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1844

抑制剂 & 化合物

127

天然产物

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Cat. No. Product Name Target Signaling Pathways
T3587 NOD-IN-1

Compound 4

NOD-like Receptor (NLR); NOD Immunology/Inflammation; NF-κB
NOD-IN-1 (Compound 4) 是核苷酸结合寡聚化结构域样受体 NOD1(IC50:5.74 μM)和 NOD2 (IC50:6.45 μM)的抑制剂。
Fr12729 1-Benzyl-4-hydroxypiperidine

1-Benzylpiperidin-4-ol

Compound Fr12729 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr12729,CAS号为 4727-72-4
T13114 CCR2 antagonist 4

Teijin compound 1

CCR Immunology/Inflammation; Microbiology/Virology
CCR2 antagonist 4 (Teijin compound 1) 是高效的、特异性的CCR2拮抗剂,对 CCR2b 的IC50为 180 nM,抑制 MCP-1 诱导的趋化作用的 IC50为 24 nM。
Fr14015 4-Methylquinolin-2-ol

2-Hydroxy-4-methylquinoline

Compound Fr14015 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr14015,CAS号为 607-66-9。
T50122 3-Ethyl-1-methyl-2-thioxoimidazolidin-4-one

3-Ethyl-1-methyl-2-thioxoimidazolidin-4-one 是一种属于咪唑烷酮类化合物的有机化合物,已被用于生命科学相关研究。
T3586 Compound 401

2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one

DNA-PK DNA Damage/DNA Repair; PI3K/Akt/mTOR signaling
Compound 401 (2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one) 是一种可靶向 mTOR 的合成 DNA-PK 抑制剂,IC50为0.28 μM。
Fr13587 7-Chloro-4-(piperazin-1-yl)quinoline

7-Chloro-4-(piperazin-1-yl)quinolone 结构是药物化学中的重要支架,它单独或与其他活性药效团混合显示出多种药理特性。7-Chloro-4-(piperazin-1-yl)quinolone 是有效的sirtuin 抑制剂,并且抑制 5-羟色胺的摄取,IC50值为 50 μM。7-Chloro-4-(piperazin-1-yl)quinolone 对恶性疟原虫 D10 和 K1 菌株表现出抗疟疾活性,IC50分别为 1.18 μM 和 0.97 μM。
FL0195 N-Boc-4-hydroxy-L-proline methyl ester

N-Boc-cis-4-hydroxy-L-proline methyl ester为不可降解(non-cleavable)的ADC linker,用于抗体药物偶联体(ADCs)合成。该化合物同时作为基于烷基链(alkyl chain)的PROTAC linker,适用于PROTAC合成。
T22678 3,5-Bis(4-nitrophenoxy)benzoic acid

3,5-二(4-硝基苯氧基)苯甲酸,Compound W

Gamma-secretase Neuroscience; Proteases/Proteasome; Stem Cells
3,5-Bis(4-nitrophenoxy)benzoic acid (Compound W) 是 γ-secretase 抑制剂。它导致 Aβ42 和 notch-1 Aβ-like peptide 25 (Nβ25) 的释放水平降低。它是母体血清中 3,3’-diiodothyronine sulfate (T2S) 的交叉反应物质,可作为胎儿甲状腺功能减退的标志物。
T6146 Dorsomorphin dihydrochloride

BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride

AMPK; Autophagy; TGF-beta/Smad Autophagy; Chromatin/Epigenetic; PI3K/Akt/mTOR signaling; Stem Cells
Dorsomorphin dihydrochloride (BML-275 2HCl) 是一种选择性和 ATP 竞争性的AMPK 抑制剂,Ki 为 109 nM。它诱导自噬,通过靶向抑制 I 型受体ALK2,ALK3和ALK6来抑制 BMP 途径。
T21000 PiB

2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇,Pittsburgh Compound-B,6-OH-BTA-1

Others Others
PiB (Pittsburgh Compound-B) 是分析 11C-PiB 的标准品。 11C-PiB 是一种用于阿尔茨海默病诊断的 β-淀粉样蛋白 PET 成像示踪剂。
T9658 DCZ3301

NPS ALX Compound 4a hydrochloride(1:1)(299433-10-6 Free base)

Others Others
DCZ3301是一种新的芳基胍抑制剂。
T9184L Compound 3344 hydrochloride

4-(2,3-dihydro-1,4-benzodioxin-5-yl)-~{N}-[3-[(dimethylamino)methyl]phenyl]-2-methoxy-aniline hydrochloride(2368246-78-8 free base),Compound 3344 hydrochloride (2368246-78-8 free base)

Ras GPCR/G Protein; MAPK
Compound 3344 hydrochloride 是 KRAS 效应相互作用的抑制剂,亲和力为 126nm。
T27757 Kv1.5-IN-IIII

Kv1.5INIIII,Kv1.5INIV,Compound IIII,Kv1.5IN4,Compound 4

Kv1.5-IN-IIII is a potent inhibitor of Kv1.5.
T19230 CCR2 antagonist 4 hydrochloride

Teijin compound 1 hydrochloride

Others Others
CCR2 antagonist 4 hydrochloride is a specific CCR2 antagonist (IC50s: 180 nM for CCR2b). It potently inhibits MCP-1-induced chemotaxis (IC50: 24 nM).
T3298 Ethyl 3-amino-1H-pyrazole-4-carboxylate

3-Amino-4-ethoxycarbonylpyrazole

T8829 2',4'-DIHYDROXYCHALCONE

2',4'-DHC,2',4'-二羟查耳酮

HSP Cytoskeletal Signaling; Metabolism
2',4'-DIHYDROXYCHALCONE (2',4'-DHC) 作为具有 Hsp90 抑制和抗真菌作用的化合物
T3681 4-Cyclohexylphenol

p-Cyclohexylphenol,4-Hydroxyphenylcyclohexane,4-环己基苯酚

Others Others
4-Cyclohexylphenol (p-Cyclohexylphenol) 是一种用于蛋白质组学研究的生化化合物。
T10337 Antimicrobial Compound 1

Antibacterial Microbiology/Virology
Antimicrobial Compound 1 是一种烷基吡啶鎓化合物,尾部为 12C,头部为 4-羧基。 Antimicrobial Compound 1 对枯草芽孢杆菌和大肠杆菌具有抗菌活性。
T67923 WIC1

Others Others
2H-1-Benzopyran-3-carboxamide, N-[4-(4-ethyl-1-piperazinyl)phenyl]-2-oxo-是 化合物,是治疗肿瘤的潜在化合物。
Fr14035 3,3-Tetramethyleneglutarimide

Compound Fr14035 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr14035,CAS号为 1075-89-4
Fr13734 Piperonylonitrile

1,3-Benzodioxole-5-carbonitrile

Compound Fr13734 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr13734,CAS号为 4421-09-4
T50084 (2E)-N-(4-methoxyphenyl)-3-[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-yl]prop-2-enamide

Others Others
(2E)-N-(4-methoxyphenyl)-3-[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-yl]prop-2-enamide 是一种用作分子结构单元的化合物,用于多种有机物的合成。
T10785 Chalcone 4 hydrate

Others; Parasite Microbiology/Virology; Others
Chalcone 4 hydrate 是一种抗寄生虫剂,可抑制 Babesia 和 Theileria 的生长。
T131725 Compound TCFN92660

Compound TCFN92660 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T131725,CAS号为 56070-89-4
T50125 Compound C749

Compound C749 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T50125,CAS号为 57-03-4
T61147 Chitin synthase inhibitor 4

Antibiotic Microbiology/Virology
Chitin synthase inhibitor 4 是一种具有抗菌活性的几丁质合成酶(CHS)抑制剂。Chitin synthase inhibitor 4 是一种基于CHS 的化合物,是一种候选的杀菌剂。
T60017 5-Bromo-4-chloro-3-indoxyl-beta-D-cellobioside

Others Others
5-Bromo-4-chloro-3-indoxyl-beta-D-cellobioside 是用于检测纤维生物水解酶的显色化合物。
T90421 2-Bromo-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine

2-Bromo-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine 是有一种有用的有机化合物,已被用于生命科学相关研究。
T40350 HPK1-IN-4

HPK1-IN-4

MAPK MAPK
HPK1-IN-4是一种HPK1(MAPK41)抑制剂,IC 50为0.061 nM。HPK1-IN-4常被作为临床前免疫治疗工具化合物。
T7038 4-Methylayapin

4-甲基-6,7-亚甲基二氧代香豆素,4-METHYL-6,7-METHYLENEDIOXYCOUMARIN

Others Others
4-Methylayapin 用作中间体。
T4675 4-Carboxyisothiazole

Others Others
4-Carboxyisothiazole 用作中间体。
T50070 1-ethyl-6-fluoro-4-oxo-7-[4-(3-phenylpropanoyl)piperazin-1-yl]-1,4-dihydroquinoline-3-carboxylic acid

Others Others
1-ethyl-6-fluoro-4-oxo-7-[4-(3-phenylpropanoyl)piperazin-1-yl]-1,4-dihydroquinoline-3-carboxylic acid 是一种用作分子结构单元的化合物,是一种SMURF1抑制剂。
T11673 IRAK4-IN-4

IRAK; cGAS Immunology/Inflammation; NF-κB
IRAK4-IN-4 (化合物 15) 是白介素-1 受体相关激酶抑制剂,IC50为 2.8 nM。它还抑制环 GMP-AM 合酶 ,IC50为 2.1 nM。
T50105 6-chloro-1-ethyl-7-(4-methylpiperazin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid

Others Others
6-chloro-1-ethyl-7-(4-methylpiperazin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid 是一种用作分子结构单元的化合物,为培氟沙星杂质。
T9872 Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-

Others Others
Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-是一种用于抗病毒活性测定的化合物。
T22364 Methyl 4-aminobutyrate HCl

4-氨基丁酸甲酯盐酸盐,Methyl 4-aminobutyrate hydrochloride,GABA methyl ester

Others Others
Methyl 4-aminobutyrate HCl (GABA methyl ester) 是一种由氨基丁酸和甲醇缩合而成的甲酯化合物。
T60124 1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea

TNF Apoptosis
1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea 是一种能够激动 TNF-α的化合物,可以诱导细胞分泌 TNF-α。
T22348 Isonipecotic acid

4-Piperidinecarboxylic acid,Hexahydroisonicotinic acid,4-哌啶甲酸,4-Carboxypiperidine

GABA Receptor Membrane transporter/Ion channel; Neuroscience
Isonipecotic acid (4-Piperidinecarboxylic acid) 是一种杂环化合物。它主要表征为 GABAA 受体部分激动剂。
T18391 N-Boc-4-pentyne-1-amine

Others; PROTAC Linker Others; PROTAC
N-Boc-4-pentyne-1-amine 是一种基于烷基链的PROTAC连结剂,用于PROTAC MG-277[1]的合成。
T3726 Erdafitinib

厄达替尼,JNJ-42756493

Apoptosis; FGFR Angiogenesis; Apoptosis; Tyrosine Kinase/Adaptors
Erdafitinib (JNJ-42756493) 是一种喹喔啉衍生物,是一种具有口服活性的FGFR 家族抑制剂,抑制FGFR1/2/3/4活性的IC50分别为1.2、 2.5、3.0和5.7 nM。
T7272 2,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE

2,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T7272,CAS号为 675602-93-4
T50028 6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole

6-氟-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚,6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole

Others Others
6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole (6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) 是一种吲哚衍生物,具有潜在抗癌活性,是开发新药的潜在先导化合物。
T4170 PKM2-IN-1

PKM2 inhibitor,compound 3k

PKM Metabolism
PKM2-IN-1 (compound 3k) 是丙酮酸激酶 M2 (PKM2) 抑制剂,其IC50=2.95 μM。
T64319 4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester

Others Others
4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester 是一种生物活性化合物,可作为中间体用于多种化合物的合成。
T9797 Benzenamine, 2-[2-(dimethylamino)ethoxy]-4-(1H-pyrazol-4-yl)-

Benzenamine, 2-[2-(dimethylamino)ethoxy]-4-(1H-pyrazol-4-yl)- 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T9797,CAS号为 1072906-07-0。
T3679 1-(4-FLUORO-PHENYL)-BUTAN-1-ONE

Others Others
1-(4-FLUORO-PHENYL)-BUTAN-1-ONE 用作中间体。
T2040 OAC1

BAS 00287861

OCT Membrane transporter/Ion channel
OAC1 (BAS 00287861) 是一种能够激活 Octamer 结合转录因子 4 的化合物。 它提高了 iPSC 重编程效率并加速重编程过程。
T19031 NBD-F

4-Fluoro-7-nitrobenzofurazan

Others Others
NBD-F (4-Fluoro-7-nitrobenzofurazan) 是一种用于氨基酸分析 (amino acid analysis) 的前荧光试剂。它能与一级或二级胺反应生成荧光产物,从而分析氨基酸和低分子量胺。
T67858 STIMA-1

2-Vinylquinazolin-4-ol,p53 Activator VII

Others Others
STIMA-1 (2-Vinylquinazolin-4-ol) 是一种活性化合物,可以恢复 p63 的活性。STIMA-1 可以刺激角质形成细胞的增殖和分化。

化合物

NOD-IN-1
Cat.No: T3587
Synonym: Compound 4
Target: NOD-like Receptor (NLR), NOD
1-Benzyl-4-hydroxypiperidine
Cat.No: Fr12729
Synonym: 1-Benzylpiperidin-4-ol
Target:
CCR2 antagonist 4
Cat.No: T13114
Synonym: Teijin compound 1
Target: CCR
4-Methylquinolin-2-ol
Cat.No: Fr14015
Synonym: 2-Hydroxy-4-methylquinoline
Target:
3-Ethyl-1-methyl-2-thioxoimidazolidin-4-one
Cat.No: T50122
Synonym:
Target:
Compound 401
Cat.No: T3586
Synonym: 2-morpholino-4H-pyrimido[2,1-a]isoquinolin-4-one
Target: DNA-PK
7-Chloro-4-(piperazin-1-yl)quinoline
Cat.No: Fr13587
Synonym:
Target:
N-Boc-4-hydroxy-L-proline methyl ester
Cat.No: FL0195
Synonym:
Target:
3,5-Bis(4-nitrophenoxy)benzoic acid
Cat.No: T22678
Synonym: 3,5-二(4-硝基苯氧基)苯甲酸,Compound W
Target: Gamma-secretase
Dorsomorphin dihydrochloride
Cat.No: T6146
Synonym: BML-275 2HCl,Compound C dihydrochloride,6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Dorsomorphin (Compound C) 2HCl,Compound C 2HCl,BML-275 dihydrochloride
Target: AMPK, Autophagy, TGF-beta/Smad
PiB
Cat.No: T21000
Synonym: 2-(4-(二甲基氨基)苯基)苯并[D]噻唑-6-醇,Pittsburgh Compound-B,6-OH-BTA-1
Target: Others
DCZ3301
Cat.No: T9658
Synonym: NPS ALX Compound 4a hydrochloride(1:1)(299433-10-6 Free base)
Target: Others
Compound 3344 hydrochloride
Cat.No: T9184L
Synonym: 4-(2,3-dihydro-1,4-benzodioxin-5-yl)-~{N}-[3-[(dimethylamino)methyl]phenyl]-2-methoxy-aniline hydrochloride(2368246-78-8 free base),Compound 3344 hydrochloride (2368246-78-8 free base)
Target: Ras
Kv1.5-IN-IIII
Cat.No: T27757
Synonym: Kv1.5INIIII,Kv1.5INIV,Compound IIII,Kv1.5IN4,Compound 4
Target:
CCR2 antagonist 4 hydrochloride
Cat.No: T19230
Synonym: Teijin compound 1 hydrochloride
Target: Others
Ethyl 3-amino-1H-pyrazole-4-carboxylate
Cat.No: T3298
Synonym: 3-Amino-4-ethoxycarbonylpyrazole
Target:
2',4'-DIHYDROXYCHALCONE
Cat.No: T8829
Synonym: 2',4'-DHC,2',4'-二羟查耳酮
Target: HSP
4-Cyclohexylphenol
Cat.No: T3681
Synonym: p-Cyclohexylphenol,4-Hydroxyphenylcyclohexane,4-环己基苯酚
Target: Others
Antimicrobial Compound 1
Cat.No: T10337
Synonym:
Target: Antibacterial
WIC1
Cat.No: T67923
Synonym:
Target: Others
3,3-Tetramethyleneglutarimide
Cat.No: Fr14035
Synonym:
Target:
Piperonylonitrile
Cat.No: Fr13734
Synonym: 1,3-Benzodioxole-5-carbonitrile
Target:
(2E)-N-(4-methoxyphenyl)-3-[3-(4-methylphenyl)-1-phenyl-1H-pyrazol-4-yl]prop-2-enamide
Cat.No: T50084
Synonym:
Target: Others
Chalcone 4 hydrate
Cat.No: T10785
Synonym:
Target: Others, Parasite
Compound TCFN92660
Cat.No: T131725
Synonym:
Target:
Compound C749
Cat.No: T50125
Synonym:
Target:
Chitin synthase inhibitor 4
Cat.No: T61147
Synonym:
Target: Antibiotic
5-Bromo-4-chloro-3-indoxyl-beta-D-cellobioside
Cat.No: T60017
Synonym:
Target: Others
2-Bromo-4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridine
Cat.No: T90421
Synonym:
Target:
HPK1-IN-4
Cat.No: T40350
Synonym: HPK1-IN-4
Target: MAPK
4-Methylayapin
Cat.No: T7038
Synonym: 4-甲基-6,7-亚甲基二氧代香豆素,4-METHYL-6,7-METHYLENEDIOXYCOUMARIN
Target: Others
4-Carboxyisothiazole
Cat.No: T4675
Synonym:
Target: Others
1-ethyl-6-fluoro-4-oxo-7-[4-(3-phenylpropanoyl)piperazin-1-yl]-1,4-dihydroquinoline-3-carboxylic acid
Cat.No: T50070
Synonym:
Target: Others
IRAK4-IN-4
Cat.No: T11673
Synonym:
Target: IRAK, cGAS
6-chloro-1-ethyl-7-(4-methylpiperazin-1-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
Cat.No: T50105
Synonym:
Target: Others
Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]-
Cat.No: T9872
Synonym:
Target: Others
Methyl 4-aminobutyrate HCl
Cat.No: T22364
Synonym: 4-氨基丁酸甲酯盐酸盐,Methyl 4-aminobutyrate hydrochloride,GABA methyl ester
Target: Others
1-(4-chloro-3-(trifluoromethyl)phenyl)-3-(7-(1-methyl-1H-pyrazol-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-yl)urea
Cat.No: T60124
Synonym:
Target: TNF
Isonipecotic acid
Cat.No: T22348
Synonym: 4-Piperidinecarboxylic acid,Hexahydroisonicotinic acid,4-哌啶甲酸,4-Carboxypiperidine
Target: GABA Receptor
N-Boc-4-pentyne-1-amine
Cat.No: T18391
Synonym:
Target: Others, PROTAC Linker
Erdafitinib
Cat.No: T3726
Synonym: 厄达替尼,JNJ-42756493
Target: Apoptosis, FGFR
2,3,5-TRIFLUORO-4-(TRIFLUOROMETHYL)PYRIDINE
Cat.No: T7272
Synonym:
Target:
6-fluoro-3-(4-1,2,5,6-tetrahydropyridyl)indole
Cat.No: T50028
Synonym: 6-氟-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚,6-fluoro-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole
Target: Others
PKM2-IN-1
Cat.No: T4170
Synonym: PKM2 inhibitor,compound 3k
Target: PKM
4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester
Cat.No: T64319
Synonym:
Target: Others
Benzenamine, 2-[2-(dimethylamino)ethoxy]-4-(1H-pyrazol-4-yl)-
Cat.No: T9797
Synonym:
Target:
1-(4-FLUORO-PHENYL)-BUTAN-1-ONE
Cat.No: T3679
Synonym:
Target: Others
OAC1
Cat.No: T2040
Synonym: BAS 00287861
Target: OCT
NBD-F
Cat.No: T19031
Synonym: 4-Fluoro-7-nitrobenzofurazan
Target: Others
STIMA-1
Cat.No: T67858
Synonym: 2-Vinylquinazolin-4-ol,p53 Activator VII
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN7210 Pseudane V

2-pentylquinolin-4-ol,Compound Z1509149676,2-n-pentyl-4-quinolinol,2-Pentylquinolin-4(1H)-one

Others Others
Pseudane V (2-pentylquinolin-4-ol) 是一种海洋来源的天然产物,存在于Pseudoalteromonas sp. M2。
TN6434 New compound 4

New compound 4是一种天然产物,属于豆科葛属,其产品编号为 TN6434。New compound 4可用作对照参考。
T21104 4-Decanol

AI3-19949,Decan-4-ol

4-Decanol (Decan-4-ol) 是一种从Valeriana jatamansi Jones 的根部和Epilobium angustifolium L.中分离出来的化合物,可能具有抗炎和抗氧化活性。
T9425 Epipinoresinol-4'-O-β-D-glucoside

Others Others
Simplocosin 是一种葡萄糖苷类化合物。
T8015 4-METHOXYCHALCONE

2-(4-Methoxybenzal)Acetophenone,4-甲氧基查耳酮

Others Others
4-METHOXYCHALCONE (2-(4-Methoxybenzal)Acetophenone) 是一种增强脂肪细胞分化的天然化合物。
TJP2865 7-methoxy-8-hydroxy-4-methylcoumarin

Others Others
7-methoxy-8-hydroxy-4-methylcoumarin 是分离自酸橙 (Citrus aurantium) 的一种化合物。
TN2883 3',4'-Dimethoxyflavone

Others; PARP Chromatin/Epigenetic; DNA Damage/DNA Repair; Others
3',4'-Dimethoxyflavone 是类黄酮化合物的参考标准,类黄酮化合物具有多种药用活性。
TN2704 2,3-Dihydroxy-4-methoxybenzoic acid

Others Others
2,3-Dihydroxy-4-methoxybenzoic acid 是从甜樱桃果实中提取分离出来的一种化合物。
TN7025 Canolol

菜籽多酚,Phenol, 4-ethenyl-2,6-dimethoxy-

COX Immunology/Inflammation; Neuroscience
Canolol (Phenol, 4-ethenyl-2,6-dimethoxy-) 是一种抗氧化酚类化合物,可用作 COX-2 抑制剂。
TN7032 4'-O-Methylpyridoxine

4-methoxymethylpyridoxine,Ginkgotoxin

Antioxidant oxidation-reduction
4'-O-Methylpyridoxine(MPN)是从银杏叶中发现的维生素类化合物,具有抗氧化活性和细胞毒性。
Fr14298 2'-Hydroxy-4'-methylacetophenone

2'-羟基-4'-甲基苯乙酮,2′-羟基-4′-甲基苯乙酮

Anti-infection Microbiology/Virology
2'-Hydroxy-4'-methylacetophenone 是一种分离自韩国当归根部得到的酚类,可用于合成 4’-methyl-2’-[(p-tolylsulfonyl) oxy] acetophenone,具有杀螨作用。
T77563 4-Ethylcatechol

DNA DNA Damage/DNA Repair
4-Ethylcatechol 存在于红葡萄酒中,可从Glechoma longituba(NaKai)Kupr 中提取。4-Ethylcatechol 在Cu(II)存在下会引起DNA 损伤。4-Ethylcatechol 是一种高效的抗血小板化合物。
T39887 (S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid

(S)-3-(4-羟苯基)乳酸,(S)-3-(4-Hydroxyphenyl)lactic acid,(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid

Others Others
(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid ((S)-3-(4-Hydroxyphenyl)lactic acid) 是分离自间肠隐球菌培养基的代谢物,具有高的 DPPH 清除自由基活性和抗氧化活性。
T7106 Menaquinone-4

四烯甲萘醌,Vitamin K2,Menaquinone K4

Others; Endogenous Metabolite Metabolism; Others
Menaquinone-4 (Vitamin K2) 是维生素 K 的一种,用作止血剂,有潜力用于骨质疏松的研究。
T5082 Calcium 2-hydroxy-4-(methylthio)butanoate

羟基蛋氨酸钙,calcium hydroxymethionine,2-Hydroxy-4-(methylthio)butyric acid calcium salt

Others; Endogenous Metabolite Metabolism; Others
Calcium 2-hydroxy-4-(methylthio)butanoate (Calcium 2-hydroxy-4-(calcium hydroxymethionine)) 是内源性代谢产物的一种。
T2A2524 2-Hydroxy-4-methoxybenzaldehyde

4-甲氧基水杨醛,4-Methoxysalicylaldehyde,2-羟基-4-甲氧基苯甲醛

Tyrosinase; Antibacterial Microbiology/Virology; Proteases/Proteasome
2-Hydroxy-4-methoxybenzaldehyde (4-Methoxysalicylaldehyde) 是一种来自三种东非药用植物,Mondia whitei、Rhus vulgaris Meikle 和Sclerocarya caffra Sond 的酪氨酸酶抑制剂。它是香兰素的异构体,可用于合成尿苷M7。
TN3029 4-(Ethoxymethyl)phenol

p-Hydroxybenzyl Et ether

Antioxidant oxidation-reduction
4-(Ethoxymethyl)phenol (p-Hydroxybenzyl Et ether) 是一种从 Amburana cearensis 中提取的小分子化合物,具有细胞毒性和抗氧化会活性。
TMO2713 4(3H)-Quinazolinone

Quinazolin-4-ol,4-Hydroxyquinazoline,4-羟基喹唑啉,4-Quinazolinol,4-Quinazolone,4-Quinazolinone

Antibacterial; Platelet aggregation Microbiology/Virology; Others
4(3H)-Quinazolinone (4-Hydroxyquinazoline) 是化学合成中的砌块,是一种生物活性氮杂环化合物。它具有多种生物学特性,如抗菌,抗真菌,抗惊厥,抗炎,抗 HIV,抗癌和缓解疼痛活性。
Fr12277 4-Hydroxy-6-methylcoumarin

Others Others
4-Hydroxy-6-methylcoumarin(4-HMC)是一种天然存在的酚类化合物,是香豆素的衍生物,存在于各种植物、真菌和细菌中,具有抗炎和抗肿瘤活性。4-HMC 在食品工业中用作调味剂、防腐剂和抗氧化剂。
TN7235 4-methoxylonchocarpin

TNF; NF-κB Apoptosis; NF-κB
4-methoxylonchocarpin 是从Abrus precatorius 的根中分离出来的以一种有效的抗炎化合物。4-methoxylonchocarpin 通过抑制LPS 与巨噬细胞的TLR4结合来抑制NF-κB 激活TNF 表达,抑制TNBS 引起的小鼠结肠炎。
T3343 5-methoxyflavone

5-methoxy-2-phenylchromen-4-one,5-甲氧基黄酮

DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair
5-methoxyflavone (5-methoxy-2-phenylchromen-4-one) 是一种类黄酮,是DNA 聚合酶 β 的抑制剂和 β-淀粉样蛋白毒性的神经保护剂。它通过调控嗜离子 GABAA 受体,起到镇静中枢神经系统的作用。
TN1950 Moracin M

PDE Metabolism
Moracin M 是桑白皮中的一种酚类成分,有效的磷酸二酯酶 4 (PDE4) 抑制剂,对于 PDE4D2,PDE4B2,PDE5A1 和 PDE9A2 的 IC50 分别为 2.9 μM,4.5 μM,> 40 μM 和 > 100 μM。Moracin M 具有抗炎活性。
T2A2486 3',​4',​5',​5,​7-​Pentamethoxyflavone

5,7,3',4',5'-Pentamethoxyflavone

Nrf2 Immunology/Inflammation
3',4',5',5,7-Pentamethoxyflavone 是从 Rutaceae 中发现的的一种天然黄铜类化合物,通过抑制Nrf2 通路克服化疗活性分子从而对癌细胞展现出耐药性。
T0562 Protocatechuic acid

3, 4-Dihydroxybenzoic acid,3,4-二羟基苯甲酸,Protocatechuate,原儿茶酸,3,4-Dihydroxybenzoic acid

Others Others
Protocatechuic acid (3, 4-Dihydroxybenzoic acid) 是天然的多酚类物质,具有神经保护活性。
T7910 4-Methoxybenzaldehyde

大茴香醛,Anisaldehyde,p-Anisaldehyde,Anisic aldehyde,4-Anisaldehyde,4-甲氧基苯甲醛,P-Methoxybenzaldehyde

Others; Endogenous Metabolite Metabolism; Others
4-Methoxybenzaldehyde (p-Anisaldehyde) 是一种天然存在的芳香酚类化合物,存在于许多植物物种中,包括辣根,茴香,八角茴香等。它是一种能够能的神经毒物,已经表现出致死亡率,吸引力和干扰宿主寻求的影响。
T67319 2',4'-Dimethylacetophenone

Endogenous Metabolite Metabolism
2',4'-Dimethylacetophenone 是一种可用于生物研究的化学物。该化合物可用于气相色谱法检测烟草化合物中的醛固酮香气,可以用于保护食品。
TN6647 4-O-Cinnamoylquinic acid

金银花

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
4-O-Cinnamoylquinic acid 是从 Casearia grewiifolia 干果中提取出来的小分子化合物,对前列腺素有抑制作用,抑制人中性粒细胞中超氧阴离子的生成。
T41095 (E)-3-(4-Methoxyphenyl)acrylic acid

(E)-3-(4-甲氧基苯基)丙烯酸

Glucosidase Metabolism
(E)-3-(4-Methoxyphenyl)acrylic acid 是从 Etlingera pavieana (Pierre ex Gagnep.) R. M. Sm. 的根茎中分离出来的一种小分子化合物。它是一种新型 α-葡萄糖苷酶抑制剂。(E)-3-(4-甲氧基苯基)丙烯酸具有保肝活性、抗失水活性、增强认知效果,并可用于降低血压血糖。
T19866 Indican

NSC-87517,3-Indoxyl-beta-D-glucopyranoside,3-吲哚基-beta-D-吡喃葡萄糖苷,NSC 87517,NSC87517,Indoxyl-β-D-glucoside

OAT; MRP Immunology/Inflammation; Membrane transporter/Ion channel
Indican (Indoxyl-β-D-glucoside) 是吲哚酚的一种糖苷,染料靛蓝和靛玉红的前体。它的主要代谢物是硫酸吲哚酚 (IS)。其中 IS 是尿毒症毒素,是有机阴离子转运蛋白1 (OAT 1)、OAT 3 和多药耐药相关蛋白4 (MRP 4) 的底物/抑制剂。
T4S21320 ISOGINKGETIN

异银杏素,4',4'''-Dimethylamentoflavone,异银杏双黄酮

MMP; Others Others; Proteases/Proteasome
ISOGINKGETIN (4',4'''-Dimethylamentoflavone) 是一种MMP9抑制剂,也是一种Pre-mRNA Splicing 抑制剂。
TCS1709 BENZYLACETONE

苄基丙酮,4-Phenylbutan-2-one,Methyl 2-phenylethyl ketone,4-Phenyl-2-butanone

Tyrosinase Proteases/Proteasome
Benzylacetone (4-Phenyl-2-butanone) 是一种从沉香木中提取的芳香族化合物。它具有增强食欲和减少运动的作用。它具有较强且可逆的抗蘑菇酪氨酸酶作用,对单酚酶和双酚酶作用的IC50值分别为 2.8 mM 和 0.6 mM。
T64353 4-tert-Octylphenol

Endogenous Metabolite Metabolism
4-tert-Octylphenol 是一种干扰内分泌的化学物质及雌激素药物,能诱导子代小鼠脑神经元祖细胞的凋亡,并通过减少溴脱氧尿苷(BrdU)、有丝分裂标志物Ki67以及磷酸组蛋白H3(p-Histone-H3)的表达,导致神经元祖细胞的增殖减少。这种物质不仅会干扰小鼠的大脑发育,还会影响其行为。
TN6985 Anhydronotoptol

4-{[(2E,5E)-3,7-dimethylocta-2,5,7-trien-1-yl]oxy}-7H-furo[3,2-g]chromen-7-one

NO Synthase Immunology/Inflammation
Anhydronotoptol (4-{[(2E,5E)-3,7-dimethylocta-2,5,7-trien-1-yl]oxy}-7H-furo[3,2-g]chromen-7-one) 是一种可从伞科植物羌活中提取得到的天然化合物。Anhydronotoptol 是一种有效的 一氧化氮生成抑制剂, 抑制 LPS 诱导的 RAW 264.7 细胞 NO 生成,其 IC50 值为 36.6 μM。
TN1861 Licoflavone C

4',5,7-Trihydroxy-8-prenylflavone

Antioxidant; Antifungal Microbiology/Virology; oxidation-reduction
Licoflavone C (4',5,7-Trihydroxy-8-prenylflavone) 是从 Glycyrrhiza inflata 的根部分离出来的异戊二烯基黄酮化合物,具有抗氧化和抗真菌活性,在培养的人类外周淋巴细胞中,它对 DAU 或 MMC 诱导的染色体损伤具有保护作用。Licoflavone C 可用于研究真菌感染。
TN1936 Mogroside III-E

罗汉果皂苷ⅢE

IL Receptor; TNF; TLR Apoptosis; Immunology/Inflammation
Mogroside IIIe 是一种葫芦烷型化合物,从罗汉果中分离得到,可抑制 NO 的释放,具有抗肺纤维化作用。
T8280 Deacetylasperulosidic Acid

去乙酰基车叶草苷酸,去乙酰车叶草苷酸,Desacetyl asperulosidic acid

IL Receptor; Interleukin Immunology/Inflammation
Deacetylasperulosidic Acid 是海巴戟果实的主要植物化学成分。它能够防止体外 4-硝基喹啉1-氧化物诱导的 DNA 损伤,抑制 IL-2的产生以及自然杀伤细胞的活化。它具有抗原活性,抑制仓鼠卵巢细胞和小鼠中染色体畸变的诱导。它可增加超氧化物歧化酶活性,从而具有抗氧化活性。
TN5263 1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one

Xanthohumol,黄腐酚

Apoptosis; BCL; PARP; HCV Protease; IAP; Caspase; HIV Protease; NMDAR; p53 Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Neuroscience; Proteases/Proteasome
1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one (Xanthohumol) 是一种从蛇麻草中提纯的具有多种生物功能的天然产物。黄腐酚对 HIV-1 有效,可能是一种有趣的先导化合物。它可能代表一种用于 HIV-1 感染的新型化疗药物。
T4S0350 Licochalcone B

甘草查尔酮 B,甘草查尔酮B

Beta Amyloid; Others Neuroscience; Others
Licochalcone B 是从Glycyrrhiza inflate 根中提取的。它能够抑制淀粉样蛋白 β 自聚集作用 (IC50=2.16 μM) ,分解预先形成的 Aβ42原纤维,并通过螯合金属离子抑制金属诱导的 Aβ42聚集。
T3S0013 Ethyl trans-caffeate

咖啡酸乙酯,Ethyl caffeate,Caffeic Acid Ethyl Ester

Others Others
Ethyl trans-caffeate (Caffeic Acid Ethyl Ester) 具有抗炎作用。 它是一种有前途的天然化合物,未来在慢性肝病中的应用。它是一种有效的化学预防化合物,可防止因太阳紫外线照射引起的皮肤癌变。它是与人胰腺α-淀粉酶复合的代表性抑制剂的高分辨率结构。 它强烈抑制 JB6 Cl41细胞的肿瘤转化,无毒性。 PI3K、ERK1/2 和 p38 激酶活性在体外通过与 HOEC 直接结合而受到抑制。
T4S1637 gamma-Mangostin

Normangostin,γ-倒捻子素

Others; 5-HT Receptor GPCR/G Protein; Neuroscience; Others
gamma-Mangostin (Normangostin) 是从药用植物山竹的果壳中提纯的一种天然产物,是一种竞争性5-HT2A 受体拮抗剂。它是运甲状腺素蛋白原纤维化抑制剂,与甲状腺素结合位点结合并稳定了 TTR 四聚体,具有抗高血压、预防结肠癌等作用。
TCS2170 2,5-Dihydroxyacetophenone

Quinacetophenone,2-Acetylhydroquinone,2-5-dihydroxyacetophenone,2 ',5'-二羟基苯乙酮,Acetylhydroquinone,2,5-二羟基苯乙酮,DHAP

ERK; NF-κB; Tyrosinase MAPK; NF-κB; Proteases/Proteasome
2,5-Dihydroxyacetophenone (Quinacetophenone) 是从熟地黄中分离出的一种天然产物,通过阻断 ERK1/2和 NF-κB 信号通路,抑制活化巨噬细胞中炎症介质的产生。
T4855 Tricosanoic acid

Tricosan-1-oic acid,二十三烷酸

Endogenous Metabolite Metabolism
Tricosanoic acid (Tricosan-1-oic acid) 是毛发生长激活剂,是长链脂肪酸。
T6S1027 Tussilagone

Others Others
Tussilagone 是Tussilago farfara 的主要活性成分,具有抗炎作用。它抑制盲肠结扎和穿刺导致脓毒症的小鼠的炎症反应,提高其生存率。它改善葡聚糖硫酸钠诱导的小鼠结肠炎的炎症反应。
T2S2264 Linalool

Linalol,(±)-Linalool,Phantol,沉香醇

Apoptosis; IL Receptor; TNF; Endogenous Metabolite; iGluR Apoptosis; Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism; Neuroscience
Linalool (Linalol) 是存在芫荽等植物中的单萜类天然产物,是竞争性NMDA 受体拮抗剂,具有抗肿瘤和抗心脏毒性的作用。它通过激活 Nrf2 诱导抗氧化防御和通过抑制 NF-κB 减少炎症反应来保护其免受 LPS/GalN 诱导的肝损伤,具有镇痛、抗菌和抗炎的特性。
T6S2099 Geraniin

Antioxidant; TNF Apoptosis; oxidation-reduction
Geraniin 是一种肿瘤坏死因子α释放抑制剂,其IC50值为 43 μM,具有抗肿瘤、抗炎和抗高血糖活性。
T5089 5-Aminovaleric acid

Others; Endogenous Metabolite Metabolism; Others
5-Aminovaleric acid 被认为是 GABA 的亚甲基同系物,是GABA 的弱激动剂。它是赖氨酸降解产物。 它既能够内源性产生,也能够通过赖氨酸的细菌分解代谢产生。
TN6605 4-Nitrocinnamic acid

4-Nitrocinnamic acid is a photosensitive compound. 4-Nitrocinnamic acid has inhibitory effects on tyrosinase.
T80958 trans-4-Hydroxy-2-nonenoic acid

trans-4-Hydroxy-2-nonenoic acid (compound 4) 为一种可从Pottsia属植物中提取的天然产物。
T19135 4-Hydroxycyclohexanecarboxylic acid

Others Others
4-Hydroxycyclohexanecarboxylic acid is a organic compounds belongs to cyclohexanol compound.
T83370 3',4'-O,O-Methylene-(+)-catechin

3',4'-O,O-Methylene-(+)-catechin (compound 10a)是Piptadenia pervillei中发现的天然化合物。
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天然产物

Pseudane V
Cat.No: TN7210
Synonym: 2-pentylquinolin-4-ol,Compound Z1509149676,2-n-pentyl-4-quinolinol,2-Pentylquinolin-4(1H)-one
Target: Others
New compound 4
Cat.No: TN6434
Synonym:
Target:
4-Decanol
Cat.No: T21104
Synonym: AI3-19949,Decan-4-ol
Target:
Epipinoresinol-4'-O-β-D-glucoside
Cat.No: T9425
Synonym:
Target: Others
4-METHOXYCHALCONE
Cat.No: T8015
Synonym: 2-(4-Methoxybenzal)Acetophenone,4-甲氧基查耳酮
Target: Others
7-methoxy-8-hydroxy-4-methylcoumarin
Cat.No: TJP2865
Synonym:
Target: Others
3',4'-Dimethoxyflavone
Cat.No: TN2883
Synonym:
Target: Others, PARP
2,3-Dihydroxy-4-methoxybenzoic acid
Cat.No: TN2704
Synonym:
Target: Others
Canolol
Cat.No: TN7025
Synonym: 菜籽多酚,Phenol, 4-ethenyl-2,6-dimethoxy-
Target: COX
4'-O-Methylpyridoxine
Cat.No: TN7032
Synonym: 4-methoxymethylpyridoxine,Ginkgotoxin
Target: Antioxidant
2'-Hydroxy-4'-methylacetophenone
Cat.No: Fr14298
Synonym: 2'-羟基-4'-甲基苯乙酮,2′-羟基-4′-甲基苯乙酮
Target: Anti-infection
4-Ethylcatechol
Cat.No: T77563
Synonym:
Target: DNA
(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid
Cat.No: T39887
Synonym: (S)-3-(4-羟苯基)乳酸,(S)-3-(4-Hydroxyphenyl)lactic acid,(S)-3-(4-Hydroxyphenyl)-2-hydroxypropionic acid
Target: Others
Menaquinone-4
Cat.No: T7106
Synonym: 四烯甲萘醌,Vitamin K2,Menaquinone K4
Target: Others, Endogenous Metabolite
Calcium 2-hydroxy-4-(methylthio)butanoate
Cat.No: T5082
Synonym: 羟基蛋氨酸钙,calcium hydroxymethionine,2-Hydroxy-4-(methylthio)butyric acid calcium salt
Target: Others, Endogenous Metabolite
2-Hydroxy-4-methoxybenzaldehyde
Cat.No: T2A2524
Synonym: 4-甲氧基水杨醛,4-Methoxysalicylaldehyde,2-羟基-4-甲氧基苯甲醛
Target: Tyrosinase, Antibacterial
4-(Ethoxymethyl)phenol
Cat.No: TN3029
Synonym: p-Hydroxybenzyl Et ether
Target: Antioxidant
4(3H)-Quinazolinone
Cat.No: TMO2713
Synonym: Quinazolin-4-ol,4-Hydroxyquinazoline,4-羟基喹唑啉,4-Quinazolinol,4-Quinazolone,4-Quinazolinone
Target: Antibacterial, Platelet aggregation
4-Hydroxy-6-methylcoumarin
Cat.No: Fr12277
Synonym:
Target: Others
4-methoxylonchocarpin
Cat.No: TN7235
Synonym:
Target: TNF, NF-κB
5-methoxyflavone
Cat.No: T3343
Synonym: 5-methoxy-2-phenylchromen-4-one,5-甲氧基黄酮
Target: DNA/RNA Synthesis
Moracin M
Cat.No: TN1950
Synonym:
Target: PDE
3',​4',​5',​5,​7-​Pentamethoxyflavone
Cat.No: T2A2486
Synonym: 5,7,3',4',5'-Pentamethoxyflavone
Target: Nrf2
Protocatechuic acid
Cat.No: T0562
Synonym: 3, 4-Dihydroxybenzoic acid,3,4-二羟基苯甲酸,Protocatechuate,原儿茶酸,3,4-Dihydroxybenzoic acid
Target: Others
4-Methoxybenzaldehyde
Cat.No: T7910
Synonym: 大茴香醛,Anisaldehyde,p-Anisaldehyde,Anisic aldehyde,4-Anisaldehyde,4-甲氧基苯甲醛,P-Methoxybenzaldehyde
Target: Others, Endogenous Metabolite
2',4'-Dimethylacetophenone
Cat.No: T67319
Synonym:
Target: Endogenous Metabolite
4-O-Cinnamoylquinic acid
Cat.No: TN6647
Synonym: 金银花
Target: Prostaglandin Receptor
(E)-3-(4-Methoxyphenyl)acrylic acid
Cat.No: T41095
Synonym: (E)-3-(4-甲氧基苯基)丙烯酸
Target: Glucosidase
Indican
Cat.No: T19866
Synonym: NSC-87517,3-Indoxyl-beta-D-glucopyranoside,3-吲哚基-beta-D-吡喃葡萄糖苷,NSC 87517,NSC87517,Indoxyl-β-D-glucoside
Target: OAT, MRP
ISOGINKGETIN
Cat.No: T4S21320
Synonym: 异银杏素,4',4'''-Dimethylamentoflavone,异银杏双黄酮
Target: MMP, Others
BENZYLACETONE
Cat.No: TCS1709
Synonym: 苄基丙酮,4-Phenylbutan-2-one,Methyl 2-phenylethyl ketone,4-Phenyl-2-butanone
Target: Tyrosinase
4-tert-Octylphenol
Cat.No: T64353
Synonym:
Target: Endogenous Metabolite
Anhydronotoptol
Cat.No: TN6985
Synonym: 4-{[(2E,5E)-3,7-dimethylocta-2,5,7-trien-1-yl]oxy}-7H-furo[3,2-g]chromen-7-one
Target: NO Synthase
Licoflavone C
Cat.No: TN1861
Synonym: 4',5,7-Trihydroxy-8-prenylflavone
Target: Antioxidant, Antifungal
Mogroside III-E
Cat.No: TN1936
Synonym: 罗汉果皂苷ⅢE
Target: IL Receptor, TNF, TLR
Deacetylasperulosidic Acid
Cat.No: T8280
Synonym: 去乙酰基车叶草苷酸,去乙酰车叶草苷酸,Desacetyl asperulosidic acid
Target: IL Receptor, Interleukin
1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one
Cat.No: TN5263
Synonym: Xanthohumol,黄腐酚
Target: Apoptosis, BCL, PARP, HCV Protease, IAP, Caspase, HIV Protease, NMDAR, p53
Licochalcone B
Cat.No: T4S0350
Synonym: 甘草查尔酮 B,甘草查尔酮B
Target: Beta Amyloid, Others
Ethyl trans-caffeate
Cat.No: T3S0013
Synonym: 咖啡酸乙酯,Ethyl caffeate,Caffeic Acid Ethyl Ester
Target: Others
gamma-Mangostin
Cat.No: T4S1637
Synonym: Normangostin,γ-倒捻子素
Target: Others, 5-HT Receptor
2,5-Dihydroxyacetophenone
Cat.No: TCS2170
Synonym: Quinacetophenone,2-Acetylhydroquinone,2-5-dihydroxyacetophenone,2 ',5'-二羟基苯乙酮,Acetylhydroquinone,2,5-二羟基苯乙酮,DHAP
Target: ERK, NF-κB, Tyrosinase
Tricosanoic acid
Cat.No: T4855
Synonym: Tricosan-1-oic acid,二十三烷酸
Target: Endogenous Metabolite
Tussilagone
Cat.No: T6S1027
Synonym:
Target: Others
Linalool
Cat.No: T2S2264
Synonym: Linalol,(±)-Linalool,Phantol,沉香醇
Target: Apoptosis, IL Receptor, TNF, Endogenous Metabolite, iGluR
Geraniin
Cat.No: T6S2099
Synonym:
Target: Antioxidant, TNF
5-Aminovaleric acid
Cat.No: T5089
Synonym:
Target: Others, Endogenous Metabolite
4-Nitrocinnamic acid
Cat.No: TN6605
Synonym:
Target:
trans-4-Hydroxy-2-nonenoic acid
Cat.No: T80958
Synonym:
Target:
4-Hydroxycyclohexanecarboxylic acid
Cat.No: T19135
Synonym:
Target: Others
3',4'-O,O-Methylene-(+)-catechin
Cat.No: T83370
Synonym:
Target:
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