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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T7740 Protease-Activated Receptor-4 diTFA

Protease-Activated Receptor-4 diTFA(245443-52-1(free base))

Protease-activated Receptor GPCR/G Protein
Protease-Activated Receptor-4 diTFA 是蛋白酶激活受体 4 (PAR4) 激动剂。
T7513 Protease-Activated Receptor-2, amide

蛋白酶活化的受体-2,酰胺,SLIGKV-NH2,H-丝氨酰亮氨酰异亮氨酰甘氨酰赖氨酰缬氨酰NH2

Protease-activated Receptor GPCR/G Protein
Protease-Activated Receptor-2, amide (SLIGKV-NH2) 是 PAR2 的激动剂,IC50为 10.4 M。
T38836L Protease-Activated Receptor-1, PAR-1 Agonist acetate

Protease-activated Receptor GPCR/G Protein
Protease-Activated Receptor-1, PAR-1 Agonist acetate 是一种选择性蛋白酶激活受体 1 (PAR-1) 激动剂肽。 它对应于 PAR1 栓系配体,可以选择性地模拟凝血酶通过该受体的作用。
TP1046 SLIGRL-NH2

Protease-Activated Receptor-2 Activating Peptide

Protease-activated Receptor GPCR/G Protein
SLIGRL-NH2 (Protease-Activated Receptor-2 Activating Peptide) 为一种蛋白酶激活受体-2 (PAR-2) 激动剂,具有诱导非组胺能性瘙痒的功能。
T10925L Cysteine Protease inhibitor hydrochloride

Cysteine Protease inhibitor hydrochloride (921625-62-9 free base)

Others Others
Cysteine Protease inhibitor hydrochloride 是一种半胱氨酸蛋白酶(cysteine protease)抑制剂。
T39729 HIV Protease Substrate 1

HIV Protease Substrate 1 is a fluorogenic compound that offers insights into the enzymatic activity of HIV protease, making it a valuable tool for studying this aspect.
T8936 Proteinase K

proteinase K for tritirachium album,Protease K,蛋白酶 K

Others Others
Proteinase K (proteinase K for tritirachium album) 是一种非特异性丝氨酸蛋白酶,可用于蛋白消化。它在有 SDS 或尿素存在的情况下,在很大 pH 值 (4-12)、盐浓度和温度单位内均有活性。
T10924 Cysteine protease inhibitor-2

Cysteine Protease Proteases/Proteasome
Cysteine protease inhibitor-2 是半胱氨酸蛋白酶抑制剂。
T10925 Cysteine Protease inhibitor

Others Others
Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease
T39503 Hepatitis Virus C NS3 Protease Inhibitor 2

Hepatitis Virus C NS3 Protease Inhibitor 2 is a peptide inhibitor derived from a product that targets the NS3 protease of the hepatitis C virus (HCV). Its inhibitory activity against the NS3 protease is characterized by a Ki value of 41 nM.
T7380 Protease-Activated Receptor-4

蛋白酶活化的受体-4

Protease-activated Receptor GPCR/G Protein
Protease-Activated Receptor-4 是蛋白酶激活受体 4 激动剂,具有抗血小板治疗。
TQ0129 TNF Protease Inhibitor 2

TAPI-2

MMP Proteases/Proteasome
TAPI-2 is a broad-spectrum inhibitor of MMP (IC50: 20 μM), tumour necrosis factorα-converting enzyme (TACE) and a disintegrin and metalloproteinase (ADAM).
T38836 Protease-Activated Receptor-1, PAR-1 Agonist

Protease-Activated Receptor-1 (PAR-1) Agonist, a selective peptide, activates the PAR-1 receptor by mimicking the specific actions of thrombin. It corresponds to the PAR1 tethered ligand, facilitating selective activation of this receptor.
T23486 ubiquitin specific protease 3 fragment

Others Others
The ubiquitin speci c protease 3 USP3 is a deubiquitinating enzyme for uH2A and uH2B.
T36288 Protease-Activated Receptor-1, PAR-1 Agonist TFA

Protease-Activated Receptor-1 (PAR-1) Agonist TFA is a selective peptide that acts as an agonist for the proteinase-activated receptor-1 (PAR-1). Corresponding to the tethered ligand of PAR-1, this compound mimics the actions of thrombin through the PAR-1 receptor[1][2].
T78363 Aspergillopepsin I

Aspergillus acid protease

Aspergillopepsin I (Aspergillus acid protease) 是一种属于天冬氨酸内肽酶类,能广泛特异性催化水解蛋白质中的肽键。
T36289 Protease-Activated Receptor-3 (PAR-3) (1-6), human TFA

Protease-Activated Receptor-3 (PAR-3) (1-6), human TFA is a peptide that acts as an agonist for the proteinase-activated receptor (PAR-3)[1].
T76155 Glutamic acid protease

谷氨酸蛋白酶仅存在于真菌中,为一种含谷氨酸残基的蛋白水解酶。
T76511 HIV Protease Substrate IV

HIV ProteaseSubstrate IV 是 HIV 蛋白酶的底物。HIV ProteaseSubstrate IV 可用于检测 HIV(人类免疫缺陷病毒)-1 蛋白酶的活性。
TP1046L PAR-2 Activating Peptide acetate

SLIGRL-NH2 acetate,PAR-2 Activating Peptide acetate(171436-38-7 free base),Protease-Activated Receptor-2 Activating Peptide acetate

Protease-activated Receptor GPCR/G Protein
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate)(171436-38-7 free base) 是 Protease-Activated Receptor-2 (PAR-2) 的激动剂。
T79277 Cysteine protease inhibitor-3

Parasite Microbiology/Virology
Cysteine protease Inhibitor-3 (Compound 15) 是抗疟作用的半胱氨酸蛋白酶抑制剂,能够有效地抑制 Pf3D7、PfW2、PfFP2 和 PfFP3,其 IC50 分别为 0.74 μM、1.05 μM、3.5 μM 和 4.9 μM。该化合物对药物敏感性和耐药性寄生虫均有效。
T76485 HIV Protease Substrate I

HIV ProteaseSubstrate I 是HIV-1蛋白酶的显色底物。HIV ProteaseSubstrate I 具有HIV 蛋白酶的裂解位点。
T36286 Protease-Activated Receptor-3 (PAR-3) (1-6), human

TFRGAP-amide, human PAR-3-derived tethered ligand sequence which does not activate PAR-3 but rather activates PAR-1 and PAR-2, either in Jurkat or in other PAR-expressing cells.
T74939 HIV protease-IN-1

HIVprotease-IN-1 (compound 1·succinate) 是一种有效的HIV 蛋白酶 (HIV protease) 非肽抑制剂,可用于艾滋病的研究。
T79493 HIV-1 protease-IN-10

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
HIV-1protease-IN-10(化合物2)显示出对HIV-1潜伏期的逆转活性,IC50值为0.22 μM。该化合物通过与PKCδC1b结构域结合展现活性,IC50值为0.69 μM。此外,HIV-1protease-IN-10对于酯酶介导的水解表现出稳定性。
T80691 β-Herpesvirus protease-IN-1

Virus Protease Microbiology/Virology
β-Herpesvirus protease-IN-1 (compound 19)为一种针对β-herpesvirus蛋白酶的抑制剂,其对HCMVPro的IC50值为2.5 μM,而对HHV6Pro的IC50值则为0.33 μM。
T76074 HIV Protease Substrate 1 TFA

HIV ProteaseSubstrate 1 TFA 是一种外源性 HIV 蛋白酶底物,可用于研究 HIV 蛋白酶的酶活性。
T64112 HIV-1 protease-IN-5

HIV-1 protease-IN-5 是一种 HIV-1 protease 抑制剂 (IC50: 1.64 nM)。HIV-1 protease-IN-5 对野生型和 DRV 耐药型 HIV-1 表现出明显的作用。
T63949 HIV-1 protease-IN-2

HIV-1 protease-IN-2 是 HIV-1 protease 的有效抑制剂 (IC50: 2.53 nM)。HIV-1 protease-IN-2 对 DRV (达芦那韦)敏感或耐药性 HIV-1 突变体均表现出抗病毒效果。
T63453 HIV-1 protease-IN-1

HIV-1 protease-IN-1 是 HIV-1 蛋白酶的有效抑制剂 (IC50: 90 pM)。HIV-1 protease-IN-1 对 B-HIV 具有抗病毒活性 (EC50: 89 nM)。HIV-1 protease-IN-1 能够作用于 C-HIV 毒株 ZM246 (EC50: 13.59 nM) 以及 C-HIV 株 Indie (EC50: 8.23 nM)。
T79536 HIV-1 protease-IN-11

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1protease-IN-11 (compound 34a) 为一抗HIV-1蛋白酶抑制剂,其IC50值为0.41 nM,并对抗耐药变异表现出显著活性。
T74942 HIV-1 protease-IN-7

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1protease-IN-7(化合物 16)作为一种HIV-1蛋白酶抑制剂,具有良好的口服活性,表现出优异的抑制效能(IC50=3.52 nM,EC50=37 nM)。
T79295 HIV-1 protease-IN-9

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1protease-IN-9 (compound 5b)为HIV-1蛋白酶抑制剂,具有0.028 nM的Ki值和66.8 nM的IC50,表现出显著的抗病毒活性。
T63733 HIV-1 protease-IN-6

HIV-1 protease-IN-6 (compound 17d) 是 HIV-1 蛋白酶 (HIV-1 protease) 的有效抑制剂 (IC50: 21 pM, Ki: 4.7 pM)。HIV-1 protease-IN-6 对 DRV (darunavir) 耐药病毒突变体具有显著的抗病毒效果 (antiviral activity),抑制强度甚至超过对野生型病毒。
T78950 HIV-1 protease-IN-8

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1protease-IN-8(compound 34b)是一款高效的HIV-1蛋白酶抑制剂,其IC50为0.32 nM。该化合物对野生型HIV-1(HIV-1NL4-3)及耐药变体(HIV-1MDR)的IC50分别为0.29 μM与1.90 μM,表明其对这两种型别均展现出显著的抗病毒效果。
T74488 HIV-1 protease-IN-4

HIV-1protease-IN-4 (Compound II-22) 是一种有效的HIV-1蛋白酶抑制剂。HIV-1protease-IN-4 是阿扎那韦的前体。HIV-1蛋白酶-IN-4 作为前体,与口服母体活性分子相比,将母体 1 输送到大鼠血浆中的 AUC 高 5 倍,C24 高 67 倍[1]。
T79537 HIV-1 protease-IN-12

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1protease-IN-12 (compound 35b)为HIV-1蛋白酶抑制剂,具有0.51 nM的IC50值,同时对HIV耐药变体也具有抑制作用。
T75902 SLIGRL-NH2 TFA

Protease-Activated Receptor-2 Activating Peptide TFA

SLIGRL-NH2 TFA(Protease-Activated Receptor-2 Activating Peptide TFA)作为PAR-2(蛋白酶激活受体-2)的激动剂,具有高度特异性。
T1307 Carmofur

HCFU,卡莫氟

Nucleoside Antimetabolite/Analog; Virus Protease; SARS-CoV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Carmofur (HCFU) 是 5-氟尿嘧啶的衍生物,是一种抗肿瘤药物。它是一种酸性神经酰胺酶抑制剂,用于治疗乳腺癌和结直肠癌。它抑制 SARS-CoV-2主要蛋白酶,还抑制 Vero E6 细胞 SARS-CoV-2,EC50为 24.3 μM。
T6327 Tubacin

Virus Protease; HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology
Tubacin 是一种高效、选择性、可逆、可渗透细胞的 HDAC6 抑制剂,IC50 为 4 nM,选择性是 HDAC1 的约 350 倍。
T62507 Protease-Activated Receptor-1 antagonist 1

Protease-Activated Receptor-1 antagonist 1 (Compound 13) 是一种蛋白酶激活受体 1 (PAR-1) 拮抗剂,通过 FLIPR 技术得到的 IC50 为 3 nM。Protease-Activated Receptor-1 antagonist 1 能够用于研究血栓性心血管、心肌梗塞和外周动脉疾病。
T64285 Protease-Activated Receptor-1 antagonist 2

Protease-Activated Receptor-1 antagonist 2 是一种选择性的、口服具有活力的蛋白酶激活受体-1 (PAR-1) 拮抗剂 (IC50: 7 nM)。Protease-Activated Receptor-1 antagonist 2 显示出良好的药代动力学特性,能够用于进行心血管疾病 (CVD) 的相关研究(如动脉粥样硬化和再狭窄)。
T74266 Protease-Activated Receptor-1 antagonist 2

Protease-Activated Receptor-1 antagonist 2 是一种选择性蛋白酶激活受体-1 (PAR-1) 拮抗剂,口服活性,IC50值为7 nM。该化合物具有优良的药代动力学特性,适用于心血管疾病 (CVD) 如动脉粥样硬化和再狭窄的研究。
T63382 Protease-Activated Receptor-1 antagonist 3

Protease-Activated Receptor-1 antagonist 3 是蛋白酶激活受体 1protease-activated receptor-1 的有效拮抗剂 (IC50: 7 nM)。Protease-Activated Receptor-1 antagonist 3 与 hERG K+通道表现出结合亲和力 (IC50: 9 μM)。
T76502 HIV-1, HIV-2 Protease Substrate

HIV-1,HIV-2Protease Substrate 是HIV-1,HIV-2蛋白酶的底物。HIV-1和HIV-2蛋白酶底物结合残基有 4 个保守取代残基。
T8350 TPCK

Proteasome Proteases/Proteasome; Ubiquitination
TPCK 是丝氨酸蛋白酶抑制剂,通过与 HPV-18 E7 蛋白的视网膜母细胞瘤蛋白 (RB) 结合核心发生反应,并能够消除其 RB 结合能力。将它添加到培养基内,可修饰活角质形成细胞中的 E7 蛋白。
T1883 Des(benzylpyridyl) Atazanavi

HIV Protease Microbiology/Virology; Proteases/Proteasome
Des(benzylpyridyl) Atazanavi 是 Atazanavir 的 N-脱烷基代谢物 (M1),一种 HIV 蛋白酶抑制剂。
T13408 ZK824190

Others; Serine Protease Others; Proteases/Proteasome
ZK824190 是具有口服活性尿激酶型纤溶酶原激活剂 (uPA) 选择性抑制剂,对 uPA,tPA 和 Plasmin 的IC50分别为 237,1600 和 1850 nM。ZK824190在多发性硬化症中有研究价值。
T13397 ZINC03129319

Virus Protease Microbiology/Virology
ZINC03129319 是有效的登革病毒 NS2B-NS3蛋白酶抑制剂,抑制常数 Ki1和 Ki3分别为 92 μM 和 20 μM。
T2244 ESI-09

cAMP; Virus Protease GPCR/G Protein; Microbiology/Virology
ESI-09是一种新型非环状核苷酸EPAC 的拮抗剂,对EPAC1和EPAC2的IC50值分别为3.2和1.4 μM。

化合物

Protease-Activated Receptor-4 diTFA
Cat.No: T7740
Synonym: Protease-Activated Receptor-4 diTFA(245443-52-1(free base))
Target: Protease-activated Receptor
Protease-Activated Receptor-2, amide
Cat.No: T7513
Synonym: 蛋白酶活化的受体-2,酰胺,SLIGKV-NH2,H-丝氨酰亮氨酰异亮氨酰甘氨酰赖氨酰缬氨酰NH2
Target: Protease-activated Receptor
Protease-Activated Receptor-1, PAR-1 Agonist acetate
Cat.No: T38836L
Synonym:
Target: Protease-activated Receptor
SLIGRL-NH2
Cat.No: TP1046
Synonym: Protease-Activated Receptor-2 Activating Peptide
Target: Protease-activated Receptor
Cysteine Protease inhibitor hydrochloride
Cat.No: T10925L
Synonym: Cysteine Protease inhibitor hydrochloride (921625-62-9 free base)
Target: Others
HIV Protease Substrate 1
Cat.No: T39729
Synonym:
Target:
Proteinase K
Cat.No: T8936
Synonym: proteinase K for tritirachium album,Protease K,蛋白酶 K
Target: Others
Cysteine protease inhibitor-2
Cat.No: T10924
Synonym:
Target: Cysteine Protease
Cysteine Protease inhibitor
Cat.No: T10925
Synonym:
Target: Others
Hepatitis Virus C NS3 Protease Inhibitor 2
Cat.No: T39503
Synonym:
Target:
Protease-Activated Receptor-4
Cat.No: T7380
Synonym: 蛋白酶活化的受体-4
Target: Protease-activated Receptor
TNF Protease Inhibitor 2
Cat.No: TQ0129
Synonym: TAPI-2
Target: MMP
Protease-Activated Receptor-1, PAR-1 Agonist
Cat.No: T38836
Synonym:
Target:
ubiquitin specific protease 3 fragment
Cat.No: T23486
Synonym:
Target: Others
Protease-Activated Receptor-1, PAR-1 Agonist TFA
Cat.No: T36288
Synonym:
Target:
Aspergillopepsin I
Cat.No: T78363
Synonym: Aspergillus acid protease
Target:
Protease-Activated Receptor-3 (PAR-3) (1-6), human TFA
Cat.No: T36289
Synonym:
Target:
Glutamic acid protease
Cat.No: T76155
Synonym:
Target:
HIV Protease Substrate IV
Cat.No: T76511
Synonym:
Target:
PAR-2 Activating Peptide acetate
Cat.No: TP1046L
Synonym: SLIGRL-NH2 acetate,PAR-2 Activating Peptide acetate(171436-38-7 free base),Protease-Activated Receptor-2 Activating Peptide acetate
Target: Protease-activated Receptor
Cysteine protease inhibitor-3
Cat.No: T79277
Synonym:
Target: Parasite
HIV Protease Substrate I
Cat.No: T76485
Synonym:
Target:
Protease-Activated Receptor-3 (PAR-3) (1-6), human
Cat.No: T36286
Synonym:
Target:
HIV protease-IN-1
Cat.No: T74939
Synonym:
Target:
HIV-1 protease-IN-10
Cat.No: T79493
Synonym:
Target: PKC
β-Herpesvirus protease-IN-1
Cat.No: T80691
Synonym:
Target: Virus Protease
HIV Protease Substrate 1 TFA
Cat.No: T76074
Synonym:
Target:
HIV-1 protease-IN-5
Cat.No: T64112
Synonym:
Target:
HIV-1 protease-IN-2
Cat.No: T63949
Synonym:
Target:
HIV-1 protease-IN-1
Cat.No: T63453
Synonym:
Target:
HIV-1 protease-IN-11
Cat.No: T79536
Synonym:
Target: HIV Protease
HIV-1 protease-IN-7
Cat.No: T74942
Synonym:
Target: HIV Protease
HIV-1 protease-IN-9
Cat.No: T79295
Synonym:
Target: HIV Protease
HIV-1 protease-IN-6
Cat.No: T63733
Synonym:
Target:
HIV-1 protease-IN-8
Cat.No: T78950
Synonym:
Target: HIV Protease
HIV-1 protease-IN-4
Cat.No: T74488
Synonym:
Target:
HIV-1 protease-IN-12
Cat.No: T79537
Synonym:
Target: HIV Protease
SLIGRL-NH2 TFA
Cat.No: T75902
Synonym: Protease-Activated Receptor-2 Activating Peptide TFA
Target:
Carmofur
Cat.No: T1307
Synonym: HCFU,卡莫氟
Target: Nucleoside Antimetabolite/Analog, Virus Protease, SARS-CoV, DNA/RNA Synthesis
Tubacin
Cat.No: T6327
Synonym:
Target: Virus Protease, HDAC
Protease-Activated Receptor-1 antagonist 1
Cat.No: T62507
Synonym:
Target:
Protease-Activated Receptor-1 antagonist 2
Cat.No: T64285
Synonym:
Target:
Protease-Activated Receptor-1 antagonist 2
Cat.No: T74266
Synonym:
Target:
Protease-Activated Receptor-1 antagonist 3
Cat.No: T63382
Synonym:
Target:
HIV-1, HIV-2 Protease Substrate
Cat.No: T76502
Synonym:
Target:
TPCK
Cat.No: T8350
Synonym:
Target: Proteasome
Des(benzylpyridyl) Atazanavi
Cat.No: T1883
Synonym:
Target: HIV Protease
ZK824190
Cat.No: T13408
Synonym:
Target: Others, Serine Protease
ZINC03129319
Cat.No: T13397
Synonym:
Target: Virus Protease
ESI-09
Cat.No: T2244
Synonym:
Target: cAMP, Virus Protease
Cat. No. Product Name Target Signaling Pathways
T5783 Rosamultin

野蔷薇苷,罗莎白素

Antioxidant; HIV Protease Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Rosamultin 是从Potentilla anserina L 分离的 19 α-羟基型三萜。它抑制 HIV-1 蛋白酶,具有抗氧化、抗炎和镇痛作用。
TN1059 Ganoderic acid B

IL Receptor; HIV Protease; JAK; STAT Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Microbiology/Virology; Proteases/Proteasome; Stem Cells
Ganoderic acid B 是从灵芝中分离的一种三萜类天然产物。它是端粒酶抑制剂,抑制 Epstein-Barr 病毒抗原的活化。它是 HIV-1 蛋白酶抑制剂。
TMO2787 Anthraquinone

dioxoanthracene,Anthradione,anthracenedione,蒽醌

Virus Protease Microbiology/Virology
Anthraquinone (Anthradione) 是常用于缓解便秘的草药中的主要活性成分,可用作染料形成前体。
T5666 Dipotassium glycyrrhizinate

Virus Protease Microbiology/Virology
Dipotassium glycyrrhizinate 是一种具有抗过敏和抗炎活性的阴离子表面活性剂。
T2741 Glycyrrhizic acid

Glycyrrhizin,甘草酸

Virus Protease; Dehydrogenase; MAO Metabolism; Microbiology/Virology; Neuroscience
Glycyrrhizic acid (Glycyrrhizin) 是甘草里面的活性成分三萜皂苷,为 HMGB1的拮抗剂,有用于肿瘤、糖尿病等研究的潜力。
T2875 Angelicin

Isopsoralen,异补骨脂素

Apoptosis; Virus Protease; Antiviral Apoptosis; Immunology/Inflammation; Microbiology/Virology
Angelicin (Isopsoralen) 是一种三环芳烃天然产物,结构上跟补骨脂素有关,具有抗癌、抗炎、抗病毒等活性。
T4S1383 Escin IA

Aescin IA,Escin IA;Aescin IA,Escin IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Escin IA (Escin IA;Aescin IA);Aescin IA 是从马蹄中七叶树分离出的一种三萜皂苷,抑制HIV-1蛋白酶,IC50值为 35 μM。它具有抗 TNBC 转移活性,其作用机制涉及通过下调 LOXL2 表达抑制上皮-间质转化过程。
T4S1387 Isoescin IA

七叶皂苷C,异七叶皂苷 IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Isoescin IA 是一种从七叶树种子中分离出来的三萜皂苷。它具有抗HIV-1蛋白酶活性。
T0254 Probucol

DH-581,普罗布考

Virus Protease; ABC; Lipid Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
Probucol (DH-581) 是一种抗高脂血症药物,可通过增加 LDL 分解代谢率来降低血液中的胆固醇水平。
T2926 Schizandrin A

P450; Virus Protease; Autophagy Autophagy; Metabolism; Microbiology/Virology
Schisandrin A 是一种从东方药物五味子中提取的主要有效成分,抑制 CYP3A 活性,IC50 分别为 6.60 μM 和 Ki 为 5.83 μM。
T0122 Bergenin

Cuscutin,Bengenin,岩白菜素

Apoptosis; IL Receptor; Virus Protease; TNF; NF-κB; Antibacterial; NOD; Autophagy; Antifungal Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology; NF-κB
Bergenin (Bengenin) 是一种在许多药用植物中发现的多酚,有细胞保护和抗氧化作用。它还具有广泛的保肝、抗炎、抗肿瘤、抗病毒、抗真菌以及免疫调节作用。
TN2082 Pinostrobin

Beta Amyloid; IL Receptor; Serine/threonin kinase; TNF Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation; Metabolism; Neuroscience
Pinostrobin 是一种 PCSK9抑制剂,可抑制 PCSK9 的催化活性。它是能够在多种植物中发现的黄酮类化合物,并具有抗氧化,抗炎,抗癌和神经保护作用。它是有前景的胆固醇调节和脂质管理剂。
T0433 Artesunate

WR-256283,青蒿琥酯

Virus Protease; Ferroptosis; STAT; Parasite Apoptosis; JAK/STAT signaling; Microbiology/Virology; Stem Cells
Artesunate (WR-256283) 是治疗疟疾的青蒿素组药物的一部分。 它是青蒿素的半合成衍生物,具有水溶性。
T5S0689 Demethylwedelolactone

去甲蟛蜞菊内酯,去甲基蟛蜞内酯

Serine Protease Proteases/Proteasome
Demethylwedelolactone 是一种分离自 Eclipta alba 中的 coumestan 天然产物。它能抑制乳腺癌细胞的移动和侵袭,是一种有效的trypsin 抑制剂(IC50:3.0 μM)。
T1717 alpha-Mangostin

α-倒捻子素,α-Mangostin,Mangostin

Apoptosis; Virus Protease; Dehydrogenase; Reactive Oxygen Species; Antibacterial; Antifungal Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
alpha-Mangostin (Mangostin) 是有多种生物活性的膳食呫吨酮。它是一种IDH1突变体的抑制剂,Ki 值为 2.85 μM。
T4850 PCL 016

2-吡啶甲酸,2-Picolinic acid

Virus Protease; Endogenous Metabolite Metabolism; Microbiology/Virology
PCL 016 (2-Picolinic acid) 是一种局部抗病毒剂,可抑制兔体内的腺病毒复制。
T8071 L-Lysine hydrochloride

赖氨酸盐酸盐,Lysine hydrochloride,L-赖氨酸盐酸盐

Virus Protease Microbiology/Virology
L-Lysine hydrochloride 是一种人类必需氨基酸,能增加钙吸收,减少糖尿病相关疾病和改善肠道健康,可用于疱疹的研究。
T2A2498 L-Lysine

Aminutrin,Lysine Acid,lysine,L-赖氨酸,赖氨酸

Virus Protease; Endogenous Metabolite; Antifection Metabolism; Microbiology/Virology
L-Lysine (Aminutrin) 是一种人类必需氨基酸,能增加钙吸收,减少糖尿病相关疾病和改善肠道健康,可用于疱疹的研究。
T3717 Hinokitiol

4-Isopropyltropolone,桧木醇,β-thujaplicin,β-桧木醇

DNA Methyltransferase; Virus Protease; Estrogen/progestogen Receptor; Nrf2 Chromatin/Epigenetic; Endocrinology/Hormones; Immunology/Inflammation; Microbiology/Virology
Hinokitiol (4-Isopropyltropolone) 是从日本扁柏中分离到的一种挥发油成分,可抑制紫外线 B 诱导的角质形成细胞凋亡,可调节雌激素受体信号传导并抑制人乳腺癌细胞的增殖。它具有抗感染、抗氧化及抗肿瘤等活性。
T6S0095 Genkwanin

7-O-Methylapigenin,Puddumetin,Apigenin 7-methyl ether,芫花素

Virus Protease Microbiology/Virology
Genkwanin (Apigenin 7-methyl ether) 是一种O-甲基化黄酮,有抗炎活性,通过被动扩散和多药耐药蛋白介导的外排机制转运。
T2718 Palmatine chloride

Others; Indoleamine 2,3-Dioxygenase (IDO); Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Others
Palmatine chloride 是口服具有活力的不可逆 IDO-1抑制剂。它能够减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,并改善 DSS 诱发的结肠炎。
T5S1923 Schisandrin C

五味子丙素,Schizandrin-C,Wuweizisu-C

Apoptosis; Others; Virus Protease Apoptosis; Microbiology/Virology; Others
Schisandrin C (Wuweizisu-C) 是从五味子中分离得到的一种植物化学木脂素。它具有抗癌、抗炎和抗氧化等多种生物活性,可研究癌症、阿尔茨海默病、肝病。
T0800 Danthron

Dantron,1,8-Dihydroxyanthraquinone,1,8-二羟基蒽醌,丹蒽醌,Chrysazin,Antrapurol

Virus Protease; Antibacterial; AMPK; Autophagy Autophagy; Chromatin/Epigenetic; Microbiology/Virology; PI3K/Akt/mTOR signaling
Danthron (Antrapurol) 是一种从中药 rhubarb 中提取的天然产物,可通过激活 AMPK 来调节葡萄糖和脂质代谢。
T6S1315 Oroxylin A

千层纸素A,6-Methoxybaicalein,Baicalein 6-methyl ether

Virus Protease; HIF/HIF Prolyl-Hydroxylase; Autophagy Autophagy; Chromatin/Epigenetic; Metabolism; Microbiology/Virology
Oroxylin A (Baicalein 6-methyl ether) 是一种有活性的黄酮,具有较强的抗癌作用。
T5S0802 Palmatine

巴马汀,Berbericinine,Burasaine

Indoleamine 2,3-Dioxygenase (IDO); AChR; AChE; Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Neuroscience
Palmatine (Burasaine) 是口服具有活力的、不可逆IDO-1抑制剂。它可以减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,从而改善DSS (Dextran Sulphate Sodium Salt) 诱发的结肠炎。它有用于结肠炎的研究潜力。
T2774 Lycorine hydrochloride

石蒜碱,Licorine hydrochloride,Galanthidine hydrochloride,Narcissine hydrochloride,Lycorine chloride,Amarylline hydrochloride,盐酸石蒜碱

Virus Protease; HCV Protease; Antibacterial; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Lycorine hydrochloride (Narcissine hydrochloride) 是黑色素瘤血管生成抑制剂,是一种来自石蒜的主要活性成分,抑制 Hey1B 细胞的有丝分裂增殖,IC50值为 1.2 μM,具有抗肿瘤活性。
TN1202 (-)-α-Pinene

左旋-α-蒎烯,左旋-alpha-蒎烯,(1S)-(-)-Alpha-Pinene

Virus Protease; GABA Receptor; Endogenous Metabolite; Antibacterial Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience
(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) 是一种单萜类化合物,通过延长 GABAergic 突触传递、作为 GABAA-BZD 受体的部分调节剂并直接与 GABAA 受体的 BZD 结合位点结合来增强 NREMS 的数量而不影响 NREMS 的强度。
T0011 2-Phenylethanol

苯乙醇,Phenethyl alcohol,2-Phenylethyl alcohol,Benzyl carbinol,Phenylethanol,Benzeneethanol

Others; Virus Protease; Antibacterial; Antibiotic Microbiology/Virology; Others
2-Phenylethanol (Phenylethanol) 是从玫瑰、风笛、阿勒颇松、桔子花等多种物种中提取得到的一种无色液体。它有一种使人感到愉悦的气味,也是一种从真菌Candida albicans 产生的自体抗生素。它可用作香皂中的防腐剂,也用作香烟添加剂。
T3759 3,4-Dimethoxycinnamic acid

Dimethylcaffeic acid,3,4-二甲氧基肉桂酸,Caffeic acid dimethyl ether,O-Methylferulic acid

Apoptosis; Virus Protease; Reactive Oxygen Species Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
3,4-Dimethoxycinnamic acid (O-Methylferulic acid) 是从 Securidaca inappendiculata Hassk 中提取和纯化的单体。 3,4-Dimethoxycinnamic acid 通过 ROS 介导的信号通路对 L-02 细胞发挥抗凋亡作用。抗凋亡作用。
T5429 Theaflavin 3,3'-digallate

茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG

Virus Protease; Antioxidant; HIV Protease; HSV Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。
T3324 Lycorine

Galanthidine,Narcissine,石蒜碱,Amarylline,Belamarine,Licorine,番石榴碱

Apoptosis; Virus Protease; Antibacterial; AChR; Fatty Acid Synthase Apoptosis; Metabolism; Microbiology/Virology; Neuroscience
Lycorine (Narcissine) 是从金眼科植物科中提取的一种天然生物碱。它是一种具有口服活性的SCAP 抑制剂,Kd 值 15.24 nM。它也是黑色素瘤血管生成抑制剂,有用于前列腺癌和代谢疾病的研究潜力。
T2732 (-)-Epicatechin gallate

表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG

Virus Protease; COX; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience
(-)-Epicatechin gallate ((-)-Epicatechin 3-O-gallate) 抑制环加氧酶-1 的IC50值为 7.5 μM。
TN1262 3-Feruloylquinic acid

3-O-阿魏酰奎尼酸,3-O-Feruloylquinic acid

Proteasome; Antifection Microbiology/Virology; Proteases/Proteasome; Ubiquitination
3-O-Feruloylquinic acid is a protease inhibitor, it exerts moderate inhibitory effect against AIV (H5N1) in vitro.
T2S0223 Isosinensetin

异橙黄酮,6-Demethoxynobiletin

Antioxidant; HIV Protease; Antibacterial; P-gp Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; oxidation-reduction; Proteases/Proteasome
Isosinensetin (6-Demethoxynobiletin) 是从青皮中提取的一种甲氧基黄酮,具有抗氧化和抑制 HIV-1 蛋白酶的活性。
T4S0181 Hinokiflavone

日本扁柏黄酮,扁柏双黄酮

MMP; BCL; E1/E2/E3 Enzyme Apoptosis; Proteases/Proteasome; Ubiquitination
Hinokiflavone 是pre-mRNA 剪接活性的新型调节剂,通过抑制剪接体装配来阻止pre-mRNA 底物的剪接,特别是阻止 B complex 的形成。它是SUMO protease 蛋白酶抑制剂,能够抑制前哨蛋白特异性蛋白酶 1 的活性。
T19503 Papain

Others; Cysteine Protease Others; Proteases/Proteasome
Papain 是一种半胱氨酸蛋白酶,是肽酶 C1 家族中一员,在食品、医药、化妆品、纺织等具有广泛的应用。
T3S0136 4'-O-Methylbavachalcone

O-Methylbroussochalcone B,4'-O-甲基补骨脂查尔酮

SARS-CoV Microbiology/Virology
4'-O-Methylbavachalcone (O-Methylbroussochalcone B) 是从补骨脂中分离得到的一种查尔酮,可抑制严重急性呼吸综合征冠状病毒木瓜样蛋白酶的活性,IC50值为 10.1 μM。
T3323 Ursonic Acid

CCRIS 7123,NSC4060,熊果酮酸,Prunol,3-Ketoursolic acid,Malol,TOS-BB-0966

Apoptosis; HIV Protease; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome
Ursonic Acid (TOS-BB-0966) 是一种天然三萜酸,属于熊果烷三萜类,其结构基于五环熊果烷骨架。 它具有作为 HIV-1 蛋白酶抑制剂的潜力。
T4915 β-Glycerophosphate disodium salt hydrate

Phosphatase; Endogenous Metabolite Metabolism
β-Glycerophosphate disodium salt hydrate 是一种磷酸酶抑制剂,是内源性代谢产物的一种。
T2O2730 L-Serine

(S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid

Endogenous Metabolite Metabolism
L-Serine (serine) 是一种人体非必需氨基酸,它存在于许多蛋白质中,并且在功能上很重要。L-Serine 也存在于丝氨酸蛋白酶类的活性位点,包括胰蛋白酶和凝乳胰蛋白酶。
T6564 Leupeptin Hemisulfate

亮肽素

Serine Protease; Cysteine Protease Proteases/Proteasome
Leupeptin hemisulfate 是一种蛋白酶抑制剂,具有细胞膜渗透性、可逆性、竞争性和口服活性。Leupeptin hemisulfate 可以抑制 Cathepsin B、Cathepsin H、Cathepsin L 的活性,阻断两性溶酶体的融合。Leupeptin hemisulfate 还具有抗炎活性。
T2768 Saikosaponin A

柴胡皂苷A,柴胡皂苷 A

NF-κB; Antibacterial; Liver X Receptor Metabolism; Microbiology/Virology; NF-κB
Saikosaponin A 是银柴胡中的主要活性成分,有抗炎活性,可上调 LXRα的表达。
T6S0071 Fraxinellone

HIF/HIF Prolyl-Hydroxylase; STAT; PD-1/PD-L1 Apoptosis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Metabolism; Stem Cells
Fraxinellone 是从白鲜的根皮中分离出来的一种天然产物,是PD-L1抑制剂,可抑制HIF-1α蛋白质合成。它通过靶向 PD-L1,有用于癌症免疫的潜力。
TN6872 Trypsin

Protease-activated Receptor GPCR/G Protein
Trypsin 是一种可从鱼类分离出的丝氨酸蛋白酶,可水解赖氨酸或精氨酸羧基侧蛋白质。Trypsin 具有抗炎活性,可通过 PDCoV 的 S 糖蛋白与 pAPN 的相互作用诱导 PDCoV 感染的细胞膜融合,可激活 PAR2 和 PAR4,促进细胞增殖和分化。Trypsin 可用于促进伤口愈合和研究神经源性炎症。
TQ0217 Gomisin G

戈米辛G,戈米辛 G

P450; HIV Protease Metabolism; Microbiology/Virology; Proteases/Proteasome
Gomisin G 是一种有抗HIV 活性的天然产物。
TN5171 Tricetin

Apoptosis; Others; Nrf2 Apoptosis; Immunology/Inflammation; Others
Tricetin 是一种从石榴中分离出的类黄酮。Tricetin 是 Keap1-Nrf2 蛋白相互作用(PPI)的强效竞争性抑制剂,通过激活 Nrf2/HO-1 信号通路和阻止线粒体依赖性细胞凋亡通路,保护帕金森病患免受 6-OHDA 诱导的神经毒性的影响。Tricetin 通过 Akt/GSK-1β途径抑制鼻咽癌的迁移和指示性蛋白酶早老素-1(PS-1)表达。Tricetin 抑制由Egr-1介导的氧化LDL 诱导的内皮炎症,保护大鼠软骨细胞免受IL-1β诱导的炎症和细胞凋亡。
T75705 Pepstatin Trifluoroacetate

Pepstatin (Pepstatin A) Trifluoroacetate 是一种由放线菌产生的特异性天冬氨酸蛋白酶(aspartic proteases)抑制剂,口服活性强。该化合物能有效抑制hemoglobin-pepsin、hemoglobin-proctase、casein-pepsin、casein-proctase、casein-acid protease和hemoglobin-acid protease的活性,其IC50值分别为4.5 nM、6.2 nM、150 nM、290 nM、520 nM和260 nM。此外,对HIV protease也有抑制作用。
TN5675 Ganomycin I

Ganomycin I inhibits the activity of HIV-1 protease.
TN4347 Jacoumaric acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
Jacoumaric acid is a lead molecule from the library or database of natural compounds as a HIV-1 protease inhibitor.
T5S0983 Absinthin

Absinthiin,Absynthin,洋艾素

HIV Protease Microbiology/Virology; Proteases/Proteasome
Absinthin (Absynthin) 是结构独特的三萜类化合物,是艾草苦味高的原因。它是苦味受体hTAS2R46的激动剂,它利用 hTAS2R46 介导的受体特异性机制抑制组胺诱导的细胞内 Ca2+升高。
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天然产物

Rosamultin
Cat.No: T5783
Synonym: 野蔷薇苷,罗莎白素
Target: Antioxidant, HIV Protease
Ganoderic acid B
Cat.No: TN1059
Synonym:
Target: IL Receptor, HIV Protease, JAK, STAT
Anthraquinone
Cat.No: TMO2787
Synonym: dioxoanthracene,Anthradione,anthracenedione,蒽醌
Target: Virus Protease
Dipotassium glycyrrhizinate
Cat.No: T5666
Synonym:
Target: Virus Protease
Glycyrrhizic acid
Cat.No: T2741
Synonym: Glycyrrhizin,甘草酸
Target: Virus Protease, Dehydrogenase, MAO
Angelicin
Cat.No: T2875
Synonym: Isopsoralen,异补骨脂素
Target: Apoptosis, Virus Protease, Antiviral
Escin IA
Cat.No: T4S1383
Synonym: Aescin IA,Escin IA;Aescin IA,Escin IA
Target: HIV Protease
Isoescin IA
Cat.No: T4S1387
Synonym: 七叶皂苷C,异七叶皂苷 IA
Target: HIV Protease
Probucol
Cat.No: T0254
Synonym: DH-581,普罗布考
Target: Virus Protease, ABC, Lipid
Schizandrin A
Cat.No: T2926
Synonym:
Target: P450, Virus Protease, Autophagy
Bergenin
Cat.No: T0122
Synonym: Cuscutin,Bengenin,岩白菜素
Target: Apoptosis, IL Receptor, Virus Protease, TNF, NF-κB, Antibacterial, NOD, Autophagy, Antifungal
Pinostrobin
Cat.No: TN2082
Synonym:
Target: Beta Amyloid, IL Receptor, Serine/threonin kinase, TNF
Artesunate
Cat.No: T0433
Synonym: WR-256283,青蒿琥酯
Target: Virus Protease, Ferroptosis, STAT, Parasite
Demethylwedelolactone
Cat.No: T5S0689
Synonym: 去甲蟛蜞菊内酯,去甲基蟛蜞内酯
Target: Serine Protease
alpha-Mangostin
Cat.No: T1717
Synonym: α-倒捻子素,α-Mangostin,Mangostin
Target: Apoptosis, Virus Protease, Dehydrogenase, Reactive Oxygen Species, Antibacterial, Antifungal
PCL 016
Cat.No: T4850
Synonym: 2-吡啶甲酸,2-Picolinic acid
Target: Virus Protease, Endogenous Metabolite
L-Lysine hydrochloride
Cat.No: T8071
Synonym: 赖氨酸盐酸盐,Lysine hydrochloride,L-赖氨酸盐酸盐
Target: Virus Protease
L-Lysine
Cat.No: T2A2498
Synonym: Aminutrin,Lysine Acid,lysine,L-赖氨酸,赖氨酸
Target: Virus Protease, Endogenous Metabolite, Antifection
Hinokitiol
Cat.No: T3717
Synonym: 4-Isopropyltropolone,桧木醇,β-thujaplicin,β-桧木醇
Target: DNA Methyltransferase, Virus Protease, Estrogen/progestogen Receptor, Nrf2
Genkwanin
Cat.No: T6S0095
Synonym: 7-O-Methylapigenin,Puddumetin,Apigenin 7-methyl ether,芫花素
Target: Virus Protease
Palmatine chloride
Cat.No: T2718
Synonym:
Target: Others, Indoleamine 2,3-Dioxygenase (IDO), Aurora Kinase
Schisandrin C
Cat.No: T5S1923
Synonym: 五味子丙素,Schizandrin-C,Wuweizisu-C
Target: Apoptosis, Others, Virus Protease
Danthron
Cat.No: T0800
Synonym: Dantron,1,8-Dihydroxyanthraquinone,1,8-二羟基蒽醌,丹蒽醌,Chrysazin,Antrapurol
Target: Virus Protease, Antibacterial, AMPK, Autophagy
Oroxylin A
Cat.No: T6S1315
Synonym: 千层纸素A,6-Methoxybaicalein,Baicalein 6-methyl ether
Target: Virus Protease, HIF/HIF Prolyl-Hydroxylase, Autophagy
Palmatine
Cat.No: T5S0802
Synonym: 巴马汀,Berbericinine,Burasaine
Target: Indoleamine 2,3-Dioxygenase (IDO), AChR, AChE, Aurora Kinase
Lycorine hydrochloride
Cat.No: T2774
Synonym: 石蒜碱,Licorine hydrochloride,Galanthidine hydrochloride,Narcissine hydrochloride,Lycorine chloride,Amarylline hydrochloride,盐酸石蒜碱
Target: Virus Protease, HCV Protease, Antibacterial, Autophagy
(-)-α-Pinene
Cat.No: TN1202
Synonym: 左旋-α-蒎烯,左旋-alpha-蒎烯,(1S)-(-)-Alpha-Pinene
Target: Virus Protease, GABA Receptor, Endogenous Metabolite, Antibacterial
2-Phenylethanol
Cat.No: T0011
Synonym: 苯乙醇,Phenethyl alcohol,2-Phenylethyl alcohol,Benzyl carbinol,Phenylethanol,Benzeneethanol
Target: Others, Virus Protease, Antibacterial, Antibiotic
3,4-Dimethoxycinnamic acid
Cat.No: T3759
Synonym: Dimethylcaffeic acid,3,4-二甲氧基肉桂酸,Caffeic acid dimethyl ether,O-Methylferulic acid
Target: Apoptosis, Virus Protease, Reactive Oxygen Species
Theaflavin 3,3'-digallate
Cat.No: T5429
Synonym: 茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG
Target: Virus Protease, Antioxidant, HIV Protease, HSV
Lycorine
Cat.No: T3324
Synonym: Galanthidine,Narcissine,石蒜碱,Amarylline,Belamarine,Licorine,番石榴碱
Target: Apoptosis, Virus Protease, Antibacterial, AChR, Fatty Acid Synthase
(-)-Epicatechin gallate
Cat.No: T2732
Synonym: 表儿茶素没食子酸酯,(−)-Epicatechin 3-gallate,Epicatechin gallate,(-)-Epicatechin 3-gallate,(-)-Epicatechin 3-O-gallate,ECG
Target: Virus Protease, COX, Autophagy
3-Feruloylquinic acid
Cat.No: TN1262
Synonym: 3-O-阿魏酰奎尼酸,3-O-Feruloylquinic acid
Target: Proteasome, Antifection
Isosinensetin
Cat.No: T2S0223
Synonym: 异橙黄酮,6-Demethoxynobiletin
Target: Antioxidant, HIV Protease, Antibacterial, P-gp
Hinokiflavone
Cat.No: T4S0181
Synonym: 日本扁柏黄酮,扁柏双黄酮
Target: MMP, BCL, E1/E2/E3 Enzyme
Papain
Cat.No: T19503
Synonym:
Target: Others, Cysteine Protease
4'-O-Methylbavachalcone
Cat.No: T3S0136
Synonym: O-Methylbroussochalcone B,4'-O-甲基补骨脂查尔酮
Target: SARS-CoV
Ursonic Acid
Cat.No: T3323
Synonym: CCRIS 7123,NSC4060,熊果酮酸,Prunol,3-Ketoursolic acid,Malol,TOS-BB-0966
Target: Apoptosis, HIV Protease, Endogenous Metabolite
β-Glycerophosphate disodium salt hydrate
Cat.No: T4915
Synonym:
Target: Phosphatase, Endogenous Metabolite
L-Serine
Cat.No: T2O2730
Synonym: (S)-Serine,L-丝氨酸,丝氨酸,serine,(-)-Serine,(S)-2-Amino-3-hydroxypropanoic acid
Target: Endogenous Metabolite
Leupeptin Hemisulfate
Cat.No: T6564
Synonym: 亮肽素
Target: Serine Protease, Cysteine Protease
Saikosaponin A
Cat.No: T2768
Synonym: 柴胡皂苷A,柴胡皂苷 A
Target: NF-κB, Antibacterial, Liver X Receptor
Fraxinellone
Cat.No: T6S0071
Synonym:
Target: HIF/HIF Prolyl-Hydroxylase, STAT, PD-1/PD-L1
Trypsin
Cat.No: TN6872
Synonym:
Target: Protease-activated Receptor
Gomisin G
Cat.No: TQ0217
Synonym: 戈米辛G,戈米辛 G
Target: P450, HIV Protease
Tricetin
Cat.No: TN5171
Synonym:
Target: Apoptosis, Others, Nrf2
Pepstatin Trifluoroacetate
Cat.No: T75705
Synonym:
Target:
Ganomycin I
Cat.No: TN5675
Synonym:
Target:
Jacoumaric acid
Cat.No: TN4347
Synonym:
Target: HIV Protease
Absinthin
Cat.No: T5S0983
Synonym: Absinthiin,Absynthin,洋艾素
Target: HIV Protease
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