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48

抑制剂 & 化合物

48

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T22426	Sodium carbonate 碳酸钠,Soda Ash,Disodium carbonate,Carbonic acid disodium salt	Others	Others
	Sodium carbonate (Soda Ash) 又称碳酸二钠、纯碱、碳酸二钠盐，是具有碱化性能的碳酸二钠盐。
T1371	1H-1,2,4-Triazole-3-carboxylic acid	Others	Others
	1H-1,2,4-Triazole-3-carboxylic acid，具有 isoprenyl transferases 抑制蛋白质的特性。
T8520	Tetrazole 1H-TETRAZOLE,1H-四唑	Antibacterial	Microbiology/Virology
	Tetrazole (1H-TETRAZOLE) 是羧酸的生物等排体，具有相当的抗菌性能。
T1144L	Lidocaine Hydrochloride hydrate	EGFR; Sodium Channel	Angiogenesis; JAK/STAT signaling; Membrane transporter/Ion channel; Tyrosine Kinase/Adaptors
	Lidocaine Hydrochloride hydrate 是一种酰胺类局部麻醉剂，具有抗炎作用。
T0457	Probenecid Benemid,丙磺舒	HIV Protease; Antibacterial; TRP/TRPV Channel	Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
	Probenecid (Benemid) 是一种苯甲酸衍生物，具有抗高尿酸特性。它也是一种选择性瞬时受体电位香草酸受体通道 2 激动剂，还可抑制pannexin 1通道。
T7313	Enclomiphene citrate 恩氯米芬柠檬酸盐,Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate	Estrogen Receptor/ERR	Endocrinology/Hormones
	Enclomiphene citrate (trans-Clomiphene citrate) 是口服具有活力的 oestrogen receptor 拮抗剂，具有抗雌激素活性。
T18890	5-ROX 5-羧基-X-罗丹明,5-Carboxy-X-rhodamine	Others	Others
	5-ROX (5-Carboxy-X-rhodamine) 是罗丹明染料的一种，λexit 为 580 nm (ε=3.6×104M-1cm-1)，λemit 为 604 nm (ϕ=0.94)。
TP1554L	HPV16 E7 (86-93) acetate HPV16 E7 (86-93) acetate(160212-93-1 Free base)	Others	Others
	HPV16 E7 (86-93) acetate 是人源白细胞抗原 A2.1 限制性 HPV16 E7 的衍生肽，在宫颈癌中具有免疫原性。
T65133	3-Hydroxybutyric acid sodium β-Hydroxybutyric acid sodium
	3-Hydroxybutyric acid sodium (β-Hydroxybutyric acid sodium) 是一种存在 I 型糖尿病患者体内的一种代谢物，具有调节膜脂的性质。
T1425	Pemirolast potassium BMY 26517,TWT-8152,吡嘧司特钾	Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Neuroscience
	Pemirolast potassium (TWT-8152) 是 H1组胺受体拮抗剂和肥大细胞稳定剂，是一种具有抗过敏特性的嘧啶酮衍生物。
T12950	Sodium laureth sulfate Sodium lauryl polyoxyethylene ether sulfate,月桂醇聚氧乙烯醚硫酸酯钠盐	Others	Others
	Sodium laureth sulfate (Sodium lauryl polyoxyethylene ether sulfate) 是一种阴离子活性剂，具有优良的去污，分散，乳化，润湿等性能。
T10239	Acolbifene 阿考比芬,EM-652,SCH 57068	Estrogen Receptor/ERR	Endocrinology/Hormones
	Acolbifene (SCH 57068) 是一种选择性雌激素受体拮抗剂，对雌二醇诱导的 ERα 和 ERβ 转录活性的 IC50 分别为 2 nM 和 0.4 nM。 Acolbifene 显示出抗癌特性。
T2592	Ropinirole hydrochloride SKF 101468 hydrochloride,SKF-101468A,Ropinirole HCl,盐酸罗匹尼罗	Dopamine Receptor	GPCR/G Protein; Neuroscience
	Ropinirole hydrochloride (SKF-101468A) 是D3/D2受体激动剂，对 D2受体的Ki=29 nM。它对 hD2，hD3和 hD4受体的pEC50分别为 7.4、8.4 和 6.8。它对 D1受体没有亲和力。它对帕金森氏病具有潜在的研究价值。
T9560	MAO-B-IN-2
	MAO-B-IN-2 是一种选择性和竞争性的MAO-B 和 BChE 抑制剂，其IC50值分别为 0.51 和 7.00 μM。MAO-B-IN-2 通过良好的 ROS 清除特性减轻 H2O2 诱导的细胞损伤。
T7000	Tiagabine hydrochloride NO328 hydrochloride,盐酸噻加宾,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Tiagabine hydrochloride (NO050328 hydrochloride) 是具有抗惊厥特性的选择性GABA 再摄取抑制剂，在突触体、神经元和神经胶质中，能够抑制 [3H]GABA 的重摄取，IC50值分别为 67、446 和 182 nM。
T29457L	5-Hydroxydecanoate sodium	Potassium Channel	Membrane transporter/Ion channel
	5-Hydroxydecanoate sodium 是一种选择性 ATP 敏感的 K+ (KATP) 通道阻滞剂，IC50 约为 30 μM。它是线粒体外膜酰基辅酶A 合成酶的底物，具有抗氧化性。
T1435	Praziquantel 吡喹酮,Pyquiton,Droncit,Biltricide	Calcium Channel; Antibiotic; Parasite	Membrane transporter/Ion channel; Metabolism; Microbiology/Virology
	Praziquantel (Droncit) 是一种外消旋混合物，由 (R)-Praziquantel 和 (S)-Praziquantel 组成。它可研究血吸虫病。
T2546	Pimozide R6238,匹莫奇特,匹莫齐特	Potassium Channel; Dopamine Receptor; Adrenergic Receptor; STAT	GPCR/G Protein; JAK/STAT signaling; Membrane transporter/Ion channel; Neuroscience; Stem Cells
	Pimozide (R6238) 是多巴胺受体拮抗剂，对多巴胺 D1、D2 和 D3 受体的 Ki 值分别为 588、1.4 和 2.5 nM。它也是STAT3和STAT5的抑制剂，对 α1 肾上腺素受体也有较高亲和性，Ki 值为 39 nM。
T0018	Procainamide hydrochloride Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺	DNA Methyltransferase; Sodium Channel; AChR; Autophagy	Autophagy; Chromatin/Epigenetic; Membrane transporter/Ion channel; Neuroscience
	Procainamide hydrochloride (Procapan) 是一种用于研究心律失常的抗心律失常制剂。
T6686	Sulconazole mononitrate Exelderm,Sulconazole Nitrate,RS 44872,硝酸硫康唑	Antibacterial; Antibiotic; Antifungal	Microbiology/Virology
	Sulconazole mononitrate (Exelderm) 是一种咪唑类广谱杀菌剂。它可研究皮肤真菌病，花斑糠疹病，皮肤念珠菌病。
T1281	Tropicamide Ro 1-7683,托吡卡胺	AChR	Neuroscience
	Tropicamide (Ro 1-7683) 是一种选择性的 M4毒蕈碱乙酰胆碱受体拮抗剂，作为滴眼剂使用时，会产生短效瞳孔扩张和睫状肌麻痹。
T0893	Tinidazole 替硝唑,CP12574	Antibacterial; Antibiotic	Microbiology/Virology
	Tinidazole (CP12574) 是一种对厌氧菌和原生动物具有选择性抗菌活性的 5-硝基咪唑，是一种具有口服活性的抗菌剂。
T6602	Naratriptan hydrochloride Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride	5-HT Receptor	GPCR/G Protein; Neuroscience
	Naratriptan hydrochloride (GR-85548A hydrochloride) 是一种5-HT1受体激动剂，有抗偏头疼特性。它还可以通过刺激三叉神经系统感觉神经末梢上的 5-HT1D/1B 受体来发挥其作用，从而减少促炎神经肽的释放。
T27183	Diproteverine
	Diproteverine is a calcium antagonist, it has antianginal property.
T16268	Namitecan ST-1968	Others	Others
	Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.
T27276	Epeleuton
	Epeleuton has anti-inflammatory property.
T0149	Pheneticillin	Others	Others
	Pheneticillin 是一种具有抗菌性的抗生素。
T39190	ATX-002
	ATX-002 is a property-tunable lipid for RNA drug delivery.
T15166	DPM-1001	Phosphatase	Metabolism
	DPM-1001 is an orally bioavailable and non-competitive protein-tyrosine phosphatase (PTP1B) inhibitor (IC50: 100 nM) with the anti-diabetic property.
T68937	Carbidopa hydrochloride
	Carbidopa hydrochloride is a drug given to people with Parkinson's disease in order to inhibit peripheral metabolism of levodopa. This property is significant in that it allows a greater proportion of peripheral levodopa to cross the blood–brain barrier for central nervous system effect.
T18932	Calcein tetraethyl ester 钙黄绿素四乙酯,Fluorexon tetraethyl ester	Others	Others
	Calcein tetraethyl ester, a fluorescent dye, is utilized in biological studies for its ability to penetrate cellular membranes into living cells. This property renders it valuable for assessing cell viability and short-term cell labeling.
T39128	Pro-Phe-Phe
	Pro-Phe-Phe, a highly aggregation-prone tripeptide composed of natural amino acids, exhibits the formation of distinctive helical-like sheets that engage in aromatic dry interfaces. This property makes Pro-Phe-Phe an excellent candidate for the development of modular super-helical self-assembling nanostructures.
T25170	Botryodiplodin Cytostipin,Antibiotic PSX 1
	Botryodiplodin, an antibiotic, has antileukemic activity from Botryodiplodia theobromae. It has the property of turning the skin of the individual in various shades of pink 2-3 hrs after application. It is a toxic metabolite of Penicillium carneo-lutescen
T28618	RS-93522 RS 93522
	RS-93522 is an antagonist of calcium channel. RS-93522 had the additional property of inhibiting phosphodiesterase activity in myocardial homogenates (IC50 = 1.6 x 10(-5)M), the potency and efficacy of phosphodiesterase inhibition was similar to that for
T79086	MC4171	Histone Acetyltransferase	Chromatin/Epigenetic
	MC4171（化合物34）作为KAT8选择性抑制剂，IC50值为8.1 µM。该化合物在多种癌症细胞系中（包括NSCLC和AML）展现中等微摩尔级别抗增殖效果，显示出其研究治疗癌症的可能性。
T76497	KRFK
	KRFK是一种源自TSP-1的多肽，具备激活TGF-β的能力。通过独立于TSP受体（例如CD47和CD36）的方式，KRFK能够促进TGF-β介导的信号传递以及其下游效应的发生，可作为慢性眼表炎症疾病研究的工具。
T81403	Priliximab cM-T412,CEN 000029
	Priliximab (CEN 000029) 是一种针对CD4的人源化单克隆抗体。其与T细胞表面CD4的结合作用可引起循环中CD4+T细胞的显著并持久的减少，适用于类风湿性关节炎 (RA) 研究。
T77280	DSPE-succinic acid
	DSPE-succinic acid是一种具有羧酸末端的磷脂，能够通过其羧酸部分与胺发生反应，形成稳定的酰胺键。该化合物常用于纳米颗粒或脂质体的制备，用作活性分子的纳米载体。
T80487	MmTx2 toxin Micrurotoxin 2	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	MmTx2 toxin作为一种GABAA受体调节剂，具有提升GABAA受体对激动剂反应敏感性的作用。该毒素来源于珊瑚蛇的毒液，并在神经系统相关疾病（例如癫痫、精神分裂症及慢性疼痛）的研究中发挥重要用途。
T70897	Zotiraciclib HCl
	Zotiraciclib, also known as TG02 and SB1317, is a novel small molecule potent CDK/JAK2/FLT3 inhibitor. Zotiraciclib may be useful for the treatment of cancer that crosses the blood brain barrier and acts by depleting Myc through the inhibition of cyclin-dependent kinase 9 (CDK9). It is one of a number of CDK inhibitors under investigation; others targeting CDK9 for the treatment of acute myeloid leukemia include alvocidib and atuveciclib. Myc overexpression is a known factor in many cancers, w...
T81305	ReAsH-EDT2
	ReAsH-EDT2为膜透性红色荧光染料，专用于蛋白质标记。作为二砷化合物，其通过共价结合至四半胱氨酸序列实现蛋白质成像，并可监测其定位与转运。(λex=530 nm，λem=592 nm)。
T77158	Diridavumab
	Diridavumab为一种针对HA茎的单克隆抗体。它能稳定HA的融合前结构，阻断细胞膜与病毒膜在核内体内因pH变化引起的融合。此抗体主要用于H2流感病毒研究。
T78391	DAUDA
	DAUDA (11-(dansylamino) undecanoic acid)是一种荧光脂肪酸类似物，对环境变化敏感。该分子通过调整其发射强度和荧光光谱与结合蛋白发生相互作用。在研究中，DAUDA用于评估天然脂肪酸与曼氏血吸虫Sm14脂肪酸结合蛋白多晶型的相对亲和力。
T0204	Protriptyline hydrochloride 盐酸普罗替林,Protriptyline HCl	5-HT Receptor; AChE	GPCR/G Protein; Neuroscience
	Protriptyline hydrochloride (Protriptyline HCl) 是一种含有一个仲胺的三环结构抗抑郁试剂，可以用于抑郁和 ADHD 的相关研究。它使动物精力充沛起激励作用，并且有时用于嗜睡症的相关研究。
T60782	THK-5470
	THK-5470 是具有高选择性和高亲和力的单胺氧化酶B 的成像探针，可用于研究神经系统疾病。THK-5470 对MAO-B 表现出显著的高结合亲和力，IC50值为 4.2 nM，其对tau 的结合亲和力较低，IC50值为 4462 nM。
T77252	Dihydrorhodamine 6G
	Dihydrorhodamine 6G (DHR 6G) 为 Rhodamine 6G 的还原型，作为线粒体荧光染料而被广泛应用。该化合物在原状态下无荧光性，但能轻易渗透大部分细胞，并由氧化物或细胞的氧化还原系统氧化为具有荧光的 Rhodamine 6G，进而在线粒体膜中累积。Dihydrorhodamine 6G 主要用于活性氧 (ROS) 的检测，包括超氧化物。
T64640	Melanin probe-2
	Melanoma is a lethal skin cancer. The early detection of melanoma using positron emission tomography (PET) probes is critical for improving the survival of melanoma patients. Melanin probe-2 is a non-radioactive bromo-picolinamide precursor that has been used for the synthesis of18F-picolinamides based PET probe (melanin probe-1). The tumor-targeting efficacy and imaging property of three melanin probes were evaluated in B16F10 tumor-bearing mice.18F-1 and18F-3 had much lower tumor uptake compar...
T76255	Certepetide
	Certepetide (CEND-1)，即双功能环肽（a.k.a. iRGD），是一种具有穿透肿瘤功能的多肽。通过与α-V整联蛋白（alphav-integrins）的RGD motif相互作用，以及激活神经纤毛蛋白1（NRP-1），Certepetide能够将实体瘤微环境转化成临时的活性分子通道，从而在肿瘤中累积。该化合物在胰腺癌和其他实体瘤的研究中具有应用潜力。

化合物

Sodium carbonate

Cat.No: T22426

Synonym: 碳酸钠,Soda Ash,Disodium carbonate,Carbonic acid disodium salt

Target: Others

1H-1,2,4-Triazole-3-carboxylic acid

Cat.No: T1371

Target: Others

Cat.No: T8520

Synonym: 1H-TETRAZOLE,1H-四唑

Target: Antibacterial

Lidocaine Hydrochloride hydrate

Cat.No: T1144L

Target: EGFR, Sodium Channel

Cat.No: T0457

Synonym: Benemid,丙磺舒

Target: HIV Protease, Antibacterial, TRP/TRPV Channel

Enclomiphene citrate

Cat.No: T7313

Synonym: 恩氯米芬柠檬酸盐,Enclomifene citrate,(E)-Clomiphene citrate,trans-Clomiphene citrate

Target: Estrogen Receptor/ERR

Cat.No: T18890

Synonym: 5-羧基-X-罗丹明,5-Carboxy-X-rhodamine

Target: Others

HPV16 E7 (86-93) acetate

Cat.No: TP1554L

Synonym: HPV16 E7 (86-93) acetate(160212-93-1 Free base)

Target: Others

3-Hydroxybutyric acid sodium

Cat.No: T65133

Synonym: β-Hydroxybutyric acid sodium

Pemirolast potassium

Cat.No: T1425

Synonym: BMY 26517,TWT-8152,吡嘧司特钾

Target: Histamine Receptor

Sodium laureth sulfate

Cat.No: T12950

Synonym: Sodium lauryl polyoxyethylene ether sulfate,月桂醇聚氧乙烯醚硫酸酯钠盐

Target: Others

Cat.No: T10239

Synonym: 阿考比芬,EM-652,SCH 57068

Target: Estrogen Receptor/ERR

Ropinirole hydrochloride

Cat.No: T2592

Synonym: SKF 101468 hydrochloride,SKF-101468A,Ropinirole HCl,盐酸罗匹尼罗

Target: Dopamine Receptor

Cat.No: T9560

Tiagabine hydrochloride

Cat.No: T7000

Synonym: NO328 hydrochloride,盐酸噻加宾,NO050328 hydrochloride,TGB hydrochloride,Gabitril,Gabitril hydrochloride

Target: GABA Receptor

5-Hydroxydecanoate sodium

Cat.No: T29457L

Target: Potassium Channel

Cat.No: T1435

Synonym: 吡喹酮,Pyquiton,Droncit,Biltricide

Target: Calcium Channel, Antibiotic, Parasite

Cat.No: T2546

Synonym: R6238,匹莫奇特,匹莫齐特

Target: Potassium Channel, Dopamine Receptor, Adrenergic Receptor, STAT

Procainamide hydrochloride

Cat.No: T0018

Synonym: Procapan,Procainamide HCl,Pronestyl,Procanbid,盐酸普鲁卡因胺

Target: DNA Methyltransferase, Sodium Channel, AChR, Autophagy

Sulconazole mononitrate

Cat.No: T6686

Synonym: Exelderm,Sulconazole Nitrate,RS 44872,硝酸硫康唑

Target: Antibacterial, Antibiotic, Antifungal

Cat.No: T1281

Synonym: Ro 1-7683,托吡卡胺

Target: AChR

Cat.No: T0893

Synonym: 替硝唑,CP12574

Target: Antibacterial, Antibiotic

Naratriptan hydrochloride

Cat.No: T6602

Synonym: Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride

Target: 5-HT Receptor

Cat.No: T27183

Cat.No: T16268

Synonym: ST-1968

Target: Others

Cat.No: T27276

Cat.No: T0149

Target: Others

Cat.No: T39190

Cat.No: T15166

Target: Phosphatase

Carbidopa hydrochloride

Cat.No: T68937

Calcein tetraethyl ester

Cat.No: T18932

Synonym: 钙黄绿素四乙酯,Fluorexon tetraethyl ester

Target: Others

Cat.No: T39128

Cat.No: T25170

Synonym: Cytostipin,Antibiotic PSX 1

Cat.No: T28618

Synonym: RS 93522

Cat.No: T79086

Target: Histone Acetyltransferase

Cat.No: T76497

Cat.No: T81403

Synonym: cM-T412,CEN 000029

DSPE-succinic acid

Cat.No: T77280

Cat.No: T80487

Synonym: Micrurotoxin 2

Target: GABA Receptor

Zotiraciclib HCl

Cat.No: T70897

Cat.No: T81305

Cat.No: T77158

Cat.No: T78391

Protriptyline hydrochloride

Cat.No: T0204

Synonym: 盐酸普罗替林,Protriptyline HCl

Target: 5-HT Receptor, AChE

Cat.No: T60782

Dihydrorhodamine 6G

Cat.No: T77252

Melanin probe-2

Cat.No: T64640

Cat.No: T76255

Cat. No.	Product Name	Target	Signaling Pathways
TN1353	N-Benzyllinoleamide (9Z,12Z)-N-Benzyloctadeca-9,12-dienamide,N-苄基-(9Z,12Z)-十八碳二烯酰胺	Others	Others
	N-Benzyllinoleamide ((9Z,12Z)-N-Benzyloctadeca-9,12-dienamide) 是一种分离自 Lepidium meyeniiWalp，能够抗运动性疲劳的药物。
TN7113	Methacrylamide	Others	Others
	Methacrylamide 是一种具有染色性的天然产物。
T0144	Ftaxilide Histanorm,安息香酸,伏保克西里	Antibacterial	Microbiology/Virology
	Ftaxilide (Histanorm) 是新型抗结核剂。
TN1432	Bacopasaponin C (-)-假马齿苋皂苷 C,假马齿苋皂苷C	Anti-infection; GABA Receptor; NMDAR	Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
	Bacopasaponin C 是一种分离自Bacopa monniera 中的天然糖苷，具有抗肿瘤和抗利什曼原虫作用。
TMA1603	Parishin C 巴利森苷 C,巴利森苷C	Antioxidant	oxidation-reduction
	Parishin C 是一种从天麻中分离出的 Parishin 衍生物，可能具有抗氧化作用。
T0938	Thiabendazole 2-(4-Thiazolyl)benzimidazole,噻菌灵	Microtubule Associated; Mitochondrial Metabolism; Parasite	Cytoskeletal Signaling; Metabolism; Microbiology/Virology
	Thiabendazole (2-(4-Thiazolyl)benzimidazole) 是具有驱虫特性的苯并咪唑衍生物。
TN1005	Parishin E 巴利森苷E,巴利森苷 E	Others	Others
	Parishin E 是一种分离自天麻的 Parishin 衍生物，可能具有抗氧化活性。
T4S2164	Narirutin Naringenin-7-O-rutinoside,Isonaringin,芸香柚皮苷,柚皮芸香苷	Others; Antibacterial	Microbiology/Virology; Others
	Narirutin (Naringenin-7-O-rutinoside) 是从Citrus unshiu 中分离的活性成分之一，具有抗氧化和抗炎活性。它是一种具有抗结核效力的shikimate 激酶抑制剂。
T0416	Gluconate sodium Sodium D-gluconate,Sodium gluconate,葡萄糖酸钠,D-Gluconic acid sodium salt,D-Gluconate sodium salt	Others; Endogenous Metabolite	Metabolism; Others
	Gluconate sodium (Sodium D-gluconate) 是一种阻垢缓蚀剂。
TN1513	Clitorin 碟豆宁,碟豆素	PKC; Antifection	Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology
	Clitorin 是一种山奈酚糖苷，分离自 Acalypha indica 的花和叶，表现出抗氧化活性。
T3948	Undecanoic acid Hendecanoic acid,十一烷酸,Undecylic acid	Others; Endogenous Metabolite; Antifungal	Metabolism; Microbiology/Virology; Others
	Undecanoic acid (Hendecanoic acid) 是一种具有抗真菌特性的一元羧酸，可抑制红色葡萄球菌中细胞外角蛋白酶、脂肪酶的产生和几种磷脂的生物合成。
T4241	Rubiadin 1,3-Dihydroxy-2-Methylanthracene-9,10-Dione,茜根定,茜草素	Free radical scavengers; PARP; Caspase	Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; oxidation-reduction; Proteases/Proteasome
	Rubiadin (1,3-Dihydroxy-2-Methylanthracene-9,10-Dione) 是一种二羟基蒽醌，提取自茜草，具有抗氧化剂作用。
T13350	Wushanicaritin	Others	Others
	Wushanicaritin 在 DPPH 自由基清除活性测试中显示出显著的抗氧化活性，其IC50值为35.3 μM，具有抗肿瘤作用和抗炎活性。
T1045	Trimipramine maleate Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐	Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor	GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
	Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂，对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。
TN1892	Lusianthridin	Others; c-Myc	Cell Cycle/Checkpoint; Others
	Lusianthridin 是来自石斛 Dendrobium venustum 的天然产物。 Lusianthridin 在无毒浓度下表现出抗迁移特性。 Lusianthridin 通过抑制 Src-STAT3 信号传导增强 c-Myc 降解。
Fr14298	2'-Hydroxy-4'-methylacetophenone 2'-羟基-4'-甲基苯乙酮,2′-羟基-4′-甲基苯乙酮	Anti-infection	Microbiology/Virology
	2'-Hydroxy-4'-methylacetophenone 是一种分离自韩国当归根部得到的酚类，可用于合成 4’-methyl-2’-[(p-tolylsulfonyl) oxy] acetophenone，具有杀螨作用。
TN1644	Flavanomarein	Others	Others
	Flavanomarein 是Coreopsis tinctoria Nutt 的主要黄酮类化合物，对糖尿病性肾病具有保护作用。它具有很好的抗氧化，降糖，降压和降血脂作用。
T3771	Methyl protodioscin 山药,Smilax saponin B,NSC-698790	Apoptosis	Apoptosis
	Methyl protodioscin (Smilax saponin B) 是一种甾二糖苷，能诱导细胞周期阻滞，具有抗肿瘤活性。
T3787	Didymin Isosakuranetin-7-O-rutinoside,Neoponcirin,香风草甙	Apoptosis; Others	Apoptosis; Others
	Didymin (Neoponcirin) 从柑橘类水果中提取的一种膳食类黄酮苷，具有抗氧化特性。它通过抑制 N-Myc 和上调 RKIP 诱导凋亡。
T3S0218	Thonningianin A	Apoptosis; Others	Apoptosis; Others
	Thonningianin A 是从非洲草药通宁宁的甲醇提取物中，分离得到的一种鞣花素，具有抗癌和抗氧化性，涉及自由基清除、抗超氧化物形成和金属螯合。
T3816	Velutin	NF-κB; HIF/HIF Prolyl-Hydroxylase	Chromatin/Epigenetic; Metabolism; NF-κB
	Velutin 是一种苷元，提取自槲寄生中，能够抑制黑色素生物合成。它利用 NF-κB 途径减少破骨细胞分化和下调 HIF-1α。
T1468	Lornoxicam Ro 13-9297,Chlortenoxicam,TS110,氯诺昔康	COX; Endogenous Metabolite	Immunology/Inflammation; Metabolism; Neuroscience
	Lornoxicam (Chlortenoxicam) 是一种新型非甾体抗炎药，是高活性 COX-1 和 COX-2 抑制剂，IC50 分别为 5 和 8 nM。
TJS0314	5,7-Dihydroxy-4-methylcoumarin Methyl-2H-Chromen-2-One,5,7-二羟基-4-甲基香豆素,4-Methyllimetol,4-Methyl-5,7-Dihydroxycoumarin	Others; Antibacterial; Antifungal	Microbiology/Virology; Others
	5,7-Dihydroxy-4-methylcoumarin (Methyl-2H-Chromen-2-One) 是墨西哥龙蒿中的一种香豆素衍生物。它抑制人类中性粒细胞氧化代谢和弹性蛋白酶活性，有抗真菌和抗细菌活性。
T6480	D-Pantothenic acid vitamin B5,pantothenate,D-泛酸	Others	Others
	D-Pantothenic acid (vitamin B5) 是必需的微量营养素，是辅酶 A 的前体，在很多生物过程中发挥关键作用，如调节碳水化合物，脂质，蛋白和核酸代谢。
T6S1784	Brazilin Natural Red 24,巴西苏木素;苏枋精,Braziletto,Brasilin,Superbresiline,巴西苏木素	Apoptosis; Others; AMPK; Autophagy	Apoptosis; Autophagy; Chromatin/Epigenetic; Others; PI3K/Akt/mTOR signaling
	Brazilin (Braziletto) 是来自几种热带硬木的心材的一种红色染料前体，有软骨保护和抗炎活性。它抑制细胞增殖，促进细胞凋亡并通过 AMPK/mTOR 途径诱导自噬。
T4S0867	Pogostone DHELWANGIN,广藿香酮	Apoptosis; Antibacterial; Autophagy	Apoptosis; Autophagy; Microbiology/Virology
	Pogostone (DHELWANGIN) 是从薄荷中分离出，对革兰氏阴性菌、革兰氏阳性菌、大肠埃希菌等具有强效抗菌、抗真菌活性。它诱导细胞凋亡和自噬。
T7032	Eupatorin	Others; P450	Metabolism; Others
	Eupatorin 是天然存在的黄酮，可捕获 G2-M 细胞周期，激活多个 caspase、细胞色素 C 的释放、多聚 (ADP-核糖) 聚合酶的裂解，促使凋亡细胞死亡。
T3795	Corilagin	Apoptosis; TLR; Reverse Transcriptase; Antibacterial; Autophagy	Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology
	Corilagin 是一种鞣酸，有抑制 RNA 肿瘤病毒逆转录酶的活性。它抑制金黄色葡萄球菌的生长，MIC 为 25 μg/mL。它有抗肿瘤活性，可用于肝癌和卵巢癌。
T6S1699	Shogaol [6]-Shogaol,姜烯酚,6-姜烯酚,6-Shogaol	Lipoxygenase; Autophagy	Autophagy; Metabolism
	6-Shogaol (6-Shogaol) 是从生姜中分离的一种天然产物，具有抗癌、抗炎和抗氧化的多种生物活性。
T6S1917	Schisandrol B Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B	P450; Reactive Oxygen Species; Autophagy	Autophagy; Immunology/Inflammation; Metabolism; NF-κB
	Schisandrol B (Besigomsin) 是华中五味子的主要活性成分，具有保肝、抗炎、抗糖尿病和抗氧化的作用。它抑制活性氧的产生，也抑制 P-糖蛋白和CYP3A 的活性。
TN4777	Physalin G	Others	Others
	Physalin G has antinociceptive property.
TN6456	N-trans-caffeoyloctopamine
	N-trans-Caffeoyltyramine has both arginase inhibitory property and antioxidant capacity.
TN4414	Laricitrin 3-O-glucoside	Others	Others
	Laricitrin 3-O-glucoside has antioxidant property.
T72794	Millmerranone A
	Millmerranone A 具有抑制乙酰胆碱酯酶的特性。
TN1760	Icariside E5 淫羊藿次甙E5,淫羊藿次甙 E5	Others	Others
	Icariside E5 may have antioxidant property that strengthen the importance of peppers in the Mediterranean diet.
TN3113	5-Heptadecylresorcinol 芒果	Others	Others
	5-Heptadecylresorcinol has strong inhibitory property against the growth of PC3 cells.
TN1811	Jionoside D	Others	Others
	Jionoside D exhibits antioxidant property.
T28834	Spirolaxine
	Spirolaxine, a natural product isolated from Sporotrichum laxum ATCC 15155, has shown a variety of biological activities including promising anti-Helicobacter pylori property.
TN3836	Desacetylmatricarin	Others	Others
	Desacetylmatricarin has anti-allergic property, it shows a potent inhibitory activity upon the beta-hexosaminidase release from RBL-2H3 cells in a dose-dependent manner and the IC50 of 7.5 microM.
TN1931	Methyllinderone	Antifection	Microbiology/Virology
	Methyllinderone is a human chymase inhibitor, it has antioxidant property, it also shows moderate to weak antifungal activities against various pathogenic fungi.
TN3133	5-O-Methylgenistein	Others	Others
	5-O-Methylgenistein may show free radical scavenging activity, it also may have hepatoprotective property on the model of toxic hepatitis induced by carbon tetrachloride damage.
TN1484	Cheilanthifoline	NF-κB; Antifection	Microbiology/Virology; NF-κB
	Cheilanthifoline has anti-osteoclastogenic property, it gives significant inhibitions on receptor activator of nuclear factor-κB ligand-induced differentiation of mouse bone marrow-derived macrophages into multinucleated osteoclasts.
T5S0313	Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷	Others; TNF	Apoptosis; Others
	Liquiritin apioside has antioxidant property by inducing glutathione (GSH) biosynthesis via the inhibition of cytokines and protected lung epithelial cells against cigarette smoke-mediated oxidative stress, might be as protective agent against epithelial
T69369	Cladosporin
	Cladosporin 是一种真菌代谢物，在 Cladosporium cladosporioid 的菌丝体中产生。含浓度 75 μg/mL Cladosporin 的琼脂培养基可完全抑制多种皮肤癣菌的生长。
TN4223	Homopterocarpin	Antifection	Microbiology/Virology
	Homopterocarpin and Pterocarpus extract offer gastroprotection against indomethacin- induced ulcer by antioxidative mechanism and the modulation of gastric homeostasis, homopterocarpin may be responsible for, or contribute to the antiulcerogenic property
TN1104	Cyanidin 3-sambubioside chloride 矢车菊素-3-桑布双糖苷,Cyanidin-3-O-sambubioside chloride	NF-κB; ROS	Immunology/Inflammation; NF-κB
	Cyanidin-3-O-sambubioside chloride is inhibitors of BPDE-induced NF-kB activity. It inhibits the enzyme activity by competing with the substrate for the active site. Cyanidin-3-O-sambubioside chloride has antioxidant activity and free-radical-scavenging p
TN3525	Boehmenan	ERK; Phosphatase; EGFR; PARP; MEK; Wnt/beta-catenin; Akt; Caspase; STAT; p53	Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; JAK/STAT signaling; MAPK; Metabolism; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
	(±)-Boehmenan shows potent protein-tyrosine phosphatase 1B (PTP1B) inhibitory activity in vitro with the IC(50) values of 43.5 uM, it inhibits PTP1B activity in a competitive manner. Boehmenan exhibits the potent cytotoxic effects against many cancer cell
T35751	Violacein
	Violacein is a bacterial metabolite originally isolated from C. violaceum that has antibacterial and antiprotozoal activities.[1] [2] It is produced by C. violaceum as a purple pigment in response to N-hexanoyl homoserine lactone , a property that has been modified to create a strain of C. violaceum used in detecting quorum-sensing molecules.[3] Violacein is active against Gram-positive bacteria, including B. subtilis and S. aureus (MICs = 0.8 and 1.6 &#181M, respectively). It is also active aga...

天然产物

N-Benzyllinoleamide

Cat.No: TN1353

Synonym: (9Z,12Z)-N-Benzyloctadeca-9,12-dienamide,N-苄基-(9Z,12Z)-十八碳二烯酰胺

Target: Others

Cat.No: TN7113

Target: Others

Cat.No: T0144

Synonym: Histanorm,安息香酸,伏保克西里

Target: Antibacterial

Bacopasaponin C

Cat.No: TN1432

Synonym: (-)-假马齿苋皂苷 C,假马齿苋皂苷C

Target: Anti-infection, GABA Receptor, NMDAR

Cat.No: TMA1603

Synonym: 巴利森苷 C,巴利森苷C

Target: Antioxidant

Cat.No: T0938

Synonym: 2-(4-Thiazolyl)benzimidazole,噻菌灵

Target: Microtubule Associated, Mitochondrial Metabolism, Parasite

Cat.No: TN1005

Synonym: 巴利森苷E,巴利森苷 E

Target: Others

Cat.No: T4S2164

Synonym: Naringenin-7-O-rutinoside,Isonaringin,芸香柚皮苷,柚皮芸香苷

Target: Others, Antibacterial

Gluconate sodium

Cat.No: T0416

Synonym: Sodium D-gluconate,Sodium gluconate,葡萄糖酸钠,D-Gluconic acid sodium salt,D-Gluconate sodium salt

Target: Others, Endogenous Metabolite

Cat.No: TN1513

Synonym: 碟豆宁,碟豆素

Target: PKC, Antifection

Undecanoic acid

Cat.No: T3948

Synonym: Hendecanoic acid,十一烷酸,Undecylic acid

Target: Others, Endogenous Metabolite, Antifungal

Cat.No: T4241

Synonym: 1,3-Dihydroxy-2-Methylanthracene-9,10-Dione,茜根定,茜草素

Target: Free radical scavengers, PARP, Caspase

Cat.No: T13350

Target: Others

Trimipramine maleate

Cat.No: T1045

Synonym: Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐

Target: Dopamine Receptor, 5-HT Receptor, Antibacterial, Adrenergic Receptor, Norepinephrine, Histamine Receptor

Cat.No: TN1892

Target: Others, c-Myc

2'-Hydroxy-4'-methylacetophenone

Cat.No: Fr14298

Synonym: 2'-羟基-4'-甲基苯乙酮,2′-羟基-4′-甲基苯乙酮

Target: Anti-infection

Cat.No: TN1644

Target: Others

Methyl protodioscin

Cat.No: T3771

Synonym: 山药,Smilax saponin B,NSC-698790

Target: Apoptosis

Cat.No: T3787

Synonym: Isosakuranetin-7-O-rutinoside,Neoponcirin,香风草甙

Target: Apoptosis, Others

Thonningianin A

Cat.No: T3S0218

Target: Apoptosis, Others

Cat.No: T3816

Target: NF-κB, HIF/HIF Prolyl-Hydroxylase

Cat.No: T1468

Synonym: Ro 13-9297,Chlortenoxicam,TS110,氯诺昔康

Target: COX, Endogenous Metabolite

5,7-Dihydroxy-4-methylcoumarin

Cat.No: TJS0314

Synonym: Methyl-2H-Chromen-2-One,5,7-二羟基-4-甲基香豆素,4-Methyllimetol,4-Methyl-5,7-Dihydroxycoumarin

Target: Others, Antibacterial, Antifungal

D-Pantothenic acid

Cat.No: T6480

Synonym: vitamin B5,pantothenate,D-泛酸

Target: Others

Cat.No: T6S1784

Synonym: Natural Red 24,巴西苏木素;苏枋精,Braziletto,Brasilin,Superbresiline,巴西苏木素

Target: Apoptosis, Others, AMPK, Autophagy

Cat.No: T4S0867

Synonym: DHELWANGIN,广藿香酮

Target: Apoptosis, Antibacterial, Autophagy

Cat.No: T7032

Target: Others, P450

Cat.No: T3795

Target: Apoptosis, TLR, Reverse Transcriptase, Antibacterial, Autophagy

Cat.No: T6S1699

Synonym: [6]-Shogaol,姜烯酚,6-姜烯酚,6-Shogaol

Target: Lipoxygenase, Autophagy

Cat.No: T6S1917

Synonym: Gomisin A,TJN-101,Besigomsin,五味子醇乙,Gamma-Schisandrin,戈米辛A,Schizandrol B,Wuweizi alcohol-B

Target: P450, Reactive Oxygen Species, Autophagy

Cat.No: TN4777

Target: Others

N-trans-caffeoyloctopamine

Cat.No: TN6456

Laricitrin 3-O-glucoside

Cat.No: TN4414

Target: Others

Millmerranone A

Cat.No: T72794

Cat.No: TN1760

Synonym: 淫羊藿次甙E5,淫羊藿次甙 E5

Target: Others

5-Heptadecylresorcinol

Cat.No: TN3113

Synonym: 芒果

Target: Others

Cat.No: TN1811

Target: Others

Cat.No: T28834

Desacetylmatricarin

Cat.No: TN3836

Target: Others

Methyllinderone

Cat.No: TN1931

Target: Antifection

5-O-Methylgenistein

Cat.No: TN3133

Target: Others

Cheilanthifoline

Cat.No: TN1484

Target: NF-κB, Antifection

Liguiritigenin-7-O-D-apiosyl-4'-O-D-glucoside

Cat.No: T5S0313

Synonym: Liquiritin apioside,甘草苷元-7-O-D-芹糖-4'-O-D-葡萄糖苷

Target: Others, TNF

Cat.No: T69369

Homopterocarpin

Cat.No: TN4223

Target: Antifection

Cyanidin 3-sambubioside chloride

Cat.No: TN1104

Synonym: 矢车菊素-3-桑布双糖苷,Cyanidin-3-O-sambubioside chloride

Target: NF-κB, ROS

Cat.No: TN3525

Target: ERK, Phosphatase, EGFR, PARP, MEK, Wnt/beta-catenin, Akt, Caspase, STAT, p53

Cat.No: T35751

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