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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2492 |
Perifosine
NSC 639966,D21266,KRX-0401,哌立福新 |
Apoptosis; Akt; Autophagy | Apoptosis; Autophagy; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Perifosine (KRX-0401) 是一种具有口服活性的烷基磷酸胆碱 Akt 抑制剂,具有抗肿瘤活性。 | |||
T1484 |
Perindoprilat
Perindoprilate,培哚普利 |
RAAS; MRP; AChR | Endocrinology/Hormones; Immunology/Inflammation; Neuroscience |
Perindoprilat (Perindoprilate) 是一种血管紧张素转换酶抑制剂。 | |||
T15034 |
Roluperidone
CYR-101,MIN-101,MT-210 |
Sigma receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Roluperidone (CYR-101) 是一种新型环酰胺衍生物,对5-HT2A 和sigma-2受体具有高亲和力,Ki 分别为 7.53 和 8.19 nM。 | |||
T1484L |
Perindopril erbumine
培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt |
Apoptosis; RAAS; MRP | Apoptosis; Endocrinology/Hormones; Immunology/Inflammation |
Perindopril erbumine (S9490-3) 是一种长效血管紧张素转换酶抑制剂。 | |||
T40111L |
BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride
|
PD-1/PD-L1 | Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation |
BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 是一种基于间苯二酚二Ph醚支架的程序性细胞死亡-1(PD-1)/程序性细胞死亡配体1(PD-L1)抑制剂, 抑制 PD-1/PD-L1 相互作用,IC50 值为 39.2 nM.BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 包含靶蛋白 PD-1/PD-L1 配体和 PROTAC linker。BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 可用于合成 PROTAC PD-1/PD-L1 degrader-1。BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 具有抗癌活性。BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 可作为稀释剂,用于用于直接压缩制备片剂。 | |||
T0990 |
Droperidol
氟派利多,NSC 169874,Dehydrobenzperidol,氟哌啶 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Droperidol (Dehydrobenzperidol) 是丁酰苯类多巴胺-2受体拮抗剂。 | |||
T17222 |
Velneperit
韦利贝特,S2367 |
Neuropeptide Y Receptor | GPCR/G Protein; Neuroscience |
Velneperit (S2367) 是一种有效且选择性的神经肽 Y (NPY) Y5 受体,有用于治疗肥胖症的研究潜力。 | |||
T66256 |
Ethyl 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
|
Factor Xa | Metabolism |
Ethyl 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate 对凝血因子Xa具有抑制作用,可用于研究血栓性静脉炎、动脉粥样硬化、脑栓塞、中风、肺栓塞。 | |||
T34921L1 |
Tresperimus TFA
Tresperimus TFA(160677-67-8 Free base) |
Others | Others |
Tresperimus TFA 可作为一种免疫制剂使用,可用于研究视网膜炎。 | |||
Fr13199 |
4-(4-chlorophenyl)piperidin-4-ol
|
||
Compound Fr13199 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr13199,CAS号为 39512-49-7。 | |||
T0082 |
Domperidone
R33812,多潘立酮 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Domperidone (R33812) 是多巴胺 2 受体拮抗剂,能够影响胃和小肠的化学感受器触发区和运动功能,具有止吐和促动力作用。 | |||
T8501 |
3-Phenyl-N-[1-(phenylmethyl)-4-piperidinyl]-tricyclo[3.3.1.13,7]decane-1-carboxamide
|
Influenza Virus | Microbiology/Virology |
3-Phenyl-N-[1-(phenylmethyl)-4-piperidinyl]-tricyclo[3.3.1.13,7]decane-1-carboxamide 具有抗埃博拉病毒的抗病毒活性靶向表面暴露的糖蛋白并抑制病毒进入宿主细胞。 Vero 细胞的体外研究表明,该化合物抑制病毒复制,EC50 为 0.38 μM。 | |||
T40018 |
4-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione
|
Others | Others |
4-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione 具有抗癌、治疗帕金森病的前药和抗炎药的潜力。 | |||
T7405 |
Piperidolate
二苯哌酯,哌立度酯 |
AChR | Neuroscience |
Piperidolate 是一种抗毒蕈碱药,可抑制乙酰胆碱引起的异常活性,能抑制大鼠和狗的肠痉挛。 | |||
T0025 |
Haloperidol
Aloperidin,氟哌啶醇,Serenace,Haldol |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Haloperidol (Serenace) 是一种安定药,是一种dopamine D2 receptor 拮抗剂。 | |||
T77598 |
Anisole-piperazine-methanone-benzothiazole-p-methylpiperidine
(4-(4-methoxyphenyl)piperazin-1-yl)(2-(4-methylpiperidin-1-yl)benzo[d]thiazol-6-yl)methanone |
Others | Others |
Anisole-piperazine-methanone-benzothiazole-p-methylpiperidine ((4-(4-methoxyphenyl)piperazin-1-yl)(2-(4-methylpiperidin-1-yl)benzo[d]thiazol-6-yl)methanone) 是一种生物合成的原材料,可用于合成多种化合物。 | |||
T7555 |
Piperidolate hydrochloride
|
AChR | Neuroscience |
Piperidolate hydrochloride 是一种抗毒蕈碱药,可抑制乙酰胆碱引起的异常活性,能抑制大鼠和狗的肠痉挛。 | |||
T16472 |
Pericyazine
Propericiazine,氰噻嗪,RP 8909 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Pericyazine (Propericiazine) 是第一代抗精神病药物,是一种选择性的 D2 多巴胺受体 (D2-dopamine receptor) 拮抗剂,具有肾上腺溶解、抗胆碱能和锥体外系作用,被用作短期管理严重焦虑状态和精神病的辅助药物。 | |||
Fr12729 |
1-Benzyl-4-hydroxypiperidine
1-Benzylpiperidin-4-ol |
||
Compound Fr12729 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr12729,CAS号为 4727-72-4。 | |||
T14083 |
Abaperidone
|
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Abaperidone 是一种有效的 5-HT2A 受体和多巴胺 D2 受体拮抗剂,对 5-HT2A 受体的 IC50 为 6.2 nM,对多巴胺 D2 受体的IC50 为 17 nM。Abaperidone是一种潜在的非典型抗精神化合物,可降低大鼠纹状体和前额叶皮层中的基础hsp70 mRNA表达。 | |||
T30077L |
Anisperimus HCl
LF 150195 HCl,Anisperimus HCl(170368-04-4 Free base) |
Others | Others |
Anisperimus HCl (LF 150195 HCl)是一种小分子免疫制剂,可用于研究自身免疫性疾病。 | |||
T50072 |
3-amino-1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one dihydrochloride
|
Others | Others |
3-amino-1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one dihydrochloride 用于多种化合物的合成。 | |||
T9361 |
5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione
5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione |
Others | Others |
5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione (5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione) 是一种合成化合物。它已被用作催化剂以及酶动力学研究中的工具;还被用于酶抑制的研究,以及药物受体相互作用的研究。 | |||
T9385 |
2-(2,6-dioxopiperidin-3-yl)-4-((7-hydroxyheptyl)oxy)isoindoline-1,3-dione
|
Others | Others |
2-(2,6-dioxopiperidin-3-yl)-4-((7-hydroxyheptyl)oxy)isoindoline-1,3-dione 是 protac。 | |||
T77687 |
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one
|
Others | Others |
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one 在人结肠癌细胞系中显示出抗肿瘤活性,可能用于防治血栓。 | |||
T64319 |
4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester
|
Others | Others |
4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester 是一种生物活性化合物,可作为中间体用于多种化合物的合成。 | |||
T9773 |
Thioquinapiperifil dihydrochloride
KF-31327 |
PDE | Metabolism |
Thioquinapiperifil dihydrochloride 是一种磷酸二酯酶(PDE-5)抑制剂(IC50: 0.074 nM),具有有效性、选择性和非竞争性,可用于研究性成熟。 | |||
T12152 |
N-piperidine Ibrutinib hydrochloride
|
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
N-piperidine Ibrutinib hydrochloride 是一种强效的 BTK 抑制剂,是BTK 配体,抑制 WT BTK 和 C481S BTK ,可用于合成一系列 PROTAC 分子。N-piperidine Ibrutinib hydrochloride具有潜在的抗癌活性,可抑制癌细胞的生长和增殖。 | |||
T0511 |
Tolperisone hydrochloride
盐酸托哌酮,Muscalm,Midocalm,托哌酮盐酸盐,Tolperisone HCl |
Sodium Channel | Membrane transporter/Ion channel |
Tolperisone hydrochloride (Muscalm) 是中枢作用肌肉松弛剂,可用于研究神经疾病引起的病理性横纹肌硬化(锥体束损伤、脊髓病、多发性硬化症、脑脊髓炎)、痉挛性麻痹及其他肌肉张力障碍相关的脑病。 | |||
T5007 |
Benproperine phosphate
磷酸苯丙哌林,Blascorid,Pirexyl phosphate |
Others; Microtubule Associated | Cytoskeletal Signaling; Others |
Benproperine phosphate (Pirexyl phosphate) 是一种具有口服活性的,肌动蛋白相关蛋白 2/3 复合亚基 2 (ARPC2) 抑制剂。它通过削弱 Arp2/3 功能来减弱肌动蛋白的聚合反应速率。它可抑制癌细胞迁移和肿瘤转移,有用于治疗止咳的潜力。 | |||
T25487 |
Haloperidol decanoate
KD 16,KD-136,KD 136,Neoperidole,Haldol |
Others | Others |
Haloperidol decanoate (KD 16) 是一种典型的抗精神病药物,用作精神分裂症和情绪障碍的维持治疗,配制成用于肌肉注射的酯。 | |||
T26360 |
Benperidol
R4584,R-4584,Anquil,McN-JR-4584,R 4584 |
||
Benperidol (Anquil)是一种具有抗精神病和安定作用的丁酮类化合物,在阻断 D2 受体方面具有很好的疗效。Benperidol可用于正电子发射断层扫描(PET)测量体内 D(2)类多巴胺受体的结合情况。 | |||
T68087 |
Inaperisone
|
Others | Others |
Inaperisone 是一种新型的中枢作用的肌肉松弛剂,对排尿反射有抑制作用。Inaperisone 可能通过间接作用于脑干的GABAB 受体来抑制排尿反射。 | |||
T3497 |
Ocaperidone
奥卡哌酮,Ocaperidona,R79598 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Ocaperidone (Ocaperidona) 是5-HT2和多巴胺D2的拮抗剂,也是5-HT1A 的激动剂,有安定作用。 | |||
T50060 |
2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid
|
Others | Others |
2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid (trifluoroacetic acid) 主要用于化合物的合成。 | |||
T9386 |
2-(2,6-dioxopiperidin-3-yl)-4-((9-hydroxynonyl)oxy)isoindoline-1,3-dione
|
Others | Others |
2-(2,6-dioxopiperidin-3-yl)-4-((9-hydroxynonyl)oxy)isoindoline-1,3-dione 是一种 PROTAC 接头,可用于 PROTAC 的合成。 | |||
T8636 |
Ibrutinib deacryloylpiperidine
IBT4A,5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyriMidin-4-ylaMine,伊布替尼中间体N-2 |
BTK | Angiogenesis; Tyrosine Kinase/Adaptors |
Ibrutinib deacryloylpiperidine (IBT4A) 是 Ibrutinib 的杂质之一。它是一种不可逆的、选择性的 Btk 抑制剂 (IC50:0.5 nM)。 | |||
T7788 |
2-Phenyl-2-(1-piperidinyl)propane
|
Others | Others |
2-Phenyl-2-(1-piperidinyl)propane 是一种具有可逆性、选择性的人 CYP2B6抑制剂,其 IC50为 5.1 μM,Ki 为 5.6。它对 CYP2D6 、CYP3A 均有抑制作用,且 IC50值分别为74 μM、200 μM。 | |||
T11894 |
Lusaperidone
R107474 |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Lusaperidone (R107474) 是一种有效的α2肾上腺素受体 (adrenergic receptor) 拮抗剂,是 α (2)-肾上腺素受体的潜在放射性配体,对 α2A和α2C 具有抑制作用, Ki 值分别为0.13和0.15 nM。 | |||
T0351 |
Risperidone
Risperidal,R 64 766,利培酮 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; P-gp | GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience |
Risperidone (R 64 766) 是5-HT2受体阻断剂、P-糖蛋白抑制剂和多巴胺 D2受体的拮抗剂,对 5-HT2A 和多巴胺 D2受体的 Ki 值分别为 4.8 和 5.9 nM。 | |||
T1539 |
Iloperidone
伊潘立酮,HP 873 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Iloperidone (HP 873) 是一种D2/5-HT2受体拮抗剂,是非典型抗精神病药,可治疗精神分裂症。 | |||
T14830 |
Bromperidol
溴哌利多,R-11333 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Bromperidol (R-11333) 是一种苯丁酮衍生物,是一种强效长效精神安定药。它被用作治疗精神分裂症的抗精神病药。 | |||
T28778 |
Silperisone HCl
RGH5002,SILA336,RGH-5002,Silperisone hydrochloride,SILA-336 |
||
Silperisone HCl (RGH-5002) 阻断细胞中的钠和钙通道,使肌肉细胞的兴奋度和收缩度降低,降低外周张力,充当肌肉松弛剂和外周血管扩张剂。 Silperisone HCl 可用于治疗脊髓损伤引起的复发性疼痛性肌阵挛、脑血管病引起的异常高肌张力、肌张力症状、锥体紧张综合征、多发性硬化症肌痉挛和脊髓炎。Silperisone 是钠通道蛋白2型α通道阻滞剂。Silperisone 是一种类似于tolperisone 的有机硅化合物,具有中枢作用的肌肉松弛剂特性。 | |||
T30077 |
Anisperimus
LF 150195,LF-150195,LF 15-0195,LF-15-0195,LF15-0195 |
Caspase | Apoptosis; Proteases/Proteasome |
Anisperimus (LF 15-0195) 是一种免疫抑制剂,通过促进 DISC 水平的 caspase-8 和 caspase-10 激活来增强激活诱导的 T 细胞死亡,通过促进表达 Foxp3 的调节性 CD4 T 细胞的发育来预防中枢神经系统自身免疫。 | |||
T9968 |
3-Piperidinyl(1-pyrrolidinyl)methanone hydrochloride
|
Others | Others |
3-Piperidinyl(1-pyrrolidinyl)methanone hydrochloride 可用于合成 MCH-R1 拮抗剂 piperidin-4-yl-urea 衍生物。 | |||
T26235 |
Sulfaperin
磺胺培林,Methylsulfadiazin,Archisulfa,Chemiopen,Demosulfan,Anastaf,Isosulfamerazine |
Antibacterial | Microbiology/Virology |
Sulfaperin (Chemiopen) 是一种磺胺类抗菌剂。 | |||
T50083 |
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide
|
Others | Others |
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide 可用作分子结构单元,用于多种化合物的合成。 | |||
T7843 |
4-phenoxypiperidine
|
Others | Others |
4-phenoxypiperidine 具有肌肉松弛和抗惊厥活性。 | |||
TP1220L |
Carperitide acetate
醋酸卡培立肽,Carperitide acetate (89213-87-6 Free base),Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate |
Endothelin Receptor | GPCR/G Protein |
Carperitide acetate (Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate) 是一种由 28 个氨基酸组成的激素,由心脏产生并分泌,以响应心脏损伤和机械拉伸。Carperitide acetate 抑制内皮素-1 (endothelin-1) 分泌。 | |||
T62461 |
Benzyl-piperazine-CO-benzothiazole-4-methylpiperidine
|
Others | Others |
Benzyl-piperazine-CO-benzothiazole-4-methylpiperidine 可用于改变真核生物寿命。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2S1992 |
Perillartine
Perilla sugar,Peryllartine,紫苏葶,DL-Perillartine |
Others; Endogenous Metabolite | Metabolism; Others |
Perillartine (DL-Perillartine) 是甜味剂,能够激活味觉受体 1 型成员 2 。 | |||
TN2054 |
Periplocymarin
|
Calcium Channel | Membrane transporter/Ion channel; Metabolism |
Periplocymarin 是一种强心苷,从 Periploca sepium 和 Periploca graeca 中分离得到,具有抗癌潜力。 | |||
TN2213 |
Imperialine 3-β-D-glucoside
Sipeimine-3-beta-D-glucoside,西贝母碱苷 |
Others | Others |
Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) 是 Imperialine 的糖苷。它对多重耐药肿瘤细胞表现出抗肿瘤特性。 | |||
T5S1982 |
Periplocin
Periplocoside,杠柳毒苷 |
Apoptosis; Others | Apoptosis; Others |
Periplocin (Periplocoside) 是从黑龙骨中分离出的一种强心类固醇。它可促进肿瘤细胞凋亡并抑制肿瘤生长。它通过激活 Na/K-ATPase 介导的 Src/ERK 和 PI3K/Akt 途径,具有促进伤口愈合的潜力。 | |||
T4S1983 |
Periplogenin
5-beta-Hydroxydigitoxigenin,Desoxostrophanthidin,杠柳苷元 |
Others | Others |
Periplogenin (Desoxostrophanthidin) 是一种天然呋喃香豆素,存在于白芷根中,可以诱导脂肪细胞分化,具有高抗银屑病作用。 | |||
T6377 |
Aloperine
|
Apoptosis; Virus Protease; HIV Protease; Antibiotic; Autophagy | Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome |
Aloperine 是一种在苦参类植物中的生物碱,其具有抗癌,抗炎、抗肿瘤和抗病毒特性,可用于研究过敏性接触性皮炎湿疹和其他皮肤炎症。 | |||
T1035 |
Hesperidin
橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷 |
Apoptosis; Reactive Oxygen Species; Endogenous Metabolite; Autophagy | Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB |
Hesperidin (Cirantin) 是一种广泛存在于柑橘类水果中黄烷酮糖苷,具有减少炎症介质并发挥重要的抗氧化作用,还有抗肿瘤和抗过敏活性。 | |||
T6S0923 |
Hypericin
Hypericine,金丝桃素,Cyclosan |
Apoptosis; Antiviral; Influenza Virus; Tyrosine Kinases; Antibacterial; PKC | Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Tyrosine Kinase/Adaptors |
Hypericin (Cyclosan) 是贯叶连翘的提取物,有抗菌、抗病毒、抗肿瘤和抗抑郁作用。 | |||
T3S2381 |
Perillene
3-Isohexenylfuran,紫苏烯,Perillen |
Others; Antibacterial | Microbiology/Virology; Others |
Perillene (3-Isohexenylfuran) 是促进肠蠕动的药物中的活性成分,它对金黄色葡萄球菌和大肠杆菌具有很强的抗药性。 | |||
TN2108 |
Protohypericin
|
Others | Others |
Protohypericin 是一种从贯叶连翘中提取的天然石脑粉。放射性碘化 Protohypericin 能用于肿瘤坏死靶向放射研究。 | |||
T0076 |
Paliperidone
9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Paliperidone (9-hydroxyrisperidone) 是 Risperidone 的主要活性代谢产物,是多巴胺 D2 拮抗剂和5-HT2A 拮抗剂。它用作非典型抗精神病药,用于精神分裂症的急性及维持治疗。它对α1和α2肾上腺素能受体和 H1组胺能受体也有拮抗作用。 | |||
T29756 |
1-piperoylpiperidine
AI3 01439,胡椒碱,AI3-01439,AI 3-01439,piperine |
Others | Others |
1-piperoylpiperidine (AI3-01439) 是一种生化物质。 | |||
T0228 |
Methyl-Hesperidin
甲基橙皮甙 |
Akt; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling |
Methyl hesperidin 是一种血管扩张剂。 | |||
T13495 |
3-Amino-2-piperidinone
Cyclo-ornithine |
Endogenous Metabolite | Metabolism |
3-Amino-2-piperidinone 是来自生物体的代谢物,可用作环状鸟氨酸类似物。 | |||
T3314 |
Perillyl alcohol
Isocarveol,Perilla alcohol,紫苏醇 |
Apoptosis; Endogenous Metabolite | Apoptosis; Metabolism |
Perillyl alcohol (Isocarveol) 是一种单萜,可在不影响正常细胞的情况下诱导肿瘤细胞凋亡。 | |||
T2767 |
Neohesperidin Dihydrochalcone
NHDC,新橙皮苷二氢查尔酮,新橙皮苷二氢查耳酮,Neohesperidin DC,NCI-c60764 |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Neohesperidin Dihydrochalcone (Neohesperidin DC) 是一种合成的糖苷查耳酮,可用作低热量人造甜味剂,添加到各种食品和饮料中。 | |||
T6S0920 |
2"-O-Galloylhyperin
2”-O-没食子酰基金丝桃苷,2''-O-Galloylhyperin,Q-100605,FT-0689359 |
Others | Others |
2"-O-Galloylhyperin (FT-0689359) 是一种分离自Pyrola incarnateFisch. 中的活性化合物,具有抗氧化和抗炎作用,对氧化应激诱导的肝损伤具有肝保护作用。 | |||
T3002 |
Piperine
胡椒碱,1-Piperoylpiperidine,Bioperine |
P450; Endogenous Metabolite; P-gp; Autophagy | Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience |
Piperine (Bioperine) 是从胡椒中分离的一种生物碱,可以抑制P-糖蛋白和 CYP3A4 的活性,在HeLa 细胞中的IC50值为61.94±0.054 μg/mL。它已用于研究治疗多发性骨髓瘤和吞咽障碍的试验。 | |||
T8282 |
(S)-(−)-Perillyl alcohol
Perillyl alcohol,(-)-Perillyl Alcohol,L-紫苏醇 |
Apoptosis; Endogenous Metabolite | Apoptosis; Metabolism |
(S)-(−)-Perillyl alcohol (Perillyl alcohol) 是一种在薰衣草中发现的单萜,可抑制 Ras 的法尼基化,上调 6-磷酸甘露糖受体并诱导细胞凋亡。 它还具有抗癌活性。 | |||
T5786 |
TETRAHYDROPIPERINE
四氢胡椒碱,Cosmoperine |
P450; TRP/TRPV Channel | Membrane transporter/Ion channel; Metabolism |
Tetrahydropiperine (Cosmoperine) 是胡椒碱的环己基类似物,也是一种天然芳基戊酰胺,从Piper longum 分离得到。它对细胞色素 P450 (CYP) 同工型 CYP1A1/芳基烃羟化酶 (AHH;IC50=23 µM)具有抑制作用。 | |||
T8256 |
piperitone
胡椒酮,3甲基-6-(1-甲基乙基)-2-环己烯-1-酮 |
Others | Others |
Piperitone 是强大的驱虫剂和抗食欲剂。它对 Cymbopogon schoenanthus(C. schoenanthus) 成虫、新产卵和新生幼虫有很大的毒性。 | |||
TN1819 |
Kaempferol 3-neohesperidoside
Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷 |
GSK-3; MEK; PI3K | MAPK; PI3K/Akt/mTOR signaling; Stem Cells |
Kaempferol 3-neohesperidoside (Kaempferol 3-O-neohesperidoside) 是一种类黄酮,对大鼠比目鱼肌具有拟胰岛素作用。 | |||
T2737 |
Neohesperidin
Hesperetin 7-O-neohesperidoside,NSC 31048,新橙皮苷 |
Antioxidant | oxidation-reduction |
Neohesperidin (NSC-31048) 是一种类黄酮化合物,存在于葫芦科植物中,具有抗氧化和抗炎活性。 | |||
TN1164 | 1-(3,4-Dimethoxycinnamoyl)piperidine | Others | Others |
1-(3,4-Dimethoxycinnamoyl)piperidine is a natural product | |||
T9112 | (-)-Perillaldehyde | AhR; ROS; Nrf2 | Immunology/Inflammation; Metabolism |
L-Perillaldehyde 是紫苏草精油的主要成分,吸入后经由嗅觉神经功能表现出抗抑郁功能。 | |||
TN2055 |
Periplogenin 3-[O-β-glucopyranosyl-(1→4)-β-sarmentopyranoside]
4)-beta-sarmentopyranoside]'>Periplogenin 3-[O-beta-glucopyranosyl-(1->4)-beta-sarmentopyranoside],异杠柳毒苷 |
Others | Others |
Periplogenin 3-[O-beta-glucopyranosyl-(1->4)-beta-sarmentopyranoside] is a natural product from Periploca sepiumBge. | |||
TN2109 | Protopseudohypericin | Others | Others |
Protopseudohypericin is a natural product | |||
TN5312 |
Periplocogenin
|
||
Periplocogenin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5312,CAS号为 112899-63-5。 | |||
TN4751 |
Periglaucine B
|
HBV | Microbiology/Virology |
Periglaucine B can inhibit hepatitis B virus (HBV) surface antigen (HBsAg) secretion in Hep G2.2.15 cells. | |||
TN1044 |
Quercetin 3-O-neohesperidoside
|
Others | Others |
Quercetin 3-O-neohesperidoside shows anti-atherosclerosis, and antiplatelet aggregation activities. | |||
T40252 |
Peritassine A
|
||
Peritassine A, an alkaloid derived from Tripterygium wilfordii Hook. f., exhibits anti-HIV properties. | |||
T40640 |
Glycoperine
|
||
Glycoperine is a alkaloid from haplophyllum perforatum. | |||
TN2758 |
2-Ethyl-2,6,6-trimethylpiperidin-4-one
|
Others | Others |
2-Ethyl-2,6,6-trimethylpiperidin-4-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2758,CAS号为 133568-79-3。 | |||
TN4148 | Glyasperin C | Tyrosinase; Antifection | Microbiology/Virology; Proteases/Proteasome |
Glyasperin C acts as a partial estrogen antagonist, it shows tyrosinase inhibitory activity (IC (50) = 0.13 +/- 0.01 microg/mL), it could be a promising candidate in the design of skin-whitening agents. Glyasperin C shows potent anti-vancomycin-resistant | |||
TN4750 | Periglaucine A | HBV | Microbiology/Virology |
Periglaucine A inhibits hepatitis B virus (HBV) surface antigen (HBsAg) secretion in Hep G2.2.15 cells. | |||
TN4372 |
Kaempferol-7-O-neohesperidoside
|
Others | Others |
Kaempferol-7-O-neohesperidoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4372,CAS号为 17353-03-6。 | |||
T83353 |
3'-Methoxy-3,5,4'-trihydroxyflavone-7-neohesperidoside
|
||
3'-Methoxy-3,5,4'-triHydroxyflavone-7-neheesperidoside,一种从Cleome droserifolia中分离的黄酮类化合物,显示出中等程度的保肝活性。 | |||
TN4825 |
Prenylpiperitol
|
Others | Others |
Prenylpiperitol是一种天然产物,属于芸香科石南芸木属,其产品编号为 TN4825,CAS号为 157659-20-6。Prenylpiperitol可用作对照参考。 | |||
TN2056 |
Perisesaccharide B
|
Others | Others |
Perisesaccharide B is a natural product | |||
TN4149 |
Glyasperin F
|
Others | Others |
Glyasperin F has antinociceptive, and anti-inflammatory effects, it could inhibit NO production in RAW 264.7 macrophages to some extent. Glyasperin F displayed cytotoxic effects against the four tested cancer cell lines with IC50values below 85 μM. | |||
TN3806 |
Dehydroglyasperin C
|
ERK; IκB/IKK; p38 MAPK; TNF; NF-κB; Akt; COX; PI3K; NADPH; DNA/RNA Synthesis; Nrf2; JNK; Autophagy | Apoptosis; Autophagy; Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Immunology/Inflammation; MAPK; Metabolism; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling |
Dehydroglyasperin C is a potent NAD(P)H:oxidoquinone reductase (NQO1) and phase 2 enzyme inducer. Dehydroglyasperin C possesses potent antioxidant, cancer chemopreventive, and neuroprotective activities, it has protective effects against chronic diseases | |||
TN4147 |
Glyasperin A
|
Others | Others |
Glyasperin A has cytotoxic properties against P-388 cells, its IC50 values being 6.0 microM. | |||
T4110 |
Perivine
Perivin,派利文碱 |
Others | Others |
Perivine (Perivin) 以视网膜母细胞瘤相关蛋白 (RbAp48) 为靶点,能够解决 RbAp48-FOG-1 复合物的不稳定性。Perivine 可用于研究阿尔茨海默病。 | |||
T7980 |
Hesperidin methylchalcone
|
NF-κB | NF-κB |
Hesperidin methylchalcone 抑制氧化应激,细胞因子产生和NF-κB 活化。它能够抑制炎症和疼痛,具有血管保护作用。 | |||
TN7049 |
6''-Acetylhyperin
|
||
6''-Acetylhyperin 在生命科学相关研究中具有广泛的应用。 | |||
TN3810 | Dehydroperilloxin | COX | Immunology/Inflammation; Neuroscience |
Dehydroperilloxin possesses inhibitory activity against cyclooxygenase-1, with the IC(50) value of 30.4 microM. | |||
TN2052 | Periplocoside M | Others | Others |
Periplocoside M possesses observably antitumor activity against SMMC-7721( IC 50=12.9 ng/L),Hela( IC 50=8.63 ng/L) and MCF-7( IC 50=18.5 ng/L) cancer cell lines. | |||
TN5315 |
Periplocoside F
Periploside F |
||
Periplocoside F 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5315,CAS号为 119902-17-9。 | |||
TN2084 |
Piperitol
|
Others | Others |
Piperitol has in vitro antioxidant potential, it also exhibits a stronger CNS depressant effect than that of M. rotundifolia. | |||
TN1356 |
Acetyl Perisesaccharide C
乙酰杠柳寡糖 C,乙酰杠柳寡糖C |
Others | Others |
Acetyl Perisesaccharide C is a natural product | |||
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Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPY-01613 |
Periostin/OSF-2 Protein, Mouse, Recombinant (His)
A630052E07Rik,OSF-2,Osf2,PLF,AI747096,peri,PN,p... |
Mouse | HEK293 Cells |
Periostin/OSF-2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 89 kDa and the accession number is Q62009-2. | |||
TMPY-01020 |
Periostin/OSF-2 Protein, Human, Recombinant (His)
PN,OSF-2,OSF2,periostin,periostin, osteobl... |
Human | HEK293 Cells |
Periostin/OSF-2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 86.4 kDa and the accession number is Q15063-3. | |||
TMPK-01032 |
Periostin/OSF-2 Protein, Mouse, Recombinant (aa 24-811, His)
POSTN,OSF2,Periostin,TRIF52,PNRP11-412K4.1,PN,Fasci... |
Mouse | HEK293 Cells |
Periostin/OSF-2 Protein, Mouse, Recombinant (aa 24-811, His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 88.7 kDa and the accession number is Q62009-1. | |||
TMPK-00973 |
Periostin/OSF-2 Protein, Human, Recombinant (aa 22-836, His)
Periostin,POSTN,Fasciclin I-like,TRIF52,OSF-2,PNRP1... |
Human | HEK293 Cells |
Periostin/OSF-2 Protein, Human, Recombinant (aa 22-836, His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 92.1 kDa and the accession number is Q15063. | |||
TMPY-05190 |
Per a 1 Protein, Periplaneta americana, Recombinant (His)
|
Periplaneta americana | E. coli |
Per a 1 Protein, Periplaneta americana, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 27.2 kDa and the accession number is Q9TZR6. | |||
TMPY-04853 |
TSHR Protein, Human, Recombinant (His)
TSHR,hTSHR-I,TSH Receptor,LGR3,CHNG1 |
Human | Baculovirus Insect Cells |
Thyroid-stimulating hormone (TSH) is secreted by the pituitary gland and promotes thyroid growth and function, with increased TSH levels typically associated with hypothyroidism. Immunohistochemical analysis revealed predominantly nuclei/peri-nuclei localization of TSHR in cancerous tissues but cell membrane localization in non-cancerous parts. Overexpression of TSHR was found in a great majority of HCC tissues and associated with unfavorable prognosis. |