: 柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate
Target: ATP Citrate Lyase, HIF/HIF Prolyl-Hydroxylase, HIF
Ciprofloxacin hydrochloride monohydrate
Cat.No: T8130
Synonym: Oftacilox,Ciprofloxacin hydrochloride hydrate,Bay-09867 hydrochloride monohydrate,环丙沙星盐酸盐一水合物,Ceprimax,盐酸环丙沙星(一水物),Ciloxan
Target: Antibacterial, Antibiotic
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Daunorubicin hydrochloride
Cat.No: T1511
Synonym: Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin
Target: Apoptosis, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic, Autophagy
Cynaroside
Cat.No: T3376
Synonym: 朝蓟糖甙,Luteoloside,Luteolin 7-β-D-Glucopyranoside,Luteolin 7-O-Glucoside,Luteolin 7-O-β-D-glucoside,木犀草苷,Luteolin 7-glucoside
Target: Others, Influenza Virus, DNA/RNA Synthesis
Benzoyleneurea
Cat.No: T8020
Synonym: 亚苯甲酰基脲,2,4-喹唑啉二酮
Target: Antibacterial
Macranthoside B
Cat.No: T5787
Synonym: 金银花,灰毡毛忍冬次皂苷乙
Target: Antibacterial
Xanthyletin
Cat.No: TN2316
Synonym: 花椒树皮素甲,美洲花椒素
Target: MMP, ERK, Antifungal
Nitrofurantoin
Cat.No: T1313
Synonym: Furadantine,呋喃妥因,Macrodantin,Furadonine
Target: Antibacterial, Antibiotic
Pseudoginsenoside RT5
Cat.No: T4S1519
Synonym: 拟人参皂苷RT5
Target: Others
Epibetulinic acid
Cat.No: T2S0765
Synonym:
Target: NO Synthase, Prostaglandin Receptor
Oridonin
Cat.No: T2790
Synonym: NSC-250682,Rubescenin,冬凌草甲素,Isodonol,Rubescensin A
Target: Akt, Antibacterial
Bakuchiol
Cat.No: T3400
Synonym:
Target: p38 MAPK, DNA/RNA Synthesis, Autophagy
4'-Hydroxy-2,4-dimethoxychalcone
Cat.No: TN3033
Synonym:
Target: Antibacterial, Parasite, Antifungal
Ginsenoside C-K
Cat.No: T3811
Synonym: 20(S)-人参皂苷 C-K,Ginsenoside compound K,Ginsenoside K,人参皂苷 C-K
Target: P450, cell cycle arrest, COX, NO Synthase
Ermanin
Cat.No: TN1622
Synonym: 堪非醇3,4'-二-O-甲醚
Target: NOS, Influenza Virus, COX, HIV Protease, Antibacterial, Antibiotic
Saikosaponin A
Cat.No: T2768
Synonym: 柴胡皂苷A,柴胡皂苷 A
Target: NF-κB, Antibacterial, Liver X Receptor
Auraptene
Cat.No: T4115
Synonym: 橙皮油内酯,7-geranyloxycoumarin,橙皮油素
Target: MMP, BACE
Licochalcone C
Cat.No: T7028
Synonym: LICOCHALCONEC,甘草查尔酮C
Target: Phosphatase, Antioxidant, Glucosidase
Pogostone
Cat.No: T4S0867
Synonym: DHELWANGIN,广藿香酮
Target: Apoptosis, Antibacterial, Autophagy
Linalool
Cat.No: T2S2264
Synonym: Linalol,(±)-Linalool,Phantol,沉香醇
Target: Apoptosis, IL Receptor, TNF, Endogenous Metabolite, iGluR
Macrocarpal H
Cat.No: TN4478
Synonym:
Target: Antifection
Macrocarpal I
Cat.No: TN4479
Synonym:
Target: Antifection
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