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272

抑制剂 & 化合物

51

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Cat. No. Product Name Target Signaling Pathways
T14033 3BDO

Apoptosis; mTOR; Autophagy Apoptosis; Autophagy; PI3K/Akt/mTOR signaling
3BDO 是新型的mTOR 激活剂,对自噬有抑制作用。
T3514 CZ415

mTOR PI3K/Akt/mTOR signaling
CZ415 是高选择性的mTOR 抑制剂,其 pIC50=8.07。它对mTORC1和mTORC2复合体具有抑制作用。
T12123 mTOR inhibitor-3

mTOR PI3K/Akt/mTOR signaling
mTOR inhibitor-3 是有效的 mTOR 抑制剂(Ki= 1.5 nM)。在细胞实验及体内实验中,mTOR inhibitor-3 均抑制 mTORC1 和 mTORC2。
T21246 Metsulfuron-methyl

Others Others
Metsulfuron-methyl 是一种内吸传导选择性麦田高效磺酰脲类除草剂,主要防治麦田大多数阔叶杂草和禾本科杂草。
T6045 Torin 1

DNA-PK; PI3K; mTOR; Autophagy Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Torin 1 是一种有效的 mTOR 抑制剂,IC50为 3 nM。它抑制 mTORC1/2复合物的 IC50值在 2 和 10 nM 之间,还诱导自噬。
T5472 PQR620

mTOR PI3K/Akt/mTOR signaling
PQR620 是一种可透过血脑屏障的,具有口服活性的mTORC1/2选择性抑制剂。
T12270 NV-5138

mTOR PI3K/Akt/mTOR signaling
NV-5138 是一种具有选择性的、口服活性的脑内mTORC1激动剂,能够与 Sestrin2 结合。它是一种亮氨酸类似物。它可用于抗抑郁的生物研究。
T6030 XL388

P450; PI3K; mTOR Metabolism; PI3K/Akt/mTOR signaling
XL388 是高效的、 ATP 竞争性的 mTOR 抑制剂,其 IC50=9.9 nM。它能够抑制 mTORC1和 mTORC2。
T40351 MHY-1685

mTOR PI3K/Akt/mTOR signaling
MHY-1685 is a mammalian target of rapamycin (mTOR) inhibitor and a senescence inhibitor that can rejuvenate senile hCSCs by modulating autophagy.
T2475 KU-0063794

mTOR PI3K/Akt/mTOR signaling
KU0063794 是一种特异性的,有效的 mTOR 抑制剂,能够抑制 mTORC1和 mTORC2,IC50值均约为 10 nM。
T7343 PF-04979064

PI3K; mTOR PI3K/Akt/mTOR signaling
PF-04979064 是一种选择性 PI3K/mTOR 双重激酶抑制剂,能够抑制 PI3Kα (Ki=0.13 nM) 和 mTOR (Ki=1.42 nM)。
T1859 AZD-8055

Apoptosis; mTOR; Autophagy Apoptosis; Autophagy; PI3K/Akt/mTOR signaling
AZD-8055 是一种选择性、具有口服活性和 ATP 竞争性的 mTOR 抑制剂,IC50为 0.8 nM。AZD-8055 抑制 mTORC1和 mTORC2。
T5338 mTOR inhibitor-1

mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
mTOR inhibitor-1是一种新型 ATP 竞争性 mTOR 抑制剂,可抑制细胞生长和增殖,诱导自噬。
T7166 GNE-493

PI3K; mTOR PI3K/Akt/mTOR signaling
GNE-493 是选择性的PI3K/mTOR 抑制剂,能够抑制 PI3Kα (IC50:3.4 nM),PI3Kβ (IC50:12 nM),PI3Kδ (IC50:16 nM),PI3Kγ (IC50:16 nM) 和 mTOR (IC50:32 nM)。
T1908 MHY1485

mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
MHY1485 是一种 mTOR 激活剂。它通过抑制自噬体和溶酶体之间的融合来抑制自噬过程,导致 LC3II 蛋白的积累和自噬体增大。
T16355 NSC781406

PI3K; mTOR PI3K/Akt/mTOR signaling
NSC781406是一种高效PI3K 和mTOR 抑制剂,其PI3Kα的IC50值为2 nM。
T6100 Torin 2

Apoptosis; ATM/ATR; DNA-PK; mTOR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Torin 2 是一种特异性 mTOR 抑制剂,IC50值为0.25 nM,并改善了药代动力学特性。它抑制 ATM/ATR/DNA-PK 的 EC50 分别为 28 nM/35 nM/118 nM。
T16567 PQR530

PQR-530

PI3K; mTOR PI3K/Akt/mTOR signaling
PQR530 是一具有口服活性,种 ATP 竞争性的,可透过血脑屏障的 PI3K/mTORC1/2双重抑制剂,对于 PI3Kα 和 mTOR (分别为 0.84 和 0.33 nM) 的Kd 为亚摩尔。它具有抗肿瘤作用。
T1961 Vistusertib

AZD2014

Apoptosis; Akt; PI3K; S6 Kinase; mTOR; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
Vistusertib (AZD2014) 是一种ATP 竞争性的mTOR 抑制剂,IC50为 2.81 nM。它抑制mTORC1和mTORC2复合物。
T2414 Torkinib

PP 242

Apoptosis; Mitophagy; PI3K; mTOR; Autophagy Apoptosis; Autophagy; PI3K/Akt/mTOR signaling
Torkinib (PP 242) 是一种选择性,ATP 竞争型的mTOR 抑制剂,IC50为 8 nM。它也抑制mTORC1和mTORC2,IC50分别为 30 nM 和 58 nM。
T2084 ETP-46464

ATM/ATR; DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
ETP-46464 是一种有效且特异性的 ATR 抑制剂,IC50为 25 nM。
T6845 GNE-317

GNE317

PI3K; mTOR PI3K/Akt/mTOR signaling
GNE-317 是一种可透过血脑屏障 (BBB)的 PI3K/mTOR 抑制剂。
T3692 GNE-477

GNE 477

PI3K; mTOR PI3K/Akt/mTOR signaling
GNE-477 是一种高效的双重PI3K(IC50=4 nM)、mTOR(Ki=21 nM) 抑制剂。
T2357 GSK1059615

GSK 1059615,GSK-1059615

Apoptosis; PI3K; mTOR Apoptosis; PI3K/Akt/mTOR signaling
GSK1059615 是一种 PI3Kα/β/δ/γ可逆的抑制剂,同时也抑制 mTOR,IC50值分别为 0.4 nM/0.6 nM/2 nM/5 nM 和 12 nM,已用于研究淋巴瘤、实体瘤、子宫内膜癌、实体瘤癌和转移性乳腺癌治疗的试验。
T3541 CC-115

CC 115

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
CC-115 是一种双重 mTOR/DNA-PK 的抑制剂,IC50分别为 21 nM 和 13 nM,可阻断mTORC1和mTORC2信号通路。
T36083 DS-7423

PI3K; mTOR PI3K/Akt/mTOR signaling
DS-7423 是PI3K 和mTOR 的有效抑制剂,抑制PI3Kα 和 mTOR 的IC50分别为15.6 nM 和 34.9 nM。DS-7423表现出抗癌活性。
T6510 GDC-0349

RG-7603

PI3K; mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
GDC-0349 (RG-7603) 是一种ATP 竞争性的选择性mTOR 抑制剂,Ki 值为 3.8 nM。它对 PI3Kα 和其他 266 种激酶的抑制作用是 790 倍,可抑制mTORC1和mTORC2复合体。
T22339 GNE-490

Others; PI3K Others; PI3K/Akt/mTOR signaling
GNE-490 是一种有效的 pan-PI3K 抑制剂,对 PI3Kα、PI3Kβ、PI3Kδ 和 PI3Kγ 的 IC50 分别为 3.5 nM、25 nM、5.2 nM、15 nM。 GNE-490 对 mTOR 具有 >200 倍的特异性(IC50 = 750 nM)。
T6251 PF-04691502

PF4691502

Akt; PI3K; mTOR; Autophagy Autophagy; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
PF-04691502 是一种有效的选择性 PI3K 和 mTOR 激酶抑制剂,具有抗肿瘤活性。它与人 PI3Kα、β、δ、γ和 mTOR 结合的 Ki 分别为1.8、2.1、1.6、1.9和16 nM。
T6557 KU-0060648

KU0060648

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
KU-0060648 是一种 PI3K 和 DNA-PK 的双重抑制剂,对 PI3Kα、PI3Kβ、PI3Kδ、PI3Kγ 和 DNA-PK 的 IC50值分别为 4 nM、0.5 nM、0.1 nM、0.59 nM 和 8.6 nM。
T4199 Desmethyl-VS-5584

PI3K; mTOR PI3K/Akt/mTOR signaling
Desmethyl-VS-5584 是 VS-5584 的二甲基类似物。其中VS-5584 是mTOR/PI3K 抑制剂,专门针对于吡啶 [2,3-d] 嘧啶结构。
T6319 OSI-027

ASP4786,OSI027

DNA-PK; PI3K; mTOR; Autophagy Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
OSI-027 (ASP4786) 是一种选择性、可口服和 ATP 竞争性的mTOR 激酶活性抑制剂,IC50为 4 nM。它抑制mTORC1和mTORC2,IC50分别为 22 nM 和 65 nM。
T6143 PI-103

PI103,PI 103

Apoptosis; DNA-PK; PI3K; mTOR; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
PI-103 是一种 PI3K 和 mTOR 抑制剂,抑制 p110α、p110β、p110δ、p110γ、mTORC1和 mTORC2,IC50分别为 8 nM、88 nM、48 nM、150 nM、20 nM 和 83 nM。它可诱导自噬,还抑制 DNA-PK,IC50为 2 nM。
T2415 PP121

Apoptosis; VEGFR; Bcr-Abl; PDGFR; Src; mTOR; Hck Angiogenesis; Apoptosis; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
PP121是一种多靶点激酶抑制剂,抑制 PDGFR、Hck、mTOR、VEGFR2、Src、Abl、DNK-PK 的 IC50值分别为2、8、10、12、14、18、60 nM。
T3351 Onatasertib

CC223,CC 223,CC-223

Apoptosis; c-Fms; DNA-PK; FLT; PI3K; mTOR Angiogenesis; Apoptosis; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Onatasertib (CC223) 是一种口服有效的mTOR 激酶抑制剂,抑制mTOR 激酶,IC50为 16 nM。它抑制mTORC1和mTORC2。
T6334 Ridaforolimus

AP23573,Deforolimus,MK-8669

mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Ridaforolimus (AP23573) 是亲脂性大环内酯类抗生素雷帕霉素的小分子非前药类似物,具有潜在的抗肿瘤活性。它是一种有效和选择性的 mTOR 抑制剂,在 HT-1080 细胞中抑制 S6 磷酸化的 IC50值为 0.2 nM。
T25399 ETP-45658

ETP45658,ETP 45658

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
ETP-45658 (ETP45658) 是一种PI3K 抑制剂,抑制PI3Kα、PI3Kδ、PI3Kβ和PI3Kγ的IC50值分别为 22.0、39.8、129.0 和 717.3 nM。它可研究癌症,还抑制DNA-PK 和mTOR,IC50分别为70.6 和 152 nM。
T12459 PI3K/mTOR Inhibitor-2

PI3K; mTOR PI3K/Akt/mTOR signaling
PI3K/mTOR Inhibitor-2 是一种有效的 PI3K 和 mTOR 泛抑制剂,对 PI3Kα、PI3Kβ、PI3Kδ、PI3Kγ 和 mTOR 的 IC50 分别为 3.4、34、16,1 和 4.7 nM。 PI3K/mTOR Inhibitor-2 具有抗肿瘤活性。
T2706 Palomid 529

P529,SG 00529

Apoptosis; mTOR Apoptosis; PI3K/Akt/mTOR signaling
Palomid 529 (SG 00529) 是一种mTORC1和mTORC2复合体抑制剂,已用于研究治疗年龄相关性黄斑变性的试验。
T6111 Selisistat

EX-527,司来司他,SEN0014196

Sirtuin Chromatin/Epigenetic; DNA Damage/DNA Repair
Selisistat (EX-527) 是一种去乙酰化酶 SIRT1 的抑制剂 (IC50=38 nM),具有有效性和特异性。Selisistat 可以用于神经系统疾病如亨廷顿舞蹈病的研究。
T1861 Omipalisib

GSK458,GSK2126458

PI3K; mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Omipalisib (GSK2126458) 是一种磷脂酰肌醇 3-激酶(PI3K) 的小分子吡啶磺酰胺抑制剂,具有抗肿瘤活性。它抑制 p110α/β/δ/γ,mTORC1/2 的活性,Ki 值分别为 0.019 nM/0.13 nM/0.024 nM/0.06 nM 和 0.18 nM/0.3 nM。
T1784 Everolimus

依维莫司,RAD001,SDZ-RAD

Apoptosis; Others; mTOR; Autophagy Apoptosis; Autophagy; Others; PI3K/Akt/mTOR signaling
Everolimus (SDZ-RAD) 是 Rapamycin 的衍生物,也是一种口服活性的mTOR1选择性抑制剂。它与FKBP-12结合可产生免疫抑制复合物,还抑制肿瘤细胞增殖并诱导细胞凋亡和自噬,有免疫抑制和抗癌活性。
T7014 Voxtalisib

XL765,SAR245409

DNA-PK; PI3K; mTOR DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Voxtalisib (XL765) 是一种PI3K 抑制剂,抑制p110α,p110β,p110γ和p110δ。它抑制mTORC1和mTORC2,IC50s 分别为 160 和 910 nM。它也抑制 DNA-PK (其 IC50=150 nM) 和 mTOR (其 IC50=157 nM)。
T6103 VS-5584

SB2343,VS 5584,VS5584

PI3K; mTOR PI3K/Akt/mTOR signaling
VS-5584 (SB2343) 是pan-PI3K/mTOR 激酶抑制剂。它能够阻断mTORC2和mTORC1。它能够抑制 PI3Kα, PI3Kβ, PI3Kδ, PI3Kγ 和 mTOR,IC50分别为 16 nM, 68 nM, 42 nM, 25 nM 和 37 nM。
T2145 Temsirolimus

NSC 683864,CCI-779,西罗莫司脂化物

Apoptosis; mTOR; Autophagy Apoptosis; Autophagy; PI3K/Akt/mTOR signaling
Temsirolimus (CCI-779) 是一种mTOR 抑制剂,IC50值为 1.76 μM。它能激活自噬,可防止心脏功能恶化。
T16409 OSMI-1

Others; Acyltransferase Metabolism; Others
OSMI-1 是一种 O-GlcNAc 转移酶 (OGT) 抑制剂 (IC50=2.7 μM),具有口服活性和细胞渗透性。OSMI-1 可以抑制蛋白质 O-GlcNA 酰化,而不会定性地改变细胞表面 N- 或 O- 连接的聚糖。
T6883 Samotolisib

GTPL8918,LY3023414

DNA-PK; PI3K; mTOR; Autophagy Autophagy; DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Samotolisib (LY3023414) 在低纳摩尔浓度下,有效抑制mTORC1/2。它选择性地有效抑制PI3Kα、PI3Kβ、PI3Kδ、PI3Kγ、DNA-PK 和mTOR,IC50分别为 6.07 nM、77.6 nM、38 nM、23.8 nM、4.24 nM 和 165 nM。它可用于多种肿瘤和癌症的试验。
T6072L BGT226

BGT226 free base,NVP-BGT226

PI3K; mTOR; Autophagy Autophagy; PI3K/Akt/mTOR signaling
BGT226 (NVP-BGT226) 是一种PI3K/mTOR 双抑制剂,对PI3Kα、PI3Kβ和PI3Kγ的IC50分别是4 nM、63 nM 和38 nM。它有效抑制人头颈癌细胞的生长。
T1970 Gedatolisib

PF-05212384,PKI-587

PI3K; mTOR PI3K/Akt/mTOR signaling
Gedatolisib (PF-05212384) 是一种高效的双重 PI3Kα (IC50:0.4 nM),PI3Kγ (IC50:5.4 nM) 和 mTOR (IC50:1.6 nM)抑制剂。它在 mTOR 复合物mTORC1和mTORC2中同样有效。
T16156 MT 63-78

Apoptosis; AMPK; mTOR Apoptosis; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling
MT 63-78 是一种有效的直接AMPK 激活剂,EC50为 25 μM。它诱导细胞有丝分裂阻滞和细胞凋亡,通过抑制脂肪生成和mTORC1途径来阻止前列腺癌的生长,具有抗肿瘤作用。

化合物

3BDO
Cat.No: T14033
Synonym:
Target: Apoptosis, mTOR, Autophagy
CZ415
Cat.No: T3514
Synonym:
Target: mTOR
mTOR inhibitor-3
Cat.No: T12123
Synonym:
Target: mTOR
Metsulfuron-methyl
Cat.No: T21246
Synonym:
Target: Others
Torin 1
Cat.No: T6045
Synonym:
Target: DNA-PK, PI3K, mTOR, Autophagy
PQR620
Cat.No: T5472
Synonym:
Target: mTOR
NV-5138
Cat.No: T12270
Synonym:
Target: mTOR
XL388
Cat.No: T6030
Synonym:
Target: P450, PI3K, mTOR
MHY-1685
Cat.No: T40351
Synonym:
Target: mTOR
KU-0063794
Cat.No: T2475
Synonym:
Target: mTOR
PF-04979064
Cat.No: T7343
Synonym:
Target: PI3K, mTOR
AZD-8055
Cat.No: T1859
Synonym:
Target: Apoptosis, mTOR, Autophagy
mTOR inhibitor-1
Cat.No: T5338
Synonym:
Target: mTOR, Autophagy
GNE-493
Cat.No: T7166
Synonym:
Target: PI3K, mTOR
MHY1485
Cat.No: T1908
Synonym:
Target: mTOR, Autophagy
NSC781406
Cat.No: T16355
Synonym:
Target: PI3K, mTOR
Torin 2
Cat.No: T6100
Synonym:
Target: Apoptosis, ATM/ATR, DNA-PK, mTOR, Autophagy
PQR530
Cat.No: T16567
Synonym: PQR-530
Target: PI3K, mTOR
Vistusertib
Cat.No: T1961
Synonym: AZD2014
Target: Apoptosis, Akt, PI3K, S6 Kinase, mTOR, Autophagy
Torkinib
Cat.No: T2414
Synonym: PP 242
Target: Apoptosis, Mitophagy, PI3K, mTOR, Autophagy
ETP-46464
Cat.No: T2084
Synonym:
Target: ATM/ATR, DNA-PK, PI3K, mTOR
GNE-317
Cat.No: T6845
Synonym: GNE317
Target: PI3K, mTOR
GNE-477
Cat.No: T3692
Synonym: GNE 477
Target: PI3K, mTOR
GSK1059615
Cat.No: T2357
Synonym: GSK 1059615,GSK-1059615
Target: Apoptosis, PI3K, mTOR
CC-115
Cat.No: T3541
Synonym: CC 115
Target: DNA-PK, PI3K, mTOR
DS-7423
Cat.No: T36083
Synonym:
Target: PI3K, mTOR
GDC-0349
Cat.No: T6510
Synonym: RG-7603
Target: PI3K, mTOR, Autophagy
GNE-490
Cat.No: T22339
Synonym:
Target: Others, PI3K
PF-04691502
Cat.No: T6251
Synonym: PF4691502
Target: Akt, PI3K, mTOR, Autophagy
KU-0060648
Cat.No: T6557
Synonym: KU0060648
Target: DNA-PK, PI3K, mTOR
Desmethyl-VS-5584
Cat.No: T4199
Synonym:
Target: PI3K, mTOR
OSI-027
Cat.No: T6319
Synonym: ASP4786,OSI027
Target: DNA-PK, PI3K, mTOR, Autophagy
PI-103
Cat.No: T6143
Synonym: PI103,PI 103
Target: Apoptosis, DNA-PK, PI3K, mTOR, Autophagy
PP121
Cat.No: T2415
Synonym:
Target: Apoptosis, VEGFR, Bcr-Abl, PDGFR, Src, mTOR, Hck
Onatasertib
Cat.No: T3351
Synonym: CC223,CC 223,CC-223
Target: Apoptosis, c-Fms, DNA-PK, FLT, PI3K, mTOR
Ridaforolimus
Cat.No: T6334
Synonym: AP23573,Deforolimus,MK-8669
Target: mTOR, Autophagy
ETP-45658
Cat.No: T25399
Synonym: ETP45658,ETP 45658
Target: DNA-PK, PI3K, mTOR
PI3K/mTOR Inhibitor-2
Cat.No: T12459
Synonym:
Target: PI3K, mTOR
Palomid 529
Cat.No: T2706
Synonym: P529,SG 00529
Target: Apoptosis, mTOR
Selisistat
Cat.No: T6111
Synonym: EX-527,司来司他,SEN0014196
Target: Sirtuin
Omipalisib
Cat.No: T1861
Synonym: GSK458,GSK2126458
Target: PI3K, mTOR, Autophagy
Everolimus
Cat.No: T1784
Synonym: 依维莫司,RAD001,SDZ-RAD
Target: Apoptosis, Others, mTOR, Autophagy
Voxtalisib
Cat.No: T7014
Synonym: XL765,SAR245409
Target: DNA-PK, PI3K, mTOR
VS-5584
Cat.No: T6103
Synonym: SB2343,VS 5584,VS5584
Target: PI3K, mTOR
Temsirolimus
Cat.No: T2145
Synonym: NSC 683864,CCI-779,西罗莫司脂化物
Target: Apoptosis, mTOR, Autophagy
OSMI-1
Cat.No: T16409
Synonym:
Target: Others, Acyltransferase
Samotolisib
Cat.No: T6883
Synonym: GTPL8918,LY3023414
Target: DNA-PK, PI3K, mTOR, Autophagy
BGT226
Cat.No: T6072L
Synonym: BGT226 free base,NVP-BGT226
Target: PI3K, mTOR, Autophagy
Gedatolisib
Cat.No: T1970
Synonym: PF-05212384,PKI-587
Target: PI3K, mTOR
MT 63-78
Cat.No: T16156
Synonym:
Target: Apoptosis, AMPK, mTOR
Cat. No. Product Name Target Signaling Pathways
T2717 Salidroside

红景天苷,Rhodioloside

Apoptosis; mTOR Apoptosis; PI3K/Akt/mTOR signaling
Salidroside (Rhodioloside) 是一种从红景天中分离出来的具有生物活性的酚苷化合物,是一种脯氨酰内肽酶抑制剂。它能通过激活 mTOR 信号缓解肿瘤恶病质小鼠模型中的恶病质症状,还能通过增强 PINK1/Parkin 介导的线粒体自噬来保护多巴胺能神经元。
T2998 Dihydromyricetin

Ampelopsin,Ampeloptin,二氢杨梅素

Influenza Virus; GABA Receptor; DNA/RNA Synthesis; mTOR; Autophagy Autophagy; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling
Dihydromyricetin (Ampelopsin) 是一种来自 Ampelopsis Grossedentata 的天然抗氧化剂类黄酮,是二氢嘧啶酶抑制剂,IC50 为 48 μM。它通过抑制mTOR 信号从而激活自噬。它还是流感依赖 RNA 的RNA 聚合酶抑制剂,IC50为 22 μM。
T5S0506 Rotundic acid

Rutundic acid,铁冬青酸

Apoptosis; Others; p38 MAPK; Akt; mTOR Apoptosis; Cytoskeletal Signaling; MAPK; Others; PI3K/Akt/mTOR signaling
Rotundic acid (Rutundic acid) 是一种从圆形肠球菌中获得的三萜类天然产物,具有抗炎和保护心脏的能力。它可通过 AKT/mTOR 和 MAPK 途径在肝细胞癌中诱导 DNA 损伤和细胞凋亡。
T3O2749 L-Leucine

(S)-Leucine,Leu,L-亮氨酸,亮氨酸

mTOR PI3K/Akt/mTOR signaling
L-Leucine ((S)-Leucine) 是必需的支链氨基酸,能够激活 mTOR 信号通路。
T3895 Polyphyllin I

重楼皂苷I,重楼皂甙

Apoptosis; Akt; JNK; PDK; mTOR; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
Polyphyllin I 是从七叶一枝花中提取的生物活性成分,具有很强的抗肿瘤活性。它是 JNK 信号通路的激活剂,也是 PDK1/Akt/mTOR 信号传导的抑制剂。它诱导自噬,G2/M 期阻滞和细胞凋亡。
T6354 (+)-Usnic acid

D-Usnic Acid,松萝酸,(+)-Usniacin,(+)-地衣酸

Antiviral; Antibacterial; mTOR Immunology/Inflammation; Microbiology/Virology; PI3K/Akt/mTOR signaling
(+)-Usnic acid (D-Usnic Acid) 是地衣中的二苯并呋喃衍生物,可结合 mTOR 的 ATP 结合口袋,抑制 mTORC1/2的活性。它诱导自噬,有抗菌和抗肿瘤活性。
TN1405 Arnicolide D

山金车内酯 D,山金车内酯D

Akt; Caspase; PI3K; STAT; mTOR Apoptosis; Cytoskeletal Signaling; JAK/STAT signaling; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells
Arnicolide D 是从石胡荽中分离出的一种倍半萜内酯,以浓度和时间依赖性方式抑制鼻咽癌细胞活力。它调节细胞周期,激活 caspase 信号通路并抑制 PI3K/AKT/mTOR 和 STAT3 信号通路。
T5740 25(R,S)-Ruscogenin

(25RS)鲁斯可皂苷元,(25RS)-Ruscogenin

Others; HIF Angiogenesis; Chromatin/Epigenetic; Others
25(R,S)-Ruscogenin 能够调节 PI3K/Akt/mTOR 信号通路,抑制 MMP-2、MMP-9、uPA、VEGF 和 HIF-1α 的表达,阻碍肝癌转移。 它能够抑制 TLR4信号通路,减轻 LPS 诱导的肺内皮细胞凋亡。
T2974 Cyclovirobuxine D

黄杨碱,CVB-D,Bebuxine,Cyclovirobuxin D,环维黄杨星D

Apoptosis; Others; Akt; mTOR; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling
Cyclovirobuxine D (Bebuxine) 是中药黄杨的主要活性成分,可诱导自噬并减弱Akt 和mTOR 的磷酸化。它通过抑制细胞周期进程和诱导线粒体介导的细胞凋亡抑制癌细胞的增殖,有用于心肌梗死引起的心力衰竭的研究潜力。
T2P2806 Hederacolchiside A1

黑海常春藤苷A1,革叶常春藤皂苷 A1,Raddeanoside R13

Apoptosis; ERK; MEK; Akt; PI3K; Parasite; mTOR Apoptosis; Cytoskeletal Signaling; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling
Hederacolchiside A1 (Raddeanoside R13) 是从白头翁中分离的一种有抗利什曼原虫和抗肿瘤增殖活性的天然产物。
T1537 Rapamycin

Sirolimus,AY 22989,雷帕霉素,NSC-2260804

Others; Endogenous Metabolite; Antibiotic; mTOR; Autophagy; Antifungal Autophagy; Metabolism; Microbiology/Virology; Others; PI3K/Akt/mTOR signaling
Rapamycin (AY 22989) 属于大环内酯类天然产物,是一种 mTOR 抑制剂,具有特异性(HEK293 细胞:IC50=0.1 nM)。Rapamycin 具有免疫抑制活性,并能诱导自噬。
T2851 Daphnetin

7,8-Dihydroxycoumarin,Daphnetol,瑞香素

EGFR; PKA; PKC; Parasite; Autophagy Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物,有抗氧化、抗炎、抗疟疾和解热作用,可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。
T4759 Urocanic acid

4-Imidazoleacrylic acid,尿刊酸

Others; Endogenous Metabolite Metabolism; Others
Urocanic acid (4-Imidazoleacrylic acid), synthesized in the epidermis, functions as a primary absorber of ultraviolet (UV) radiation in mammalian skin.
T21205 Ponasterone A

坡那甾酮A,AI3-44686

Others Others
Ponasterone A (AI3-44686) 是一种蜕皮激素,能够高度亲和蜕皮激素受体。它能够使报告基因能够快速打开和关闭,是细胞和转基因动物中基因表达的有效调节剂。
T13802 Oleamide

Oleic acid amide

Others; Endogenous Metabolite Metabolism; Others
Oleamide (Oleic acid amide) 是一种内源性脂肪酸酰胺,可用于哺乳动物神经系统的从头合成。
T4730 Thymidine-5'-monophosphate disodium salt

胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT

Others; Endogenous Metabolite Metabolism; Others
Thymidine-5'-monophosphate disodium salt (TMP DISODIUM SALT) 是内源性代谢产物的一种。
T5145 Oxytocin acetate

Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素

Oxytocin Receptor Endocrinology/Hormones; GPCR/G Protein
Oxytocin acetate (α-Hypophamine acetate) 是哺乳动物的神经垂体激素,是多效的下丘脑肽,是催产素受体的配体,有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子,具有抗炎、抗氧化剂和保护作用。
T5514 Epibrassinolide

24-Epibrassinolide,B1105,表油菜素内酯,BP55

Apoptosis Apoptosis
Epibrassinolide (BP55) 是一种广泛存在的植物生长激素,具有缓解植物重金属和农药胁迫潜力。它在各种癌细胞中是一种潜在的凋亡诱导剂。
T0344L Miconazole nitrate

NSC 169434 Nitrate,硝酸咪康唑,R18134 nitrate

Antibacterial; Antibiotic; Antifungal Microbiology/Virology
Miconazole nitrate (R18134 nitrate) 是咪唑类可抗菌的抗真菌剂。
T4514 N-Acetyl-D-Glucosamine

N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc

Endogenous Metabolite Metabolism
N-Acetyl-D-Glucosamine (NAG) 是葡萄糖的单糖衍生物。
TMA0507 Tomatidine

NF-κB; JNK; Autophagy Autophagy; MAPK; NF-κB
Tomatidine 通过阻断 NF-κB 和 JNK 信号传导而发挥抗炎作用。它在哺乳动物细胞或秀丽隐杆线虫中激活自噬。
T5026 Oxytocin

催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)

Oxytocin Receptor Endocrinology/Hormones; GPCR/G Protein
Oxytocin (Oxytocin (Syntocinon)) 是哺乳动物的神经垂体激素,是多效的下丘脑肽,是催产素受体的配体,有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子,具有抗炎、抗氧化剂和保护作用。
T5086 Pharmatose DCL 14

D-乳糖一水合物,D-Lactose monohydrate

Others; Endogenous Metabolite Metabolism; Others
Pharmatose DCL 14 (D-Lactose monohydrate) 是内源性代谢产物的一种。
T2O2707 D-(+)-Fucose

Others Others
D-(+)-Fucose 是一种 l-阿拉伯糖的非代谢类似物,也是 β-甲基半乳糖苷透皮酶诱导剂。它能够抑制 l-阿拉伯糖操纵子的诱导,阻断大肠杆菌 B/r 在矿物盐培养基上加 l-阿拉伯糖的生长。
T5645 Nerol

Cis-Geraniol,橙花醇,Neryl alcohol

Apoptosis; Reactive Oxygen Species; Mitochondrial Metabolism; Endogenous Metabolite; Antifungal Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Nerol (Neryl alcohol) 是橙花油的一种单萜, 它通过增强 Ca2+和ROS 来触发线粒体功能障碍并诱导凋亡,具有抗真菌活性。它可减轻哺乳动物心脏中哇巴因引发的心律失常的严重程度。
T2596 N-Acetyl-β-Asp-Glu

Others Others
N-Acetyl-β-Asp-Glu 是一种肽类神经递质,是哺乳动物神经系统中第三常见的神经递质。 NAAG 由通过肽键偶联的 N-乙酰天冬氨酸 (NAA) 和谷氨酸组成。
T5663 α-Lactose

D-乳糖单水合物,Lactose

Others Others
α-Lactose 是牛奶中的主要的糖。它一般以 α 和 β 两个异构体的形式存在,其中α 形式通常以一水合物的形式结晶。
T5915 D-chiro-Inositol

D-手性肌醇,D-(+)-CHIRO-INOSITOL

Endogenous Metabolite Metabolism
D-chiro-Inositol (D-(+)-CHIRO-INOSITOL) 是肌醇差向异构体,存在于某些哺乳动物糖基磷脂酰肌醇蛋白锚和具有胰岛素样生物特性的肌醇磷脂聚糖中。它能够抑制高血糖,改善胰岛素抵抗。它用于多囊卵巢综合征和糖尿病的相关研究。
T4814 (R)-5-Oxopyrrolidine-2-carboxylic acid

D-Pyroglutamic acid,(R)-(+)-2-Pyrrolidone-5-carboxylic acid,D-焦谷氨酸

Others; Endogenous Metabolite Metabolism; Others
(R)-5-Oxopyrrolidine-2-carboxylic acid (D-Pyroglutamic acid) 是内源性代谢产物的一种。
T4875 Palatinose hydrate

6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物

Others; Endogenous Metabolite Metabolism; Others
Palatinose hydrate (6-O-α-D-Glucopyranosyl-D-fructose, Isoma) 是内源性代谢产物的一种。
T1009 Estrone

Oestrone,雌酮,Fluoroethyl,Aquacrine

Estrogen Receptor/ERR; Estrogen/progestogen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Estrone (Aquacrine) 是内源性雌激素的主要代表,由多种组织产生,尤其是脂肪组织。它是脂肪细胞中雄烯二酮芳构化过程的结果。
T1638 N-Acetylneuraminic acid

唾液酸,Acide aceneuramique,N-乙酰神经氨酸,NeuAc,Lactaminic acid

Others; Influenza Virus; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
N-Acetylneuraminic acid (Acide aceneuramique) 是一种九碳唾液酸单糖,通常存在于细胞膜上的糖蛋白和哺乳动物细胞中的神经节苷脂等糖脂中。它可用于神经传递、白细胞外渗、病毒或细菌感染以及碳水化合物-蛋白质识别。
T2S1792 Lycobetaine

石蒜内胺,Ungeremine,石蒜醋胺,石蒜碱内铵盐

Antibacterial Microbiology/Virology
Lycobetaine (Ungeremine) 是一种潜在的抗罗克福尔青霉和黑曲霉的生物杀菌剂。它对柱状黄杆菌有很强的抗菌活性。它有效地靶向哺乳动物以及细菌I 型和II 型拓扑异构酶。它显示出强烈的乙酰胆碱酯酶抑制活性(IC(50) 值为 0.35 microM)。 它具有抗原生动物活性,在体外试验中对Trypanosoma brucei rhodesiense、T. cruzi 表现出良好的活性。
T4716 Pyrrole-2-carboxylic acid

吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline

Endogenous Metabolite Metabolism
Pyrrole-2-carboxylic acid (Minaline) 是一种天然生物碱类,从海洋细菌Pelomonas puraquaesp. Nov 中分离得到。
T37974 (S)-Coriolic acid

13(S)-HODE

Lipoxygenase; Mitochondrial Metabolism; PPAR DNA Damage/DNA Repair; Metabolism
(S)-Coriolic acid (13(S)-HODE) 是一种重要的细胞内信号剂,是亚油酸与植物和哺乳动物脂氧合酶反应生成的,在各种生物系统中参与细胞增殖和分化。(S)-Coriolic acid 在 1 μM 左右时,它能抑制肿瘤细胞与血管内皮的粘附,能下调 IRGpIIb/IIIa 受体的表达。(S)-Coriolic acid 是15-脂氧合酶 (15-LOX) 代谢产物,常作为内源性配体激活 PPARγ。(S)-Coriolic acid 诱导线粒体功能障碍 和气道上皮损伤。
TN5040 Soyasaponin IV

Others Others
Soyasaponin IV has hepatoprotective activity.It also has antimutagenic activity in mammalian cells.
T13297 Verruculogen

Others Others
Verruculogen is a toxin produced mainly by Penicillium and Aspergillus spp. Verruculogen inhibits Ca2+-activated K+ channels, and is an M phase inhibitor of the mammalian cell cycle.
T15094 Dehydroaltenusin

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
Dehydroaltenusin is a selective eukaryotic DNA polymerase α inhibitor and a type of antibiotic produced by a fungus (IC50: 0.68 μM). Dehydroaltenusin inhibits mammalian pol α activity.
T14548 Beta-Zearalanol

Others Others
Beta-Zearalenol, a derivative of zearalenone (ZEA) capable of conjugating with glucuronic acid[2], is a mycotoxin produced by Fusarium spp. It induces apoptosis and oxidative stress in mammalian reproductive cells[1].
T20123 L-Carnitine hydrochloride

L-Carnitine chloride,LC 80,Levocarnitine chloride,(R)-Carnitine hydrochloride,LC-80,LC80

Carnitine is a quaternary amine that occurs naturally in most mammalian tissue. Carnitine is present in relatively high concentrations in skeletal muscle and heart where it is involved in regulating energy metabolism. It has also been used to allow the en
TN5190 Tryprostatin A

Topoisomerase; Antifection DNA Damage/DNA Repair; Microbiology/Virology
Tryprostatin A is an inhibitor of breast cancer resistance protein. Tryprostatin A and tryprostatin B are indole alkaloid-based fungal products that inhibit mammalian cell cycle at the G2/M phase.
TN6059 Demethoxyfumitremorgin C

Demethoxyfumitremorgin C and tryprostatin B are fungal inhibitors of mammalian cell cycle progression at the G(2)/M transition. Demethoxyfumitremorgin C inhibits the proliferation of PC3 human prostate cancer cells via the intrinsic (mitochondrial) and ex
T81029 Tazettine

Tazettine为一生物碱,其对哺乳动物细胞系具有较低的细胞毒性(CC50 >100 μg/mL)。
TCA2511 11Beta-hydroxyprogesterone

Sodium Channel Membrane transporter/Ion channel
The progesterone derivatives 11 alpha- and 11 beta-hydroxyprogesterone are potent inhibitors of 11 beta-hydroxysteroid dehydrogenase (isoforms 1 and 2) in vitro and can confer mineralocorticoid activity on corticosterone in the rat in vivo. 11beta-Hydroxyprogesterone acts as a mineralocorticoid agonist in stimulating Na+ absorption in mammalian principal cortical collecting duct cells.
T36560 (±)9-HpODE

(±)9-HpODE is a racemic mixture of the fatty acid hydroperoxide product (9(S)-HpODE) formed from lipoxygenase action on linoleic acid. It shows antimicrobial activity against various fungal and bacterial pathogens and thus may play a role in plant defense. In mammalian species, monocyte-induced oxidization of LDL generates significant amounts of esterified 9-HpODE, which is rapidly reduced to 9-HODE.
T28379 PF-1163B

PF1163B,(-)-PF1163B,PF 1163B

PF-1163B is an antifungal agent form Penicillium sp. II. PF-1163B inhibits ergosterol (ERG) synthesis with IC50 value of 34 ng/ml. PF-1163B showed potent growth inhibitory activity against pathogenic fungal strain Candida albicans but did not show cytotox
T82032 Isoglobotriaose

Gala-3Galb-4Glc

Isoglobotriaose (Gala-3Galb-4Glc)是哺乳动物组织中的一种糖鞘脂,属于球状三脂糖的类似物。其神经节苷脂衍生物isoglobotriaosylceramide特定分布于小肠非上皮细胞的残基中,而globotriaosylceramide则在两种细胞隔室中都有分布。
T83582 (±)-Pantothenic acid

(±)-Vitamin B5,(±)-Pantothenate

(±)-Pantothenic acid ((±)-Pantothenate) 作为 B 组维生素的一员,对于哺乳动物细胞中辅酶 A (CoA) 的生物合成是不可或缺的。此外,该化合物能防护丙戊酸 (VPA) 在 CD-1 小鼠中引起的神经管缺陷 (NTD)。
T78506 α-Lactose hydrate

α-D-Lactose hydrate

α-Lactose (hydrate)(α-D-Lactose (hydrate))是哺乳动物乳汁的主要碳水化合物,由葡萄糖和半乳糖构成,并有α和β两种异构体。它广泛应用于食品和制药行业,常作为松散剂或凝聚剂,也用于稀释色素、香料或酶。
T35415 α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)

α-D-Glucose-1,6-bisphosphate is abis-phosphorylated derivative of α-D-glucose that has roles in carbohydrate metabolism.1It is the product of the reaction of glucose-1- or 6-phosphate with glucose-1,6-bisphosphate synthase (PGM2LI) in the conversion of 1,3-bisphosphoglycerate to 3-phosphoglycerate.2It is also a cofactor for the bacterial enzyme phosphopentomutase.3,4α-D-Glucose-1,6-bisphosphate has been used in the study of carbohydrate metabolism. 1.Beitner, R.Regulation of carbohydrate metabol...
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天然产物

Salidroside
Cat.No: T2717
Synonym: 红景天苷,Rhodioloside
Target: Apoptosis, mTOR
Dihydromyricetin
Cat.No: T2998
Synonym: Ampelopsin,Ampeloptin,二氢杨梅素
Target: Influenza Virus, GABA Receptor, DNA/RNA Synthesis, mTOR, Autophagy
Rotundic acid
Cat.No: T5S0506
Synonym: Rutundic acid,铁冬青酸
Target: Apoptosis, Others, p38 MAPK, Akt, mTOR
L-Leucine
Cat.No: T3O2749
Synonym: (S)-Leucine,Leu,L-亮氨酸,亮氨酸
Target: mTOR
Polyphyllin I
Cat.No: T3895
Synonym: 重楼皂苷I,重楼皂甙
Target: Apoptosis, Akt, JNK, PDK, mTOR, Autophagy
(+)-Usnic acid
Cat.No: T6354
Synonym: D-Usnic Acid,松萝酸,(+)-Usniacin,(+)-地衣酸
Target: Antiviral, Antibacterial, mTOR
Arnicolide D
Cat.No: TN1405
Synonym: 山金车内酯 D,山金车内酯D
Target: Akt, Caspase, PI3K, STAT, mTOR
25(R,S)-Ruscogenin
Cat.No: T5740
Synonym: (25RS)鲁斯可皂苷元,(25RS)-Ruscogenin
Target: Others, HIF
Cyclovirobuxine D
Cat.No: T2974
Synonym: 黄杨碱,CVB-D,Bebuxine,Cyclovirobuxin D,环维黄杨星D
Target: Apoptosis, Others, Akt, mTOR, Autophagy
Hederacolchiside A1
Cat.No: T2P2806
Synonym: 黑海常春藤苷A1,革叶常春藤皂苷 A1,Raddeanoside R13
Target: Apoptosis, ERK, MEK, Akt, PI3K, Parasite, mTOR
Rapamycin
Cat.No: T1537
Synonym: Sirolimus,AY 22989,雷帕霉素,NSC-2260804
Target: Others, Endogenous Metabolite, Antibiotic, mTOR, Autophagy, Antifungal
Daphnetin
Cat.No: T2851
Synonym: 7,8-Dihydroxycoumarin,Daphnetol,瑞香素
Target: EGFR, PKA, PKC, Parasite, Autophagy
Urocanic acid
Cat.No: T4759
Synonym: 4-Imidazoleacrylic acid,尿刊酸
Target: Others, Endogenous Metabolite
Ponasterone A
Cat.No: T21205
Synonym: 坡那甾酮A,AI3-44686
Target: Others
Oleamide
Cat.No: T13802
Synonym: Oleic acid amide
Target: Others, Endogenous Metabolite
Thymidine-5'-monophosphate disodium salt
Cat.No: T4730
Synonym: 胸苷酸二钠,Thymidine 5'-monophosphate disodium salt,TMP DISODIUM SALT
Target: Others, Endogenous Metabolite
Oxytocin acetate
Cat.No: T5145
Synonym: Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素
Target: Oxytocin Receptor
Epibrassinolide
Cat.No: T5514
Synonym: 24-Epibrassinolide,B1105,表油菜素内酯,BP55
Target: Apoptosis
Miconazole nitrate
Cat.No: T0344L
Synonym: NSC 169434 Nitrate,硝酸咪康唑,R18134 nitrate
Target: Antibacterial, Antibiotic, Antifungal
N-Acetyl-D-Glucosamine
Cat.No: T4514
Synonym: N-乙酰-D-氨基葡萄糖,NAG,N-Acetyl-2-amino-2-deoxyglucose,Marine Sweet,N-Acetyl-2-amino-2-deoxy-D-glucose,N-乙酰氨基葡萄糖,GlcNAc
Target: Endogenous Metabolite
Tomatidine
Cat.No: TMA0507
Synonym:
Target: NF-κB, JNK, Autophagy
Oxytocin
Cat.No: T5026
Synonym: 催产素,α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)
Target: Oxytocin Receptor
Pharmatose DCL 14
Cat.No: T5086
Synonym: D-乳糖一水合物,D-Lactose monohydrate
Target: Others, Endogenous Metabolite
D-(+)-Fucose
Cat.No: T2O2707
Synonym:
Target: Others
Nerol
Cat.No: T5645
Synonym: Cis-Geraniol,橙花醇,Neryl alcohol
Target: Apoptosis, Reactive Oxygen Species, Mitochondrial Metabolism, Endogenous Metabolite, Antifungal
N-Acetyl-β-Asp-Glu
Cat.No: T2596
Synonym:
Target: Others
α-Lactose
Cat.No: T5663
Synonym: D-乳糖单水合物,Lactose
Target: Others
D-chiro-Inositol
Cat.No: T5915
Synonym: D-手性肌醇,D-(+)-CHIRO-INOSITOL
Target: Endogenous Metabolite
(R)-5-Oxopyrrolidine-2-carboxylic acid
Cat.No: T4814
Synonym: D-Pyroglutamic acid,(R)-(+)-2-Pyrrolidone-5-carboxylic acid,D-焦谷氨酸
Target: Others, Endogenous Metabolite
Palatinose hydrate
Cat.No: T4875
Synonym: 6-O-α-D-Glucopyranosyl-D-fructose, Isoma,帕拉金糖水合物
Target: Others, Endogenous Metabolite
Estrone
Cat.No: T1009
Synonym: Oestrone,雌酮,Fluoroethyl,Aquacrine
Target: Estrogen Receptor/ERR, Estrogen/progestogen Receptor, Endogenous Metabolite
N-Acetylneuraminic acid
Cat.No: T1638
Synonym: 唾液酸,Acide aceneuramique,N-乙酰神经氨酸,NeuAc,Lactaminic acid
Target: Others, Influenza Virus, Endogenous Metabolite
Lycobetaine
Cat.No: T2S1792
Synonym: 石蒜内胺,Ungeremine,石蒜醋胺,石蒜碱内铵盐
Target: Antibacterial
Pyrrole-2-carboxylic acid
Cat.No: T4716
Synonym: 吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline
Target: Endogenous Metabolite
(S)-Coriolic acid
Cat.No: T37974
Synonym: 13(S)-HODE
Target: Lipoxygenase, Mitochondrial Metabolism, PPAR
Soyasaponin IV
Cat.No: TN5040
Synonym:
Target: Others
Verruculogen
Cat.No: T13297
Synonym:
Target: Others
Dehydroaltenusin
Cat.No: T15094
Synonym:
Target: DNA/RNA Synthesis
Beta-Zearalanol
Cat.No: T14548
Synonym:
Target: Others
L-Carnitine hydrochloride
Cat.No: T20123
Synonym: L-Carnitine chloride,LC 80,Levocarnitine chloride,(R)-Carnitine hydrochloride,LC-80,LC80
Target:
Tryprostatin A
Cat.No: TN5190
Synonym:
Target: Topoisomerase, Antifection
Demethoxyfumitremorgin C
Cat.No: TN6059
Synonym:
Target:
Tazettine
Cat.No: T81029
Synonym:
Target:
11Beta-hydroxyprogesterone
Cat.No: TCA2511
Synonym:
Target: Sodium Channel
(±)9-HpODE
Cat.No: T36560
Synonym:
Target:
PF-1163B
Cat.No: T28379
Synonym: PF1163B,(-)-PF1163B,PF 1163B
Target:
Isoglobotriaose
Cat.No: T82032
Synonym: Gala-3Galb-4Glc
Target:
(±)-Pantothenic acid
Cat.No: T83582
Synonym: (±)-Vitamin B5,(±)-Pantothenate
Target:
α-Lactose hydrate
Cat.No: T78506
Synonym: α-D-Lactose hydrate
Target:
α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)
Cat.No: T35415
Synonym:
Target:
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