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1059

抑制剂 & 化合物

313

天然产物

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Cat. No. Product Name Target Signaling Pathways
TP1527 CEF8, Influenza Virus NP (383-391)

CEF8, Influenza Virus NP 383-391

Others Others
CEF8, Influenza Virus NP (383-391) 是一种甲型流感病毒核蛋白,含有 383-391 残基,是甲型流感病毒核蛋白中重要的 HLA-B*2705 限制性表位,与细胞毒性 T 淋巴细胞介导的免疫逃逸有关。
TP1267L CEF27, Epstein-Barr Virus BRLF-1 lytic 148-156 acetate

CEF27, Epstein-Barr Virus BRLF-1 lytic 148-156 acetate(254110-79-7 free base)

Others Others
CEF27, Epstein-Barr Virus BRLF-1 lytic 148-156 acetate(254110-79-7 free base) 对应于 BRLF1 的氨基酸 148-156。 BRLF1 是一种转录激活因子,可直接与一些 Epstein-Barr 病毒 (EBV) 裂解基因启动子中的富含 GC 的基序结合。
T39335 Anti-virus agent 1

Anti-virus agent 1,Remdesivir isopropyl ester analog

Anti-virus agent 1 (compound 4i), a phosphoramidate prodrug of GS-5734, exhibits potent antiviral efficacy. It is primarily utilized in the study of coronavirus and Ebola virus (EBOV).
TP1520 Hepatitis B Virus Core (128-140)

Hepatitis B Virus Core 128-140

The hepatitis B virus (HBV) core protein has been found in the nucleus, the cytoplasm, or both of HBV-infected hepatocytes. nuclear localization of the HBV core protein is negatively regulated by phosphorylation during the cell cycle.
TP1596 CEF7, Influenza Virus NP (380-388)

CEF7, Influenza Virus NP 380-388

HLA-B*08 restricted influenza virus nucleoprotein epitope.
TP1268 CEF19, Epstein-Barr Virus latent NA-3A (458-466)

CEF19,Epstein-Barr Virus latent NA-3A 458-466

CEF19, Epstein-Barr Virus latent NA-3A (458-466) is a single peptide epitope, YPLHEQHGM, representing residues 458-466 of the type 1 Epstein-Barr Virus (EBV) nuclear antigen 3A protein (B95.8 strain).
TP1267 CEF27, Epstein-Barr Virus BRLF-1 lytic (148-156)

CEF27,Epstein-Barr Virus BRLF-1 lytic 148-156

HLA-A*0301-restricted epitope from Epstein-Barr Virus , EBV BRLF-1 (148-156).
T39778 Influenza A virus-IN-1

Influenza A virus-IN-1, a dihydropyrrolidones derivative, is a highly effective inhibitor of various subtypes of influenza A virus (IAV) with IC 50 values ranging from 3.11 μM to 7.13 μM. It effectively suppresses IAV replication and enhances the expression of key antiviral cytokines, such as IFN-β, and the antiviral protein MxA.
TP1871 Rabies Virus Glycoprotein

Rabies Virus Glycoprotein is a 29 amino acid fragment generated from rabies virus glycoprotein (RVG). This peptide specifically binds to the acetylcholine receptor expressed by neuronal cells.
TP1871L Rabies Virus Glycoprotein acetate

Rabies Virus Glycoprotein acetate 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 TP1871L。
T13046 Syncytial Virus Inhibitor-1

Others Others
Syncytial Virus Inhibitor-1 is a potent and orally bioavailable inhibitor of respiratory syncytial virus (RSV) fusion(EC50s of 0.002 μM, 0.004 μM, and 0.002 μM for RSV Long, RSV A2, and RSV B strains, respectively).
TP1553 Rabies Virus Glycoprotein TFA

Rabies Virus Glycoprotein (TFA) is a kind of by the Rabies Virus Glycoprotein 29 - amino acid derived cell penetrating peptides, it can pass the blood brain barrier (BBB) into the brain cells.
T22868 Influenza A virus fragment

Others Others
Influenza A virus fragment has the RNA sequence of Leu-Lys-Phe-Ala-Phe-Ser-Met-Met.
T39503 Hepatitis Virus C NS3 Protease Inhibitor 2

Hepatitis Virus C NS3 Protease Inhibitor 2 is a peptide inhibitor derived from a product that targets the NS3 protease of the hepatitis C virus (HCV). Its inhibitory activity against the NS3 protease is characterized by a Ki value of 41 nM.
TP2231 HBcAg [Hepatitis B virus] (18-27)

Others Others
HBcAg (core antigen) is a hepatitis B viral protein. It is an indicator of active viral replication; this means the person infected with Hepatitis B can likely transmit the virus on to another person.
T22838 hemagglutinin (332-340) [Influenza A virus]

Others Others
Influenza hemagglutinin is a type of hemagglutinin found on the surface of the influenza viruses. It is an antigenic glycoprotein. It is responsible for binding the virus to the cell that is being infected. Influenza hemagglutinin proteins bind to cells w
T23407 surface antigen (208-215) [Hepatitis B Virus]

Others Others
The nucleocapsid of the hepatitis B virus is covered by an envelope of HBV surface antigen (HBsAg), which has the common, group-specific determinant a. The four major subtypes of HBsAg, adw, adr, ayw and ayr, are generated, and they have been proposed to
T9231 Mbx2329

Antiviral Immunology/Inflammation
MBX2329 是一种流感病毒抑制剂,能特异性地抑制血凝素介导的病毒进入,HIV/HA(H5) 的 IC90值为8.6 μM。它能够有效地抑制多种甲型流感病毒。
T7785 T-1105

Influenza Virus Microbiology/Virology
T-1105 是 T-705 的结构类似物,是一种广谱病毒聚合酶抑制剂,在转化为核糖核苷三磷酸代谢物后抑制 RNA 病毒的聚合酶,有抗病毒活性。
TP2230 Fusion glycoprotein (92-106) [Human respiratory syncytial virus]

Others Others
Fusion glycoprotein (92-106) [Human respiratory syncytial virus] is a peptide with the sequence H2N-Glu-Leu-Gln-Leu-Leu-Met-Gln-Ser-Thr-Pro-Pro-Thr-Asn-Asn-Arg-OH, MW= 1741.96.
TP2232 hemagglutinin precursor (114-122) amide [Influenza A virus]

Others Others
Partial antigenic glycoprotein
T80338 RVG

Rabies Virus Glycoprotein-29,RVG29,RDP

RVG (RVG29) 是从狂犬病病毒糖蛋白衍生的肽,它能够结合到神经元细胞的烟碱乙酰胆碱受体 (AchR) α-7 亚基上。此外,RVG 促进了结核分枝杆菌抗原向抗原呈递细胞的递送效率。
T12953 Sodium copper chlorophyllin B

Influenza Virus; HIV Protease Microbiology/Virology; Proteases/Proteasome
Sodium copper chlorophyllin B 对流感病毒和HIV 有抗病毒活性,IC50s 值都是 50 到 100 μM。
T38514 PMEDAP

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
PMEDAP 是有效的人类免疫缺陷病毒 (HIV) 复制抑制剂。它具有抗小鼠巨细胞病毒活性。它有效抑制莫罗尼鼠肉瘤病毒诱导的肿瘤形成和相关死亡率。
T61953 Zika virus-IN-2

Zika virus-IN-2 (Compd 3) 是Zika 病毒的抑制剂(EC50= 7.4 μM)。
T61762 Zika virus-IN-3

Zika virus-IN-3 (Compd 7) 是Zika 病毒的抑制剂,其EC50值为 3.4 μM。
T60697 Influenza virus-IN-1

Influenza virus-IN-1 (compound 14) 具有抗甲型流感病毒活性,它是甲型流感病毒的有效抑制剂,其CC50值 >200 μM,EC50值为 2.46 μM。Influenza virus-IN-1 对 PAN 核酸内切酶显示出浓度依赖性的抑制活性 (EC50 = 312.36 nM)。
T76517 Herpes virus inhibitor 2

Herpes virus inhibitor 2 为一种疱疹病毒抑制剂,专门破坏疱疹病毒的核糖核苷酸还原酶四级结构,从而抑制病毒复制。
T62837 Influenza virus-IN-3

Influenza virus-IN-3 (compound 9) 是一种选择性流感病毒的有效抑制剂,能够作用于 H5N1 (IC50: 0.88 μM)、H5N2 (IC50: 0.10 μM)、H5N6 (IC50: 5.5 μM)、H5N8 (IC50: 0.51 μM)。Influenza virus-IN-3 具有抗病毒和 NA (神经氨酸酶) 抑制作用,且细胞毒性低 (CC50>200 μM)。
T75166 Influenza virus-IN-7

Influenza virus-IN-7 (Example 16) 是一种口服活性的帽依赖性核酸内切酶抑制剂,适用于流感病毒感染疾病的研究。
T62216 Influenza virus-IN-5

Influenza virus-IN-5 (Compound 5f) 是一种流感病毒血球凝集素 (hemagglutinin (HA)) 抑制剂,能够作用于 A/H3N2 病毒 (EC50: 1 nM)。
T62197 Influenza virus-IN-4

Influenza virus-IN-4 (compound 11e) 是一种流感病毒神经氨酸酶的有效抑制剂,能够作用于 H5N1 (IC50: 3.4 μM)、H5N2 (IC50: 0.094 μM)、H5N6 (IC50: 0.79 μM)、H5N8 (IC50: 0.077 μM)。Influenza virus-IN-4 能够抑制 NA(神经氨酸酶),并具有低细胞毒性(CC50>200 μM)。Influenza virus-IN-4 在1500 mg/kg 时,对小鼠没有明显的毒性。
T76515 Herpes virus inhibitor 1

Herpes virus inhibitor 1 是一种抑制疱疹病毒的化合物,能破坏疱疹病毒的核糖核苷酸还原酶四级结构,从而抑制病毒复制。
T72450 Influenza virus-IN-6

Influenza Virus Microbiology/Virology
Influenza virus-IN-6 (Compound 35) 是一种针对流感病毒聚合酶酸性蛋白亚基内切酶N端结构域(PAN)的高效抑制剂,展现出0.20 μM的IC50值。
T38239 2'-Deoxy-2'-fluorouridine

2'-Deoxy-2'-fluorouridine 是合成抗流感病毒试剂的中间体。
T63586 Zika virus-IN-1

Zika virus-IN-1 是一种 Zika 病毒的抑制剂 (EC50: 1.56 μM)。
T60810 Influenza virus-IN-2

Influenza virus-IN-2 (compound 19) 具有抗甲型流感病毒活性,是有效的流感病毒抑制剂,CC50值为 150.85 μM,EC50值为 2.58 μM,。Influenza virus-IN-2 浓度依赖性的抑制 PAN 核酸内切酶,EC50为 489.39 nM。
T1848 Dynasore

Dynamin Inhibitor I

Dynamin; Virus Protease; Autophagy; HSV Autophagy; Cytoskeletal Signaling; Microbiology/Virology
Dynasore (Dynamin Inhibitor I) 是一种可渗透细胞的化学物质,可逆且非竞争性地抑制 dynamin 1/2 的 GTPase 活性。 它还抑制线粒体动力蛋白 Drp1,对其他小 GTPase 没有影响。
T6846 Vesatolimod

GS-9620,维沙莫德

Apoptosis; HCV Protease; HBV; TLR; HIV Protease Apoptosis; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Vesatolimod (GS-9620) 是一种选择性 Toll 样受体 7 口服激动剂,EC50值为291 nM。
T16366 NVR 3-778

HBV Microbiology/Virology
NVR 3-778 是一种 SBA 类的口服有效HBV CAM 衣壳组装调制剂,具有抗 HBV 活性。
T74762 Influenza A virus-IN-8

Influenza A virus-IN-8 (S5) 为一种大环肽,无细胞毒性,并作为甲型流感病毒 (IAV) 的有效抑制剂,显示出较好的蛋白酶稳定性。其对 H1 和 H5 变体的IC50值分别低至 6.7 nM 和 6.6 nM。此外,Influenza A virus-IN-8 能够与 HA 茎的一个保守区域结合,特别是对 H1 变体展现出 1.0 nM 的高亲和性Kd 值。
T62059 Influenza A virus-IN-6

Influenza A virus-IN-6 (compound 16j) 是有效的选择性甲型流感病毒抑制剂(IC50= 3.88 μM, CC50= 36.64 μM)。Influenza A virus-IN-6 显示出抗 IAV 活性和较低的细胞毒性。
T16276 NBD-556

HIV Protease Microbiology/Virology; Proteases/Proteasome
NBD-556是一种 CD4 模拟物,识别 HIV-1 包膜蛋白 gp120 并诱导 gp120 重组,类似于 CD4 结合,可阻断 gp120-CD4 的相互作用。
T11669 IR415

HBV Microbiology/Virology
IR415 选择性地与 HBx 相互作用 (Kd=2 nM) 并阻断 HBV 介导的 RNAi 抑制,逆转 HBx 蛋白对 Dicer 核糖核酸内切酶活性的抑制作用。IR415 具有抗 HBV 的活性。
T6327 Tubacin

Virus Protease; HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology
Tubacin 是一种高效、选择性、可逆、可渗透细胞的 HDAC6 抑制剂,IC50 为 4 nM,选择性是 HDAC1 的约 350 倍。
T38236 2′-Deoxy-2′-fluoroguanosine

Nucleoside Antimetabolite/Analog; Influenza Virus Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
2′-Deoxy-2′-fluoroguanosine 是一种核苷类似物,有效抑制流感病毒,抑制A 型和B 型流感病毒的EC90值 <0.35 μM。2′-Deoxy-2′-fluoroguanosine 显著抑制流感病毒在上呼吸道中的复制,从而改善鼻腔炎症和发烧。
T79921 Moloney murine leukemia virus RT

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Moloney murine leukemia virus RT为源自Moloney小鼠白血病病毒的逆转录酶,作为复制聚合酶在逆转录病毒生命周期中扮演关键角色。
T62888 Influenza A virus-IN-7

Influenza A virus-IN-7 (compound 16r) 是一种有效的、口服具有活力的甲型流感病毒抑制剂 (IC50: 3.43 μM, CC50>100 μM)。Influenza A virus-IN-7 具有抗 IAV 作用,细胞毒性低,对病毒 RNA 的转录和复制表现出抑制作用。
T61877 Influenza A virus-IN-5

Influenza A virus-IN-5 (Compound 16e) is a highly potent and orally active agent against the influenza A virus (IAV), exhibiting an IC 50 of 1.29 μM. It effectively inhibits the transcription and replication of viral RNA while maintaining acceptable levels of cytotoxicity [1].
T61557 Influenza A virus-IN-4

Influenza A virus-IN-4 (compound 23b), a derivative of Oseltamivir, is a highly effective neuraminidase inhibitor. It exerts potent inhibitory effects on influenza viruses [1].

化合物

CEF8, Influenza Virus NP (383-391)
Cat.No: TP1527
Synonym: CEF8, Influenza Virus NP 383-391
Target: Others
CEF27, Epstein-Barr Virus BRLF-1 lytic 148-156 acetate
Cat.No: TP1267L
Synonym: CEF27, Epstein-Barr Virus BRLF-1 lytic 148-156 acetate(254110-79-7 free base)
Target: Others
Anti-virus agent 1
Cat.No: T39335
Synonym: Anti-virus agent 1,Remdesivir isopropyl ester analog
Target:
Hepatitis B Virus Core (128-140)
Cat.No: TP1520
Synonym: Hepatitis B Virus Core 128-140
Target:
CEF7, Influenza Virus NP (380-388)
Cat.No: TP1596
Synonym: CEF7, Influenza Virus NP 380-388
Target:
CEF19, Epstein-Barr Virus latent NA-3A (458-466)
Cat.No: TP1268
Synonym: CEF19,Epstein-Barr Virus latent NA-3A 458-466
Target:
CEF27, Epstein-Barr Virus BRLF-1 lytic (148-156)
Cat.No: TP1267
Synonym: CEF27,Epstein-Barr Virus BRLF-1 lytic 148-156
Target:
Influenza A virus-IN-1
Cat.No: T39778
Synonym:
Target:
Rabies Virus Glycoprotein
Cat.No: TP1871
Synonym:
Target:
Rabies Virus Glycoprotein acetate
Cat.No: TP1871L
Synonym:
Target:
Syncytial Virus Inhibitor-1
Cat.No: T13046
Synonym:
Target: Others
Rabies Virus Glycoprotein TFA
Cat.No: TP1553
Synonym:
Target:
Influenza A virus fragment
Cat.No: T22868
Synonym:
Target: Others
Hepatitis Virus C NS3 Protease Inhibitor 2
Cat.No: T39503
Synonym:
Target:
HBcAg [Hepatitis B virus] (18-27)
Cat.No: TP2231
Synonym:
Target: Others
hemagglutinin (332-340) [Influenza A virus]
Cat.No: T22838
Synonym:
Target: Others
surface antigen (208-215) [Hepatitis B Virus]
Cat.No: T23407
Synonym:
Target: Others
Mbx2329
Cat.No: T9231
Synonym:
Target: Antiviral
T-1105
Cat.No: T7785
Synonym:
Target: Influenza Virus
Fusion glycoprotein (92-106) [Human respiratory syncytial virus]
Cat.No: TP2230
Synonym:
Target: Others
hemagglutinin precursor (114-122) amide [Influenza A virus]
Cat.No: TP2232
Synonym:
Target: Others
RVG
Cat.No: T80338
Synonym: Rabies Virus Glycoprotein-29,RVG29,RDP
Target:
Sodium copper chlorophyllin B
Cat.No: T12953
Synonym:
Target: Influenza Virus, HIV Protease
PMEDAP
Cat.No: T38514
Synonym:
Target: Others, HIV Protease
Zika virus-IN-2
Cat.No: T61953
Synonym:
Target:
Zika virus-IN-3
Cat.No: T61762
Synonym:
Target:
Influenza virus-IN-1
Cat.No: T60697
Synonym:
Target:
Herpes virus inhibitor 2
Cat.No: T76517
Synonym:
Target:
Influenza virus-IN-3
Cat.No: T62837
Synonym:
Target:
Influenza virus-IN-7
Cat.No: T75166
Synonym:
Target:
Influenza virus-IN-5
Cat.No: T62216
Synonym:
Target:
Influenza virus-IN-4
Cat.No: T62197
Synonym:
Target:
Herpes virus inhibitor 1
Cat.No: T76515
Synonym:
Target:
Influenza virus-IN-6
Cat.No: T72450
Synonym:
Target: Influenza Virus
2'-Deoxy-2'-fluorouridine
Cat.No: T38239
Synonym:
Target:
Zika virus-IN-1
Cat.No: T63586
Synonym:
Target:
Influenza virus-IN-2
Cat.No: T60810
Synonym:
Target:
Dynasore
Cat.No: T1848
Synonym: Dynamin Inhibitor I
Target: Dynamin, Virus Protease, Autophagy, HSV
Vesatolimod
Cat.No: T6846
Synonym: GS-9620,维沙莫德
Target: Apoptosis, HCV Protease, HBV, TLR, HIV Protease
NVR 3-778
Cat.No: T16366
Synonym:
Target: HBV
Influenza A virus-IN-8
Cat.No: T74762
Synonym:
Target:
Influenza A virus-IN-6
Cat.No: T62059
Synonym:
Target:
NBD-556
Cat.No: T16276
Synonym:
Target: HIV Protease
IR415
Cat.No: T11669
Synonym:
Target: HBV
Tubacin
Cat.No: T6327
Synonym:
Target: Virus Protease, HDAC
2′-Deoxy-2′-fluoroguanosine
Cat.No: T38236
Synonym:
Target: Nucleoside Antimetabolite/Analog, Influenza Virus
Moloney murine leukemia virus RT
Cat.No: T79921
Synonym:
Target: DNA/RNA Synthesis
Influenza A virus-IN-7
Cat.No: T62888
Synonym:
Target:
Influenza A virus-IN-5
Cat.No: T61877
Synonym:
Target:
Influenza A virus-IN-4
Cat.No: T61557
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T4S1718 Punicalin

HBV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Punicalin 是从Punica granatumL. 或Terminalia catappaL. 的叶子中分离的,一种可水解的单宁,具有抗炎活性。它是一种抗乙型肝炎病毒药物。
T8187 Tetrahydroepiberberine

Others; Influenza Virus; Antifungal Microbiology/Virology; Others
Tetrahydroepiberberine 是从Corydalis impatiens(Pall) 中分离得到的一种异喹啉生物碱,具有抗真菌和选择性抑制 PI-3 病毒活性的作用。
TN1482 Chamaechromone

P450; HBV Metabolism; Microbiology/Virology
Chamaechromone 是从 Stellera chamaejasme L. 的根中分离出来的天然产物。 Chamaechromone 具有抗 HBV 和杀虫活性。
T3S0872 Paederoside

Antiviral; HBV Immunology/Inflammation; Microbiology/Virology
Paederoside 是从Paederia pertomentosa 分离的一种单萜 S-甲基硫代碳酸酯。它抑制 Epstein-Barr 病毒的激活,有抗肿瘤促进作用。
T3S1852 Cephaeline hydrochloride

Others; Virus Protease; Influenza Virus Microbiology/Virology; Others
Cephaeline hydrochloride 是 Indian Ipecac 中的一种酚类生物碱。它有效抑制病毒 ZIKV 和 EBOV 感染。
TN1103 Diphyllin

山荷叶素,二叶草素

ATPase; Proton pump; Influenza Virus; HIV Protease Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Diphyllin 是一种从Justicia procumbens 中分离的芳基萘木脂素,是HIV-1的有效抑制剂,IC50 为 0.38 μM。它是V-ATPase 抑制剂,IC50值为 17 nM,可抑制人破骨细胞中的溶酶体酸化。它抑制NO 产生,IC50值为 50 μM ,具有抗癌和抗炎活性。
T2945 Germacrone

P450; Antiviral; Influenza Virus Immunology/Inflammation; Metabolism; Microbiology/Virology
Germacrone 提取自姜黄,具有抗炎、抗雄激素和抗病毒活性。 它还通过促进细胞凋亡来抑制胶质瘤细胞的增殖。
T0775 Coumarin

Factor Xa; Influenza Virus Metabolism; Microbiology/Virology
Coumarin 是中国北沙参中的一种主要生物活性成分,具有抗癌、抗炎和抗病毒等活性。它作为几种抗凝剂的前体具有临床价值,尤其是华法林。
T5S1708 Dendrobine

Others; Influenza Virus Microbiology/Virology; Others
Dendrobine 是从石斛中分离的一种生物碱,对甲型流感病毒具有抗病毒活性。
TQ0248 Alisol F

泽泻醇 F,泽泻醇F

HBV Microbiology/Virology
Alisol F 是从泽泻中分离得到的一种三萜,具有免疫抑制和抗病毒功能。
T3905 Isomangiferin

芒果

Free radical scavengers; Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology; oxidation-reduction
Isomangiferin 是一种天然产物,具有抗病毒的作用。它还具有抗氧化和自由基清除活性。
TN1788 Isookanin

Amylase Metabolism
Isookanin 在多种疾病领域有研究价值,包括肿瘤,皮疹,蛇和昆虫叮咬,糖尿病,腹泻。它可作为抗病毒剂对抗 HSV 和水痘带状疱疹病毒。它也具有抗氧化特性。
T2780 Catalpol

梓醇,Catalpinoside,Digitalis purpurea L

Others; HBV Microbiology/Virology; Others
Catalpol (Catalpinoside) 是一种在Rehmannia glutinosa 中发现的鸢尾花苷,具有神经保护、降血糖、抗癌、抗痉挛、抗氧化、抗HBV 和抗肝炎病毒作用。
T7602 Theaflavin

Influenza Virus; Endogenous Metabolite Metabolism; Microbiology/Virology
Theaflavin 是在红茶中发现的一种多酚类黄酮,具有如抗氧化、抗癌、抗炎和抗病毒多种生物活性。
T2942 Psoralen

Ficusin,Furocoumarin,补骨脂素,psoralene

Apoptosis; Influenza Virus; HIV Protease; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
Psoralen (Ficusin) 是从补骨脂种子中提取的一种香豆素。它具有如抗癌、抗氧化、抗抑郁、抗癌、抗菌、抗病毒等多种生物学特性。
T5712 zerumbone

花薑酮,球姜酮

Antioxidant; HSV Microbiology/Virology; oxidation-reduction
Zerumbone 是从Zingiber zerumbetSmith 的根茎中分离的一种单环倍半萜烯,可有效抑制Epstein-Barr 病毒的激活,IC50为 0.14 mM,具有抗癌、抗炎、抗氧化和抗增殖的作用。
TN1480 Cephaeline

吐根鹼,吐根酚碱

Virus Protease; Influenza Virus; HIF Angiogenesis; Chromatin/Epigenetic; Microbiology/Virology
Cephaeline 对受保护的原代 CLL 细胞具有高度活性(相对 IC50 为 35nM),并通过抑制 HIF-1α± 和扰乱细胞内氧化还原稳态发挥作用。
T2S0257 Dehydroandrographolide succinate

Others; Influenza Virus Microbiology/Virology; Others
Dehydroandrographolide succinate 是从中药穿心莲中提取的一种天然产物,具有免疫刺激、抗感染和抗炎作用,有潜力研究病毒性肺炎和病毒性上呼吸道感染。
T3342 Xanthohumol

Apoptosis; Others; Influenza Virus; COX; Acyltransferase; HSV Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience; Others
Xanthohumol 是从啤酒花中分离到的黄酮类化合物,可抑制 COX-1 和 COX-2 活性,具有抗肿瘤,抗血管生成的作用,还具有抗多种病毒的活性。
TN2331 Eleutheroside B1

刺五加苷B1

Influenza Virus Microbiology/Virology
Eleutheroside B1是具有广谱抗人流感病毒的一种香豆素。它抑制多种趋化因子基因和流感病毒核蛋白基因的 mRNA 表达。它具有抗病毒、抗流感和抗炎活性,且细胞毒性小。
TN2283 Tripterifordin

HIV Protease Microbiology/Virology; Proteases/Proteasome
Tripterifordin 在 H9 淋巴细胞中显示出抗 HIV 复制活性,EC50值为 3100 nM。
TMO2787 Anthraquinone

dioxoanthracene,Anthradione,anthracenedione,蒽醌

Virus Protease Microbiology/Virology
Anthraquinone (Anthradione) 是常用于缓解便秘的草药中的主要活性成分,可用作染料形成前体。
T6377 Aloperine

Apoptosis; Virus Protease; HIV Protease; Antibiotic; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Aloperine 是一种在苦参类植物中的生物碱,其具有抗癌,抗炎、抗肿瘤和抗病毒特性,可用于研究过敏性接触性皮炎湿疹和其他皮肤炎症。
T2738 Dehydroandrographolide

NOS; Influenza Virus Immunology/Inflammation; Microbiology/Virology
Dehydroandrographolide 是从草药穿心莲中提取的一种天然产物。它通过使 iNOS 失活来降低 LPS 诱导的急性肺损伤中的氧化应激,有抗感染活性。
T2957 Arctigenin

牛蒡苷元,牛蒡子苷元,(-)-Arctigenin

Apoptosis; MMP; Influenza Virus; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Arctigenin ((-)-Arctigenin) 是一种存在于牛蒡中的木脂素,具有抗氧化、抗肿瘤、抗炎和抗病毒活性。它可研究代谢紊乱和中枢神经系统功能障碍。
T5666 Dipotassium glycyrrhizinate

Virus Protease Microbiology/Virology
Dipotassium glycyrrhizinate 是一种具有抗过敏和抗炎活性的阴离子表面活性剂。
T2854 Phillyrin

Forsythin,连翘苷

P450; Influenza Virus; AMPK Chromatin/Epigenetic; Metabolism; Microbiology/Virology; PI3K/Akt/mTOR signaling
Phillyrin (Forsythin) 是从连翘中分离出来的一种天然产物,具有抗甲型流感病毒的活性,以及抗菌和消炎作用。
T1131 Ivermectin

MK-933,伊维菌素

Mitophagy; GluCls; P2X Receptor; SARS-CoV; HIV Protease; Antibiotic; Parasite; Autophagy; HSV Autophagy; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ivermectin (MK-933) 是谷氨酸门控氯离子通道激活剂,具有抗寄生虫活性。它特异性抑制Impα/β1 介导的核导入,还抑制牛疱疹病毒 1 复制并抑制BoHV-1DNA 聚合酶的核输入。它具有很强的抗病毒活性。它也是P2X4和 α7nAChRs 的正异构效应物。
T2741 Glycyrrhizic acid

Glycyrrhizin,甘草酸

Virus Protease; Dehydrogenase; MAO Metabolism; Microbiology/Virology; Neuroscience
Glycyrrhizic acid (Glycyrrhizin) 是甘草里面的活性成分三萜皂苷,为 HMGB1的拮抗剂,有用于肿瘤、糖尿病等研究的潜力。
T2875 Angelicin

Isopsoralen,异补骨脂素

Apoptosis; Virus Protease; Antiviral Apoptosis; Immunology/Inflammation; Microbiology/Virology
Angelicin (Isopsoralen) 是一种三环芳烃天然产物,结构上跟补骨脂素有关,具有抗癌、抗炎、抗病毒等活性。
TQ0180 Chebulagic acid

SARS-CoV; Influenza Virus; Lipoxygenase; COX Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
Chebulagic acid 是从 Terminalia chebula Retz 中分离出来的一种 COX-LOX 双重抑制剂,有抗炎和抗感染作用。它抑制 SARS-CoV-2病毒的复制,EC50值为 9.76 μM。它还是 M2(S31N)抑制剂和抗流感病毒剂。
T8286 Harringtonine

三尖杉酯碱,三尖杉脂碱

Others; Influenza Virus Microbiology/Virology; Others
Harringtonine 是一种天然的 Cephalotaxus 生物碱,可抑制蛋白质合成,有抗基孔肯雅病毒活性,EC50为 0.24 μM。
T5429 Theaflavin 3,3'-digallate

茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG

Virus Protease; Antioxidant; HIV Protease; HSV Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。
T2718 Palmatine chloride

Others; Indoleamine 2,3-Dioxygenase (IDO); Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Others
Palmatine chloride 是口服具有活力的不可逆 IDO-1抑制剂。它能够减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,并改善 DSS 诱发的结肠炎。
T5S0802 Palmatine

巴马汀,Berbericinine,Burasaine

Indoleamine 2,3-Dioxygenase (IDO); AChR; AChE; Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Neuroscience
Palmatine (Burasaine) 是口服具有活力的、不可逆IDO-1抑制剂。它可以减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,从而改善DSS (Dextran Sulphate Sodium Salt) 诱发的结肠炎。它有用于结肠炎的研究潜力。
T6523 Guanosine

鸟苷,DL-Guanosine,Vernine,Guanozin

Endogenous Metabolite; HSV Metabolism; Microbiology/Virology
Guanosine (DL-Guanosine) 是由鸟嘌呤与核糖环组成的一种核苷,两者之间由 β-N9-配糖键相连,具有抗HSV 的活性。
T6677 Sophocarpine

ERK; p38 MAPK; NF-κB; TLR; COX; HER; JNK; STAT Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; MAPK; Neuroscience; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Sophocarpine 是一种从传统草药苦参中提取的重要生物碱。苦参具有抗病毒、抗肿瘤和抗炎等多种药理作用。它通过多种机制显著抑制癌细胞的生长,具有抗肿瘤活性。
T5S1598 Mulberroside C

桑皮苷 C,桑皮苷C

Antioxidant; HCV Protease Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Mulberroside C 是桑树中的主要生物活性成分之一,可抑制 HCV 复制,具有抗病毒活性。
TQ0217 Gomisin G

戈米辛G,戈米辛 G

P450; HIV Protease Metabolism; Microbiology/Virology; Proteases/Proteasome
Gomisin G 是一种有抗HIV 活性的天然产物。
T2212 Geniposide

栀子苷,京尼平甙

Beta Amyloid; Influenza Virus Microbiology/Virology; Neuroscience
Geniposide 是从栀子花中提取的一种环烯醚萜甙,具有如神经保护、抗糖尿病、抗增殖和抗氧化多种生物活性。 它可调节 Nrf2 易位。
T2926 Schizandrin A

P450; Virus Protease; Autophagy Autophagy; Metabolism; Microbiology/Virology
Schisandrin A 是一种从东方药物五味子中提取的主要有效成分,抑制 CYP3A 活性,IC50 分别为 6.60 μM 和 Ki 为 5.83 μM。
T4S1335 Daphnoretin

Dephnoretin,西瑞香素,Thymelol

Influenza Virus; Caspase; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
Daphnoretin (Thymelol) 是从了哥王中提取得到的一种天然产物,具有抗癌和抗病毒活性。它通过在 G2/M 期连续阻断细胞并激活 caspase-3 通路导致 HOS 细胞死亡。
T6S0232 Eriodictyol

圣草酚,Huazhongilexone

Influenza Virus; DNA/RNA Synthesis; Nrf2; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology
Eriodictyol (Huazhongilexone) 是从中草药中得到的一种黄酮类天然产物,具有抗氧化、抗炎和抗糖尿病作用。它还是一种流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 18 nM。它可诱导Nrf2信号通路。
T10835 Cletoquine

Desethylhydroxychloroquine

Parasite; Antifection Microbiology/Virology
Cletoquine 是 Hydroxychloroquine 的主要活性代谢物。 Cletoquine 具有对抗基孔肯雅病毒 (CHIKV) 的能力。 Cletoquine 具有抗疟作用,并具有治疗自身免疫性疾病的潜力。
T3750 4-Hydroxyacetophenone

对羟基苯乙酮,4-Acetylphenol,Piceol,p-Acetylphenol,4'-Hydroxyacetophenone

HBV; Xanthine Oxidase Metabolism; Microbiology/Virology
4-Hydroxyacetophenone (4-Acetylphenol) 是蒿属植物和木香属植物中的一种黄嘌呤氧化酶抑制剂,具有保肝促胆、抗乙型肝炎病毒和抗炎作用。
T0122 Bergenin

Cuscutin,Bengenin,岩白菜素

Apoptosis; IL Receptor; Virus Protease; TNF; NF-κB; Antibacterial; NOD; Autophagy; Antifungal Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology; NF-κB
Bergenin (Bengenin) 是一种在许多药用植物中发现的多酚,有细胞保护和抗氧化作用。它还具有广泛的保肝、抗炎、抗肿瘤、抗病毒、抗真菌以及免疫调节作用。
T13229 Tunicamycin

Influenza Virus; Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Tunicamycin 是一种抗生素的混合物,通过阻断 GlcNAc 磷酸转移酶 (GPT),抑制 N-连接糖基化。Tunicamycin 具有抗肿瘤活性,还具有抗细菌、抗真菌和抗病毒活性。
T3273 Bifendate

联苯双酯,Bifendatatum

HBV; Reverse Transcriptase Microbiology/Virology
Bifendate (Bifendatatum) 是 Schisandrin C 的合成中间体,在慢性 B 型肝炎的研究中具有抗HBV 功效,用于治疗病毒性肝炎和药物性肝损伤引起的转氨酶升高。
TN1025 3,29-O-Dibenzoyloxykarounidiol

Others Others
3,29-O-Dibenzoyloxykarounidiol 是一种苯甲酸三萜烯酯,从 Momordica grosvenori 果实中提取。它能够抑制肿瘤启动子 TPA 诱导的 EB 病毒早期抗原活化。
T0433 Artesunate

WR-256283,青蒿琥酯

Virus Protease; Ferroptosis; STAT; Parasite Apoptosis; JAK/STAT signaling; Microbiology/Virology; Stem Cells
Artesunate (WR-256283) 是治疗疟疾的青蒿素组药物的一部分。 它是青蒿素的半合成衍生物,具有水溶性。
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天然产物

Punicalin
Cat.No: T4S1718
Synonym:
Target: HBV, HIV Protease
Tetrahydroepiberberine
Cat.No: T8187
Synonym:
Target: Others, Influenza Virus, Antifungal
Chamaechromone
Cat.No: TN1482
Synonym:
Target: P450, HBV
Paederoside
Cat.No: T3S0872
Synonym:
Target: Antiviral, HBV
Cephaeline hydrochloride
Cat.No: T3S1852
Synonym:
Target: Others, Virus Protease, Influenza Virus
Diphyllin
Cat.No: TN1103
Synonym: 山荷叶素,二叶草素
Target: ATPase, Proton pump, Influenza Virus, HIV Protease
Germacrone
Cat.No: T2945
Synonym:
Target: P450, Antiviral, Influenza Virus
Coumarin
Cat.No: T0775
Synonym:
Target: Factor Xa, Influenza Virus
Dendrobine
Cat.No: T5S1708
Synonym:
Target: Others, Influenza Virus
Alisol F
Cat.No: TQ0248
Synonym: 泽泻醇 F,泽泻醇F
Target: HBV
Isomangiferin
Cat.No: T3905
Synonym: 芒果
Target: Free radical scavengers, Antiviral, Influenza Virus
Isookanin
Cat.No: TN1788
Synonym:
Target: Amylase
Catalpol
Cat.No: T2780
Synonym: 梓醇,Catalpinoside,Digitalis purpurea L
Target: Others, HBV
Theaflavin
Cat.No: T7602
Synonym:
Target: Influenza Virus, Endogenous Metabolite
Psoralen
Cat.No: T2942
Synonym: Ficusin,Furocoumarin,补骨脂素,psoralene
Target: Apoptosis, Influenza Virus, HIV Protease, DNA/RNA Synthesis
zerumbone
Cat.No: T5712
Synonym: 花薑酮,球姜酮
Target: Antioxidant, HSV
Cephaeline
Cat.No: TN1480
Synonym: 吐根鹼,吐根酚碱
Target: Virus Protease, Influenza Virus, HIF
Dehydroandrographolide succinate
Cat.No: T2S0257
Synonym:
Target: Others, Influenza Virus
Xanthohumol
Cat.No: T3342
Synonym:
Target: Apoptosis, Others, Influenza Virus, COX, Acyltransferase, HSV
Eleutheroside B1
Cat.No: TN2331
Synonym: 刺五加苷B1
Target: Influenza Virus
Tripterifordin
Cat.No: TN2283
Synonym:
Target: HIV Protease
Anthraquinone
Cat.No: TMO2787
Synonym: dioxoanthracene,Anthradione,anthracenedione,蒽醌
Target: Virus Protease
Aloperine
Cat.No: T6377
Synonym:
Target: Apoptosis, Virus Protease, HIV Protease, Antibiotic, Autophagy
Dehydroandrographolide
Cat.No: T2738
Synonym:
Target: NOS, Influenza Virus
Arctigenin
Cat.No: T2957
Synonym: 牛蒡苷元,牛蒡子苷元,(-)-Arctigenin
Target: Apoptosis, MMP, Influenza Virus, Autophagy
Dipotassium glycyrrhizinate
Cat.No: T5666
Synonym:
Target: Virus Protease
Phillyrin
Cat.No: T2854
Synonym: Forsythin,连翘苷
Target: P450, Influenza Virus, AMPK
Ivermectin
Cat.No: T1131
Synonym: MK-933,伊维菌素
Target: Mitophagy, GluCls, P2X Receptor, SARS-CoV, HIV Protease, Antibiotic, Parasite, Autophagy, HSV
Glycyrrhizic acid
Cat.No: T2741
Synonym: Glycyrrhizin,甘草酸
Target: Virus Protease, Dehydrogenase, MAO
Angelicin
Cat.No: T2875
Synonym: Isopsoralen,异补骨脂素
Target: Apoptosis, Virus Protease, Antiviral
Chebulagic acid
Cat.No: TQ0180
Synonym:
Target: SARS-CoV, Influenza Virus, Lipoxygenase, COX
Harringtonine
Cat.No: T8286
Synonym: 三尖杉酯碱,三尖杉脂碱
Target: Others, Influenza Virus
Theaflavin 3,3'-digallate
Cat.No: T5429
Synonym: 茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG
Target: Virus Protease, Antioxidant, HIV Protease, HSV
Palmatine chloride
Cat.No: T2718
Synonym:
Target: Others, Indoleamine 2,3-Dioxygenase (IDO), Aurora Kinase
Palmatine
Cat.No: T5S0802
Synonym: 巴马汀,Berbericinine,Burasaine
Target: Indoleamine 2,3-Dioxygenase (IDO), AChR, AChE, Aurora Kinase
Guanosine
Cat.No: T6523
Synonym: 鸟苷,DL-Guanosine,Vernine,Guanozin
Target: Endogenous Metabolite, HSV
Sophocarpine
Cat.No: T6677
Synonym:
Target: ERK, p38 MAPK, NF-κB, TLR, COX, HER, JNK, STAT
Mulberroside C
Cat.No: T5S1598
Synonym: 桑皮苷 C,桑皮苷C
Target: Antioxidant, HCV Protease
Gomisin G
Cat.No: TQ0217
Synonym: 戈米辛G,戈米辛 G
Target: P450, HIV Protease
Geniposide
Cat.No: T2212
Synonym: 栀子苷,京尼平甙
Target: Beta Amyloid, Influenza Virus
Schizandrin A
Cat.No: T2926
Synonym:
Target: P450, Virus Protease, Autophagy
Daphnoretin
Cat.No: T4S1335
Synonym: Dephnoretin,西瑞香素,Thymelol
Target: Influenza Virus, Caspase, PKC
Eriodictyol
Cat.No: T6S0232
Synonym: 圣草酚,Huazhongilexone
Target: Influenza Virus, DNA/RNA Synthesis, Nrf2, Endogenous Metabolite
Cletoquine
Cat.No: T10835
Synonym: Desethylhydroxychloroquine
Target: Parasite, Antifection
4-Hydroxyacetophenone
Cat.No: T3750
Synonym: 对羟基苯乙酮,4-Acetylphenol,Piceol,p-Acetylphenol,4'-Hydroxyacetophenone
Target: HBV, Xanthine Oxidase
Bergenin
Cat.No: T0122
Synonym: Cuscutin,Bengenin,岩白菜素
Target: Apoptosis, IL Receptor, Virus Protease, TNF, NF-κB, Antibacterial, NOD, Autophagy, Antifungal
Tunicamycin
Cat.No: T13229
Synonym:
Target: Influenza Virus, Antibacterial, Antibiotic, Antifungal
Bifendate
Cat.No: T3273
Synonym: 联苯双酯,Bifendatatum
Target: HBV, Reverse Transcriptase
3,29-O-Dibenzoyloxykarounidiol
Cat.No: TN1025
Synonym:
Target: Others
Artesunate
Cat.No: T0433
Synonym: WR-256283,青蒿琥酯
Target: Virus Protease, Ferroptosis, STAT, Parasite
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