85
67
11
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T6273 |
Vadimezan
DMXAA,伐地美生,5,6-Dimethylxanthenone-4-acetic Acid,NSC 640488,ASA-404 |
Influenza Virus; VDA; STING; IFNAR | Angiogenesis; Immunology/Inflammation; Microbiology/Virology |
Vadimezan (DMXAA) 是一种血管破坏剂,一种鼠 STING 激动剂,也是一种细胞因子如 I 型 IFN 的诱导剂。Vadimezan 具有抗肿瘤活性,可以诱导肿瘤中的血流快速停止,但不影响正常组织中的血流。 | |||
T0005 |
Aspirin
阿司匹林,Acetylsalicylate,Acetylsalicylic Acid,邻乙酰水杨酸,ASA |
Mitophagy; Virus Protease; COX; Autophagy | Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Aspirin (Acetylsalicylic Acid) 是一种选择性 COX 抑制剂,具有多种药理活性。它是组蛋白去乙酰化酶抑制剂,可上调细胞周期阻滞蛋白 p21,抑制携带 COX-1 的卵巢 Y 细胞。 它还抑制 HUVEC 和新生大鼠心室心肌细胞中 COX-2 的表达,分别减少 PG 的产生和 ERK 和 NF-KB 的下调。 | |||
T6254 |
Idasanutlin
RG7388,Ro 5503781,依达奴林 |
Mdm2; E1/E2/E3 Enzyme | Apoptosis; Ubiquitination |
Idasanutlin (Ro 5503781) 是一种有效且特异性的 p53-MDM2 抑制剂 ,IC50值为 6 nM。 | |||
T22303 |
Dasatinib hydrochloride
BMS-354825 HCl |
Bcr-Abl; Src; c-Kit | Angiogenesis; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors |
Dasatinib hydrochloride (BMS-354825 HCl) (BMS-354825) hydrochloride 是一种具有口服活性的,ATP 竞争性的,双重 Src/Bcr-Abl 抑制剂,具有有效的抗肿瘤活性。对 Src 和 Bcr-Abl 的 Ki 值分别为 16 pM 和 30 pM。Dasatinib hydrochloride hydrochloride 抑制 Bcr-Abl 和 Src 的IC50 分别为 <1.0 nM 和 0.5 nM。Dasatinib hydrochloride hydrochloride 还诱导凋亡 (apoptosis) 和自噬 (autophagy)。 | |||
T6962 |
Rasagiline Mesylate
TVP1012,甲磺酸雷沙吉兰,AGN1135,Azilect |
Apoptosis; MAO; Autophagy; Monoamine Oxidase | Apoptosis; Autophagy; Metabolism; Neuroscience |
Rasagiline Mesylate (AGN1135) 是一种高效的,不可逆的选择性线粒体单胺氧化酶 (MAO) 抑制剂,抑制大鼠脑 MAO B 和 MAO A 的IC50分别为 4.43 nM 和 412 nM。 | |||
T3608 |
Carbasalate calcium
Rheomin,Omegin,Alcacyl,Iromin,卡巴匹林钙,Solupsan,Carbasalate Calcium |
Platelet aggregation | Others |
Carbasalate calcium (Rheomin) 是抗炎和解热剂,可用于研究疼痛的缓解。 | |||
T12361 |
Parcetasal
MR-897 |
Others | Others |
Parcetasal (MR-897) 是一种非甾类体抗炎剂,在缓解疼痛方面具有研究价值。 | |||
T6090 |
Belnacasan
VX-765 |
Caspase | Apoptosis; Proteases/Proteasome |
Belnacasan (VX-765) 是一种具有口服活性的 IL 转换酶/caspase-1 抑制剂,是 VRT-043198 的口服生物活性前药,作用于外周血单核细胞,可抑制 LPS 诱导的 IL-1β 和 IL-18 释放。 | |||
T9407 |
Rasarfin
|
Others; Ras | GPCR/G Protein; MAPK; Others |
Rasarfin 是Ras 和ARF6双抑制剂。 | |||
T1448L |
Dasatinib monohydrate
达沙替尼,BMS-354825 Monohydrate |
Apoptosis; Bcr-Abl; Src; c-Kit; Ephrin Receptor; Autophagy | Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors |
Dasatinib monohydrate (BMS-354825 Monohydrate) 是一种具有口服活性的,ATP 竞争性的双重Src/Bcr-Abl 抑制剂,有抗肿瘤活性,还诱导凋亡和自噬。它抑制Src 和Bcr-Abl 的IC50分别为 0.5 nM 和 <1.0 nM,Ki 值分别为 16 pM 和 30 pM。 | |||
T3510 |
Olumacostat Glasaretil
|
Acetyl-CoA Carboxylase | Metabolism |
Olumacostat glasaretil 是乙酰辅酶A 羧化酶的有效抑制剂。 | |||
T18595 |
Dasatinib carbaldehyde
PROTAC ABL binding moiety 4,BMS-354825 carbaldehyde |
Others; Ligands for Target Protein for PROTAC | Others; PROTAC |
Dasatinib carbaldehyde (PROTAC ABL binding moiety 4) 基于 ABL 抑制剂达沙替尼,通过接头与 IAP 配体结合,形成 SNIPER [1]。 | |||
T2322 |
Fimasartan
非马沙坦,BR-A-657,Kanarb |
Apoptosis; RAAS | Apoptosis; Endocrinology/Hormones |
Fimasartan (BR-A-657) 是血管紧张素受体 AT1 非肽类拮抗剂,用于研究高血压和心力衰竭。 | |||
T0907 |
Sulfasalazine
柳氮磺吡啶,NSC 667219,Azulfidine |
Apoptosis; Ferroptosis; NF-κB; COX; Antibacterial; Antibiotic; Autophagy | Apoptosis; Autophagy; Immunology/Inflammation; Microbiology/Virology; Neuroscience; NF-κB |
Sulfasalazine (Azulfidine) 是一种合成的水杨酸衍生物,对含有弹性蛋白的结缔组织具有亲和力,并配制成前药。 | |||
T6826 |
Emricasan
PF 03491390,恩利卡生,IDN-6556 |
Influenza Virus; Caspase | Apoptosis; Microbiology/Virology; Proteases/Proteasome |
Emricasan (IDN-6556) 是一种泛的 caspase 抑制剂,具有不可逆性。Emricasan 具有抗炎和抗凋亡活性,可以用于治疗感染和肝衰竭等。Emricasan 还可以抑制 Zika 病毒感染。 | |||
T5386 |
Asapiprant
|
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
Asapiprant 是一种强选择性DP1受体拮抗剂,Ki 值为 0.44 nM,对DP1受体表现出高亲和力和选择性。 | |||
T18750 |
N-Deshydroxyethyl Dasatinib
N-Deshydroxyethyl BMS-354825 |
Others; IAP; Drug Metabolite | Apoptosis; Metabolism; Others |
N-Deshydroxyethyl Dasatinib (N-Deshydroxyethyl BMS-354825) 是 Dasatinib 的代谢物,是以达沙替尼为基础的分子,通过连接体与 IAP 配体结合,形成 SNIPER,从而降解 ABL。N-Deshydroxyethyl Dasatinib 可用于研究癌症和免疫疾病。 | |||
T27122 |
Dasantafil
SCH446132,SCH-446132,SCH 446132 |
PDE | Metabolism |
Dasantafil (SCH446132) 是一种小分子磷酸二酯酶-5A(PDE5A)抑制剂,可用于治疗泌尿生殖系统疾病和研究勃起功能障碍。 | |||
T1119 |
Rasagiline
雷沙吉兰,AGN1135,TVP1012 |
BCL; MAO; Monoamine Oxidase | Apoptosis; Metabolism; Neuroscience |
Rasagiline (AGN1135) 是不可逆的、高效的、选择性的线粒体单胺氧化酶 (MAO) 抑制剂,抑制大鼠脑 MAO B 和 MAO A 的 IC50分别为 4.43 nM 和 412 nM。 | |||
T37600 | Dasatinib N-oxide | Others | Others |
Dasatinib N-oxide 是 Dasatinib 的一种次要代谢物。Dasatinib 是口服有效的 Src/Bcr-Abl 抑制剂。 | |||
T6816 |
DASA-58
|
PKM | Metabolism |
DASA58 是一种有效的丙酮酸激酶M2 (PKM2) 活化剂,其中AC90=680 nM,AC50=38 nM。 | |||
T15198 |
Edasalonexent
CAT-1004 |
NF-κB | NF-κB |
Edasalonexent (CAT-1004) 是一种可口服的 NF-κB 抑制剂,可用于改善杜氏肌营养不良症。 | |||
T3489 |
Dasabuvir
ABT-333,达塞布韦 |
HCV Protease | Microbiology/Virology; Proteases/Proteasome |
Dasabuvir (ABT-333) 是丙型肝炎病毒非结构蛋白 5B 的非核苷抑制剂,是一种 RNA 依赖性 RNA 聚合酶,具有抗 HCV 的潜在活性。 | |||
T1448 |
Dasatinib
BMS-354825,达沙替尼 |
Apoptosis; Bcr-Abl; Src; c-Kit; Autophagy | Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Tyrosine Kinase/Adaptors |
Dasatinib (BMS-354825) 是一种酪氨酸激酶抑制剂,抑制 Src 和 Bcr-Abl (Ki=16/30 pM),具有口服活性和 ATP 竞争性。Dasatinib 具有抗肿瘤活性,用于治疗白血病和淋巴瘤等。 | |||
T31845 |
Forasartan
SC52458,SC 52458,SC-52458 |
||
Forasartan is a non - peptide angiotensin II receptor antagonist with antihypertensive activity. Forasartan and angiotensin II compete to bind AT1 receptor subtypes in vascular smooth muscle, thereby blocking angiotensin II-mediated vasoconstriction, lead | |||
T125742 | Herniariasaponin 3 | ||
Herniariasaponin 3 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125742,CAS号为 155179-16-1。 | |||
T125158 | Schidigerasaponin A3 | ||
Schidigerasaponin A3 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125158,CAS号为 266997-31-3。 | |||
T74424 | Masavibart | ||
Masavibart (ZRC3308-A7) 是一种靶向SARS-CoV-2的单克隆抗体 (IgG1 型)。Masavibart 对SARS-CoV-2穗状蛋白的RBD 上的非竞争性表位显示出良好的结合亲和力。Masavibart 可按 1:1 与ZRC3308-B10 联合使用,对 COVID-19 的预防以及尚未发展为严重疾病的早期 COVID-19 有效。 | |||
T126294 |
Kaikasaponin I
|
||
Kaikasaponin I 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126294,CAS号为 117210-04-5。 | |||
T126349 |
Cynarasaponin H
|
||
Cynarasaponin H 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126349,CAS号为 114006-82-5。 | |||
T124217 |
Soyasaponin A1
|
||
Soyasaponin A1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124217,CAS号为 78693-94-4。 | |||
T13252L |
(S)-Rasagiline mesylate
TVP1022 (mesylate),(S)-雷沙吉兰甲磺酸,S-PAI mesylate |
Others | Others |
(S)-Rasagiline mesylate is rasagiline S-isomer, and is an agent of anti-Parkinson. | |||
T124469 |
Primulasaponin 1
|
||
Primulasaponin 1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124469,CAS号为 65312-86-9。 | |||
T68390 |
Nivocasan
|
||
Nivocasan, also known as GS-9450 and LB-84451, a novel caspase-inhibitor has demonstrated hepatoprotective activity in fibrosis/apoptosis animal models. GS-9450 treatment induced significant reductions in ALT levels in NASH patients. | |||
T125712 |
Eclalbasaponin III
|
||
Eclalbasaponin III 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125712,CAS号为 158511-60-5。 | |||
T125629 |
Schidigerasaponin A1
|
||
Schidigerasaponin A1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125629,CAS号为 167221-10-5。 | |||
T80607 |
Eblasakimab
CSL-334,ASLAN004 |
||
Eblasakimab (ASLAN004; CSL-334)是一种人源化IgG4单克隆抗体,特异性针对IL13RA1,主要通过CHO-K1细胞生产表达。 | |||
T126030 |
Gypsophilasaponin G4
|
||
Gypsophilasaponin G4 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126030,CAS号为 133632-80-1。 | |||
T125155 |
Schidigerasaponin F1
|
||
Schidigerasaponin F1 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125155,CAS号为 266998-42-9。 | |||
T126123 |
Wistariasaponin B2
|
||
Wistariasaponin B2 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126123,CAS号为 126594-46-5。 | |||
T28039 |
Milfasartan
LR-B081,LRB-081,LR-B-081,LRB 081,LR-B 081 |
||
Milfasartan is a potent, selective antagonist of AT1 receptor with oral activity. It markedly lowers the blood-pressure in conscious renal and spontaneously hypertensive rats. | |||
T30151 |
Asafan
Asaphan |
||
Asafan is a bioactive chemical. | |||
T125711 |
Eclalbasaponin IV
|
||
Eclalbasaponin IV 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125711,CAS号为 158511-61-6。 | |||
T125718 |
Herniariasaponin 2
|
||
Herniariasaponin 2 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125718,CAS号为 157446-62-3。 | |||
T4358 |
Vosilasarm
Testolone,RAD140 |
Androgen Receptor | Endocrinology/Hormones |
Testolone 是一种有效的、非甾体的、具有口服活性的、选择性雄激素受体调节剂 (SARM),Ki 为 7 nM。它对雄激素受体的选择性比其他类固醇激素核受体高。 | |||
T126276 | Cynarasaponin E | ||
Cynarasaponin E 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126276,CAS号为 117804-11-2。 | |||
T29235 |
Zolasartan
GR-117289,GR 117289,GR 117289C,GR117289,GR-117289C |
||
Zolasartan is a potent, specific, selective and insurmountable antagonist at angiotensin AT, receptors. | |||
T13252 |
(S)-Rasagiline
TVP1022,(S)-雷沙吉兰,S-PAI |
Others | Others |
(S)-Rasagiline is rasagiline S-isomer, and is an agent of anti-Parkinson. | |||
T16570 |
Pralnacasan
VX-740,HMR 3480 |
Others | Others |
Pralnacasan inhibits proinflammatory cytokines IL-18, IL-1β , and IFN-γ. Pralnacasan is an effective, non-peptide, and orally active interleukin-1β converting enzyme inhibitor (Ki: 1.4 nM). Pralnacasan has the potential for osteoarthritis and rheumatoid a | |||
T72319 |
Lewis y tetrasaccharide
Lewis y |
||
Lewis Y tetrasaccharide (Lewis Y, LeY) 是Lewis X trisaccharide 的四糖衍生物。Lewis Y tetrasaccharide 是一种与恶性卵巢癌转移和预后不良相关的抗原。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T0646 |
5-Aminosalicylic Acid
Mesalazine,5-ASA,5-氨基水杨酸,Mesalamine |
NF-κB; Lipoxygenase; COX; Glutathione Peroxidase; Endogenous Metabolite; PAK; PPAR | Cytoskeletal Signaling; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB |
5-Aminosalicylic Acid (5-ASA) 是一种特异性的PPARγ激动剂,还抑制 p21-激活激酶1(PAK1) 和NF-κB,具有抗炎活性。 | |||
TN2232 |
Soyasaponin Ab
|
NOS; NF-κB; COX | Immunology/Inflammation; Neuroscience; NF-κB |
Soyasaponin Ab 是一种大豆皂苷。Soyasaponin Ab 在 3T3-L1 脂肪细胞中通过下调 PPARγ 产生抗肥胖的作用。 | |||
T15716 |
Lasalocid sodium
拉沙洛西钠,拉沙里菌素,Ionophore X-537A sodium,Antibiotic X-537A sodium,Lasalocid-A sodium |
Antibacterial; Antibiotic; Autophagy | Autophagy; Microbiology/Virology |
Lasalocid sodium (Lasalocid-A sodium) 是一种抗菌剂。 | |||
T3765 |
L-asarinin
細辛素,(-)-Episesamin |
Others | Others |
L-asarinin ((-)-Episesamin) 降低外周血 IL-12 浓度并抑制 CXCR3 和 TLR4 的表达,这意味着 Asarinin 可能在 TLR4 通路中发挥作用,并延长同种异体心脏的存活时间。 | |||
T3S0601 |
Buddlejasaponin IVb
醉鱼草皂苷IVb,Saikosaponin 1b |
Others | Others |
Buddlejasaponin IVb (Saikosaponin 1b) 是一种三萜皂苷,从Clinopodium chinense (Benth.) O. Kuntze 中分离得到,能够缩短凝血时间,具有止血作用。 | |||
T0771 |
Casanthranol
美鼠李皮蒽酚苷,鼠李蒽酚 |
Others | Others |
Casanthranol是从Rhamnus p.的干燥树皮(通常称为cascara sagrada)提取的高浓度的蒽酚苷混合物。Casanthranol 主要用于缓解便秘。Casanthranol通过其对肠壁的作用,促进肌肉收缩的增加,从而帮助肠道运动。 | |||
T2733 |
Sarsasapogenin
Parigenin,知母皂苷元,Sarsagenin |
Apoptosis; NF-κB; Endogenous Metabolite | Apoptosis; Metabolism; NF-κB |
Sarsasapogenin (Parigenin) 是一种甾体皂苷元,从中草药知母中分离到,具有抗糖尿病、抗氧化、抗癌、抗炎等作用。 | |||
T3345 |
Hederasaponin B
常春藤皂苷B,Eleutheroside M,刺五加叶中,Hederacoside B |
Others; Virus Protease | Microbiology/Virology; Others |
Hederasaponin B (Hederacoside B) 是从Hedera helix 中分离的,有广谱抗病毒活性。 | |||
T3S0687 |
Ecliptasaponin D
|
Others | Others |
Ecliptasaponin D 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 T3S0687,CAS号为 206756-04-9。 | |||
T11680 |
Isoasatone A
|
P450 | Metabolism |
Isoasatone A 是一种具有抗虫作用的天然产物,分离自Heterotropa takaoiM。它作用于细胞色素 P450 单加氧酶和谷胱甘肽转移酶,产生抗S. litura 作用。 | |||
TQ0036 |
Anemarrhenasaponin I
|
Others | Others |
Anemarrhenasaponin I 是一种对血小板聚集有显著的抑制作用的传统中药。 | |||
TN1600 |
Eclalbasaponin I
|
Others | Others |
Eclalbasaponin I 分离自鳢肠中,具有抗肿瘤作用,能够抑制肝癌细胞 smmc-7721 的增殖(IC50:111.1703 μg/ml)。 | |||
T5S1959 |
(-)-Asarinin
Fagarol,Sesamin,细辛脂素,Pseudocubebin,Eleutheroside B4,Episesamin,Asarinin |
Antibacterial | Microbiology/Virology |
(-)-Asarinin (Eleutheroside B4) 是一种主要从 Zanthoxylum armatum 根部提取到的木脂素。 | |||
TN6931 |
Anemarrhenasaponin Ia
知母皂苷IA,(2S,3R,4S,5S,6R)-2-{[(2R,3R,4S,5R,6R)-4,5-dihydroxy-2-{[(1R,3R,4R,7S,9S,12S,13S,16S,18R)-3-hydroxy-6-methoxy-7,9,13-trimethyl-6-(3-methylbutyl)-5-oxapentacyclo[10.8.0.02,?.0?,?.013,1?]icosan-16-yl]oxy}-6-(hydroxymethyl)oxan-3-yl]oxy}-6-(hydroxymethyl)oxan |
Others | Others |
Anemarrhenasaponin Ia ((2S,3R,4S,5S,6R)-2-{[(2R,3R,4S,5R,6R)-4,5-dihydroxy-2-{[(1R,3R,4R,7S,9S,12S,13S,16S,18R)-3-hydroxy-6-methoxy-7,9,13-trimethyl-6-(3-methylbutyl)-5-oxapentacyclo[10.8.0.02,?.0?,?.013,1?]icosan-16-yl]oxy}-6-(hydroxymethyl)oxan-3-yl]oxy}-6-(hydroxymethyl)oxan) 具有抗炎活性。Anemarrhenasaponin Ia 具有抗炎作用,从知母根茎中分离得到。 Anemarrhenasaponin Ia 抑制 N-甲酰-甲硫氨酰-亮氨酰-苯丙氨酸 (fMLP) 诱导的超氧化物的进一步产生。 | |||
T3S0335 |
Soyasaponin Bb
Soyasaponin I,大豆皂苷Bb |
NF-κB; Caspase | Apoptosis; NF-κB; Proteases/Proteasome |
Soyasaponin Bb (Soyasaponin I) 是一种分离自菜豆科中的大豆皂苷,可用作醛糖还原酶差异抑制剂。 | |||
T3826 |
Polygalasaponin F
异牡荆苷,瓜子金皂苷己 |
NF-κB; TLR; Akt; PI3K | Cytoskeletal Signaling; Immunology/Inflammation; NF-κB; PI3K/Akt/mTOR signaling |
Polygalasaponin F 是从瓜子金中提取的齐墩果烷型三萜皂苷,可通过调节TLR4-PI3K/AKT-NF-kB 信号通路减少神经炎症细胞因子的分泌,能降低炎性细胞因子肿瘤坏死因子 α 的释放。 | |||
T4S0675 |
Polygalasaponin V
瓜子金皂苷V,瓜子金皂苷 V |
Others | Others |
Polygalasaponin V 是一种三萜皂苷,分离自Polygala japonica 的地上部分。其中Polygala japonica 是民间的药用植物,在中国南方用作祛痰、抗菌、抗炎、抗抑郁药。 | |||
T75675 |
Nepasaikosaponin K
|
Antiviral | Immunology/Inflammation |
Nepasaikosaponin K 是一种从柴胡根中分离出来小分子化合物,具有抗流感和抗病毒活性,可用于研究病毒感染。 | |||
T15717 |
Lasalocid
Lasalocid-A,Antibiotic X-537A,Ionophore X-537A |
Antibacterial | Microbiology/Virology |
Lasalocid (Lasalocid-A) 是一种由链霉菌产生的离子载体抗生素,具有抗菌和寄生虫作用,常添加进饲料中。 | |||
T2826 |
Asaraldehyde
Asarylaldehyde,2,4,5-trimethoxy-Benzaldehyde,Asaronaldehyde,细辛醛 |
COX | Immunology/Inflammation; Neuroscience |
Asaraldehyde (2,4,5-trimethoxy-Benzaldehyde) 是COX-2抑制剂,能够明显降低环加氧酶 II (COX-2) 的活性(IC50:100 μg/mL)。 | |||
T2S0690 |
Ecliptasaponin A
早莲苷 A,旱莲苷A,Echinocystic acid-3-o-glucoside |
Others | Others |
Ecliptasaponin A (Echinocystic acid-3-o-glucoside) 是一种墨旱莲 (Eclipta prostrate) 中分离得到的五环三萜皂苷。其中墨旱莲是一种具有多效作用的滋补草药,如抗炎、保肝、抗氧化和免疫调节。 | |||
TN1432 |
Bacopasaponin C
(-)-假马齿苋皂苷 C,假马齿苋皂苷C |
Anti-infection; GABA Receptor; NMDAR | Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience |
Bacopasaponin C 是一种分离自Bacopa monniera 中的天然糖苷,具有抗肿瘤和抗利什曼原虫作用。 | |||
T3698 |
alpha-Asarone
α-Asarone,trans-Asarone,α-细辛脑 |
P450; GABA Receptor; HMG-CoA Reductase | Membrane transporter/Ion channel; Metabolism; Neuroscience |
alpha-Asarone (trans-Asarone) 是来自胡萝卜的一种天然产物,具有抗抑郁等功效。 | |||
TN2230 |
Soyasaponin Ba
大豆皂苷 BA,大豆皂苷Ba |
Others | Others |
Soyasaponin Ba 是一种大豆皂苷,分离自菜豆类,可用作醛糖还原酶抑制剂。 | |||
TN2043 |
Pasakbumin B
13-alpha-(21)-Epoxyeurycomanone,13ALPHA(21)-环氧宽缨酮 |
Others | Others |
Pasakbumin B (13-alpha-(21)-Epoxyeurycomanone) 是一种从 Eurycoma longifoliaJack 中获得的具有生物活性的化合物,显示出抗溃疡作用。 | |||
T10383 |
Asatone
|
NF-κB | NF-κB |
Asatone 是一种从细辛中分离到的活性成分,通过活化 NF-κB 及下调 p-MAPK (ERK,JNK 和 p38) 通路起作用,具有抗炎作用。 | |||
T4S1962 |
beta-Asarone
β-细辛脑,(Z)-1,2,4-三甲氧基-5-丙烯基苯;顺式细辛脑,Cis-Isoasarone,Cis-Asarone,Cis-Isoelemicin |
NF-κB; JNK | MAPK; NF-κB |
beta-Asarone (Cis-Isoelemicin) 是一种石菖蒲中的主要成分,具有免疫抑制、促进安定、中枢神经系统抑制、降温等功能。它可透过血脑屏障,能够预防帕金森病。 | |||
TN2225 |
Soyasapogenol B
大豆甾醇 B,大豆甾醇B |
Apoptosis; Autophagy | Apoptosis; Autophagy |
Soyasapogenol B 是大豆的一种成分,具有降胆固醇、抗补体和保肝作用。它抑制培养的 Hep-G2 的增殖,可触发内质网应激反应,其介导结肠直肠癌中的细胞凋亡和自噬。 | |||
TN2224 |
Soyasapogenol A
大豆甾醇A,大豆甾醇 A |
TNF | Apoptosis |
Soyasapogenol A shows estrogenic and hepatoprotective activities, it directly prevents apoptosis of hepatocytes, and secondly, inhibits the elevation of plasma TNF-α±, which consequently resulted in the prevention of liver damage in the concanavalin A-induced hepatitis model. | |||
TN6531 |
Polygalasaponin E
|
||
Polygalasaponin E 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6531,CAS号为 882664-72-4。 | |||
TN1382 |
Anemarrhenasaponin III
|
Others | Others |
Anemarrhenasaponin III is a natural product | |||
T82539 |
DL-Asarinin
|
||
DL-Asarinin(化合物88)是Cinnamomum camphora中的一种天然产物。 | |||
TN2227 |
Soyasapogenol D
大豆皂甙元 D,大豆甾醇D |
Others | Others |
Soyasapogenol D is a natural product | |||
TN5040 | Soyasaponin IV | Others | Others |
Soyasaponin IV has hepatoprotective activity.It also has antimutagenic activity in mammalian cells. | |||
T39042 |
Tarasaponin IV
|
||
Tarasaponin IV, an oleanane-type triterpene saponin, is derived from the bark of Aralia elata and holds potential for cancer research. | |||
TN1636 |
Eupteleasaponin I
|
Others | Others |
Eupteleasaponin I is a natural product from Euptelea polyandra Sieb. et Zucc. | |||
T82855 |
Blood group A pentasaccharide
A-Pentasaccharide |
||
A-Pentasaccharide 是一种尿液中的寡糖,具有抑制抗 A 抗体与 A 型血物质结合的功能。 | |||
TN6805 |
Dehydrosoyasaponin I
|
||
Dehydrosoyasaponin I is a natural product. | |||
T11555 |
Heptasaccharide Glc4Xyl3
|
Others | Others |
Heptasaccharide Glc4Xyl3 is a covalent inhibitor of endo-xyloglucanases. It used for the identification and analysis of diverse xyloglucan-active enzymes in nature. | |||
TN6273 |
Soyasapogenol A 21-O-α-L-rhamnopyranoside
|
||
Soyasapogenol A 21-O-α-L-rhamnopyranoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN6273,CAS号为 2067321-88-2。 | |||
TN2231 |
Soyasaponin II
|
Influenza Virus; HIV Protease; HSV | Microbiology/Virology; Proteases/Proteasome |
Soyasaponin II has antiviral effects, it can inhibit the replication of human cytomegalovirus, influenza virus, and human immunodeficiency virus type 1. | |||
T81429 |
Polygalasaponin LII
|
||
Polygalasaponin LII,一种三萜皂苷,由Polygala japonica Houtt的根中提取。 | |||
TN2229 |
Soyasaponin Ac
|
Others | Others |
Soyasaponin Ac can decrease the drug resistance via EMT pathway and weaken the migration ability of ovarian cancer cells. | |||
T82747 |
Centellasaponin A
|
||
Centellasaponin A (compound 10)为五环三萜皂苷类化合物,可通过积雪草甲醇提取物进行分离提取。 | |||
T83463 |
11(α)-Hydroxynepasaikosaponin k
|
||
11(α)-Hydroxynepasaikosaponin k(HOSSc)是B. scorzonerifolium Willd中的一种柴胡皂苷。 | |||
T80995 |
Theasaponin E2
|
||
Theasaponin E2, 一种从茶树分离得到的化合物,对K562和HL60细胞表现出显著的细胞毒性,其半抑制浓度(IC50)为14.7 μg/mL。 | |||
T38552 |
Dehydrosoyasaponin I methyl ester
大豆皂苷BE甲酯,Soyasaponin Be methyl ester,DHS-Imethylester |
||
Dehydrosoyasaponin I methyl ester, also known as Soyasaponin Be methyl ester, is a saponin compound that is naturally occurring in Trifolium alexandrinum. | |||
T80996 |
Theasaponin E1
|
||
Theasaponin E1,一种可从茶籽分离的茶皂苷,对人肿瘤细胞系K562和HL60展示了抗肿瘤潜能。此外,Theasaponin E1具备醌还原酶(QR)诱导活性,有助于作为抗癌预防药物的研究。 | |||
T24242 |
Kaikasaponin III
|
||
Kaikasaponin III is isolated from Abrus Cantoniensis. It also has an antihepatotoxic activity. | |||
T13082 |
Tarasaponin VI
|
Others | Others |
Tarasaponin VI 是从 Aralia elata 中分离出来的,对乙醇吸收具有有效的抑制活性。 | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPH-02398 |
ASA dehydrogenase Protein, Legionella pneumophila, Recombinant (His)
Aspartate-beta-semialdehyde dehydrogenase,asd,Aspartate-semi... |
Legionella pneumophila | E. coli |
Catalyzes the NADPH-dependent formation of L-aspartate-semialdehyde (L-ASA) by the reductive dephosphorylation of L-aspartyl-4-phosphate. | |||
TMPY-00670 |
ARSA Protein, Mouse, Recombinant (His)
arylsulfatase A,TISP73,AW212749,As-2,AS-A,ASA,As2 |
Mouse | HEK293 Cells |
ARSA Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 53.5 kDa and the accession number is P50428. | |||
TMPY-00964 |
ASAM Protein, Human, Recombinant (His)
ACAM,CXADR-like membrane protein,CSBM,ASAM,CSBS |
Human | HEK293 Cells |
ASAM Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.8 kDa and the accession number is Q9H6B4. | |||
TMPH-02490 |
ASAH1 Protein, Mouse, Recombinant (GST & His & Myc)
Acid CDase,HSD-33,Acid ceramidase,N-acylsphingosine amidohyd... |
Mouse | E. coli |
ASAH1 Protein, Mouse, Recombinant (GST & His & Myc) is expressed in E. coli expression system with N-10XHis-GST and C-Myc tag. The predicted molecular weight is 43.8 kDa and the accession number is Q9WV54. | |||
TMPH-01985 |
ASAH2B Protein, Human, Recombinant (His)
ASAH2L,ASAH2B,Putative inactive non-lysoso... |
Human | E. coli |
N/A. ASAH2B Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 23.0 kDa and the accession number is P0C7U1. | |||
TMPH-00880 |
ASAH1 Protein, Human, Recombinant (His & SUMO)
AC,Acid CDase,HSD33,Acylsphingosine deacylase,N-acylsphingos... |
Human | E. coli |
ASAH1 Protein, Human, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 58.7 kDa and the accession number is Q13510. | |||
TMPY-02998 |
ASAM Protein, Rat, Recombinant (His)
ACAM,CXADR-like membrane protein,Asam,Ol16 |
Rat | HEK293 Cells |
ASAM Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.6 kDa and the accession number is Q8K1G0. | |||
TMPH-01771 |
ASAH2 Protein, Human, Recombinant (His)
HNAC1,LCDase (hCD),BCDase,Non-lysosomal ceramidase,Neutral c... |
Human | E. coli |
ASAH2 Protein, Human, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 25.2 kDa and the accession number is Q9NR71. | |||
TMPY-00963 |
ASAH2 Protein, Mouse, Recombinant (His)
N-acylsphingosine amidohydrolase (non-lysosomal ceramidase) ... |
Mouse | HEK293 Cells |
ASAH2 (N-acylsphingosine amidohydrolase 2), also known as neutral ceramidase, is a type II integral membrane protein that can be cleaved to produce a soluble secreted protein. The enzyme is abundant in the brush border membranes of the intestine, and also expressed in several tissues such as kidney, brain and liver. The primary structure of ASAH2/neutral ceramidase is highly conserved from bacteria to humans, however, there is a clear difference in the molecular architecture. The murine ASAH2 po... | |||
TMPH-03176 |
LasA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO)
|
Pseudomonas aeruginosa | E. coli |
LasA Protein, Pseudomonas aeruginosa, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 36.0 kDa and the accession number is P14789. | |||
TMPY-01698 |
ASAM Protein, Mouse, Recombinant (His)
ACAM,AW557819,CXADR-like membrane protein,9030425E11Rik,ASP5 |
Mouse | HEK293 Cells |
ASAM Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 25.6 kDa and the accession number is Q8R373-1. |