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465

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T38514 PMEDAP

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
PMEDAP 是有效的人类免疫缺陷病毒 (HIV) 复制抑制剂。它具有抗小鼠巨细胞病毒活性。它有效抑制莫罗尼鼠肉瘤病毒诱导的肿瘤形成和相关死亡率。
T11539 HCV-IN-29

HCV Protease Microbiology/Virology; Proteases/Proteasome
HCV-IN-29 是一种丙型肝炎病毒抑制剂。
T38237 2′-O-Methylcytidine

Nucleoside Antimetabolite/Analog; HCV Protease Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
2'-O-Methylcytidine 是 2'-代核苷,可抑制 HCV 复制。 它在体外抑制 NS5B 催化的 RNA 合成,其抑制方式是与底物核苷三磷酸竞争。
T11541 HCV-IN-30

Others; HCV Protease Microbiology/Virology; Others; Proteases/Proteasome
HCV-IN-30 是 HCV NS5A 复制复合物的抑制剂(基因型 1a 和 1b 复制子的 IC50 = 901 和 102 nM)。
T14495 Baloxavir

Baloxavir acid,S-033447

Influenza Virus Microbiology/Virology
Baloxavir (S-033447) 是衍生自前药 Baloxavir marboxil,是流感病毒聚合酶 PA 亚基的一流帽依赖性核酸内切酶抑制剂。它抑制病毒 RNA 的转录和复制,具有强大的抗病毒活性。
T9212 IMB-301

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
IMB-301是根据 hA3G 模型通过虚拟筛选的一种小分子抑制剂。
T8354 Triazavirin

Nucleoside Antimetabolite/Analog; Influenza Virus; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Triazavirin 是一种核酸的核苷类似物和抗病毒剂,通过抑制病毒 RNA 和 DNA 的合成以及基因组片段的复制而起作用。在流感传播阶段,它可作为保护剂。
T8371 ML188

Virus Protease; SARS-CoV Microbiology/Virology
ML188是一种选择性非共价 SARS-CoV3CLpro 抑制剂,具有抗病毒活性,IC50为 1.5 μM。
T6738 Z-FA-FMK

SARS-CoV; Cysteine Protease Microbiology/Virology; Proteases/Proteasome
Z-FA-FMK 是一种广谱的卤代甲基酮抑制剂,可抑制冠状病毒蛋白酶3CL,Ki 为 25.7 μM。它可以不可逆地抑制半胱氨酸蛋白酶,也可以抑制效应半胱天冬酶。
T11669 IR415

HBV Microbiology/Virology
IR415 选择性地与 HBx 相互作用 (Kd=2 nM) 并阻断 HBV 介导的 RNAi 抑制,逆转 HBx 蛋白对 Dicer 核糖核酸内切酶活性的抑制作用。IR415 具有抗 HBV 的活性。
T11538 Hck-IN-1

HIV Protease; Src; Hck Angiogenesis; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Hck-IN-1 是二苯基吡唑啉化合物,选择性的 Nef 依赖性 Hck 抑制剂。它是广泛的 HIV-1 Nef 直接拮抗剂,对于野生型 HIV-1 复制的IC50为 100-300 nM。它结合口袋残基 Asn126,具有抗逆转录病毒活性。
T9716 Ensitrelvir

S-217622

SARS-CoV Microbiology/Virology
Ensitrelvir (S-217622) 是首个口服有效的、非共价的、非肽的SARS-CoV-2 3CL 蛋白酶抑制剂,IC50为13 nM。
T4527 Seclidemstat

SP-2577

Histone Demethylase Chromatin/Epigenetic
Seclidemstat (SP-2577) 是非竞争性可逆KDM1A (LSD1)抑制剂,可用于尤文肉瘤的研究。它促进 SWI/SNF 复合物突变卵巢癌的抗肿瘤免疫,并抑制病毒产生、病毒 DNA 复制和晚期基因表达。
T7318 Elimusertib

BAY-1895344

ATM/ATR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Elimusertib (BAY-1895344) 是一种可口服的选择性ATR 抑制剂,IC50值为 7 nM。它具有抗肿瘤活性,可研究实体瘤和淋巴瘤。
T9350 IMP-1088

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
IMP-1088 是一种人N-肉豆蔻酰基转移酶NMT1和NMT2双重抑制剂,对 HsNMT1 和 HsNMT2 的IC50小于1 nM,对 HsNMT1 的Kd 小于210 pM。它有保护宿主细胞免受病毒感染的细胞毒作用,通过阻断鼻病毒的 N-肉豆蔻酰化蛋白来阻断鼻病毒的复制。
T0220 Foscarnet sodium

Phosphonoformate,膦甲酸钠

Virus Protease; Reverse Transcriptase; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Foscarnet sodium (Phosphonoformate) 是一种病毒 DNA 聚合酶活性抑制剂,可逆地抑制病毒复制。它是一种用于治疗巨细胞病毒性视网膜炎的抗病毒剂。
T7330 Nucleozin

[4-(2-氯-4-硝基苯基)-1-哌嗪基](5-甲基-3-苯基-4-异噁唑基)-甲酮

Influenza Virus Microbiology/Virology
Nucleozin 靶向流感 A 核蛋白,这是一种病毒复制所必需的多功能 RNA 结合蛋白。
T39477 Calcium trinatrium diethylenetriaminepentaacetic acid hydrate

Ca-DTPA trisodium salt hydrate

Others Others
Calcium trinatrium diethylenetriaminepentaacetic acid hydrate (Ca-DTPA trisodium salt hydrate) 是螯合剂和有用的解毒剂,如急性镉中毒。它是一种无毒的 CMV 复制抑制剂。
T9567 Samatasvir

ATOLIHZIXHZSBA-BTSKBWHGSA-N,IDX719

HCV Protease Microbiology/Virology; Proteases/Proteasome
Samatasvir (ATOLIHZIXHZSBA-BTSKBWHGSA-N) 是 NS5A HCV 复制抑制剂。它能够有效的选择复制子及感染性 HCV,在基因型 1至5 复制子中,EC50= 2~24 pM。
T6439 Cetylpyridinium Chloride

西吡氯铵,Cetamium,Pristacin,Hexadecylpyridinium Chloride

Others; HBV; Antibacterial Microbiology/Virology; Others
Cetylpyridinium Chloride (Hexadecylpyridinium Chloride) 是阳离子季铵,是一种广谱抗菌剂。它有效抑制 HBV 衣壳装配,IC50为 2.5 μM。它被用于杀虫剂和各种漱口水以及其他个人护理产品中。
T1623 Lopinavir

ABT-378,洛匹那韦

SARS-CoV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Lopinavir (ABT-378) 是一种选择性肽模拟 HIV-1 蛋白酶的高效抑制剂。它通过阻止 HIV-1 的成熟而起作用,从而阻断其感染性。它也是 SARS-CoV 3CLpro 的抑制剂。
T14968 Cinanserin hydrochloride

SQ 10643

Influenza Virus; 5-HT Receptor GPCR/G Protein; Microbiology/Virology; Neuroscience
Cinanserin hydrochloride (SQ 10643) 是一种高亲和力拮抗剂,对 5-HT2 受体的Ki 值为 41 nM。它也是严重急性呼吸综合征冠状病毒的 3C 样蛋白酶抑制剂。
T11281L FGI-106 tetrahydrochloride

Virus Protease; HCV Protease; Influenza Virus; HIV Protease Microbiology/Virology; Proteases/Proteasome
FGI-106 tetrahydrochloride 对多种病毒具有抑制活性,有抗埃博拉病毒,裂谷病毒和登革热病毒的 EC50分别为 100 nM,800 nM 和 400-900 nM,抑制非失血性发热病毒HCV 和HIV-1的EC50分别为 200 nM 和 150 nM 。
T7055 Bz-RS-ISer(3-Ph)-Ome

Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) 是紫杉醇衍生物,在低细胞毒性下抑制 HSV 复制周期,阻断 Vero 细胞的有丝分裂,影响 M-MSV 诱导的肿瘤大小,并通过抑制 PHA 诱导的 T 淋巴细胞增殖而影响免疫应答。
T4327 Prexasertib dihydrochloride

LY2606368 (dihydrochloride),Prexasertib HCl,LY2606368

Apoptosis; Chk; S6 Kinase Apoptosis; Cell Cycle/Checkpoint; MAPK; PI3K/Akt/mTOR signaling
Prexasertib dihydrochloride (LY2606368) 是一种选择性的,ATP 竞争性的细胞周期检测点激酶 1 抑制剂,Ki 为 0.9 nM,IC50为 <1 nM。它抑制 CHK2(IC50=8 nM) 和 RSK1 (IC50=9 nM)。它引起双链 DNA 断裂和复制突变,导致细胞凋亡,有抗肿瘤活性。
T4686 Simeprevir

TMC435,西咪匹韦,TMC-435350,Olysio

HCV Protease; SARS-CoV Microbiology/Virology; Proteases/Proteasome
Simeprevir (TMC435) 是一种有效的 HCV NS3/4A 蛋白酶抑制剂,抑制 HCV 复制,EC50 为 7.8 nM。它也是 SARS-CoV-2 3CLpro 抑制剂。
T9854 HIV-1 inhibitor-6 

3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) 是一种有效的HIV-1 pre-mRNA 选择性剪接抑制剂,可以阻断HIV 复制。
T0688 Ganciclovir

BW 759,更昔洛韦,RS-21592,2'-Nor-2'-deoxyguanosine

Nucleoside Antimetabolite/Analog; Others; Antibiotic; Antifection; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ganciclovir (2'-Nor-2'-deoxyguanosine) 是核苷类似物和口服抗病毒药物,对CMV 具有抗病毒活性。它用于治疗与艾滋病相关的巨细胞病毒感染的并发症。
T4310 Prexasertib

5-[[5-[2-(3-氨基丙氧基)-6-甲氧基苯基]-1H-吡唑-3-基]氨基]-2-吡嗪甲腈,LY2606368

Apoptosis; Chk Apoptosis; Cell Cycle/Checkpoint
Prexasertib (LY2606368) 是一种具有潜在抗肿瘤活性的检查点激酶 1 抑制剂。它可引起双链 DNA 断裂和复制突变,导致细胞凋亡。
T22337 Ganciclovir sodium

RS-21592 sodium,Cytovene IV sodium,2'-Nor-2'-deoxyguanosine sodium,BW 759 sodium,更昔洛韦钠

Nucleoside Antimetabolite/Analog; Others; Antifection; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Others
Ganciclovir sodium (Cytovene IV sodium) 是核苷类似物和口服抗病毒药物,具有抗病毒活性,尤其是针对巨细胞病毒和单纯疱疹病毒 1 型。
TQ0162 R-1479

4'-Azidocytidine

HCV Protease Microbiology/Virology; Proteases/Proteasome
R-1479 (4'-Azidocytidine) 是一种 RdRp 抑制剂,对于 HCV 亚基因组复制子系统中的 HCV RNA 复制,IC50 值为 1.28 μM。
T16088 MK-0608

HCV Protease Microbiology/Virology; Proteases/Proteasome
MK-0608 是一种可口服的体外 HCV 复制抑制剂。在亚基因组复制子测定中,EC50值为 0.3 μM,EC90值为 1.3 μM。
T1822L Clemizole hydrochloride

克立咪唑盐酸,盐酸克立咪唑

HCV Protease; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Clemizole hydrochloride 是一种 TRPC5通道的抑制剂。它还是一种 H1 组胺受体拮抗剂,抑制 HCV 复制。
T15235 Enocitabine

Nucleoside Antimetabolite/Analog; HCV Protease; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
Enocitabine 是一种核苷类似物,抑制 DNA 复制剂。Enocitabine 抑制人巨细胞病毒的复制,显示出抗白血病和抗病毒活性。
T9331 Bemnifosbuvir hemisulfate

AT-527

HCV Protease; SARS-CoV Microbiology/Virology; Proteases/Proteasome
Bemnifosbuvir hemisulfate (AT-527) 是一种 HCV 病毒复制抑制剂。
T67753 Trifluoromethyl-tubercidin

Influenza Virus Microbiology/Virology
Trifluoromethyl-tubercidin (TFMT)可抑制宿主Mtr1并抑制病毒复制。TFMT 通过其S-adenosyl-l-methionine 结合袋相互作用抑制Mtr1,限制流感病毒复制。TFMT 能有效抑制病毒在小鼠体内的复制,毒性很小。
T6244 Cidofovir

HPMPC,GS 0504,西多福韦,(S)-HPMPC

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Cidofovir ((S)-HPMPC) 通过特异性抑制病毒 DNA 合成来抑制病毒复制。
T8736 Cidofovir dihydrate

HPMPC,(S)-HPMPC,GS 0504,西多福韦二水合物

Others Others
Cidofovir dihydrate (HPMPC) 是注射型巨细胞病毒 DNA 聚合酶抑制剂,通过选择性抑制病毒 DNA 聚合酶来抑制 CMV 复制,从而阻止病毒复制和转录。
T0085 Entecavir monohydrate

SQ 34676,BMS-200475,Entecavir hydrate,恩替卡韦 (1水合物),恩替卡韦一水合物

HBV Microbiology/Virology
Entecavir monohydrate (BMS-200475) 是一种选择性HBV 抑制剂,在HepG2细胞中的EC50值为3.75 nM。
T1095 Sparfloxacin

AT-4140,PD 131501,Zagam,司帕沙星,CI-978

DNA gyrase; Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Sparfloxacin (CI-978) 是一种氟喹诺酮类抗菌素。
T0711 Niclosamide

BAY2353,Niclocide,氯硝柳胺

Antibiotic; STAT; Parasite JAK/STAT signaling; Microbiology/Virology; Stem Cells
Niclosamide (Niclocide) 是一种口服生物可利用的氯化水杨酰苯胺。它通过抑制 DNA 复制,具有驱虫和潜在的抗肿瘤活性。
T35719 T2AA

T2AA,4-[4-[(2S)-2-amino-3-hydroxypropyl]-2,6-diiodophenoxy]phenol,ZINC95605533

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
T2AA (4-[4-[(2S)-2-amino-3-hydroxypropyl]-2,6-diiodophenoxy]phenol) 是一种增殖细胞核抗原 (PCNA) 抑制剂,对 PCNA/PIP-box 肽相互作用的 IC50 为 1 μM。 T2AA 通过停止 DNA 复制叉和抑制 PCNA 与 DNA 聚合酶 δ 的相互作用来引起 DNA 复制压力并抑制癌细胞生长。
T4311 HAMNO

NSC111847

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
HAMNO (NSC-111847) 是一种复制蛋白 A 的新型蛋白质相互作用抑制剂。
T1822 Clemizole

克立咪唑,吡咯咪唑

HCV Protease; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Clemizole 是一种 H1 组胺受体拮抗剂,可抑制 NS4B 的 RNA 结合和丙型肝炎病毒复制。它也是TRP5通道抑制剂。
T3117 Marbofloxacin

马波沙星,Marbofloxacine,Zeniquin,Marbocyl

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Marbofloxacin (Zeniquin) 是一种具有口服活性的氟喹诺酮类广谱抗菌剂。它可研究革兰氏阳性和革兰氏阴性细菌以及支原体引起的感染。
T11025 hDHODH-IN-3

DHODH-IN-2

Dehydrogenase Metabolism
hDHODH-IN-3 是人二氢乳清酸脱氢酶的抑制剂,pMIC50 值为 8.6。 hDHODH-IN-3 可以抑制麻疹病毒的复制。
T4536 Pleconaril

VP 63843,Win 63843,Picovir,普可那利

Virus Protease; Antiviral Immunology/Inflammation; Microbiology/Virology
Pleconaril (VP 63843) 是一种有潜力研究肠病毒的衣壳抑制剂,, 它可有效抑制复制, IC50值为 50 nM。
T10343 AOH1160

N-(2-Oxo-2-(2-phenoxyphenylamino)ethyl)-1-naphthamide

Apoptosis; DNA/RNA Synthesis Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair
AOH1160 是增殖细胞核抗原 (PCNA) 的抑制剂。 AOH1160 通过干扰 DNA 复制导致细胞周期停滞并诱导细胞凋亡。
T1087 Valacyclovir hydrochloride

Valaciclovir hydrochloride,盐酸伐昔洛韦,盐酸万乃洛韦,Valaciclovir HCl

DNA/RNA Synthesis; Antibiotic; HSV Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Valacyclovir hydrochloride (Valaciclovir hydrochloride) 是一种口服有效的抗病毒药物,能抑制疱疹 B,单纯疱疹和带状疱疹。它抑制 HSV-1W,IC50为2.9 μg/ml。它是 Aciclovir 的前药。
T0425L Pefloxacin Mesylate Dihydrate

Pefloxacinium mesylate dihydrate,1589 RB,甲磺酸培氟沙星二水合物

Topoisomerase; Antibacterial; Antibiotic DNA Damage/DNA Repair; Microbiology/Virology
Pefloxacin Mesylate Dihydrate (1589 RB) 是一种抗菌素,能通过抑制DNA 旋转酶阻断细菌DNA 复制。

化合物

PMEDAP
Cat.No: T38514
Synonym:
Target: Others, HIV Protease
HCV-IN-29
Cat.No: T11539
Synonym:
Target: HCV Protease
2′-O-Methylcytidine
Cat.No: T38237
Synonym:
Target: Nucleoside Antimetabolite/Analog, HCV Protease
HCV-IN-30
Cat.No: T11541
Synonym:
Target: Others, HCV Protease
Baloxavir
Cat.No: T14495
Synonym: Baloxavir acid,S-033447
Target: Influenza Virus
IMB-301
Cat.No: T9212
Synonym:
Target: Others, HIV Protease
Triazavirin
Cat.No: T8354
Synonym:
Target: Nucleoside Antimetabolite/Analog, Influenza Virus, DNA/RNA Synthesis
ML188
Cat.No: T8371
Synonym:
Target: Virus Protease, SARS-CoV
Z-FA-FMK
Cat.No: T6738
Synonym:
Target: SARS-CoV, Cysteine Protease
IR415
Cat.No: T11669
Synonym:
Target: HBV
Hck-IN-1
Cat.No: T11538
Synonym:
Target: HIV Protease, Src, Hck
Ensitrelvir
Cat.No: T9716
Synonym: S-217622
Target: SARS-CoV
Seclidemstat
Cat.No: T4527
Synonym: SP-2577
Target: Histone Demethylase
Elimusertib
Cat.No: T7318
Synonym: BAY-1895344
Target: ATM/ATR
IMP-1088
Cat.No: T9350
Synonym:
Target: Others, DNA/RNA Synthesis
Foscarnet sodium
Cat.No: T0220
Synonym: Phosphonoformate,膦甲酸钠
Target: Virus Protease, Reverse Transcriptase, DNA/RNA Synthesis
Nucleozin
Cat.No: T7330
Synonym: [4-(2-氯-4-硝基苯基)-1-哌嗪基](5-甲基-3-苯基-4-异噁唑基)-甲酮
Target: Influenza Virus
Calcium trinatrium diethylenetriaminepentaacetic acid hydrate
Cat.No: T39477
Synonym: Ca-DTPA trisodium salt hydrate
Target: Others
Samatasvir
Cat.No: T9567
Synonym: ATOLIHZIXHZSBA-BTSKBWHGSA-N,IDX719
Target: HCV Protease
Cetylpyridinium Chloride
Cat.No: T6439
Synonym: 西吡氯铵,Cetamium,Pristacin,Hexadecylpyridinium Chloride
Target: Others, HBV, Antibacterial
Lopinavir
Cat.No: T1623
Synonym: ABT-378,洛匹那韦
Target: SARS-CoV, HIV Protease
Cinanserin hydrochloride
Cat.No: T14968
Synonym: SQ 10643
Target: Influenza Virus, 5-HT Receptor
FGI-106 tetrahydrochloride
Cat.No: T11281L
Synonym:
Target: Virus Protease, HCV Protease, Influenza Virus, HIV Protease
Bz-RS-ISer(3-Ph)-Ome
Cat.No: T7055
Synonym: Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate
Target: Others, HIV Protease
Prexasertib dihydrochloride
Cat.No: T4327
Synonym: LY2606368 (dihydrochloride),Prexasertib HCl,LY2606368
Target: Apoptosis, Chk, S6 Kinase
Simeprevir
Cat.No: T4686
Synonym: TMC435,西咪匹韦,TMC-435350,Olysio
Target: HCV Protease, SARS-CoV
HIV-1 inhibitor-6 
Cat.No: T9854
Synonym: 3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-
Target: HIV Protease
Ganciclovir
Cat.No: T0688
Synonym: BW 759,更昔洛韦,RS-21592,2'-Nor-2'-deoxyguanosine
Target: Nucleoside Antimetabolite/Analog, Others, Antibiotic, Antifection, HSV
Prexasertib
Cat.No: T4310
Synonym: 5-[[5-[2-(3-氨基丙氧基)-6-甲氧基苯基]-1H-吡唑-3-基]氨基]-2-吡嗪甲腈,LY2606368
Target: Apoptosis, Chk
Ganciclovir sodium
Cat.No: T22337
Synonym: RS-21592 sodium,Cytovene IV sodium,2'-Nor-2'-deoxyguanosine sodium,BW 759 sodium,更昔洛韦钠
Target: Nucleoside Antimetabolite/Analog, Others, Antifection, HSV
R-1479
Cat.No: TQ0162
Synonym: 4'-Azidocytidine
Target: HCV Protease
MK-0608
Cat.No: T16088
Synonym:
Target: HCV Protease
Clemizole hydrochloride
Cat.No: T1822L
Synonym: 克立咪唑盐酸,盐酸克立咪唑
Target: HCV Protease, Histamine Receptor
Enocitabine
Cat.No: T15235
Synonym:
Target: Nucleoside Antimetabolite/Analog, HCV Protease, DNA/RNA Synthesis
Bemnifosbuvir hemisulfate
Cat.No: T9331
Synonym: AT-527
Target: HCV Protease, SARS-CoV
Trifluoromethyl-tubercidin
Cat.No: T67753
Synonym:
Target: Influenza Virus
Cidofovir
Cat.No: T6244
Synonym: HPMPC,GS 0504,西多福韦,(S)-HPMPC
Target: Others, DNA/RNA Synthesis
Cidofovir dihydrate
Cat.No: T8736
Synonym: HPMPC,(S)-HPMPC,GS 0504,西多福韦二水合物
Target: Others
Entecavir monohydrate
Cat.No: T0085
Synonym: SQ 34676,BMS-200475,Entecavir hydrate,恩替卡韦 (1水合物),恩替卡韦一水合物
Target: HBV
Sparfloxacin
Cat.No: T1095
Synonym: AT-4140,PD 131501,Zagam,司帕沙星,CI-978
Target: DNA gyrase, Topoisomerase, Antibacterial, Antibiotic
Niclosamide
Cat.No: T0711
Synonym: BAY2353,Niclocide,氯硝柳胺
Target: Antibiotic, STAT, Parasite
T2AA
Cat.No: T35719
Synonym: T2AA,4-[4-[(2S)-2-amino-3-hydroxypropyl]-2,6-diiodophenoxy]phenol,ZINC95605533
Target: DNA/RNA Synthesis
HAMNO
Cat.No: T4311
Synonym: NSC111847
Target: DNA/RNA Synthesis
Clemizole
Cat.No: T1822
Synonym: 克立咪唑,吡咯咪唑
Target: HCV Protease, Histamine Receptor
Marbofloxacin
Cat.No: T3117
Synonym: 马波沙星,Marbofloxacine,Zeniquin,Marbocyl
Target: Topoisomerase, Antibacterial, Antibiotic
hDHODH-IN-3
Cat.No: T11025
Synonym: DHODH-IN-2
Target: Dehydrogenase
Pleconaril
Cat.No: T4536
Synonym: VP 63843,Win 63843,Picovir,普可那利
Target: Virus Protease, Antiviral
AOH1160
Cat.No: T10343
Synonym: N-(2-Oxo-2-(2-phenoxyphenylamino)ethyl)-1-naphthamide
Target: Apoptosis, DNA/RNA Synthesis
Valacyclovir hydrochloride
Cat.No: T1087
Synonym: Valaciclovir hydrochloride,盐酸伐昔洛韦,盐酸万乃洛韦,Valaciclovir HCl
Target: DNA/RNA Synthesis, Antibiotic, HSV
Pefloxacin Mesylate Dihydrate
Cat.No: T0425L
Synonym: Pefloxacinium mesylate dihydrate,1589 RB,甲磺酸培氟沙星二水合物
Target: Topoisomerase, Antibacterial, Antibiotic
Cat. No. Product Name Target Signaling Pathways
TN2283 Tripterifordin

HIV Protease Microbiology/Virology; Proteases/Proteasome
Tripterifordin 在 H9 淋巴细胞中显示出抗 HIV 复制活性,EC50值为 3100 nM。
T1068 Dithranol

1,8,9-trihydroxyanthracene,cignoline,蒽林,Anthralin

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Dithranol (cignoline) 是蒽醌衍生物,可破坏线粒体功能和结构,用于治疗皮肤病。
TWP2911 Thymidine

beta-胸苷,5-Methyldeoxyuridine,Deoxyribothymidine,DThyd,NSC 21548,Thymidin

Others; DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Others
Thymidine (DThyd) 是一种细胞同步剂,是脱氧核糖核酸的特殊前体。它可在 DNA 复制前在 G1/S 边界阻滞细胞,是DNA 合成抑制因子。
T6S2391 L-Chicoric Acid

(-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸,是一种选择性可逆的 HIV-1 整合酶抑制剂,IC50约为 100 nM。它还可抑制 HIV-1 复制。
T5429 Theaflavin 3,3'-digallate

茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG

Virus Protease; Antioxidant; HIV Protease; HSV Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。
T4850 PCL 016

2-吡啶甲酸,2-Picolinic acid

Virus Protease; Endogenous Metabolite Metabolism; Microbiology/Virology
PCL 016 (2-Picolinic acid) 是一种局部抗病毒剂,可抑制兔体内的腺病毒复制。
T2143 Bergapten

5-Methoxypsoralen,佛手柑内酯,香柑内酯

P450; Autophagy Autophagy; Metabolism
Bergapten (5-Methoxypsoralen) 是白芷中的一种香豆素,也是一种补骨脂素,可抑制细胞复制。
T7607 PSI-6130

R 1656,2'-去氧-2'-氟-2'-C-甲基胞苷

HCV Protease Microbiology/Virology; Proteases/Proteasome
PSI-6130 (R 1656) 是高效选择性 HCV NS5B 聚合酶抑制剂,抑制 HCV 复制,IC50值为 0.6 μM。
TL0006 Cichoric Acid

菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。
T40834 5-Hydroxymethyl-2'-deoxycytidine

5hmdC,2'-脱氧-5-(羟甲基)胞啶

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
5-Hydroxymethyl-2'-deoxycytidine 是 DNA 中 5-methyl-2'-deoxycytidine (5-mdC) 的氧化衍生物,引起DNA损伤反应,染色体畸变,复制叉损伤和细胞活力丧失。5-Hydroxymethyl-2’-deoxycytidine 复制叉不稳定性与染色质上聚(ADP-核糖)聚合酶1(PARP1)的存在有关。
T37635 2'-Deoxyadenosine-5'-triphosphate trisodium

dATP trisodium

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
2'-Deoxyadenosine-5'-triphosphate trisodium (dATP trisodium) 是一种核苷酸,是 DNA 聚合酶的底物,在细胞中用于 DNA 合成或复制。
T4S1521 1,4-Dicaffeoylquinic acid

1,4-二咖啡酰奎宁酸,洋蓟素

HIV Protease Microbiology/Virology; Proteases/Proteasome
1,4-Dicaffeoylquinic acid 是一种苯丙素类物质,从苍耳子中获得,可以减少 LPS 诱导的 TNF-α 的生成,具有抗炎活性。
T1511 Daunorubicin hydrochloride

Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin

Apoptosis; DNA/RNA Synthesis; Topoisomerase; Antibacterial; Antibiotic; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Daunorubicin hydrochloride (Rubidomycin hydrochloride) 是一种蒽环类氨基糖苷类抗肿瘤药物,可抑制 DNA 复制和修复以及 RNA 和蛋白质合成。
T3905 Isomangiferin

芒果

Free radical scavengers; Antiviral; Influenza Virus Immunology/Inflammation; Microbiology/Virology; oxidation-reduction
Isomangiferin 是一种天然产物,具有抗病毒的作用。它还具有抗氧化和自由基清除活性。
TN1068 Tricin

Others; CDK Cell Cycle/Checkpoint; Others
Tricin 是米糠中大量存在的一种天然类黄酮。它通过抑制 CDK9 来抑制HCMV 的复制。它通过上调 FAK 靶向 microRNA-7 的表达来抑制 C6 胶质瘤细胞的增殖和侵袭。
T7004 Tubercidin

结核菌素,杀结核菌素,Sparsomycin A,7-Deazaadenosine

Influenza Virus; DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Tubercidin (Sparsomycin A) 是从Streptomyces tubercidicus 得到的抗生素,抑制粪链球菌生长的IC50值为 0.02 μM。它是腺苷磷酸化酶的弱抑制剂,并干扰腺苷和 AMP 的磷酸化。它有抗病毒作用。
T1591 Ancitabine hydrochloride

NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C

Others; DNA/RNA Synthesis; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Ancitabine hydrochloride (NSC 145668 HCl) 是一种天然的抗白血病药物。
T40179 Sodium Camptothecin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Sodium Camptothecin 是一种植物生物碱,具有抗肿瘤活性。它是可逆 RNA 合成抑制剂,可以抑制腺病毒的复制。它能抑制 DNA 合成,并引起细胞内预形成的病毒 DNA 断裂。
T4S1335 Daphnoretin

Dephnoretin,西瑞香素,Thymelol

Influenza Virus; Caspase; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome
Daphnoretin (Thymelol) 是从了哥王中提取得到的一种天然产物,具有抗癌和抗病毒活性。它通过在 G2/M 期连续阻断细胞并激活 caspase-3 通路导致 HOS 细胞死亡。
T7961 N4-Benzoyl-2′-deoxycytidine

N-苯甲酰-2'-脱氧胞苷

Others Others
N4-Benzoyl-2′-deoxycytidine 是天然核苷脱氧胞苷(dC)的合成核苷类似物,是一种DNA 聚合酶的竞争性抑制剂。体外研究表明,它可以抑制病毒、细菌和真核细胞的复制。在动物模型中,它也被证明可以抑制肿瘤细胞的生长。
T0884 1-Docosanol

Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol

Antifection; HSV Microbiology/Virology
1-Docosanol (Behenic alcohol) 是一种具有抗病毒活性的饱和 22 碳脂肪醇,局部用于治疗复发性单纯性唇疱疹发作并缓解相关疼痛并可能有助于更快地治愈疮。
TN3500 beta-Amyrone

β-Amyron,β-香树脂酮

COX; AChR; PPAR; Antifection DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; Neuroscience
beta-Amyrone (β-Amyron) 对基孔肯雅病毒复制具有抗真菌活性,EC50 为 86 uM。 beta-Amyrone 通过抑制 COX-2 的表达而具有抗炎活性。 beta-Amyrone 表现出抗α-葡萄糖苷酶抑制活性和中等 AChE 活性。 β-Amyrone 可用于炎症、感染和肥胖等疾病的研究。
T35455 N-Nitrosodiethylamine

Diethylnitrosamine,NDEA

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
N-Nitrosodiethylamine (NDEA) 是致癌物质二烷基硝胺。它主要存在于水、烟草烟雾、腌制食品、油炸食品以及许多酒精饮料中。它与 DNA 修复/复制相关的核酶的变化相关。
T0486L Irinotecan Hydrochloride

盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride

Topoisomerase; Autophagy Autophagy; DNA Damage/DNA Repair
Irinotecan Hydrochloride (CPT-11 hydrochloride) 是喜树碱半合成衍生物的盐酸盐,是一种拓扑异构酶 I 抑制剂,可研究结肠癌和直肠癌。
T2973 Astragaloside IV

AST-IV,黄芪甲苷IV,AS-IV,黄芪皂苷 IV

MMP; ERK; Estrogen/progestogen Receptor; JNK Endocrinology/Hormones; MAPK; Proteases/Proteasome
Astragaloside IV (AS-IV) 是从黄芪中分离得到的一种皂苷,抑制ERK1/2和JNK 激活,在乳腺癌细胞 MDA-MB-231 中,下调(MMP)-2和(MMP)-9的信号通路。
T21251 OSW-1

OSW1

OSW-1 is a natural broad-range inhibitor to inhibits replication of enterovirus.
TN1668 Ganoderic acid Y

灵芝酸Y

Antifection Microbiology/Virology
Ganoderic acid Y significantly inhibits the replication of the viral RNA (vRNA) of EV71 replication through blocking EV71 uncoating.
T26953 Carubicin hydrochloride

NSC 275649,Karminomycin hydrochloride,Carubicin HCl

Carubicin HCl is an anthracycline antineoplastic antibiotic. Through intercalates into DNA and interacts with topoisomerase II, Carubicin inhibits DNA replication and repair and RNA and protein synthesis.
TN1767 InteriotherinA

Interiotherin A,内南五味子酯A

HIV Protease Microbiology/Virology; Proteases/Proteasome
Interiotherin A inhibits HIV replication with the EC50 value of 3.1 micrograms/mL.
T26111 Robustaflavone

Robustaflavone is a naturally occurring biflavanoid isolated from Rhus succedanea and is a hepatitis B virus replication inhibitor.
T21328 Carubicin

carminomycin,Carminomycin I,Carminomicin I,Antibiotic R 588A,Demethyldaunomycin

Carubicin is an anthracycline antineoplastic antibiotic isolated from the bacterium Actinomadura carminata. Carubicin intercalates into DNA and interacts with topoisomerase II, thereby inhibiting DNA replication and repair and RNA and protein synthesis.
TN6395 Citrusin B

Citrusin B exhibits moderate in vitro inhibitory effect on tobacco mosaic virus replication with IC50 values 0.26 mmol L⁻1.
TN2231 Soyasaponin II

Influenza Virus; HIV Protease; HSV Microbiology/Virology; Proteases/Proteasome
Soyasaponin II has antiviral effects, it can inhibit the replication of human cytomegalovirus, influenza virus, and human immunodeficiency virus type 1.
TN4646 Neotripterifordin

HIV Protease Microbiology/Virology; Proteases/Proteasome
Neotripterifordin shows potent anti-HIV replication activity in H9 lymphocyte cells with an EC50 of 25 nM and TI of 125.
T17270 Yatein

Others Others
Yatein inhibits herpes simplex virus type 1 replication by interruption the immediate-early gene expression. Yatein is a lignan isolated from A. chilensis. It also has antiproliferative activity.
TN3809 Dehydrojuncusol

HCV Protease Microbiology/Virology; Proteases/Proteasome
Dehydrojuncusol, a new inhibitor of hepatitis C virus RNA replication, it inhibits infection of different HCV genotypes by targeting the NS5A protein and is active against resistant HCV variants frequently found in patients with treatment failure.
TN4934 Salaspermic acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
Salaspermic acid is an inhibitor of HIV reverse transcriptase and HIV replication in H9 lymphocyte cells.
TN1632 Euparin

Antifection Microbiology/Virology
Euparin exhibits a moderate antioxidant activity, it also exhibits antifungal activity against Trichophyton mentagrophytes. Euparin has antiviral activity, it exerts its effect during the early events of the replication cycle, from the virus adsorption to
T16719 Radicicol

根赤壳菌素,Monorden

HSP Cytoskeletal Signaling; Metabolism
Radicicol is an antifungal antibiotic, impairs mitochondrial replication by targeting P. falciparum topoisomerase VIB. Radicicol is an inhibitor of Hsp90 (IC50: 1 μM). Radicicol binds to the ATPase domain of Hsp90 and prevents maturation of Hsp90 clients,
TN5012 Shizukaol C

HIV Protease; Antifection Microbiology/Virology; Proteases/Proteasome
1. Shizukaol C shows anti-HIV-1 replication activities in both wild-type HIV-1 and two NNRTIs-resistant strains. <br/> 2. Shizukaol C has significant cytotoxicities against C8166 cells. <br/>
T11837 Leptomycin A

CRM1 Membrane transporter/Ion channel
Leptomycin A, a metabolite derived from Streptomyces, acts as an inhibitor of CRM1 (exportin 1) and effectively suppresses HIV-1 replication. Compared to Leptomycin B, it exhibits lesser potency. Leptomycin A hampers the interaction between CRM1 and nuclear export signals, effectively hindering the nuclear export of a wide array of proteins.
T83401 2′-O-Methylphloretin

2′-O-Methylphloretin是一种从Melodorum siamensis叶子中分离出的类黄酮衍生物,具有抑制肿瘤细胞系复制的生物活性。
TN5880 Mesuol

Mesuol has antioxidant activity, it shows very high scavenging activity against DPPH radical; it also has immunomodulatory activity, can potentiate percentage neutrophil adhesion in neutrophil adhesion test in rats and phagocytosis in carbon clearance assay. Mesuol can suppress HIV-1 replication in Jurkat T cells, it inhibits TNFα-induced HIV-1-LTR transcriptional activity by targeting the nuclear factor-κB (NF-κB) pathway.
TN6014 Norcepharadione B

鱼腥草

Norcepharadione B shows good inhibitory activity against the replication of HSV-1, it also shows antimalarial activity with EC50 values of 7.5mug/ml. Norcepharadione B exhibits significant cytotoxicity against five human tumor cell lines (A-549, SK-OV-3,
TN1194 16beta,17-Dihydroxy-ent-kaurane-19-oic acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
16beta,17-Dihydroxy-ent-kaurane-19-oic acid as an anti-HIV principle, it showed significant activity against HIV replication in H9 lymphocyte cells with an EC50 value of 0.8 microgram/mL. It also possesses the activities of decompression and blood viscosi
T38015 Herquline A

Herquline A is an alkaloid fungal metabolite originally isolated from P. herquei. It inhibits cell death induced by influenza A strain A/PR/8/34 in MDCK cells with an IC50 value of 10 μg/ml and inhibits viral replication in a plaque assay in a concentration-dependent manner. Herquline A also inhibits platelet aggregation induced by ADP and platelet-activating factor (PAF) in vitro (IC50s = 180 and 240 μM, respectively).
T73758 Glycolithocholic acid 3-sulfate

Glycolithocholic acid 3-sulfate (SLCG) 为一种胆汁酸衍生物及甘胆酸的代谢产物,具有抑制HIV-1复制的作用。该化合物在HIV感染和胆囊疾病的研究中有潜在应用价值。
T75692 Hypoglaunine D

Hypoglaunine D 是 Triptonine B 的类似物,是一种抗HIV 的化合物,Hypoglaunine D 抑制 H9 淋巴细胞中HIV 病毒复制的EC50值为 22 μg/ml。
T80002 Wulfenioidin F

Virus Protease Microbiology/Virology
Wulfenioidin F是从Orthosiphon wulfenioides全草分离的二萜类化合物。该化合物对抗寨卡病毒(ZIKV)活性显著,其半数有效浓度(EC50)为8.07 μM。Wulfenioidin F的抗病毒机制通过抑制ZIKV包膜(E)蛋白的表达,从而干扰病毒复制。
TN4490 Manassantin B

ERK; BCL; p38 MAPK; TNF; NF-κB; JNK; STAT; Antifection Apoptosis; JAK/STAT signaling; MAPK; Microbiology/Virology; NF-κB; Stem Cells
Manassantin B is a potent inhibitor of NF-κB activation by the suppression of transciptional activity of RelA/p65 subunit of NF-κB. It also possesses anti-EBV lytic replication activity. Manassantin B inhibits interleukin-6-induced signal transducer and activator of transcription 3 activation in Hep3B cells, it has potential as a potent anti-inflammatory drug for use in pathological processes such as sepsis or acute lung injury. Manassantin B exerts antifibrotic activity in HSC-T6 cells, in pa...
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天然产物

Tripterifordin
Cat.No: TN2283
Synonym:
Target: HIV Protease
Dithranol
Cat.No: T1068
Synonym: 1,8,9-trihydroxyanthracene,cignoline,蒽林,Anthralin
Target: Others, DNA/RNA Synthesis
Thymidine
Cat.No: TWP2911
Synonym: beta-胸苷,5-Methyldeoxyuridine,Deoxyribothymidine,DThyd,NSC 21548,Thymidin
Target: Others, DNA/RNA Synthesis, Endogenous Metabolite
L-Chicoric Acid
Cat.No: T6S2391
Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸
Target: Others, HIV Protease
Theaflavin 3,3'-digallate
Cat.No: T5429
Synonym: 茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG
Target: Virus Protease, Antioxidant, HIV Protease, HSV
PCL 016
Cat.No: T4850
Synonym: 2-吡啶甲酸,2-Picolinic acid
Target: Virus Protease, Endogenous Metabolite
Bergapten
Cat.No: T2143
Synonym: 5-Methoxypsoralen,佛手柑内酯,香柑内酯
Target: P450, Autophagy
PSI-6130
Cat.No: T7607
Synonym: R 1656,2'-去氧-2'-氟-2'-C-甲基胞苷
Target: HCV Protease
Cichoric Acid
Cat.No: TL0006
Synonym: 菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid
Target: Reactive Oxygen Species, HIV Protease
5-Hydroxymethyl-2'-deoxycytidine
Cat.No: T40834
Synonym: 5hmdC,2'-脱氧-5-(羟甲基)胞啶
Target: PARP
2'-Deoxyadenosine-5'-triphosphate trisodium
Cat.No: T37635
Synonym: dATP trisodium
Target: DNA/RNA Synthesis, Endogenous Metabolite
1,4-Dicaffeoylquinic acid
Cat.No: T4S1521
Synonym: 1,4-二咖啡酰奎宁酸,洋蓟素
Target: HIV Protease
Daunorubicin hydrochloride
Cat.No: T1511
Synonym: Daunomycin HCl,盐酸佐柔比星,盐酸柔红霉素,RP-13057 Hydrochloride,Rubidomycin hydrochloride,Daunorubicin HCl,Daunomycin
Target: Apoptosis, DNA/RNA Synthesis, Topoisomerase, Antibacterial, Antibiotic, Autophagy
Isomangiferin
Cat.No: T3905
Synonym: 芒果
Target: Free radical scavengers, Antiviral, Influenza Virus
Tricin
Cat.No: TN1068
Synonym:
Target: Others, CDK
Tubercidin
Cat.No: T7004
Synonym: 结核菌素,杀结核菌素,Sparsomycin A,7-Deazaadenosine
Target: Influenza Virus, DNA/RNA Synthesis, Antibacterial, Antibiotic
Ancitabine hydrochloride
Cat.No: T1591
Synonym: NSC 145668 HCl,盐酸环胞苷,Cyclocytidine hydrochloride,Cyclo-CMP hydrochloride,Cyclocytidine HCl,Cyclo-C
Target: Others, DNA/RNA Synthesis, Autophagy
Sodium Camptothecin
Cat.No: T40179
Synonym:
Target: DNA/RNA Synthesis
Daphnoretin
Cat.No: T4S1335
Synonym: Dephnoretin,西瑞香素,Thymelol
Target: Influenza Virus, Caspase, PKC
N4-Benzoyl-2′-deoxycytidine
Cat.No: T7961
Synonym: N-苯甲酰-2'-脱氧胞苷
Target: Others
1-Docosanol
Cat.No: T0884
Synonym: Behenic alcohol,Behenyl alcohol,n-Docosanol,二十二醇,Docosanol
Target: Antifection, HSV
beta-Amyrone
Cat.No: TN3500
Synonym: β-Amyron,β-香树脂酮
Target: COX, AChR, PPAR, Antifection
N-Nitrosodiethylamine
Cat.No: T35455
Synonym: Diethylnitrosamine,NDEA
Target: DNA/RNA Synthesis
Irinotecan Hydrochloride
Cat.No: T0486L
Synonym: 盐酸伊立替康,伊立替康盐酸盐,Camptothecin 11 hydrochloride,CPT-11 hydrochloride
Target: Topoisomerase, Autophagy
Astragaloside IV
Cat.No: T2973
Synonym: AST-IV,黄芪甲苷IV,AS-IV,黄芪皂苷 IV
Target: MMP, ERK, Estrogen/progestogen Receptor, JNK
OSW-1
Cat.No: T21251
Synonym: OSW1
Target:
Ganoderic acid Y
Cat.No: TN1668
Synonym: 灵芝酸Y
Target: Antifection
Carubicin hydrochloride
Cat.No: T26953
Synonym: NSC 275649,Karminomycin hydrochloride,Carubicin HCl
Target:
InteriotherinA
Cat.No: TN1767
Synonym: Interiotherin A,内南五味子酯A
Target: HIV Protease
Robustaflavone
Cat.No: T26111
Synonym:
Target:
Carubicin
Cat.No: T21328
Synonym: carminomycin,Carminomycin I,Carminomicin I,Antibiotic R 588A,Demethyldaunomycin
Target:
Citrusin B
Cat.No: TN6395
Synonym:
Target:
Soyasaponin II
Cat.No: TN2231
Synonym:
Target: Influenza Virus, HIV Protease, HSV
Neotripterifordin
Cat.No: TN4646
Synonym:
Target: HIV Protease
Yatein
Cat.No: T17270
Synonym:
Target: Others
Dehydrojuncusol
Cat.No: TN3809
Synonym:
Target: HCV Protease
Salaspermic acid
Cat.No: TN4934
Synonym:
Target: HIV Protease
Euparin
Cat.No: TN1632
Synonym:
Target: Antifection
Radicicol
Cat.No: T16719
Synonym: 根赤壳菌素,Monorden
Target: HSP
Shizukaol C
Cat.No: TN5012
Synonym:
Target: HIV Protease, Antifection
Leptomycin A
Cat.No: T11837
Synonym:
Target: CRM1
2′-O-Methylphloretin
Cat.No: T83401
Synonym:
Target:
Mesuol
Cat.No: TN5880
Synonym:
Target:
Norcepharadione B
Cat.No: TN6014
Synonym: 鱼腥草
Target:
16beta,17-Dihydroxy-ent-kaurane-19-oic acid
Cat.No: TN1194
Synonym:
Target: HIV Protease
Herquline A
Cat.No: T38015
Synonym:
Target:
Glycolithocholic acid 3-sulfate
Cat.No: T73758
Synonym:
Target:
Hypoglaunine D
Cat.No: T75692
Synonym:
Target:
Wulfenioidin F
Cat.No: T80002
Synonym:
Target: Virus Protease
Manassantin B
Cat.No: TN4490
Synonym:
Target: ERK, BCL, p38 MAPK, TNF, NF-κB, JNK, STAT, Antifection
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