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2063

抑制剂 & 化合物

178

天然产物

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Cat. No. Product Name Target Signaling Pathways
T4356 POL1-IN-1

Compound 3A

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
POL1-IN-1 (Compound 3A) 是一种RNA 聚合酶 1 POL1抑制剂,IC50值低于 0.5 uM。 它能有效抑制A375恶性黑色素瘤细胞系中RNA 聚合酶I 的转录。
T11942 MAP4K4-IN-3

Compound 17

MAPK MAPK
MAP4K4-IN-3 (Compound 17) 是 MAP4K4选择性抑制剂,在激酶实验中 IC50为 14.9 nM,在细胞实验中 IC50为 470 nM。具有抗糖尿病作用。
T11035 diABZI STING agonist-1 (Tautomerism)

diABZI STING agonist (Compound 3)

STING Immunology/Inflammation
diABZI STING agonist-1 (Tautomerism) (diABZI STING agonist (Compound 3)) 是一个选择性的干扰素基因刺激受体 (STING) 的激动剂,其在人和小鼠中的 EC50 值分别为 130 nM 和 186 nM。。
T13017 STL127705

Compound L,7-[[2-(3,4-Dimethoxyphenyl)ethyl]amino]-3-(3-fluorophenyl)pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione

DNA-PK; Others DNA Damage/DNA Repair; Others; PI3K/Akt/mTOR signaling
STL127705 (Compound L) 是一种有效的 Ku 70/80 异二聚体蛋白抑制剂,抑制 Ku70/80-DNA 相互作用,IC50 为 3.5 μM。 它抑制 Ku 依赖性 DNA-PKCS 激酶的激活,IC50 为 2.5 μM。
T10608 BRD5648

(R)-BRD0705

GSK-3 PI3K/Akt/mTOR signaling; Stem Cells
BRD5648 ((R)-BRD0705) 是 BRD0705 的 阴性对照,BRD0705 是旁系选择性和口服有效的 GSK3α 抑制剂,Kd 为 4.8 μM,IC50为 66 nM。与 GSK3β (IC50为 515 nM) 相比,BRD0705 对 GSK3α 的选择性更高 (8 倍)。BRD0705 可用于急性髓细胞性白血病。
T7944 VPS34 inhibitor 1 (Compound 19, PIK-III analogue)

PIK-III analogue

PI3K PI3K/Akt/mTOR signaling
VPS34 inhibitor 1 (Compound 19, PIK-III analogue) (PIK-III analogue) 是一种有效的选择性 VPS34抑制剂( IC50 : 15 nM)。
T9184L Compound 3344 hydrochloride

4-(2,3-dihydro-1,4-benzodioxin-5-yl)-~{N}-[3-[(dimethylamino)methyl]phenyl]-2-methoxy-aniline hydrochloride(2368246-78-8 free base),Compound 3344 hydrochloride (2368246-78-8 free base)

Ras GPCR/G Protein; MAPK
Compound 3344 hydrochloride 是 KRAS 效应相互作用的抑制剂,亲和力为 126nm。
T6146 Dorsomorphin dihydrochloride

BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride

AMPK; Autophagy; TGF-beta/Smad Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Stem Cells
Dorsomorphin dihydrochloride (BML-275 2HCl) 是一种选择性和 ATP 竞争性的AMPK 抑制剂,Ki 为 109 nM。它诱导自噬,通过靶向抑制 I 型受体ALK2,ALK3和ALK6来抑制 BMP 途径。
T9658 DCZ3301

NPS ALX Compound 4a hydrochloride(1:1)(299433-10-6 Free base)

Others Others
DCZ3301是一种新的芳基胍抑制剂。
T9537 N'-Nitro-D-arginine

N'-Nitro-D-arginine,H-D-Arg(NO2)-OH,(R)-2-Amino-5-(3-nitroguanidino)pentanoic acid,N'-硝基-D-精氨酸

Others Others
N'-Nitro-D-arginine (N'-Nitro-D-arginine) 是一种砌块。
T8055 TFEB activator 1

(1E,4E)-1,5-Bis(2-Methoxyphenyl)penta-1,,Curcumin analog compound C1,Curcumin analog C1,(1E,4E)-1,5(2 -甲氧基苯基)-1,4-戊二烯-3-酮,RPN77612

Others; Autophagy Autophagy; Others
TFEB activator 1 (Curcumin analog compound C1) 是转录因子 EB 的一种激活剂,有望预防或治疗阿尔茨海默病。
T64349 Necroptosis-IN-3

Cyclohexanecarboxamide, N-(2-thienylmethyl)-

Necroptosis Apoptosis
Necroptosis-IN-3 (Cyclohexanecarboxamide, N-(2-thienylmethyl)-)(Compound 69) 是一种坏死性凋亡 (necroptosis) 抑制剂,抑制 TNF-α 诱导的坏死性凋亡。Necroptosis-IN-3(Compound 69) 也抑制 11β-HSD1。
T64350 Casein kinase 1δ-IN-3

Casein Kinase Metabolism; Stem Cells
Casein kinase 1δ-IN-3 (Casein kinase 1δ-IN-3) (Compound 23a) 是一种酪蛋白激酶 1δ (CK1d) 抑制剂,pIC50 为 6.5376。
Fr12380 Benzothiazole-6-carboxylic acid

Compound Fr12380 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr12380,CAS号为 3622-35-3
T67696 1-(2-fluorophenyl)-3-[5-(2-methoxyphenyl)-1,3,4-thiadiazol-2-yl]urea

Others Others
1-(2-fluorophenyl)-3-[5-(2-methoxyphenyl)-1,3,4-thiadiazol-2-yl]urea 是一种化合物。
Fr13623 Benzofuran-2-carboxylic acid

Compound Fr13623 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr13623,CAS号为 496-41-3
T60158 PBRM1-BD2-IN-3

Epigenetic Reader Domain Chromatin/Epigenetic
PBRM1-BD2-IN-3 (compound 12) 是一种有效的 PBRM1-BD2 抑制剂,IC50 为 1.1 μM。PBRM1-BD2 Inhibitor 可用于抗癌研究。
T14264 Aminooxy-PEG3-azide

Others Others
Aminooxy-PEG3-azide is a 3-unit PEG-based azide linker compound employed in the synthesis of antibody-drug conjugates (ADCs)[1]. Additionally, Aminooxy-C2-PEG3-azide is a PEG-based PROTAC linker compound used in the synthesis of PROTACs[2].
T60485 DIF-3

DIF-3 is a chemical compound that acts by activating GSK-3β to facilitate the degradation of cyclin D1 and c-Myc, resulting in reduced expression levels of these proteins. In addition, DIF-3 inhibits Wnt/β-catenin signaling pathway-related proteins in DLD-1 cells. This compound exerts a potent antiproliferative effect on the HeLa human cervical cancer cell line by inducing cyclin D1 degradation and inhibiting cyclin D1 mRNA expression [1].
T20163 Acetyltrialanine

Acetyltrialanine 是一种二肽化合物,在 Tb+3-胰腺弹性蛋白酶复合物上的两个位点结合,可做为氮源使用。
T67777 Flaviviruses-IN-3

WAY-324593

Virus Protease Microbiology/Virology
Flaviviruses-IN-3(化合物87)是flaviviruse 的有效抑制剂。Flaviviruses-IN-3可降低西尼罗河病毒(WNV)蛋白酶活性,抑制率为54%。
T50084 (2E)-N-(4-methoxyphenyl)-3-[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-yl]prop-2-enamide

Others Others
(2E)-N-(4-methoxyphenyl)-3-[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-yl]prop-2-enamide 是一种用作分子结构单元的化合物,用于多种有机物的合成。
T60017 5-Bromo-4-chloro-3-indoxyl-beta-D-cellobioside

Others Others
5-Bromo-4-chloro-3-indoxyl-beta-D-cellobioside 是用于检测纤维生物水解酶的显色化合物。
T60124 1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea

TNF Apoptosis
1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea 是一种能够激动 TNF-α的化合物,可以诱导细胞分泌 TNF-α。
T9872 Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-

Others Others
Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-是一种用于抗病毒活性测定的化合物。
T50070 1-ethyl-6-fluoro-4-oxo-7-[4-(3-phenylpropanoyl)piperazin-1-yl]-1,4-dihydroquinoline-3-carboxylic acid

Others Others
1-ethyl-6-fluoro-4-oxo-7-[4-(3-phenylpropanoyl)piperazin-1-yl]-1,4-dihydroquinoline-3-carboxylic acid 是一种用作分子结构单元的化合物,是一种SMURF1抑制剂。
Fr21265 2-Methyl-2H-indazole-3-carboxylic acid

2-Methyl-2H-indazole-3-carboxylic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr21265,CAS号为 34252-44-3
T4581 3-hydroxycephem

Others Others
3-hydroxycephem 是各类头孢中间体。
T5151 5-Methoxyindole-3-carboxaldehyde

Others Others
5-Methoxyindole-3-carboxaldehyde 用作中间体。
T22432 SU5208

3-[(Thien-2-yl)methylene]-2-indolinone

VEGFR Angiogenesis; Tyrosine Kinase/Adaptors
SU5208 (3-[(Thien-2-yl)methylene]-2-indolinone) 对血管内皮生长因子受体2具有抑制作用。
T64347 ALDH1A3-IN-3

Dehydrogenase Metabolism
ALDH1A3-IN-3 (化合物 16) 是一种有效的 ALDH1A3 抑制剂,IC50 值为 0.26 μM。ALDH1A3-IN-3 也是 ALDH3A1 的底物。ALDH1A3-IN-3 可用于前列腺癌的研究。
T77681 3-Methoxy-9H-Carbazole

Apoptosis Apoptosis
3-methoxy-9H-carbazole 是一种光敏剂,是来自克劳塞纳七叶植物和克劳塞纳籼稻的天然化合物。3-methoxy-9H-carbazole具有抗乳腺癌活性,可诱导细胞凋亡。
T75005 TGFβ1-IN-3

Others Others
TGFβ1-IN-3 是一种二芳基酰基腙衍生物,对成纤维细胞的活化和增殖有抑制作用。TGFβ1-IN-3 是治疗特发性肺纤维化 (IPF) 的候选化合物。
T3726 Erdafitinib

厄达替尼,JNJ-42756493

Apoptosis; FGFR Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Erdafitinib (JNJ-42756493) 是一种喹喔啉衍生物,是一种具有口服活性的FGFR 家族抑制剂,抑制FGFR1/2/3/4活性的IC50分别为1.2、 2.5、3.0和5.7 nM。
T10162 5-HT3 antagonist 3

5-HT Receptor GPCR/G Protein; Neuroscience
5-HT3 antagonist 3 是一种高亲和力的 5-HT3 受体拮抗剂。5-HT3 antagonist 3 结合到大鼠脑皮质膜中的 5-HT3 受体,Ki 为 0.25 nM。
T60812 Cathepsin X-IN-1

Cysteine Protease Proteases/Proteasome
Cathepsin X-IN-1 (compound 25) 降低人前列腺癌细胞 PC-3 的迁移且具有较低的细胞毒性,它是组织蛋白酶 X 的有效抑制剂 (IC50 = 7.13 μM)。
T50028 6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole

6-氟-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚,6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole

Others Others
6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole (6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) 是一种吲哚衍生物,具有潜在抗癌活性,是开发新药的潜在先导化合物。
T67923 WIC1

Others Others
2H-1-Benzopyran-3-carboxamide, N-[4-(4-ethyl-1-piperazinyl)phenyl]-2-oxo-是 化合物,是治疗肿瘤的潜在化合物。
T50051 1,3-diethyl 2-(3-methoxyphenyl)propanedioate

Others Others
1,3-diethyl 2-(3-methoxyphenyl)propanedioate 是一种用作分子结构单元的化合物,可用于多种化合物的合成。
T39805 LDHA-IN-3

PSTMB,1-(phenylseleno)-4-(trifluoromethyl) benzene

Dehydrogenase Metabolism
LDHA-IN-3 (1-(phenylseleno)-4-(trifluoromethyl) benzene) 是一种有效的非竞争性乳酸脱氢酶(LDHA) 抑制剂,IC50值为 145.2 nM。LDHA-IN-3 是一种硒苯化合物,可用于研究癌症。
T63909 GLP-1R agonist 3

Glucagon Receptor GPCR/G Protein
GLP-1R agonist 3 是增稠的咪唑衍生物化合物,是 GLP-1R 的有效激动剂。其中胰高血糖素样肽-1 (GLP-1) 是一种肠道降血糖激素,由下消化道 L 细胞分泌。GLP-1R agonist 3 对糖尿病表现出研究潜力。
T13965 Watermelon ketone

7-Methyl-2H-1,5-benzodioxepin-3(4H)-one,西瓜酮

Others Others
Watermelon ketone (7-Methyl-2H-1,5-benzodioxepin-3(4H)-one) 是一种具有特殊气味的香料,已广泛应用于香水行业。
T90421 2-Bromo-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine

2-Bromo-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 是有一种有用的有机化合物,已被用于生命科学相关研究。
T9795 INT. 2

INT. 2 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T9795,CAS号为 210193-42-3
T9798 2H-1-Benzopyran-3-carboxylic acid, 3,4-dihydro-6-Methoxy-, (3S)-

(S)-6-methoxychroman-3-carboxylic acid is a synthetic compound with a molecular formula of C11H10O5. It is a member of the chroman family of compounds, which are characterized by a seven-membered ring with one oxygen and one carbon atom.
T9856 FLT3-IN-10

2-Oxazolamine, 5-(4-fluorophenyl)-N-phenyl-

FLT Angiogenesis; Tyrosine Kinase/Adaptors
FLT3-IN-10 (2-Oxazolamine, 5-(4-fluorophenyl)-N-phenyl-) (compound 7c) 是有效的 FMS 样酪氨酸激酶 3 (FLT3) 抑制剂。FLT3-IN-10 具有治疗 FLT3 突变的急性髓性白血病 (AML) 的潜力。
T50122 3-Ethyl-1-methyl-2-thioxoimidazolidin-4-one

3-Ethyl-1-methyl-2-thioxoimidazolidin-4-one 是一种属于咪唑烷酮类化合物的有机化合物,已被用于生命科学相关研究。
T65090 Copper(II) gluconate

Copper(II) gluconate 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T65090,CAS号为 527-09-3
TNU0060 3’-O-Methyladenosine

Antiviral; Adenosine deaminase Immunology/Inflammation; Metabolism
3’-O-Methyladenosine 是一种抗病毒化合物,对西尼罗河病毒具有抑制作用,可用于治疗病毒感染。3’-O-Methyladenosine 对腺苷脱氨酶VII型具有抑制作用,Ki 值为 493 µM。
T67747 CB2R/FAAH modulator-3

Cannabinoid Receptor; FAAH GPCR/G Protein; Metabolism; Neuroscience
CB2R/FAAH modulator-3 (compound 27) 是一种双重靶点的调节剂,是 CB2R 的激动剂, 也是FAAH 的抑制剂, 作用于 CB2R 和 CB1R 的 Ki 值分别是 20.1 和 67.6 nM,作用于 FAAH 的IC50值为 3.4 μM。CB2R/FAAH modulator-3 可用于癌症、神经退行性疾病中发生的有害炎症级联反应以及 COVID-19 感染相关研究。

化合物

POL1-IN-1
Cat.No: T4356
Synonym: Compound 3A
Target: DNA/RNA Synthesis
MAP4K4-IN-3
Cat.No: T11942
Synonym: Compound 17
Target: MAPK
diABZI STING agonist-1 (Tautomerism)
Cat.No: T11035
Synonym: diABZI STING agonist (Compound 3)
Target: STING
STL127705
Cat.No: T13017
Synonym: Compound L,7-[[2-(3,4-Dimethoxyphenyl)ethyl]amino]-3-(3-fluorophenyl)pyrimido[4,5-d]pyrimidine-2,4(1H,3H)-dione
Target: DNA-PK, Others
BRD5648
Cat.No: T10608
Synonym: (R)-BRD0705
Target: GSK-3
VPS34 inhibitor 1 (Compound 19, PIK-III analogue)
Cat.No: T7944
Synonym: PIK-III analogue
Target: PI3K
Compound 3344 hydrochloride
Cat.No: T9184L
Synonym: 4-(2,3-dihydro-1,4-benzodioxin-5-yl)-~{N}-[3-[(dimethylamino)methyl]phenyl]-2-methoxy-aniline hydrochloride(2368246-78-8 free base),Compound 3344 hydrochloride (2368246-78-8 free base)
Target: Ras
Dorsomorphin dihydrochloride
Cat.No: T6146
Synonym: BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride
Target: AMPK, Autophagy, TGF-beta/Smad
DCZ3301
Cat.No: T9658
Synonym: NPS ALX Compound 4a hydrochloride(1:1)(299433-10-6 Free base)
Target: Others
N'-Nitro-D-arginine
Cat.No: T9537
Synonym: N'-Nitro-D-arginine,H-D-Arg(NO2)-OH,(R)-2-Amino-5-(3-nitroguanidino)pentanoic acid,N'-硝基-D-精氨酸
Target: Others
TFEB activator 1
Cat.No: T8055
Synonym: (1E,4E)-1,5-Bis(2-Methoxyphenyl)penta-1,,Curcumin analog compound C1,Curcumin analog C1,(1E,4E)-1,5(2 -甲氧基苯基)-1,4-戊二烯-3-酮,RPN77612
Target: Others, Autophagy
Necroptosis-IN-3
Cat.No: T64349
Synonym: Cyclohexanecarboxamide, N-(2-thienylmethyl)-
Target: Necroptosis
Casein kinase 1δ-IN-3
Cat.No: T64350
Synonym:
Target: Casein Kinase
Benzothiazole-6-carboxylic acid
Cat.No: Fr12380
Synonym:
Target:
1-(2-fluorophenyl)-3-[5-(2-methoxyphenyl)-1,3,4-thiadiazol-2-yl]urea
Cat.No: T67696
Synonym:
Target: Others
Benzofuran-2-carboxylic acid
Cat.No: Fr13623
Synonym:
Target:
PBRM1-BD2-IN-3
Cat.No: T60158
Synonym:
Target: Epigenetic Reader Domain
Aminooxy-PEG3-azide
Cat.No: T14264
Synonym:
Target: Others
DIF-3
Cat.No: T60485
Synonym:
Target:
Acetyltrialanine
Cat.No: T20163
Synonym:
Target:
Flaviviruses-IN-3
Cat.No: T67777
Synonym: WAY-324593
Target: Virus Protease
(2E)-N-(4-methoxyphenyl)-3-[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-yl]prop-2-enamide
Cat.No: T50084
Synonym:
Target: Others
5-Bromo-4-chloro-3-indoxyl-beta-D-cellobioside
Cat.No: T60017
Synonym:
Target: Others
1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea
Cat.No: T60124
Synonym:
Target: TNF
Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-
Cat.No: T9872
Synonym:
Target: Others
1-ethyl-6-fluoro-4-oxo-7-[4-(3-phenylpropanoyl)piperazin-1-yl]-1,4-dihydroquinoline-3-carboxylic acid
Cat.No: T50070
Synonym:
Target: Others
2-Methyl-2H-indazole-3-carboxylic acid
Cat.No: Fr21265
Synonym:
Target:
3-hydroxycephem
Cat.No: T4581
Synonym:
Target: Others
5-Methoxyindole-3-carboxaldehyde
Cat.No: T5151
Synonym:
Target: Others
SU5208
Cat.No: T22432
Synonym: 3-[(Thien-2-yl)methylene]-2-indolinone
Target: VEGFR
ALDH1A3-IN-3
Cat.No: T64347
Synonym:
Target: Dehydrogenase
3-Methoxy-9H-Carbazole
Cat.No: T77681
Synonym:
Target: Apoptosis
TGFβ1-IN-3
Cat.No: T75005
Synonym:
Target: Others
Erdafitinib
Cat.No: T3726
Synonym: 厄达替尼,JNJ-42756493
Target: Apoptosis, FGFR
5-HT3 antagonist 3
Cat.No: T10162
Synonym:
Target: 5-HT Receptor
Cathepsin X-IN-1
Cat.No: T60812
Synonym:
Target: Cysteine Protease
6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole
Cat.No: T50028
Synonym: 6-氟-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚,6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Target: Others
WIC1
Cat.No: T67923
Synonym:
Target: Others
1,3-diethyl 2-(3-methoxyphenyl)propanedioate
Cat.No: T50051
Synonym:
Target: Others
LDHA-IN-3
Cat.No: T39805
Synonym: PSTMB,1-(phenylseleno)-4-(trifluoromethyl) benzene
Target: Dehydrogenase
GLP-1R agonist 3
Cat.No: T63909
Synonym:
Target: Glucagon Receptor
Watermelon ketone
Cat.No: T13965
Synonym: 7-Methyl-2H-1,5-benzodioxepin-3(4H)-one,西瓜酮
Target: Others
2-Bromo-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine
Cat.No: T90421
Synonym:
Target:
INT. 2
Cat.No: T9795
Synonym:
Target:
2H-1-Benzopyran-3-carboxylic acid, 3,4-dihydro-6-Methoxy-, (3S)-
Cat.No: T9798
Synonym:
Target:
FLT3-IN-10
Cat.No: T9856
Synonym: 2-Oxazolamine, 5-(4-fluorophenyl)-N-phenyl-
Target: FLT
3-Ethyl-1-methyl-2-thioxoimidazolidin-4-one
Cat.No: T50122
Synonym:
Target:
Copper(II) gluconate
Cat.No: T65090
Synonym:
Target:
3’-O-Methyladenosine
Cat.No: TNU0060
Synonym:
Target: Antiviral, Adenosine deaminase
CB2R/FAAH modulator-3
Cat.No: T67747
Synonym:
Target: Cannabinoid Receptor, FAAH
Cat. No. Product Name Target Signaling Pathways
TC0036 Compound Lup-20(29)-en-3-yl acetate

IL Receptor; VEGFR; Others; TNF; COX Angiogenesis; Apoptosis; Immunology/Inflammation; Neuroscience; Others; Tyrosine Kinase/Adaptors
Lup-20(29)-en-3-yl acetate 是 Lupeol 的衍生物,通过下调 TNF-α、IL-1β、MCP-1、COX-2、VEGF 和颗粒酶 B 来抑制类风湿性关节炎的进展。
TN6410 New compound 3

New compound 3 可用于生命科学领域的相关研究,其产品编号为 TN6410。
TN1264 3'-O-Methylbatatasin III

Antifungal Microbiology/Virology
3'-O-Methylbatatasin III 是一种来自兰科植物白芨的天然化合物,具有抗生素活性和解痉活性。3'-O-Methylbatatasin III 具有抗真菌活性。
T5277 3-Furanoic acid

3-Furoic acid,3-糠酸,3-Carboxyfuran,3-Furancarboxylic acid

Others; Endogenous Metabolite Metabolism; Others
3-Furanoic acid (3-Carboxyfuran) 是内源性代谢产物的一种。
TN1819 Kaempferol 3-neohesperidoside

Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷

GSK-3; MEK; PI3K MAPK; PI3K/Akt/mTOR signaling; Stem Cells
Kaempferol 3-neohesperidoside (Kaempferol 3-O-neohesperidoside) 是一种类黄酮,对大鼠比目鱼肌具有拟胰岛素作用。
TN7247 Limocitrin 3-O-sophoroside

Limocitrinyle-3-O-β-D-sophoroside

Limocitrin 3-O-sophoroside 是一种可用于生物研究的化合物。
TN2883 3',4'-Dimethoxyflavone

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。
T64343 3-Methylcarbazole

NSC 10154

Others Others
3-Methylcarbazole (NSC-10154) 是具有抗癌作用的咔唑生物碱化合物。3-Methylcarbazole 对人纤维肉瘤 HT-1080 细胞具有生长抑制活性 (IC50 为 25 μg/mL)。
T5653 Cinnamyl acetate

3-Phenylallyl acetate,乙酸桂酯

Others Others
Cinnamyl acetate (3-Phenylallyl acetate) 是一种新型广谱抗菌剂,广泛应用于香料和香料工业。
T4778 3-Hydroxybenzaldehyde

Others; Dehydrogenase Metabolism; Others
3-Hydroxybenzaldehyde 是很多酚类化合物的前体分子。它是人和大鼠醛脱氢酶 (ALDH) 的底物 (substrate)。它具有血管保护的作用。
T2769 3-Aminopropionitrile fumarate (2:1)

Di-β-aminopropionitrile fumarate,3-Aminopropionitrile fumarate,3-氨基丙腈,β-Aminopropionitrile fumarate,3-Aminopropionitrile fumarate 2:1,Beta-Aminopropionitrile fumarate,β-Ammoniumpropionitrile hemifumarate

Others Others
3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) 是一种能抑制胶原蛋白(collagen)交联的山黧豆素。
T4702 (3-Carboxypropyl)trimethylammonium chloride

γ-Butyrobetaine hydrochloride,(3-羧丙基)三甲基氯化铵,(3-Carboxypropyl)trimethylammonium chlor

Endogenous Metabolite Metabolism
(3-Carboxypropyl)trimethylammonium chloride ((3-Carboxypropyl)trimethylammonium chlor) 一种血管病变性中间代谢物,是由肠道微生物代谢产生,这些微生物以红肉中的肉碱为食。
T4455 DL-3-Phenyllactic acid

DL-3-苯乳酸,3-Phenyllactic acid,2-Hydroxy-3-phenylpropanoic acid

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
DL-3-Phenyllactic acid (3-Phenyllactic acid) 是广谱抗菌化合物,对细菌和真菌具有活性。
T8002 3-Hydroxycoumarin

Lipoxygenase Metabolism
3-hydroxycoumarin 是一种 15-LOX-1的有效氧化还原抑制剂,近期被证明能保护海胆生殖细胞免受紫外线 B 的损伤。
T4939 Indole-3-pyruvic acid

3-(3-吲哚基)-2-氧代丙酸,3-(3-Indolyl)-2-oxopropanoic acid

Others Others
Indole-3-pyruvic acid (3-(3-Indolyl)-2-oxopropanoic acid) 是一种参与Indole-3-acetic acid 生物合成的化合物,Indole-3-acetic acid 是一种植物激素,在调节生长和对环境变化的反应中起重要作用。
T39887 (S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid

(S)-3-(4-羟苯基)乳酸,(S)-3-(4-Hydroxyphenyl)lactic acid,(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid

Others Others
(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid ((S)-3-(4-Hydroxyphenyl)lactic acid) 是分离自间肠隐球菌培养基的代谢物,具有高的 DPPH 清除自由基活性和抗氧化活性。
T4773 3-Ethoxy-3-oxopropanoic acid

Monoethyl malonic acid,Ethyl hydrogen malonate,丙二酸单乙酯

Others; Endogenous Metabolite Metabolism; Others
3-Ethoxy-3-oxopropanoic acid (Monoethyl malonic acid) 是内源性代谢产物的一种。
T8051 Bis(2-methyl-3-furyl)disulfide

双(2-甲基-3-呋喃基)二硫,Bis(2-methyl-3-furyl)disulphide

Others Others
Bis(2-methyl-3-furyl)disulfide 是调味剂,能够增强与牛奶相关的产品的自然感,清新感。
T2893 Muscone

3-Methylcyclopentadecanone,Methylexaltone,麝香酮

MMP; TNF; NF-κB; NOD-like Receptor (NLR); P-gp; Interleukin Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Neuroscience; NF-κB; Proteases/Proteasome
Muscone (3-Methylcyclopentadecanone) 是中药麝香的一种主要活性单体。它抑制NF-κB 和NLRP3炎性小体的活化,显著降低炎性细胞因子水平,并最终改善心脏功能和存活率。
TN1049 Ingenol-5,20-acetonide

Others Others
Ingenol-5,20-acetonide 是一种天然化合物,Ingenol 3-Angelate 的类似物,当局部用于治疗光化性角化病时具有抗肿瘤活性。
TN2125 Quercetin 3-O-β-D-(6''-p-coumaroyl)glucopyranosyl(1→2)-α-L-rhamnopyranoside

3-O-{2-O-[6-O-(P羟基-反-香豆酰)-葡萄糖基]-鼠李糖基}槲皮素,Quercetin 3-O-beta-(6''-p-coumaroyl)glucopyranosyl(1->2)-alpha-L-rhamnopyranoside

Antioxidant oxidation-reduction
Quercetin 3-O-β-D-(6''-p-coumaroyl)glucopyranosyl(1→2)-α-L-rhamnopyranoside (Quercetin 3-O-beta-(6''-p-coumaroyl)glucopyranosyl(1->2)-alpha-L-rhamnopyranoside) 是一种从银杏叶中提取出来的化合物。Quercetin 3-O-β-D-(6''-p-coumaroyl)glucopyranosyl(1→2)-α-L-rhamnopyranoside 具有抗氧化的功能。
TN1043 Keracyanin chloride

Cyanidin-3-O-rutinoside chloride,Cyanidin 3-rutinoside chloride,Cyanidin 3-O-rutinoside chloride,花青素鼠李葡糖苷

COX Immunology/Inflammation; Neuroscience
Keracyanin chloride (Cyanidin 3-rutinoside chloride) 是一种花青素,能够抑制氧化的小牛胸腺 DNA 中丙二醛的形成,具有抗氧化作用。
Fr13883 3-Methoxyphenylacetic acid

Others Others
3-Methoxyphenylacetic acid 是 m-hydroxyphenylacetic (m-OHPAA) 的衍生物,茄形假丝酵母中的一种植物毒素。它可用于针对介氧菌根腐烂的毒素介导的生物测定法的开发。
T40607 2,4,6-Trimethylphenol

Mesitol

Others Others
2,4,6-Trimethylphenol (Mesitol) 是一种与有机物 (3DOM*) 反应的探针化合物,可在水溶液中被单线态氧快速氧化。
T5274 D-​(+)​-​Phenyllactic acid

D-3-苯乳酸,D-3-Phenyllactic acid

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
D-​(+)​-​Phenyllactic acid (D-3-Phenyllactic acid) 是一种由白地霉分泌得到的抗菌剂,可抑制部分来自人类和食品的革兰氏阳性菌以及来自人类的革兰氏阴性菌。
T2A2486 3',​4',​5',​5,​7-​Pentamethoxyflavone

5,7,3',4',5'-Pentamethoxyflavone

Nrf2 Immunology/Inflammation
3',4',5',5,7-Pentamethoxyflavone 是从 Rutaceae 中发现的的一种天然黄铜类化合物,通过抑制Nrf2 通路克服化疗活性分子从而对癌细胞展现出耐药性。
T9368 3,4-(Methylenedioxy)cinnamic acid

3-(Benzo[d][1,3]dioxol-5-yl)acrylic acid,3,4-(亚甲二氧)肉桂酸

Others Others
3,4-(Methylenedioxy)cinnamic acid (3-(Benzo[d][1,3]dioxol-5-yl)acrylic acid) 是一种植物衍生化合物,首先从芦笋的根中提取,并进一步表征为一种化感化学物质。
TN7029 (2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol

Others Others
(2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol 是一种有用的研究化合物,适用于许多研究应用,包括化学领域和生命科学领域等。
T2910 Flavonol

3-羟基黄酮,3-Hydroxyflavone,3-HF,Flavon-3-ol,3-Hydroxy-2-phenylchromone

Others; Endogenous Metabolite Metabolism; Others
Flavonol (3-Hydroxyflavone) 是内源性代谢产物的一种。
T0562 Protocatechuic acid

3, 4-Dihydroxybenzoic acid,3,4-二羟基苯甲酸,Protocatechuate,原儿茶酸,3,4-Dihydroxybenzoic acid

Others Others
Protocatechuic acid (3, 4-Dihydroxybenzoic acid) 是天然的多酚类物质,具有神经保护活性。
T5S1988 Isorhamnetin-3-O-glucoside

Isorhamnetin-3-O-beta-D-Glucoside,异鼠李素-3-O-葡萄糖苷

Others Others
Isorhamnetin-3-O-glucoside (Isorhamnetin-3-O-beta-D-Glucoside) 是一种天然化合物,广泛存在于蔬菜和水稻中,经消化后可在肠道菌群中代谢。
T22308 Dimboa

2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布

Others; Antibacterial; Antibiotic; Antifungal Microbiology/Virology; Others
Dimboa (2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one) 是抗生素,是禾本科植物化学防御系统的一部分。 它对许多已研究的细菌和真菌菌株具有生长抑制特性。它表现出强大的自由基清除活性和较弱的铁 (III) 离子还原活性和有抗氧化活性。
TN5263 1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one

Xanthohumol,黄腐酚

Apoptosis; BCL; PARP; HCV Protease; IAP; Caspase; HIV Protease; NMDAR; p53 Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Neuroscience; Proteases/Proteasome
1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one (Xanthohumol) 是一种从蛇麻草中提纯的具有多种生物功能的天然产物。黄腐酚对 HIV-1 有效,可能是一种有趣的先导化合物。它可能代表一种用于 HIV-1 感染的新型化疗药物。
T41095 (E)-3-(4-Methoxyphenyl)acrylic acid

(E)-3-(4-甲氧基苯基)丙烯酸

Glucosidase Metabolism
(E)-3-(4-Methoxyphenyl)acrylic acid 是从 Etlingera pavieana (Pierre ex Gagnep.) R. M. Sm. 的根茎中分离出来的一种小分子化合物。它是一种新型 α-葡萄糖苷酶抑制剂。(E)-3-(4-甲氧基苯基)丙烯酸具有保肝活性、抗失水活性、增强认知效果,并可用于降低血压血糖。
TQ0099 20-O-Acetylingenol-3-angelate

巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1

Others Others
20-O-Acetylingenol-3-angelate (Euphorbia factor Pe1) 是一种天然化合物,存在于植物英加的叶子和茎中。它具有多种生物活性,包括抑制肿瘤生长、抗炎、抗真菌和抗氧化作用。
T5764 Alliin

蒜氨酸,(S)-3-(Allylsulphinyl)-L-alanine

NF-κB; PPAR DNA Damage/DNA Repair; Metabolism; NF-κB
Alliin ((S)-3-(Allylsulphinyl)-L-alanine) 是一种从大蒜中提取的亚砜化合物,具有口服活性,表现出降血糖、抗氧化和抗炎特性。
T2871 Quercitrin

Sophoretin,3-rhamnosyl quercetin,Quercetin 3-rhamnoside,Xanthaurine,槲皮苷,Meletin

Reactive Oxygen Species; S6 Kinase; Autophagy Autophagy; Immunology/Inflammation; MAPK; Metabolism; NF-κB; PI3K/Akt/mTOR signaling
Quercitrin (3-rhamnosyl quercetin) 是苦荞麦中的一种天然产物,具有抗炎作用,有用于心血管疾病的研究潜力。
T8105 Indole-3-carboxaldehyde

3-Formylindole,3-吲哚甲醛

Endogenous Metabolite Metabolism
Indole-3-carboxaldehyde (3-Formylindole) 是由黄化豌豆幼苗的粗酶制剂氧化降解IAA 的产物,是一种卷心菜提取物。它可用于制备吲哚类植物抗毒素环芸香素类似物。
T5238 1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine

1,2-Dipalmitoyl-sn-glycero-3-PE,L-磷脂酰乙醇胺,1,2-Dipalmitoyl-sn-glycerol-3-Phosphoethanolamine,1,2-DPPE

Others; Endogenous Metabolite Metabolism; Others
1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine (DPPE) 是内源性代谢产物的一种。
T19384 Isovalerylcarnitine

Apoptosis; Cysteine Protease Apoptosis; Proteases/Proteasome
Isovalerylcarnitine (3-methylbutyrylcarnitine) 是 L-亮氨酸分解代谢和异戊酸的积累产生的小分子化合物,也是一种具有选择性和有效性的钙蛋白酶 (calpain) 激活剂,可促使细胞凋亡,与异戊酸血症有关,可作为异戊酸血症的标志。
T5290 (S)-2-Hydroxy-3-phenylpropanoic acid

L-(−)-3-Phenyllactic acid,L-3-苯乳酸

Others; Endogenous Metabolite Metabolism; Others
(S)-2-Hydroxy-3-phenylpropanoic acid (L-(−)-3-Phenyllactic acid) 是苯丙氨酸的代谢产物。苯丙酮尿症患者体液中苯丙氨酸的水平升高。
T4768 Diethyl oxalpropionate

草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE

Others; Endogenous Metabolite Metabolism; Others
Diethyl oxalpropionate (HYL 2-METHYL-3-OXOSUCCINATE) 是一种合成 PDMMLA 的中间体。其中 PDMMLA 的衍生物可用于纳米粒子的合成和研究。
T8274 3-Methyl-L-histidine

Endogenous Metabolite Metabolism
3-Methyl-L-histidine 是一种肉类尤其是鸡肉摄入和大豆制品摄入的生物标记。
T4S0350 Licochalcone B

甘草查尔酮 B,甘草查尔酮B

Beta Amyloid; Others Neuroscience; Others
Licochalcone B 是从Glycyrrhiza inflate 根中提取的。它能够抑制淀粉样蛋白 β 自聚集作用 (IC50=2.16 μM) ,分解预先形成的 Aβ42原纤维,并通过螯合金属离子抑制金属诱导的 Aβ42聚集。
T4S21320 ISOGINKGETIN

异银杏素,4',4'''-Dimethylamentoflavone,异银杏双黄酮

MMP; Others Others; Proteases/Proteasome
ISOGINKGETIN (4',4'''-Dimethylamentoflavone) 是一种MMP9抑制剂,也是一种Pre-mRNA Splicing 抑制剂。
TCS1772 Dehydroabietic acid

Dehydroabietate,脱氢松香酸

Antifection Microbiology/Virology
Dehydroabietic acid (Dehydroabietate) 是 EBV-EA 活化抑制剂。 它是食物衍生化合物,可通过降低血浆葡萄糖、胰岛素水平、血浆甘油三酯 (TG) 和肝 TG 水平来治疗肥胖相关疾病。它的衍生物在动物模型中表现出抗分泌和抗胃蛋白酶作用。
T19866 Indican

NSC-87517,3-Indoxyl-beta-D-glucopyranoside,3-吲哚基-beta-D-吡喃葡萄糖苷,NSC 87517,NSC87517,Indoxyl-β-D-glucoside

OAT; MRP Immunology/Inflammation; Membrane transporter/Ion channel
Indican (Indoxyl-β-D-glucoside) 是吲哚酚的一种糖苷,染料靛蓝和靛玉红的前体。它的主要代谢物是硫酸吲哚酚 (IS)。其中 IS 是尿毒症毒素,是有机阴离子转运蛋白1 (OAT 1)、OAT 3 和多药耐药相关蛋白4 (MRP 4) 的底物/抑制剂。
T7452 2-methoxycinnamaldehyde

2'-甲氧基肉桂醛,O-methoxycinnamaldehyde

Apoptosis; Others Apoptosis; Others
2-methoxycinnamaldehyde 是一种肉桂中的天然产物。它能通过使线粒体膜电位 (ΔΨm) 损失 、激活 caspase-3 和 caspase-9,来抑制细胞增殖和诱导细胞凋亡,具有抗肿瘤活性。它还能抑制血小板衍生生长因子诱导的 HASMC 迁移。
TCS2170 2,5-Dihydroxyacetophenone

Quinacetophenone,2-Acetylhydroquinone,2-5-dihydroxyacetophenone,2 ',5'-二羟基苯乙酮,Acetylhydroquinone,2,5-二羟基苯乙酮,DHAP

ERK; NF-κB; Tyrosinase MAPK; NF-κB; Proteases/Proteasome
2,5-Dihydroxyacetophenone (Quinacetophenone) 是从熟地黄中分离出的一种天然产物,通过阻断 ERK1/2和 NF-κB 信号通路,抑制活化巨噬细胞中炎症介质的产生。
TN1880 Lucidenic acid B

Lucidenicacid B

Apoptosis; Caspase Apoptosis; Proteases/Proteasome
Lucidenic acid B (Lucidenicacid B) 是从灵芝中提取得到的天然化合物,可诱导caspase-9 和 caspase-3 的活化和 PARP 的裂解,可通过线粒体介导诱导人白血病细胞凋亡 。 Lucidenic acid B通过灭活MAPK / ERK信号转导途径和降低NF-kappaB和AP-1的结合活性来抑制PMA诱导的人肝癌细胞侵袭。。Lucidenic acid B 对细胞周期和坏死细胞没有影响。
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天然产物

Compound Lup-20(29)-en-3-yl acetate
Cat.No: TC0036
Synonym:
Target: IL Receptor, VEGFR, Others, TNF, COX
New compound 3
Cat.No: TN6410
Synonym:
Target:
3'-O-Methylbatatasin III
Cat.No: TN1264
Synonym:
Target: Antifungal
3-Furanoic acid
Cat.No: T5277
Synonym: 3-Furoic acid,3-糠酸,3-Carboxyfuran,3-Furancarboxylic acid
Target: Others, Endogenous Metabolite
Kaempferol 3-neohesperidoside
Cat.No: TN1819
Synonym: Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷
Target: GSK-3, MEK, PI3K
Limocitrin 3-O-sophoroside
Cat.No: TN7247
Synonym: Limocitrinyle-3-O-β-D-sophoroside
Target:
3',4'-Dimethoxyflavone
Cat.No: TN2883
Synonym:
Target: Others, PARP
3-Methylcarbazole
Cat.No: T64343
Synonym: NSC 10154
Target: Others
Cinnamyl acetate
Cat.No: T5653
Synonym: 3-Phenylallyl acetate,乙酸桂酯
Target: Others
3-Hydroxybenzaldehyde
Cat.No: T4778
Synonym:
Target: Others, Dehydrogenase
3-Aminopropionitrile fumarate (2:1)
Cat.No: T2769
Synonym: Di-β-aminopropionitrile fumarate,3-Aminopropionitrile fumarate,3-氨基丙腈,β-Aminopropionitrile fumarate,3-Aminopropionitrile fumarate 2:1,Beta-Aminopropionitrile fumarate,β-Ammoniumpropionitrile hemifumarate
Target: Others
(3-Carboxypropyl)trimethylammonium chloride
Cat.No: T4702
Synonym: γ-Butyrobetaine hydrochloride,(3-羧丙基)三甲基氯化铵,(3-Carboxypropyl)trimethylammonium chlor
Target: Endogenous Metabolite
DL-3-Phenyllactic acid
Cat.No: T4455
Synonym: DL-3-苯乳酸,3-Phenyllactic acid,2-Hydroxy-3-phenylpropanoic acid
Target: Others, Endogenous Metabolite, Antibacterial
3-Hydroxycoumarin
Cat.No: T8002
Synonym:
Target: Lipoxygenase
Indole-3-pyruvic acid
Cat.No: T4939
Synonym: 3-(3-吲哚基)-2-氧代丙酸,3-(3-Indolyl)-2-oxopropanoic acid
Target: Others
(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid
Cat.No: T39887
Synonym: (S)-3-(4-羟苯基)乳酸,(S)-3-(4-Hydroxyphenyl)lactic acid,(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid
Target: Others
3-Ethoxy-3-oxopropanoic acid
Cat.No: T4773
Synonym: Monoethyl malonic acid,Ethyl hydrogen malonate,丙二酸单乙酯
Target: Others, Endogenous Metabolite
Bis(2-methyl-3-furyl)disulfide
Cat.No: T8051
Synonym: 双(2-甲基-3-呋喃基)二硫,Bis(2-methyl-3-furyl)disulphide
Target: Others
Muscone
Cat.No: T2893
Synonym: 3-Methylcyclopentadecanone,Methylexaltone,麝香酮
Target: MMP, TNF, NF-κB, NOD-like Receptor (NLR), P-gp, Interleukin
Ingenol-5,20-acetonide
Cat.No: TN1049
Synonym:
Target: Others
Quercetin 3-O-β-D-(6''-p-coumaroyl)glucopyranosyl(1→2)-α-L-rhamnopyranoside
Cat.No: TN2125
Synonym: 3-O-{2-O-[6-O-(P羟基-反-香豆酰)-葡萄糖基]-鼠李糖基}槲皮素,Quercetin 3-O-beta-(6''-p-coumaroyl)glucopyranosyl(1->2)-alpha-L-rhamnopyranoside
Target: Antioxidant
Keracyanin chloride
Cat.No: TN1043
Synonym: Cyanidin-3-O-rutinoside chloride,Cyanidin 3-rutinoside chloride,Cyanidin 3-O-rutinoside chloride,花青素鼠李葡糖苷
Target: COX
3-Methoxyphenylacetic acid
Cat.No: Fr13883
Synonym:
Target: Others
2,4,6-Trimethylphenol
Cat.No: T40607
Synonym: Mesitol
Target: Others
D-​(+)​-​Phenyllactic acid
Cat.No: T5274
Synonym: D-3-苯乳酸,D-3-Phenyllactic acid
Target: Endogenous Metabolite, Antibacterial
3',​4',​5',​5,​7-​Pentamethoxyflavone
Cat.No: T2A2486
Synonym: 5,7,3',4',5'-Pentamethoxyflavone
Target: Nrf2
3,4-(Methylenedioxy)cinnamic acid
Cat.No: T9368
Synonym: 3-(Benzo[d][1,3]dioxol-5-yl)acrylic acid,3,4-(亚甲二氧)肉桂酸
Target: Others
(2S)-1-O-p-coumaroyl-2-O-acetyl-3-O-β-D-glucopyranosylglycerol
Cat.No: TN7029
Synonym:
Target: Others
Flavonol
Cat.No: T2910
Synonym: 3-羟基黄酮,3-Hydroxyflavone,3-HF,Flavon-3-ol,3-Hydroxy-2-phenylchromone
Target: Others, Endogenous Metabolite
Protocatechuic acid
Cat.No: T0562
Synonym: 3, 4-Dihydroxybenzoic acid,3,4-二羟基苯甲酸,Protocatechuate,原儿茶酸,3,4-Dihydroxybenzoic acid
Target: Others
Isorhamnetin-3-O-glucoside
Cat.No: T5S1988
Synonym: Isorhamnetin-3-O-beta-D-Glucoside,异鼠李素-3-O-葡萄糖苷
Target: Others
Dimboa
Cat.No: T22308
Synonym: 2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one,丁布
Target: Others, Antibacterial, Antibiotic, Antifungal
1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one
Cat.No: TN5263
Synonym: Xanthohumol,黄腐酚
Target: Apoptosis, BCL, PARP, HCV Protease, IAP, Caspase, HIV Protease, NMDAR, p53
(E)-3-(4-Methoxyphenyl)acrylic acid
Cat.No: T41095
Synonym: (E)-3-(4-甲氧基苯基)丙烯酸
Target: Glucosidase
20-O-Acetylingenol-3-angelate
Cat.No: TQ0099
Synonym: 巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1
Target: Others
Alliin
Cat.No: T5764
Synonym: 蒜氨酸,(S)-3-(Allylsulphinyl)-L-alanine
Target: NF-κB, PPAR
Quercitrin
Cat.No: T2871
Synonym: Sophoretin,3-rhamnosyl quercetin,Quercetin 3-rhamnoside,Xanthaurine,槲皮苷,Meletin
Target: Reactive Oxygen Species, S6 Kinase, Autophagy
Indole-3-carboxaldehyde
Cat.No: T8105
Synonym: 3-Formylindole,3-吲哚甲醛
Target: Endogenous Metabolite
1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine
Cat.No: T5238
Synonym: 1,2-Dipalmitoyl-sn-glycero-3-PE,L-磷脂酰乙醇胺,1,2-Dipalmitoyl-sn-glycerol-3-Phosphoethanolamine,1,2-DPPE
Target: Others, Endogenous Metabolite
Isovalerylcarnitine
Cat.No: T19384
Synonym:
Target: Apoptosis, Cysteine Protease
(S)-2-Hydroxy-3-phenylpropanoic acid
Cat.No: T5290
Synonym: L-(−)-3-Phenyllactic acid,L-3-苯乳酸
Target: Others, Endogenous Metabolite
Diethyl oxalpropionate
Cat.No: T4768
Synonym: 草酰丙酸二乙酯,HYL 2-METHYL-3-OXOSUCCINATE
Target: Others, Endogenous Metabolite
3-Methyl-L-histidine
Cat.No: T8274
Synonym:
Target: Endogenous Metabolite
Licochalcone B
Cat.No: T4S0350
Synonym: 甘草查尔酮 B,甘草查尔酮B
Target: Beta Amyloid, Others
ISOGINKGETIN
Cat.No: T4S21320
Synonym: 异银杏素,4',4'''-Dimethylamentoflavone,异银杏双黄酮
Target: MMP, Others
Dehydroabietic acid
Cat.No: TCS1772
Synonym: Dehydroabietate,脱氢松香酸
Target: Antifection
Indican
Cat.No: T19866
Synonym: NSC-87517,3-Indoxyl-beta-D-glucopyranoside,3-吲哚基-beta-D-吡喃葡萄糖苷,NSC 87517,NSC87517,Indoxyl-β-D-glucoside
Target: OAT, MRP
2-methoxycinnamaldehyde
Cat.No: T7452
Synonym: 2'-甲氧基肉桂醛,O-methoxycinnamaldehyde
Target: Apoptosis, Others
2,5-Dihydroxyacetophenone
Cat.No: TCS2170
Synonym: Quinacetophenone,2-Acetylhydroquinone,2-5-dihydroxyacetophenone,2 ',5'-二羟基苯乙酮,Acetylhydroquinone,2,5-二羟基苯乙酮,DHAP
Target: ERK, NF-κB, Tyrosinase
Lucidenic acid B
Cat.No: TN1880
Synonym: Lucidenicacid B
Target: Apoptosis, Caspase
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