10000+
1000+
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T36848 |
Combretastatin A-1
Combretastatin A1 |
Akt; Microtubule Associated | Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Combretastatin A-1 是一种有效的微管抑制剂,具有抗肿瘤和抗血管活性,通过微管蛋白解聚介导的 AKT 失活抑制 Wnt/β-catenin 通路发挥作用,可用于研究肝癌。 | |||
T12404 |
CCK-A receptor inhibitor 1
|
cholecystokinin | GPCR/G Protein |
CCK-A receptor inhibitor 1 是一种有效的缩胆囊素 A (CCK-A) 受体抑制剂(IC50:340 nM)。CCK-A receptor inhibitor 1 可用于研究与消化系统相关的疾病。 | |||
TP1179L |
Porcine dynorphin A(1-13) acetate
Dynorphin A Porcine Fragment 1-13 acetate,Porcine dynorphin A(1-13) acetate(72957-38-1 free base) |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Porcine dynorphin A(1-13) acetate (Dynorphin A Porcine Fragment 1-13 acetate)(72957-38-1 free base) 是一种有效的内源性 κ opioid 受体激动剂,在生理浓度下具有镇痛作用。暴露于强啡肽 A (1-13) 会导致单个神经元中 [Ca2+]i 的急剧增加,类似于急性 NMDA 治疗所见的增加。 | |||
T21708L |
Angiotensin 1/2 + A (2 - 8) Acetate
Angiotensin 1/2 + A (2 - 8) Acetate (51833-76-2 Free base) |
Others | Others |
Angiotensin 1/2 + A (2 - 8) Acetate 是一种血管收缩剂。 | |||
T76341L |
[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine(94596-26-6 Free base) |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
[DPro10] Dynorphin A (1-11)acetate,porcine 是一种高效的 κ-阿片受体激动剂,其 Ki 值为 0.13 nM。[DPro10] Dynorphin A (1-11), porcine 是一种 N-烷基化衍生物,具有镇痛活性。 | |||
TP1813L |
Dynorphin A 1-10 acetate(79994-24-4 free base)
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Dynorphin A 1-10 acetate(79994-24-4 free base) 是一种内源性 opioid 样物质神经肽,与 κ-opioid 样物质受体的细胞外环 2 结合。 Dynorphin A (1-10) 还阻断 NMDA 激活的电流,IC50 为 42.0 μM。 | |||
T21781 |
A-286982
|
Integrin | Cytoskeletal Signaling |
A 286982是高效的LFA-1/ICAM-1相互作用变构抑制剂,在LFA-1/ICAM-1结合和LFA-1介导的细胞粘附实验中,其IC50分别为44和35 nM。 | |||
T10927 |
Cyt-PTPε Inhibitor-1
Cyt-PTP|A Inhibitor-1 |
Phosphatase; Src | Angiogenesis; Metabolism; Tyrosine Kinase/Adaptors |
Cyt-PTPε Inhibitor-1 (A Inhibitor-1) 是胞质蛋白酪氨酸磷酸酶 ε 的抑制剂。 Cyt-PTPε Inhibitor-1 阻断 c-Src 的去磷酸化并表现出抗破骨活性。 | |||
T11373 |
GCN2-IN-1
A-92 |
Others | Others |
GCN2-IN-1 (A-92) 是一种有效的一般性调控阻遏蛋白激酶 2 抑制剂,可作为化疗药物用于癌症治疗的研究。 | |||
T36432 |
A2ti-1
|
Virus Protease | Microbiology/Virology |
A2ti-1 是一种具有高选择性的附件蛋白 A2/S100A10 杂四聚体(A2t)抑制剂(IC50 : 24 μM), 抑制ARV介导的Src和p38丝裂原活化蛋白激酶(MAPK)的激活。A2ti-1 可用于研究人类乳头瘤病毒 16 型(HPV16)感染。 | |||
T2254 |
A-205804
|
Integrin | Cytoskeletal Signaling |
A-205804 是一种选择性口服有效的先导抑制剂,抑制 E-selectin 和 ICAM-1表达,IC50分别为 20 nM 和 25 nM,可用于慢性炎症疾病的研究。 | |||
T30222 |
Avenacin A 1
|
||
Avenacin A 1 is a biochemical. | |||
T13303 |
Virginiamycin M1
Pristinamycin IIA,Ostreogrycin A |
Antibacterial | Microbiology/Virology |
Virginiamycin M1 (Pristinamycin IIA)是一种大环内酯肽类抗生素,是链菌素a 类抗生素的成员。 | |||
T38817 |
Golgicide A-1
GCA-1,Golgicide A-1 |
||
Golgicide A-1 (GCA-1) is a moderately potent cis-diastereomer variant of Golgicide A (GCA) specifically designed to inhibit mosquito reproduction. | |||
T16904 |
Smurf1-IN-A01
A01 |
Others | Others |
Smurf1-IN-A01 (A01) 是泛素连接酶 Smad 泛素化调节因子-1(Smurf1)抑制剂,其kd=3.664 nM。它能够抑制 Smurf1 介导的 Smad1/5 降解,并提高 BMP-2 的反应性。 | |||
T29787 | Ajugamarin A 1 | ||
Ajugamarin A 1 is a Neoclerodane diterpenoid. | |||
T11007L |
Levofloxacin Hydrochloride Impurity A
Levofloxacin Hydrochloride Impurity A(117707-40-1 Free base),左氧氟沙星杂质A(盐酸盐) |
Antibacterial | Microbiology/Virology |
Levofloxacin Hydrochloride Impurity A 是一种喹诺酮类药物,具有广谱抗菌作用。 | |||
TP1813 |
Dynorphin A (1-10)
Dynorphin A 1-10 |
||
Dynorphin A (1-10), an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A (1-10) also blocks NMDA-activated current with an IC50 of 42.0 μM. | |||
T10208 |
A-69412
N-1-(Fur-3-ylethyl)-N-hydroxyurea |
Lipoxygenase | Metabolism |
A-69412 (N-1-(Fur-3-ylethyl)-N-hydroxyurea) 是一种特异性的 5-脂氧合酶 (5-LO) 的可逆抑制剂。 A-69412 能用于哮喘和溃疡性结肠炎,以及其他炎症和过敏症状的研究。 | |||
T67742 |
EX-A5386
Glucocorticoid receptor modulator-1 |
Glucocorticoid Receptor | Endocrinology/Hormones |
EX-A5386 (Glucocorticoid receptor modulator-1)是一种有效的糖皮质激素受体调节剂,IC50/EC50<100nM。 | |||
T7774 |
A2793
2-[(5-氯-8-喹啉基)氧基]乙酸乙酯 |
Potassium Channel | Membrane transporter/Ion channel |
A2793 是 TWIK 相关酸敏感 K+通道 1(TASK-1)/TRESK 的双重抑制剂,对 mTRESK 的 IC50为 6.8 μM。它对 TRESK 选择性更好, 对 TREK-1 和 TALK-1 相对弱一些。 | |||
T7205 |
A-967079
(1E,3E)-1-(4-氟苯基)-2-甲基-1-戊烯-3-酮肟 |
TRP/TRPV Channel | Membrane transporter/Ion channel |
A 967079是一种有效的TRPA1受体选择性拮抗剂,对人和大鼠 TRPA1 受体的IC50分别为 67 nM 和 289 nM。A 967079具有良好的CNS 穿透性。 | |||
T60021 |
ecMetAP-IN-1
|
Others | Others |
ecMetAP-IN-1 可用作 QSAR 模型,以使用多元线性回归研究蛋氨酸氨基肽酶抑制剂作为抗癌剂。 | |||
T8562 |
A 425619
1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA |
TRP/TRPV Channel | Membrane transporter/Ion channel |
A 425619 (1-(4-(TRIFLUOROMETHYL)BENZYL)-3-(ISOQUINOLIN-5-YL)UREA) 是一种有效的 TRPV1 拮抗剂。 | |||
T30797 |
Ceramide 1 A
Linoleoyloxyheptacosanoyl-C18-phytosphingosine |
||
Ceramide 1 A 是一种蜡状脂质化合物,是顶端皮肤层的脂质。它具有特殊的分子结构,因为它含有一种与长链ω-羟基酸相连的亚油酸。 | |||
T16886 |
Sinefungin
Adenosyl-Ornithine,西奈芬净,A-9145,Antibiotic 32232RP |
Others; Histone Methyltransferase; Antibiotic; Antifungal | Chromatin/Epigenetic; Microbiology/Virology; Others |
Sinefungin (Adenosyl-Ornithine) 是病毒粒子mRNA (鸟嘌呤-7-)-甲基转移酶、 mRNA (核苷-2'-)-甲基转移酶和病毒增殖的有效抑制剂。它还抑制SET7/9,通过抑制H3K4甲基化来改善肾纤维化。 | |||
TP1845 |
Cyclosporin A-Derivative 1
|
||
Cyclosporin A-Derivative 1 is a crystalline intermediate derived from the opening of cyclosporin A. | |||
T21358 |
Dalbavancin
BI 397,BI-397,VER 001,A-A 1,BI397,VER-001,Dalbavancin HCl,达巴万星 |
Antibacterial; Antibiotic | Microbiology/Virology |
Dalbavancin (BI-397) HCl 是一种半合成的脂糖肽抗生素,对革兰氏阳性细菌有杀菌活性。Dalbavancin 抑制金黄色葡萄球菌和炭疽芽孢杆菌的 MIC90分别为 0.06 μg/mL 和 0.25 μg/mL。 | |||
T9842 |
5-HT2B antagonist-1
|
||
5-HT2B antagonist-1 是一种具有口服活性的5-HT2B 受体拮抗剂,IC50值为 33.4 nM。5-HT2B antagonist-1可用于以 5-HT2B 受体信号传导为特征的疾病研究,如肝细胞癌、心血管疾病或胃肠道疾病。 | |||
TP1179 |
Porcine dynorphin A(1-13)
Dynorphin A Porcine Fragment 1-13 |
||
Porcine dynorphin A (1-13) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiological concentrations. Exposure to dynorphin A (1-13) causes acute increases in [Ca2+]i in individual neurons similar to increases seen with acut | |||
T20403 |
Dynorphin A (1-8)
PH-8P,Dynorphin (1-8) |
||
Dynorphin (1-8) is an opioid octapeptide from the porcine hypothalamus. It comprises the N-terminal eight residues of dynorphin. | |||
T10058 |
A2B receptor antagonist 1
|
Adenosine Receptor | GPCR/G Protein; Neuroscience |
A2B receptor antagonist 1 是一个有效的 A2B 腺苷受体 (A2B adenosine receptor) 拮抗剂。 | |||
T29419 |
3'-Rhamnopiericidin A(1)
SN-198-C |
||
3'-Rhamnopiericidin A(1) is a piericidin rhamnoside from Streptomyces. | |||
T39778 |
Influenza A virus-IN-1
|
||
Influenza A virus-IN-1, a dihydropyrrolidones derivative, is a highly effective inhibitor of various subtypes of influenza A virus (IAV) with IC 50 values ranging from 3.11 μM to 7.13 μM. It effectively suppresses IAV replication and enhances the expression of key antiviral cytokines, such as IFN-β, and the antiviral protein MxA. | |||
T4288 |
hVEGF-IN-1
|
VEGFR | Angiogenesis; Tyrosine Kinase/Adaptors |
hVEGF-IN-1 是一种喹唑啉衍生物,可以特异性结合内部核糖体进入位点 A 中富含 G 的序列,并会使 G-四链体结构不稳定。在 SPR 实验中,它与 IRES-A (WT) 结合的Kd 值为 0.928 μM。它能够抑制VEGF-A 蛋白表达,阻止肿瘤细胞迁移,抑制肿瘤生长。 | |||
T40367 |
Combretastatin A-1 phosphate tetrasodium
Combretastatin A-1 phosphate tetrasodium,OXi-4503 tetrasodium |
||
Combretastatin A-1 phosphate (OXi-4503) tetrasodium, a prodrug of Combretastatin A-1, is a tubulin-binding microtubule polymerization inhibitor that targets the colchicine-binding site. By inducing tubulin depolymerization, Combretastatin A-1 phosphate tetrasodium inhibits the Wnt/β-catenin pathway and leads to the deactivation of AKT. It possesses both anti-tumor and anti-vascular properties. | |||
T7512 |
BMS-191011
BMS-A |
Potassium Channel | Membrane transporter/Ion channel |
BMS-191011 (BMS-A) 是一种大电导 Ca2+激活的钾通道 (Ca2+-activated potassium (maxi-K) channel) 激活剂,在中风模型中有研究价值。 | |||
TP1405 |
Cyclosporin A-Derivative 1 Free base
|
||
Cyclosporin A-Derivative 1 (Free base) is a crystalline intermediate derived from the opening of cyclosporin A. | |||
T0564 |
1-Indanone
1-茚酮,Alpha-Indanone,Indan-1-one |
Others | Others |
1-Indanone (Indan-1-one) 是Indinavir 的中间体。 | |||
T6365 |
A 922500
A922500,(1R,2R)-2-[[4-[[(苯基氨基)羰基]氨基][1,1-联苯]-4-基]甲酰基]环戊烷羧酸,DGAT-1 Inhibitor 4a |
Acyltransferase; Transferase | Metabolism |
A 922500 (DGAT-1 Inhibitor 4a) 是一种口服有效的二酰甘油酰基转移酶 1(DGAT-1)选择性抑制剂,抑制小鼠和人 DGAT-1 的IC50s 分别为9 nM,22 nM。 | |||
T7649 |
Tyrphostin A1
AG9,(4-甲氧基苄烯)丙二腈,Tyrphostin 1 |
EGFR; Interleukin | Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Tyrphostin A1 (Tyrphostin 1) 对巨噬细胞培养中CD40L 刺激的IL-12产生和抗原诱导的Th1细胞生成具有抑制作用。 | |||
T81825 |
Melan-A/MART-1 analog
[Leu27]-Melan-A, MART-1 (26-35) |
||
[Leu27]-Melan-A, MART-1 (26-35)是一种具有改良的HLA-A*0201结合能力和增强的免疫原性及抗原性的生物活性肽。该类似物在第27位的Leu替换了Ala,与原生Melan-A (26-35)相比表现出更佳的性能。当序列N端为谷氨酰胺(Q)或谷氨酸(E)时,肽可能会自发形成焦谷氨酰(pGlu)。Q或E到pGlu的转化是自然发生的,pGlu的疏水性γ-内酰胺环被认为可增强针对胃肠道蛋白酶的抵抗力,使得含pGlu的肽成为这类肽的正常子集,在HPLC分析中通常作为评估肽纯度的一部分。 | |||
T0550 |
Domperidone EP Impurity A
5-氯-1,3-二氢-1-(4-哌啶基)-2H-苯并咪唑-2-酮 |
Others | Others |
Domperidone EP Impurity A 用作医药中间体。 | |||
TP1423 |
Dynorphin A (1-10) TFA(79994-24-4,free)
Dynorphin A (1-10) TFA |
||
Dynorphin A (1-10) (TFA), an endogenous opioid neuropeptide, binds in the transmembrane domain of the κ-receptor. | |||
T60098 |
MSC2504877
3-(4-(2-Hydroxypropan-2-yl)phenyl)-6-methylpyrrolo[1,2-a]pyrazin-1(2H)-one |
Others | Others |
MSC2504877 是一种tankyrase 抑制剂,可增强临床CDK4/6 抑制剂的作用。 MSC2504877 抑制由 palbociclib 引起的 Cyclin D2 和 Cyclin E2 的上调,并增强对 phospho-Rb 的抑制。 | |||
T77805 |
KRAS G12C mutant protein inhibitor A-1
|
||
KRAS G12C mutant protein inhibitor A-1 可用于 Ras 相关研究。 | |||
T12247 |
NOT Receptor Modulator 1
2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol |
Others | Others |
NOT Receptor Modulator 1 (2-(3-(2-(4-chlorophenyl)imidazo[1,2-a]pyridin-6-yl)phenyl)propan-2-ol) 是核受体 NOT 调节剂。 | |||
T12282 |
Benzyl-α-GalNAc
O-glycosylation-IN-1 |
Others | Others |
Benzyl-α-GalNAc (O-glycosylation-IN-1) 是 O-糖基化的有效抑制剂,用于减少细胞表面粘蛋白的含量。它抑制人胰腺癌细胞模型黏蛋白 O-糖基化的合成。 | |||
T8436 |
Minodronic acid
Phosphonicacid,(1-hydroxy-2-imidazo(1,2-a)pyridin-3-ylethylidene)bis-,ONO-5920,YM-529 |
Apoptosis; P2X Receptor | Apoptosis; Membrane transporter/Ion channel; Neuroscience |
Minodronic acid(YM-529) 是一种 P2X2/3 受体拮抗剂, 具有抗癌活性,可直接或间接的抑制癌细胞增殖,诱导细胞凋亡。Minodronic-acid 对各种类型的癌细胞的转移具有抑制作用。Minodronic-acid 可用于研究骨质疏松。 | |||
T9264 |
ECBN HCL
1-[(4R,5R)-4,5-Dihydroxy-L-ornithine]echinocandin B hydrochloride (1:1) |
Others | Others |
ECBN HCL (A-30912A nucleus hydrochloride) 是一种 Echinocandin B 脱酰酶催化反应的产物。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN1517 |
1-(2,6-dimethoxyphenyl)-3-(4-hydroxyphenyl)propan-1-one
剑叶龙血素A,Cochinchinenin A |
Others | Others |
1-(2,6-dimethoxyphenyl)-3-(4-hydroxyphenyl)propan-1-one (Cochinchinenin A) 是龙血镇痛作用的物质基础。 | |||
TN2525 | 1-Acetyltagitinin A | Others | Others |
1-Acetyltagitinin A是一种天然产物,属于菊科肿柄菊属,其产品编号为 TN2525,CAS号为 60547-63-9。1-Acetyltagitinin A可用作对照参考。 | |||
T5715 |
(E)-Flavokawain A
(E)-1-(2-羟基-4,6-二甲氧基苯基)-3-(4-甲氧基苯基)-2-丙烯-1-酮,FLAVOKAVAIN A(P),卡瓦胡椒素A |
Apoptosis; P450 | Apoptosis; Metabolism |
(E)-Flavokawain A 是一种来自卡瓦提取物的新型查尔酮,通过参与 Bax 蛋白依赖性和线粒体依赖性凋亡途径诱导膀胱癌细胞凋亡,并抑制小鼠肿瘤生长,具有抗癌作用。 | |||
TN1136 |
Procyanidin A1
原花青素 A1,Proanthocyanidin A1,原花色素A1 |
LDL; Calcium Channel; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Membrane transporter/Ion channel; Metabolism |
Procyanidin A1 (Proanthocyanidin A1) 是一种原花青素二聚体,具有抗过敏作用,可抑制蛋白激酶 C 激活下游脱粒或 RBL-213 细胞内部储存的 Ca2+流入。 | |||
T2S2295 |
Timosaponin A1
知母皂苷A1 |
Others | Others |
Timosaponin A1 是一种黄酮类甾体皂苷,分离自知母中。 | |||
TN7157 |
(+/-)-Longamide
Pyrrolo[1,2-a]pyrazin-1(2H)-one, 6,7-dibromo-3,4-dihydro-4-hydroxy-,6,7-dibromo-4-hydroxy-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-1-one,6,7-dibromo-4-hydroxy-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-one |
Others | Others |
(+/-)-Longamide (6,7-dibromo-4-hydroxy-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-one) 是一种海洋来源的天然产物,存在于Agelas flabelliformis。 | |||
TN2332 |
Ciwujianoside A1
刺五加皂苷A1,刺五加皂苷 A1 |
Others | Others |
Ciwujianoside A1 是分离自刺五加的叶子中。 | |||
T4924 |
α-D-Glucose-1-phosphate disodium
A-D-葡萄糖-1-磷酸-二钠盐,α-D-Glucose 1-phosphate disodium salt hy,α-D-Glucopyranose 1-phosphate |
Others; Endogenous Metabolite | Metabolism; Others |
α-D-Glucose 1-phosphate disodium salt hydrate 是合成葡萄糖醛酸的起始原料。它可用作心脏病研究所必需的细胞抑制剂、抗生素、免疫抑制剂和循环系统研究材料。 | |||
TN4991 |
Senkyunolide A
(3S)-3-丁基-4,5-二氢-1(3H)-异苯并呋喃酮,洋川芎内酯 A,洋川芎内酯 |
Others | Others |
Senkyunolide 是分离自 Ligusticum chuanxiongHort 中,具有细胞保护和抗增殖活性、抗肿瘤作用。 | |||
TN7148 |
Mukanadin C
7-bromo-4-hydroxy-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-1-one |
Others | Others |
Mukanadin C (7-bromo-4-hydroxy-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-1-one) 是一种海洋来源的天然产物,存在于 Stylissa carteri。 | |||
T7090 |
Jionoside A1
焦地黄苯乙醇甙A1,焦地黄苯乙醇苷A1 |
Others | Others |
Jionoside A1 分离自Radix Rehmanniae Praeparata 中,具有剂量依赖性免疫增强作用,并对 H2O2处理的 SH-SY5Y 细胞具有中等保护活性。 | |||
T6740 |
Bafilomycin A1
巴佛洛霉素A1,巴佛洛霉素 A1 |
Apoptosis; Proton pump; Antibacterial; Antibiotic; Autophagy | Apoptosis; Autophagy; Membrane transporter/Ion channel; Microbiology/Virology |
Bafilomycin A1 属于大环内酯类抗生素,是一种 V-ATPase (IC50=0.44 nM),具有特异性和可逆性。Bafilomycin A1 是自噬晚期阶段抑制剂,阻断自噬体与溶酶体的融合。Bafilomycin A1 也诱导凋亡。 | |||
T3920 |
Pseudoginsenoside F11
Ginsenoside A1,拟人参皂苷 F11,拟人参皂苷F11 |
Others; Endogenous Metabolite | Metabolism; Others |
Pseudoginsenoside F11 (Ginsenoside A1) 从人参根和叶中分离得到。PF11在一系列心血管和中枢神经系统疾病中具有广泛的保护作用。 | |||
T2777 |
Ginsenoside Rg1
Sanchinoside C1,Panaxoside Rg1,Sanchinoside Rg1,人参皂苷Rg1,Panaxoside A,人参皂苷 Rg1,Ginsenoside A2 |
Apoptosis; Beta Amyloid; NF-κB | Apoptosis; Neuroscience; NF-κB |
Ginsenoside Rg1 (Panaxoside Rg1) 是人参的主要活性成分之一,可减少NF-κB 核易位。它改善认知功能受损,通过降低大脑Aβ水平来发挥作用。 | |||
T2P2806 |
Hederacolchiside A1
黑海常春藤苷A1,革叶常春藤皂苷 A1,Raddeanoside R13 |
Apoptosis; ERK; MEK; Akt; PI3K; Parasite; mTOR | Apoptosis; Cytoskeletal Signaling; MAPK; Microbiology/Virology; PI3K/Akt/mTOR signaling |
Hederacolchiside A1 (Raddeanoside R13) 是从白头翁中分离的一种有抗利什曼原虫和抗肿瘤增殖活性的天然产物。 | |||
TN2119 |
Pulsatilla saponin H
白头翁属皂苷H,白头翁皂苷 H,3-O-Β-D-葡萄糖( 1→4)-[ A -L-鼠李糖(1→2)]- A-L-阿拉伯糖 常春藤配基- 28-O-鼠李糖(1→4)葡萄糖(1→6)葡萄糖苷 |
Others | Others |
Pulsatilla saponin H 是一种从 Pulsatilla koreana 的根中分离出来的天然产物。 | |||
T2S1193 |
Mogroside III-A1
罗汉果苷 III-A1 |
Others | Others |
Mogroside III-A1 是一种来自罗汉果 Swingle 的三萜糖苷。 Mogroside III-A1 一种无糖甜味剂。 | |||
TN7213 |
Ellagic acid 3-O-α-L-rhamnopyranoside
|
Others | Others |
Ellagic acid 3-O-α-L-rhamnopyranoside 是一种天然产物,存在于植物鹅绒委陵菜Potentilla anserina 的块根中。 | |||
TN2117 |
Pulsatilloside E
3-O-B-D-葡萄糖( 1→4)-[ A -L-鼠李糖(1→2)]- A-L-阿拉伯糖 23-羟基羽扇豆20(29)-烯-28–酸- 28-O-鼠李糖(1→4)葡萄糖(1→6)葡萄糖苷,Pulchinenoside E,白头翁皂苷E |
Others | Others |
Pulsatilloside E (Pulchinenoside E) 是一种从毛茛科白头翁Pulsatilla chinensis (Ranunculaceae)的根中分离出来的天然产物。 | |||
T4789 |
1-Hydroxy-2-naphthoic acid
1-羟基-2-萘甲酸,ALPHA-HYDROXYNAPHTHOIC ACID |
Others; Endogenous Metabolite | Metabolism; Others |
1-Hydroxy-2-naphthoic acid (ALPHA-HYDROXYNAPHTHOIC ACID) 是内源性代谢产物的一种。 | |||
TMO2790 |
1-Naphthaleneacetic acid
Transplantone,1-Naphthylacetic acid,α-Naphthaleneacetic acid,Phyomone,1-萘乙酸 |
Phospholipase | Metabolism |
1-Naphthaleneacetic acid (Transplantone) 是一种 PLA2抑制剂,IC50=13.16 μM。它也是一种合成的植物生长素,可以促进植物生长。 | |||
T2932 |
Ginsenoside Rh1
Sanchinoside B2,人参皂苷 Rh1,人参皂苷Rh1,Prosapogenin A2,20(S)-Ginsenoside Rh1,Sanchinoside Rh1 |
IL Receptor; TNF; Endogenous Metabolite; PPAR; Interleukin | Apoptosis; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism |
Ginsenoside Rh1 (Sanchinoside B2) 是人参的一种主要成分,具有抗炎作用,抑制PPAR-γ,TNF-α,IL-6和IL-1β的表达。 | |||
T8714 |
1-Stearoyl-sn-glycero-3-phosphocholine
1-硬脂酰-SN-甘油-3-磷酰胆碱,1-stearoyl-lysophosphatidylcholine,L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY |
Others | Others |
1-Stearoyl-sn-glycero-3-phosphocholine (L-ALPHA-LYSOPHOSPHATIDYLCHOLINE, STEAROY) 是一种用于脂质代谢研究的化学物质。 | |||
T4942 |
Galactose 1-phosphate Potassium salt
D-半乳糖 1-磷酸二钾盐五水合物,α-D-Galactose-1-phosphate Dipotassium Pentahydrate |
Others; Endogenous Metabolite | Metabolism; Others |
Galactose 1-phosphate Potassium salt (α-D-Galactose-1-phosphate Dipotassium Pentahydrate) 是一种半乳糖代谢中的中间体和核苷酸糖。 | |||
TN5712 |
9,10-Didehydroeffususol A
5-(1-Methoxyethyl)-1-methylphenanthrene-2,7-diol |
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9,10-Didehydroeffususol A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5712,CAS号为 1869082-57-4。 | |||
TN5725 |
Juncatrin A
1-(3,7-Dihydroxy-2,8-dimethyl-9,10-dihydrophenanthren-1-yl)ethanone |
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Juncatrin A 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5725,CAS号为 2265925-12-8。 | |||
T41310 |
Gibberellin A1
|
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Gibberellin A1 是一种天然产物,在生命科学相关研究中具有广泛的应用。 | |||
TN5016 | Sibiricose A1 | Others | Others |
Sibiricose A1 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5016,CAS号为 139726-40-2。 | |||
T5S2139 |
Epimedin A1
朝藿定A1,Hexandraside F |
Others | Others |
Epimedin A1 (Hexandraside F) 是一种黄酮类化合物,从常用中药淫羊藿中提取得到。 | |||
T12089 |
Mogroside I A1
罗汉果苷 I A1 |
Others | Others |
Mogroside I A1 是一种非糖类甜味剂,是三萜糖苷。Mogroside 比蔗糖更甜,具有抗氧化,抗糖尿病和抗癌作用。 | |||
T35752 |
Xanthoquinodin A1
Xanthoquinodin A1 |
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Xanthoquinodin A1 is a fungal metabolite that has been found inHumicolaand has diverse biological activities.1,2It inhibitsE. tenellaschizont formation in BHK-21 cells with a minimum effective concentration (MEC) value of 0.02 μg/ml.1Xanthoquinodin A1 is active againstB. subtilis,M. luteus,S. aureus,A. laidlawii, andB. fragilisin a disc assay when used at a concentration of 1 mg/ml. It is also active againstB. cereus(MIC = 0.44 μM).2Xanthoquinodin A1 is cytotoxic to KB, MCF-7, and NCI H187 cance... | |||
T35667 |
Napyradiomycin A1
Napyradiomycin A1 |
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Napyradiomycin A1is a fungal metabolite originally isolated fromC. rubraand has diverse biological activities.1,2It is active againstS. aureus,M. luteus,B. anthracis,C. bovis, andM. smegmatis(MICs = 1.56-12.5 μg/ml).1Napyradiomycin A1is an estrogen receptor antagonist (IC50= 4.2 μM in rat uterine homogenates).2It also inhibits mitochondrial NADH:ubiquinone oxidoreductase (complex I) and succinate:ubiquinone oxidoreductase (complex II) activities in bovine heart homogenates (IC50s = 20 and 9.7 μM... | |||
T0200 |
α-Lipoic Acid
Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid,α-硫辛酸,硫辛酸 |
Apoptosis; NF-κB; HIV Protease; Mitochondrial Metabolism; Endogenous Metabolite | Apoptosis; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome |
α-Lipoic Acid (DL-α-Lipoic acid) 是线粒体酶复合物的重要辅助因子,是一种抗氧化剂,可抑制NF-κB 依赖性的HIV-1LTR 活化。它还可诱导内质网应激介导的肝癌细胞凋亡。 | |||
T17302 |
(9Z,11E)-Prodlure
(9Z,11E)-Prodlure,Litlure A,(9Z,11E)-Tetradecadien-1-yl acetate,Ferodin SL |
Others | Others |
(9Z, 11E) - Prodlure is the main component of the sex pheromone of female Spodoptera littoralis. | |||
TN2311 |
Wulignan A1
五脂素 A1 |
Antifection | Microbiology/Virology |
Wulignan A1 exhibits activity against leukemia P-388 in vitro; it also may have anti-influenza virus H1N1 and H1N1-TR (a Tamiflu drug resistant virus strain) activities. | |||
TN1713 |
Graveobioside A
木犀草素 7-芹糖(1-2)-葡萄糖苷,木犀草素7-芹糖(1-2)-葡萄糖苷 |
Others | Others |
Graveobioside A can be used in hyperuricemia and gout-resistant drugs or health foods. | |||
TN1446 |
Bisabolol oxide A
甜没药萜醇氧化物A,[S-(R*,R*)]-α’-4-二甲基-α’-(4-甲基-3-戊烯基)-3-环己烯-1-甲醇 |
Others | Others |
Bisabololoxide A induces apoptosis in rat thymocytes. | |||
T2968 |
Hyodeoxycholic acid
NSC 60672,猪去氧胆酸,α-Hyodeoxycholic Acid,HDCA |
FXR; Endogenous Metabolite; GPCR19 | GPCR/G Protein; Metabolism |
Hyodeoxycholic acid (NSC 60672) 是由肠道菌群在小肠中形成的次级胆汁酸,是TGR5(GPCR19)的激动剂, CHO 细胞中的EC50=31.6 µM。它已用于研究高胆固醇血症的治疗。 | |||
T11201 |
Enniatin A1
恩镰孢菌素 A1 |
ERK | MAPK |
Enniatin A1 possesses anticarcinogenic properties by induction of apoptosis and disruption of ERK signalling pathway. Enniatin A1 inhibits ACAT with an IC50 of 49 μM in rat liver microsomes. Enniatin A1 isolated from Fusarium mycotoxins is a cyclic hexadepsipeptide consisting of alternating D-α-hydroxyisovaleric acids and N-methyl-L-amino acids. | |||
TN2442 |
Bacoside A1
假马齿苋皂素 A1 |
Others | Others |
Bacoside A1 is a natural product from plants | |||
T81993 |
Kadsurin A analogue-1
|
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Kadsurin A analogue-1 (Compound 8) 为源自Piper argyrophylum的木脂素类化合物。 | |||
T2851 |
Daphnetin
7,8-Dihydroxycoumarin,Daphnetol,瑞香素 |
EGFR; PKA; PKC; Parasite; Autophagy | Angiogenesis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; JAK/STAT signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Daphnetin (7,8-Dihydroxycoumarin) 是从 Genus Daphne 中分离得到的香豆素衍生物,有抗氧化、抗炎、抗疟疾和解热作用,可用于凝血功能障碍、类风湿性关节炎等疾病的相关研究。 | |||
T4183 |
lavendustin A
RG-14355,NSC 678027,薰草菌素 |
EGFR; Tyrosinase | Angiogenesis; JAK/STAT signaling; Proteases/Proteasome; Tyrosine Kinase/Adaptors |
lavendustin A (RG-14355) 是从链霉菌中分离得到的一种天然产物,是细胞渗透性表皮生长因子受体 (EGFR) 酪氨酸激酶抑制剂,能抑制血管内皮生长因子诱导的血管生成,阻断 LTPGABA-A 的诱导。 | |||
T83344 |
3-O-β-D-Glucopyranosyl(1→2)-[a-Lrhamnopyranosyl(1→3)]-β-D-glucopyranosyl 28-O-β-D-glucuronopyranoside
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3-O-β-D-Glucopyranosyl(1→2)-[a-Lrhamnopyranosyl(1→3)]-β-D-glucopyranosyl 28-O-β-D-glucuronopyranoside 是Polaskia chichipeBackbg 中分离的一种皂苷,具有抑制B16黑色素瘤细胞中黑色素生物合成的活性,100 μM 浓度可达到84.2%的抑制效果。 | |||
T5S1708 |
Dendrobine
|
Others; Influenza Virus | Microbiology/Virology; Others |
Dendrobine 是从石斛中分离的一种生物碱,对甲型流感病毒具有抗病毒活性。 | |||
TN6891 |
1-Hexanol
hexan-1-ol,正己醇 |
Others | Others |
1-Hexanol (hexan-1-ol) 是一种伯醇,是一种表面活性剂,通过非质子机制解偶联线粒体呼吸,可用于增强工业过程中的界面性能。 | |||
TN6912 |
1-Nonanol
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1-Nonanol is a natural product. | |||
TN6960 |
1-Pentadecanol
pentadecan-1-ol,1-十五醇,n-Pentadecanol |
Others | Others |
1-Pentadecanol (pentadecan-1-ol) 是一种天然产物,具有抗粉刺活性。 | |||
T10233 |
Acetylarenobufagin
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HIF | Angiogenesis; Chromatin/Epigenetic |
Acetylarenobufagin 是一种类固醇缺氧诱导因子-1 (HIF-I) 调节剂。 | |||
TN5924 |
3-Hydroxy-1-(4-hydroxyphenyl)propan-1-one
3-Hydroxy-1-(4-hydroxyphenyl)-1-propanone,3-羟基-1-(4-羟基苯基)丙烷-1-酮 |
Others | Others |
3-Hydroxy-1-(4-hydroxyphenyl)propan-1-one (3-Hydroxy-1-(4-hydroxyphenyl)-1-propanone) 是植物来源的天然产物。 | |||
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