144
3
2
14
Cat. No. | Product Name | ||
---|---|---|---|
L8110 | 细胞重编程化合物库 | 1813 compounds | |
1813 种重编程信号通路相关的生物活性小分子化合物的特有集合,可用于高通量、高内涵筛选 | |||
L9860 | 抗抑郁症化合物库 | 1163 compounds | |
1163 种与抑郁症相关的化合物,可以用于高通量和高内涵筛选 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T63349 |
Treprostinil diethanolamine
UT-15C |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Treprostinil diethanolamine (UT-15C) 是EP2、DP1和IP 的有效激动剂,对EP2、DP1、IP、EP1、EP4、EP3 和 FPKi 的值分别为 3.6、4.4、32.1、212、826、2505 和 4680 nM。Treprostinil diethanolamine 能够促使 cAMP 的上调,进而维持血管系统内的稳态,并造成人肺动脉的血管扩张。 | |||
T77364 |
Sibeprenlimab
VIS649,VIS-649 |
Others | Others |
Sibeprenlimab (VIS649) 是一种抑制 APRIL 的人源化IgG 2单克隆抗体。Sibeprenlimab 对 APRIL 有抑制作用,可用于研究预防和治疗 肾病(IgAN)。 | |||
T20626 |
Esomeprazole
|
Proton pump; Cysteine Protease | Membrane transporter/Ion channel; Proteases/Proteasome |
Esomeprazole 是奥美拉唑(omeprazole) 的S-异构体,抑制溶酶体半胱氨酸蛋白酶legumain,防止癌症转移。它是一种质子泵抑制剂(PPI)。 | |||
T21746 |
Terameprocol
tetramethyl Nordihydroguaiaretic Acid,EM-1421 |
HIV Protease | Microbiology/Virology; Proteases/Proteasome |
Terameprocol (EM-1421) 是 Nordihydroguaiaretic acid 的合成衍生物,是非选择性脂氧合酶抑制剂。 | |||
T16732 |
Reproxalap
NS-2,ADX-102 |
Others | Others |
Reproxalap (NS-2) 是一种活性醛类隔离剂,可用于干眼症的研究。它能够与醛 (包括丙二醛和 4-羟基壬醛) 共价结合。 | |||
T68048 |
Cloxacepride
|
CaMK | Neuroscience |
cloxacepride 是一种CaM 拮抗剂,可用于治疗哮喘疾病。 | |||
T1651 |
Rabeprazole sodium
Dexrabeprazole Sodium,LY307640 sodium,Habeprazole Sodium,雷贝拉唑钠,Rebeprazole sodium,Aciphex Sodium |
Apoptosis; Proton pump | Apoptosis; Membrane transporter/Ion channel |
Rabeprazole sodium (Habeprazole Sodium) 是一种质子泵抑制剂,不可逆地抑制胃 H+/K+-ATPase,可研究胃溃疡和胃食管反流。它诱导细胞凋亡,也抑制尿苷核苷核糖水解酶 ,IC50为 0.3 μM。 | |||
T12883 |
Fezagepras
PBI-4050,3-戊基苯乙酸,Setogepram |
GPR | Endocrinology/Hormones; GPCR/G Protein |
Fezagepras (Setogepram) 是一种可口服的 GPR40激动剂和GPR84拮抗剂或反向激动剂。它减轻肾、肝和胰腺纤维化,具有抗纤维化、抗炎和抗增殖作用。 | |||
T31659 |
Eprociclovir
AV10,AV-10,A-5021,A 5021,A5021,AV 10 |
Antifection | Microbiology/Virology |
Eprociclovir (A-5021) 是一种新型阿昔洛韦类似物,是 EHV1 复制的强效抑制剂,可能用于治疗和/或预防该病毒感染。Eprociclovir 对大多数人类疱疹病毒都有很强的抗疱疹活性。 | |||
T78556 |
Antidepressant agent 5
|
Others | Others |
Antidepressant agent 5 是一种具有抗抑郁活性的 7-取代四氢异喹啉衍生物。Antidepressant agent 5 在研究抑郁症方面和木兰花碱作用效果类似,可用于预防和治疗抑郁症疾病。 | |||
T76727 |
Teprotumumab
R 1507,HZN 001 |
TSH Receptor; IGF-1R | GPCR/G Protein; Tyrosine Kinase/Adaptors |
Teprotumumab 是一种阻断 IGF-1 受体 (IGF-1R) 的人单克隆抗体。Teprotumumab 与 IGF-1R 的细胞外 α-亚基结构域配体结合。Teprotumumab 抑制纤维细胞中的 TSH 和 IGF-1 作用。Teprotumumab 可降低 TSH 依赖性 IL-6 和 IL-8 的表达和 Akt 的磷酸化。Teprotumumab 可用于甲状腺相关眼病的研究。 | |||
T21433 |
Stepronin
Prostenoglycine,Tiofacic,Tiase,TTPG |
Others | Others |
Stepronin (TTPG) 具有祛痰活性并抑制气道分泌。 | |||
T7808 |
Alacepril
Cetapril,阿拉普利,DU-1219 |
RAAS | Endocrinology/Hormones |
Alacepril (DU-1219) 是一种具有口服活性血管紧张素转换酶 (ACE) 抑制剂,具有长效抗高血压作用。 | |||
T19826 |
Rabeprazole
LY307640 |
Potassium Channel; STAT | JAK/STAT signaling; Membrane transporter/Ion channel; Stem Cells |
Rabeprazole (LY307640) 是一种 H+/K+-ATPase 抑制剂,通过靶向 STAT3 介导的糖酵解来抑制胃上皮细胞中的细胞增殖,可用于研究胃溃疡。 | |||
T32658L |
Leteprinim
AIT082 acid,AIT 082 acid,AIT-082 acid |
Others | Others |
Leteprinim (AIT 082 acid) 是一种次黄嘌呤衍生物,可刺激体外神经突生长和星形胶质细胞产生腺苷和神经营养因子。 | |||
T4414 |
Eprenetapopt
APR-246,PRIMA-1Met |
Apoptosis; Others; Ferroptosis; p53; Autophagy | Apoptosis; Autophagy; Others |
Eprenetapopt (PRIMA-1Met) 是一种在 TP53突变细胞中恢复野生型 p53功能的小分子,可引发肿瘤细胞凋亡,还抑制硒蛋白硫氧还蛋白还原酶 1。 | |||
T2686 |
Esomeprazole Magnesium
(S)-Omeprazole magnesium,NEXIUM,埃索美拉唑镁,(-)-Omeprazole magnesium |
ATPase; Proton pump | Membrane transporter/Ion channel |
Esomeprazole Magnesium (NEXIUM) 是一种口服有效的 H+, K+-ATPase 抑制剂,在上消化道疾病和胃食管反流疾病中具有研究价值。Esomeprazole magnesium 是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。 | |||
T15239 |
Epristeride
SKF105657,ONO-9302 |
Apoptosis; Reductase | Apoptosis; Endocrinology/Hormones; Metabolism |
Epristeride (ONO-9302) 是具有口服活性、选择性和非竞争性类固醇 5-α-还原酶亚型2抑制剂,抑制SR 同工酶 2。Episteride 可减小前列腺大小并改善良性前列腺增生男性的症状。Episteride 诱导大鼠腹侧前列腺萎缩和凋亡。 | |||
T6580 |
Meprednisone
SCH 4358,Methylprednisone,NSC 527579,Betanisona,Betapar,泼尼松 |
Glucocorticoid Receptor; Autophagy | Autophagy; Endocrinology/Hormones |
Meprednisone (Betapar) 是糖皮质激素,用于糖皮质激素受体,是泼尼松的甲基化衍生物。 | |||
T2687 |
Omeprazole sulfide
Omeprazole metabolite Omeprazole sulfide,Ufiprazole,奥美拉唑硫醚 |
Proton pump; Drug Metabolite | Membrane transporter/Ion channel; Metabolism |
Omeprazole sulfide (Ufiprazole) 是 Omeprazole 的代谢物。 | |||
T2531L |
Eprosartan
KF-108566J free base,Teveten |
RAAS | Endocrinology/Hormones |
Eprosartan (SKF-108566J free base) 是一种具有选择性和竞争性的非肽类血管紧张素II受体拮抗剂,对AT1受体亚型具有高亲和力,可用作降压剂。Eprosartan 对血管紧张素 II 受体有抑制作用,在大鼠和人类肾上腺皮质膜中的 IC50 值分别为 9.2 nM 和 3.9 nM。 | |||
T3034 |
Eprazinone dihydrochloride
Resplen,Mucitux,Eftapan,NSC 317935,盐酸依普拉酮,依普拉酮二盐酸,Eprazinone 2HCl |
Others; Neurokinin receptor | GPCR/G Protein; Neuroscience; Others |
Eprazinone dihydrochloride (NSC 317935) 是一种具有镇咳和粘液溶解作用的粘液溶解剂。它是神经激肽 1 受体的配体,可改善肺功能和动脉血氧分压,可用于慢性支气管炎的研究。 | |||
T10138 |
4-Desmethoxy Omeprazole
|
Drug Metabolite | Metabolism |
4-Desmethoxy Omeprazole 是 Omeprazole 的活性代谢物。Omeprazole 是质子泵抑制剂。Omeprazole 竞争性抑制 CYP2C19 活性,Ki=2 - 6 μM。Omeprazole 还抑制革兰氏阴性菌和革兰氏阳性菌生长。 | |||
T10221 |
Abeprazan hydrochloride
DWP14012 hydrochloride,Fexuprazan hydrochloride |
Proton pump | Membrane transporter/Ion channel |
Abeprazan hydrochloride (Fexuprazan hydrochloride) 是一种有效的、可逆的、具有口服活性的potassium-competitive acid 阻滞剂,通过竞争性的与钾离子结合抑制 H+,K+- ATPase,而无需酸激活。Abeprazan hydrochloride 是一种质子泵抑制剂(PPI),通过减少胃酸的产生而起作用,可用于治疗胃酸相关疾病,如胃食管反流病(GERD)和消化性溃疡。 | |||
T8386 |
Esomeprazole Magnesium trihydrate
埃索美拉唑镁三水合物,埃索美拉唑镁(三水),(S)-Omeprazole magnesium trihydrate |
Proton pump | Membrane transporter/Ion channel |
Esomeprazole Magnesium trihydrate ((S)-Omeprazole magnesium trihydrate) 是一种口服有效的H+, K+-ATPase 抑制剂,在上消化道疾病和胃食管反流疾病的研究中具有价值。它是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。 | |||
T15773 |
Lofepramine
Gamanil,洛非帕明,Amplit,Leo 640,Lopramine |
5-HT Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Lofepramine (Leo 640) 是一种有效的三环抗抑郁药,广泛地代谢为 Desipramine。它能够抑制摄取促进去甲肾上腺素能神经传递,以及抑制神经元摄取 5-羟色胺和色氨酸吡咯酶,增强 5-羟色胺能神经传递,进而发挥其抗抑郁作用。它还具有显著的抗焦虑效果。 | |||
T1102 |
Mifepristone
C-1073,RU486,RU 38486,米非司酮 |
Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; NO Synthase; Autophagy | Autophagy; Endocrinology/Hormones; Immunology/Inflammation; Others |
Mifepristone (C-1073) 是一种黄体酮受体和糖皮质激素受体拮抗剂,在体外实验中的 IC50值分别为 0.2 nM 和 2.6 nM。 | |||
T9417L |
gamma-preprotachykinin amide (72-92) acetate
gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base) |
Others | Others |
gamma-preprotachykinin amide (72-92) acetate 是一种 21 个氨基酸的肽,属于速激肽 (TK) 家族,在其 C 末端序列中包括神经激肽 A (NKA)。它对中枢 NK-2 受体的亲和力高于 NKA;它对 NK-1 受体的亲和力较低,但是,它有效地刺激唾液分泌,这是由 NK-1 受体激活介导的。 | |||
T5150 |
Treprostinil
LRX-15,曲前列环素,Orenitram,曲前列尼尔,Remodulin |
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Treprostinil (Orenitram) 是有效的 DP1、IP 和 EP2 激动剂,EC50分别为0.6、1.9 和 6.2 nM。 | |||
T15471 |
Hepronicate
Megrin |
Others | Others |
Hepronicate(Megrin) 是一种具有降血脂和血管扩张活性的小分子化合物。 | |||
T19722 |
Benazeprilat
CGS14831,CGS-14831,CGS 14831 |
RAAS; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Benazeprilat(CGS 14831) 是一种具有口服活性的贝那普利活性代谢物。Benazeprilat 具有高效的抗血压活性,可与其他其他类别的化合物(包括噻嗪类利尿剂和钙通道阻滞剂)联合使用来减少与心血管风险和继发性终末器官损伤相关的疾病的发生。Benazeprilat 可能用于研究急性左心室衰竭。 | |||
T5836 |
Eprinomectin
依普菌素,MK-397 |
Parasite | Microbiology/Virology |
Eprinomectin (MK-397) 是一种阿维菌素,具有驱虫,杀虫杀螨活性。 | |||
T37621 |
Ezeprogind disulfate
|
Beta Amyloid | Neuroscience |
Ezeprogind disulfate 是一种神经营养诱导剂。 Ezeprogind disulfate 针对所有神经退行性变,包括 Abeta 蛋白或 tau 蛋白。 Ezeprogind disulfate 可用于神经系统疾病相关研究,包括进行性核上性麻痹(PSP)、tau 蛋白病、阿尔茨海默病和帕金森病等。 | |||
T5391 |
Bepridil hydrochloride
CERM 1978,盐酸苄普地尔 |
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Bepridil hydrochloride (CERM 1978) 是一种钙通道阻滞剂,还抑制 Na+/Ca2+ 交换(NCX)、钠通道和心脏肌膜 KATP 通道,具有抗心绞痛的作用。 | |||
T22391 |
Omeprazole Sodium
|
P450; Proton pump; Antibacterial; Autophagy | Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Omeprazole 是有效的质子泵抑制剂,在胃肠道疾病的研究中具有价值。它竞争性抑制CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阴性菌和革兰氏阳性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。 | |||
T2686L |
Esomeprazole Sodium
埃索美拉唑钠,(S)-Omeprazole sodium |
ATPase; Proton pump | Membrane transporter/Ion channel |
Esomeprazole Sodium ((S)-Omeprazole sodium) 是一种口服有效的活性质子泵抑制剂。Esomeprazole sodium 通过抑制胃壁细胞中的 H+, K+-ATPase 来降低酸分泌,在胃食管反流疾病中有研究价值。Esomeprazole 是一种外泌体抑制剂,通过抑制 V-H+-ATPases 来阻断外泌体的释放。 | |||
T2531 |
Eprosartan Mesylate
SKF-108566J,甲磺酸依普罗沙坦 |
RAAS | Endocrinology/Hormones |
Eprosartan Mesylate (SKF-108566J) 是一种具有选择性、竞争性血管紧张素 II 受体拮抗剂,是具有口服活性的非肽。它结合血管紧张素 II 受体,在大鼠和人类肾上腺皮质膜中的IC50值分别为 9.2 nM 和 3.9 nM,可用作降压剂。 | |||
T1734 |
Rabeprazole Sulfide
雷贝拉唑相关物质E,Rabeprazole Related Compound E |
Proton pump; Antibacterial | Membrane transporter/Ion channel; Microbiology/Virology |
Rabeprazole Sulfide (Rabeprazole Related Compound E) 是 Rabeprazole 的活性代谢产物。Rabeprazole 是一种质子泵抑制剂类的抗溃疡药物,有效抑制幽门螺旋杆菌的活性,可通过与胃壁细胞中的(H+/K+)-ATPase 相互作用来抑制胃酸分泌,可研究各种消化系统疾病。 | |||
T12375 |
Fezagepras sodium
Setogepram sodium salt,PBI-4050 sodium salt |
GPR | Endocrinology/Hormones; GPCR/G Protein |
Fezagepras sodium (Setogepram sodium salt) 是口服有效的 GPR40 激动剂及 GPR84 拮抗剂或反向激动剂。Fezagepras sodium 可以减轻肝,肾和胰腺纤维化。Fezagepras sodium 具有抗炎,抗增殖和抗纤维化作用。 | |||
T0382 |
Eprodisate disodium
NC-503,伊罗地塞二钠,伊罗地塞二钠盐 |
Others | Others |
Eprodisate disodium (NC-503) 是一种带负电荷的磺化类的原纤维形成抑制剂,是口服具有活力的 Eprodisate 二钠盐形式,可用于研究淀粉样蛋白A(AA) 淀粉样变性病。 | |||
T5053 |
Eprobemide
LIS 630,依普贝胺 |
MAO; Monoamine Oxidase | Metabolism; Neuroscience |
Eprobemide (LIS 630) 是一种非竞争性的、可逆的单胺氧化酶 A 抑制剂。 | |||
T5360 |
Eprotirome
伊罗替罗,KB2115 |
Thyroid hormone receptor(THR) | Endocrinology/Hormones |
Eprotirome (KB2115) 是一种肝脏选择性甲状腺激素受体 (thyroid hormone receptor, TR) 激动剂。它对 TRβ的亲和力略高于TRα。它降低了低密度脂蛋白 (LDL) 胆固醇的浓度,可用于研究血脂异常和肥胖症。 | |||
T12309 |
Omeprazole metabolite Omeprazole sulfone
Omeprazole sulphone,Omeprazole sulfone |
Others | Others |
Omeprazole metabolite Omeprazole sulfone 是Omeprazole 的代谢物,能够抑制质子泵。 | |||
T5008 |
Teprenone
Tetraprenylacetone,Geranylgeranylacetone,替普瑞酮 |
HSP | Cytoskeletal Signaling; Metabolism |
Teprenone (Geranylgeranylacetone) 是一种热休克蛋白诱导剂,有抗溃疡作用。 | |||
T7722 |
Feprazone
Prenazone,非普拉宗,DA 2370,DA2370,DA-2370 |
Others | Others |
Feprazone (DA-2370) 具有抗炎和抗脂肪生成特性。 Feprazone 可用于治疗关节和肌肉疼痛的研究。 | |||
T71934 |
Atibeprone
|
MAO | Metabolism; Neuroscience |
Atibeprone 是 MAO-B 抑制剂,具有抗抑郁活性,可用于研究帕金森病。 | |||
T0757 |
Omeprazole
Losec,Prilosec,奥美拉唑,奥美拉挫,H 16868,Antra |
Proton pump; Phospholipase; Antibacterial; Autophagy | Autophagy; Membrane transporter/Ion channel; Metabolism; Microbiology/Virology |
Omeprazole (Losec) 是一种质子泵抑制剂,有研究胃肠道疾病的潜力。它竞争性抑制 CYP2C19活性,Ki 为 2 到 6 μM。它还抑制革兰氏阳性菌和革兰氏阴性菌生长。它是中性鞘磷脂酶的外泌体抑制剂。 | |||
T7728 |
ACEPROMAZINE MALEATE
|
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Acepromazine maleate 是一种 α 肾上腺素受体 (alpha-adrenoceptor) 拮抗剂,是一种吩噻嗪类促进安定的试剂。 | |||
T4686 |
Simeprevir
TMC435,西咪匹韦,TMC-435350,Olysio |
HCV Protease; SARS-CoV | Microbiology/Virology; Proteases/Proteasome |
Simeprevir (TMC435) 是一种有效的 HCV NS3/4A 蛋白酶抑制剂,抑制 HCV 复制,EC50 为 7.8 nM。它也是 SARS-CoV-2 3CLpro 抑制剂。 | |||
T0180 |
Benazepril hydrochloride
盐酸贝那普利,CGS 14824A HCl,Benazepril HCl,CGS14824A |
RAAS | Endocrinology/Hormones |
Benazepril hydrochloride (CGS 14824A HCl) 是一种血管紧张素转化酶(ACE)抑制剂,能够作用于高血压。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5029 |
Oxaceprol
奥沙西罗,N-Acetyl-L-hydroxyproline,N-乙酰-L-4-羟基脯氨酸 |
Others | Others |
Oxaceprol (N-Acetyl-L-hydroxyproline) 是一种可口服的、具有显著抗炎作用的 L-脯氨酸衍生物,常用于研究骨关节炎和类风湿性关节炎。 | |||
T5297 |
3-Indolepropionic acid
Indolepropionic acid,IPA,indole-3-propionic acid,吲哚-3-丙酸 |
Antioxidant; Reactive Oxygen Species; Endogenous Metabolite | Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction |
3-Indolepropionic acid (Indolepropionic acid) 是强效的抗氧化剂,具有研究阿尔兹海默症的潜能。 | |||
TN1571 | Depressine | Others | Others |
Depressine is a natural product from Gentiana depressa. |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-02166 |
Epiregulin Protein, Mouse, Recombinant (hFc)
epiregulin,EPR |
Mouse | HEK293 Cells |
Epiregulin Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 33.8 kDa and the accession number is Q61521. | |||
TMPY-03672 |
Survivin Protein, Human, Recombinant
BIRC5,IAP4,API4,baculoviral IAP repeat containing 5,EPR<... |
Human | E. coli |
BIRC5, also known as Survivin and EPR-1, is a member of theIAP family. IAP family members usually contain multiple baculovirus IAP repeat (BIR) domains, but BIRC5 has only a single BIR domain. It is expressed cell cycle-dependently and highly expressed at mitosis. As a multitasking protein, BIRC5 has dual roles in promoting cell proliferation and preventing apoptosis. Survivin is a component of a chromosome passage protein complex (CPC) which is essential for chromosome alignment and segregation... | |||
TMPK-01516 |
HLA-A*02:01&B2M&Survivin (LMLGEFLKL) Tetramer Protein, Human, MHC (His & Avi)
IAP4,survivin variant 3 alpha,BIRC5,Survivin,EPR-1,... |
Human | HEK293 Cells |
Survivin (also known as BIRC5) is an evolutionarily conserved eukaryotic protein that is essential for cell division and can inhibit cell death. Normally it is only expressed in actively proliferating cells, but is upregulated in most, if not all cancers; consequently, it has received significant attention as a potential oncotherapeutic target. | |||
TMPK-01480 |
HLA-A*02:01&B2M&Survivin (LMLGEFLKL) Monomer Protein, Human, MHC (His & Avi), Biotinylated
IAP4,Survivin,API4,BIRC5,MHC,MHC I,EPR-1,survivin v... |
Human | HEK293 Cells |
Survivin (also known as BIRC5) is an evolutionarily conserved eukaryotic protein that is essential for cell division and can inhibit cell death. Normally it is only expressed in actively proliferating cells, but is upregulated in most, if not all cancers; consequently, it has received significant attention as a potential oncotherapeutic target. | |||
TMPK-01517 |
HLA-A*02:01&B2M&Survivin (LMLGEFLKL) Monomer Protein, Human, MHC (His & Avi)
survivin variant 3 alpha,MHC I,BIRC5,EPR-1,IAP4,Sur... |
Human | HEK293 Cells |
Survivin (also known as BIRC5) is an evolutionarily conserved eukaryotic protein that is essential for cell division and can inhibit cell death. Normally it is only expressed in actively proliferating cells, but is upregulated in most, if not all cancers; consequently, it has received significant attention as a potential oncotherapeutic target. | |||
TMPY-01318 |
Meprin alpha/MEP1A Protein, Mouse, Recombinant (His)
meprin A, alpha (PABA peptide hydrolase),AW107200,M... |
Mouse | HEK293 Cells |
Meprin alpha/MEP1A Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 69 kDa and the accession number is A0A0R4J043. | |||
TMPJ-00411 |
LEPR Protein, Human, Recombinant (hFc)
LEPR,Leptin receptor,OB-R,OB receptor,OBR,CD295,DB,... |
Human | HEK293 Cells |
LEPR Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-Fc tag. The predicted molecular weight is 150-180 KDa and the accession number is P48357. | |||
TMPY-00261 |
Meprin beta Protein, Human, Recombinant (His)
meprin A, β,Meprin β,meprin A, be... |
Human | HEK293 Cells |
MEP1B (Meprin A Subunit Beta) is a Protein Coding gene. This gene encodes the beta subunit. Targeted disruption of this gene in mice affects embryonic viability, renal gene expression profiles, and distribution of the membrane-associated alpha subunit in the kidney and intestine. Meprins are cell membrane, oligomeric metalloendopeptidases composed of two distinct but evolutionarily related subunits, alpha, and beta. MEP1A is mapped to the short arm of chromosome 6 by the use of radiation and som... | |||
TMPY-01737 |
Meprin alpha/MEP1A Protein, Human, Recombinant (His)
meprin A, α (PABA peptide hydrolase),mepri... |
Human | HEK293 Cells |
Meprin alpha/MEP1A Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 67.7 kDa and the accession number is Q16819. | |||
TMPJ-00976 |
LEPR Protein, Mouse, Recombinant (His)
OBR,DB,Leptin receptor,OB receptor,CD295,OB-R,LEPR,... |
Mouse | HEK293 Cells |
LEPR Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with C-10His tag. The predicted molecular weight is 120-150 KDa and the accession number is P48356. | |||
TMPJ-00975 |
LEPR Protein, Mouse, Recombinant (hFc)
CD295,DB,HuB219,OB receptor,LEP-R,Leptin receptor,OBR,LE... |
Mouse | HEK293 Cells |
LEPR Protein, Mouse, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-Fc tag. The predicted molecular weight is 130-190 KDa and the accession number is P48356. | |||
TMPH-00644 |
Lactose operon repressor Protein, E. coli, Recombinant (His & SUMO)
|
E. coli | E. coli |
Repressor of the lactose operon. Binds allolactose as an inducer. | |||
TMPJ-00977 |
LEPR Protein, Mouse, Recombinant (mFc)
LEPR,CD295,OB-R,LEP-R,HuB219,Leptin receptor,OBR,DB... |
Mouse | HEK293 Cells |
LEPR Protein, Mouse, Recombinant (mFc) is expressed in HEK293 mammalian cells with C-mFc tag. The predicted molecular weight is 130-190 KDa and the accession number is P48356. | |||
TMPH-00646 |
LexA repressor Protein, E. coli, Recombinant (His & SUMO)
|
E. coli | E. coli |
Represses a number of genes involved in the response to DNA damage (SOS response), including recA and lexA. Binds to the 16 bp palindromic sequence 5'-CTGTATATATATACAG-3'. In the presence of single-stranded DNA, RecA interacts with LexA causing an autocatalytic cleavage which disrupts the DNA-binding part of LexA, leading to derepression of the SOS regulon and eventually DNA repair. Implicated in hydroxy radical-mediated cell death induced by hydroxyurea treatment.The SOS response controls an ap... |