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Targets Recommended: Apoptosis Akt Autophagy

242

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T2492 Perifosine

NSC 639966,D21266,KRX-0401,哌立福新

Apoptosis; Akt; Autophagy Apoptosis; Autophagy; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Perifosine (KRX-0401) 是一种具有口服活性的烷基磷酸胆碱 Akt 抑制剂,具有抗肿瘤活性。
T1484 Perindoprilat

Perindoprilate,培哚普利

RAAS; MRP; AChR Endocrinology/Hormones; Immunology/Inflammation; Neuroscience
Perindoprilat (Perindoprilate) 是一种血管紧张素转换酶抑制剂。
T15034 Roluperidone

CYR-101,MIN-101,MT-210

Sigma receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Roluperidone (CYR-101) 是一种新型环酰胺衍生物,对5-HT2A 和sigma-2受体具有高亲和力,Ki 分别为 7.53 和 8.19 nM。
T1484L Perindopril erbumine

培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt

Apoptosis; RAAS; MRP Apoptosis; Endocrinology/Hormones; Immunology/Inflammation
Perindopril erbumine (S9490-3) 是一种长效血管紧张素转换酶抑制剂。
T40111L BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride

PD-1/PD-L1 Apoptosis; Cell Cycle/Checkpoint; Immunology/Inflammation
BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 是一种基于间苯二酚二Ph醚支架的程序性细胞死亡-1(PD-1)/程序性细胞死亡配体1(PD-L1)抑制剂, 抑制 PD-1/PD-L1 相互作用,IC50 值为 39.2 nM.BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 包含靶蛋白 PD-1/PD-L1 配体和 PROTAC linker。BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 可用于合成 PROTAC PD-1/PD-L1 degrader-1。BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 具有抗癌活性。BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride 可作为稀释剂,用于用于直接压缩制备片剂。
T0990 Droperidol

氟派利多,NSC 169874,Dehydrobenzperidol,氟哌啶

Dopamine Receptor GPCR/G Protein; Neuroscience
Droperidol (Dehydrobenzperidol) 是丁酰苯类多巴胺-2受体拮抗剂。
T17222 Velneperit

韦利贝特,S2367

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Velneperit (S2367) 是一种有效且选择性的神经肽 Y (NPY) Y5 受体,有用于治疗肥胖症的研究潜力。
T66256 Ethyl 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate

Factor Xa Metabolism
Ethyl 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate 对凝血因子Xa具有抑制作用,可用于研究血栓性静脉炎、动脉粥样硬化、脑栓塞、中风、肺栓塞。
T34921L1 Tresperimus TFA

Tresperimus TFA(160677-67-8 Free base)

Others Others
Tresperimus TFA 可作为一种免疫制剂使用,可用于研究视网膜炎。
Fr13199 4-(4-chlorophenyl)piperidin-4-ol

Compound Fr13199 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr13199,CAS号为 39512-49-7。
T0082 Domperidone

R33812,多潘立酮

Dopamine Receptor GPCR/G Protein; Neuroscience
Domperidone (R33812) 是多巴胺 2 受体拮抗剂,能够影响胃和小肠的化学感受器触发区和运动功能,具有止吐和促动力作用。
T8501 3-​Phenyl-​N-​[1-​(phenylmethyl)​-​4-​piperidinyl]​-tricyclo[3.3.1.13,​7]​decane-​1-​carboxamide

Influenza Virus Microbiology/Virology
3-​Phenyl-​N-​[1-​(phenylmethyl)​-​4-​piperidinyl]​-tricyclo[3.3.1.13,​7]​decane-​1-​carboxamide 具有抗埃博拉病毒的抗病毒活性靶向表面暴露的糖蛋白并抑制病毒进入宿主细胞。 Vero 细胞的体外研究表明,该化合物抑制病毒复制,EC50 为 0.38 μM。
T40018 4-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione

Others Others
4-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione 具有抗癌、治疗帕金森病的前药和抗炎药的潜力。
T7405 Piperidolate

二苯哌酯,哌立度酯

AChR Neuroscience
Piperidolate 是一种抗毒蕈碱药,可抑制乙酰胆碱引起的异常活性,能抑制大鼠和狗的肠痉挛。
T0025 Haloperidol

Aloperidin,氟哌啶醇,Serenace,Haldol

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Haloperidol (Serenace) 是一种安定药,是一种dopamine D2 receptor 拮抗剂。
T77598 Anisole-piperazine-methanone-benzothiazole-p-methylpiperidine

(4-(4-methoxyphenyl)piperazin-1-yl)(2-(4-methylpiperidin-1-yl)benzo[d]thiazol-6-yl)methanone

Others Others
Anisole-piperazine-methanone-benzothiazole-p-methylpiperidine ((4-(4-methoxyphenyl)piperazin-1-yl)(2-(4-methylpiperidin-1-yl)benzo[d]thiazol-6-yl)methanone) 是一种生物合成的原材料,可用于合成多种化合物。
T7555 Piperidolate hydrochloride

AChR Neuroscience
Piperidolate hydrochloride 是一种抗毒蕈碱药,可抑制乙酰胆碱引起的异常活性,能抑制大鼠和狗的肠痉挛。
T16472 Pericyazine

Propericiazine,氰噻嗪,RP 8909

Dopamine Receptor GPCR/G Protein; Neuroscience
Pericyazine (Propericiazine) 是第一代抗精神病药物,是一种选择性的 D2 多巴胺受体 (D2-dopamine receptor) 拮抗剂,具有肾上腺溶解、抗胆碱能和锥体外系作用,被用作短期管理严重焦虑状态和精神病的辅助药物。
Fr12729 1-Benzyl-4-hydroxypiperidine

1-Benzylpiperidin-4-ol

Compound Fr12729 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 Fr12729,CAS号为 4727-72-4。
T14083 Abaperidone

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Abaperidone 是一种有效的 5-HT2A 受体和多巴胺 D2 受体拮抗剂,对 5-HT2A 受体的 IC50 为 6.2 nM,对多巴胺 D2 受体的IC50 为 17 nM。Abaperidone是一种潜在的非典型抗精神化合物,可降低大鼠纹状体和前额叶皮层中的基础hsp70 mRNA表达。
T30077L Anisperimus HCl

LF 150195 HCl,Anisperimus HCl(170368-04-4 Free base)

Others Others
Anisperimus HCl (LF 150195 HCl)是一种小分子免疫制剂,可用于研究自身免疫性疾病。
T50072 3-amino-1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one dihydrochloride

Others Others
3-amino-1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one dihydrochloride 用于多种化合物的合成。
T9361 5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione

5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione

Others Others
5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione (5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione) 是一种合成化合物。它已被用作催化剂以及酶动力学研究中的工具;还被用于酶抑制的研究,以及药物受体相互作用的研究。
T9385 2-(2,6-dioxopiperidin-3-yl)-4-((7-hydroxyheptyl)oxy)isoindoline-1,3-dione

Others Others
2-(2,6-dioxopiperidin-3-yl)-4-((7-hydroxyheptyl)oxy)isoindoline-1,3-dione 是 protac。
T77687 3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one

Others Others
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one 在人结肠癌细胞系中显示出抗肿瘤活性,可能用于防治血栓。
T64319 4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester

Others Others
4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester 是一种生物活性化合物,可作为中间体用于多种化合物的合成。
T9773 Thioquinapiperifil dihydrochloride

KF-31327

PDE Metabolism
Thioquinapiperifil dihydrochloride 是一种磷酸二酯酶(PDE-5)抑制剂(IC50: 0.074 nM),具有有效性、选择性和非竞争性,可用于研究性成熟。
T12152 N-piperidine Ibrutinib hydrochloride

BTK Angiogenesis; Tyrosine Kinase/Adaptors
N-piperidine Ibrutinib hydrochloride 是一种强效的 BTK 抑制剂,是BTK 配体,抑制 WT BTK 和 C481S BTK ,可用于合成一系列 PROTAC 分子。N-piperidine Ibrutinib hydrochloride具有潜在的抗癌活性,可抑制癌细胞的生长和增殖。
T0511 Tolperisone hydrochloride

盐酸托哌酮,Muscalm,Midocalm,托哌酮盐酸盐,Tolperisone HCl

Sodium Channel Membrane transporter/Ion channel
Tolperisone hydrochloride (Muscalm) 是中枢作用肌肉松弛剂,可用于研究神经疾病引起的病理性横纹肌硬化(锥体束损伤、脊髓病、多发性硬化症、脑脊髓炎)、痉挛性麻痹及其他肌肉张力障碍相关的脑病。
T5007 Benproperine phosphate

磷酸苯丙哌林,Blascorid,Pirexyl phosphate

Others; Microtubule Associated Cytoskeletal Signaling; Others
Benproperine phosphate (Pirexyl phosphate) 是一种具有口服活性的,肌动蛋白相关蛋白 2/3 复合亚基 2 (ARPC2) 抑制剂。它通过削弱 Arp2/3 功能来减弱肌动蛋白的聚合反应速率。它可抑制癌细胞迁移和肿瘤转移,有用于治疗止咳的潜力。
T25487 Haloperidol decanoate

KD 16,KD-136,KD 136,Neoperidole,Haldol

Others Others
Haloperidol decanoate (KD 16) 是一种典型的抗精神病药物,用作精神分裂症和情绪障碍的维持治疗,配制成用于肌肉注射的酯。
T26360 Benperidol

R4584,R-4584,Anquil,McN-JR-4584,R 4584

Benperidol (Anquil)是一种具有抗精神病和安定作用的丁酮类化合物,在阻断 D2 受体方面具有很好的疗效。Benperidol可用于正电子发射断层扫描(PET)测量体内 D(2)类多巴胺受体的结合情况。
T68087 Inaperisone

Others Others
Inaperisone 是一种新型的中枢作用的肌肉松弛剂,对排尿反射有抑制作用。Inaperisone 可能通过间接作用于脑干的GABAB 受体来抑制排尿反射。
T3497 Ocaperidone

奥卡哌酮,Ocaperidona,R79598

Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience
Ocaperidone (Ocaperidona) 是5-HT2和多巴胺D2的拮抗剂,也是5-HT1A 的激动剂,有安定作用。
T50060 2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid

Others Others
2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid (trifluoroacetic acid) 主要用于化合物的合成。
T9386 2-(2,6-dioxopiperidin-3-yl)-4-((9-hydroxynonyl)oxy)isoindoline-1,3-dione

Others Others
2-(2,6-dioxopiperidin-3-yl)-4-((9-hydroxynonyl)oxy)isoindoline-1,3-dione 是一种 PROTAC 接头,可用于 PROTAC 的合成。
T8636 Ibrutinib deacryloylpiperidine

IBT4A,5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyriMidin-4-ylaMine,伊布替尼中间体N-2

BTK Angiogenesis; Tyrosine Kinase/Adaptors
Ibrutinib deacryloylpiperidine (IBT4A) 是 Ibrutinib 的杂质之一。它是一种不可逆的、选择性的 Btk 抑制剂 (IC50:0.5 nM)。
T7788 2-Phenyl-2-(1-piperidinyl)propane

Others Others
2-Phenyl-2-(1-piperidinyl)propane 是一种具有可逆性、选择性的人 CYP2B6抑制剂,其 IC50为 5.1 μM,Ki 为 5.6。它对 CYP2D6 、CYP3A 均有抑制作用,且 IC50值分别为74 μM、200 μM。
T11894 Lusaperidone

R107474

Adrenergic Receptor GPCR/G Protein; Neuroscience
Lusaperidone (R107474) 是一种有效的α2肾上腺素受体 (adrenergic receptor) 拮抗剂,是 α (2)-肾上腺素受体的潜在放射性配体,对 α2A和α2C 具有抑制作用, Ki 值分别为0.13和0.15 nM。
T0351 Risperidone

Risperidal,R 64 766,利培酮

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; P-gp GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
Risperidone (R 64 766) 是5-HT2受体阻断剂、P-糖蛋白抑制剂和多巴胺 D2受体的拮抗剂,对 5-HT2A 和多巴胺 D2受体的 Ki 值分别为 4.8 和 5.9 nM。
T1539 Iloperidone

伊潘立酮,HP 873

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor GPCR/G Protein; Neuroscience
Iloperidone (HP 873) 是一种D2/5-HT2受体拮抗剂,是非典型抗精神病药,可治疗精神分裂症。
T14830 Bromperidol

溴哌利多,R-11333

5-HT Receptor GPCR/G Protein; Neuroscience
Bromperidol (R-11333) 是一种苯丁酮衍生物,是一种强效长效精神安定药。它被用作治疗精神分裂症的抗精神病药。
T28778 Silperisone HCl

RGH5002,SILA336,RGH-5002,Silperisone hydrochloride,SILA-336

Silperisone HCl (RGH-5002) 阻断细胞中的钠和钙通道,使肌肉细胞的兴奋度和收缩度降低,降低外周张力,充当肌肉松弛剂和外周血管扩张剂。 Silperisone HCl 可用于治疗脊髓损伤引起的复发性疼痛性肌阵挛、脑血管病引起的异常高肌张力、肌张力症状、锥体紧张综合征、多发性硬化症肌痉挛和脊髓炎。Silperisone 是钠通道蛋白2型α通道阻滞剂。Silperisone 是一种类似于tolperisone 的有机硅化合物,具有中枢作用的肌肉松弛剂特性。
T30077 Anisperimus

LF 150195,LF-150195,LF 15-0195,LF-15-0195,LF15-0195

Caspase Apoptosis; Proteases/Proteasome
Anisperimus (LF 15-0195) 是一种免疫抑制剂,通过促进 DISC 水平的 caspase-8 和 caspase-10 激活来增强激活诱导的 T 细胞死亡,通过促进表达 Foxp3 的调节性 CD4 T 细胞的发育来预防中枢神经系统自身免疫。
T9968 3-Piperidinyl(1-pyrrolidinyl)methanone hydrochloride

Others Others
3-Piperidinyl(1-pyrrolidinyl)methanone hydrochloride 可用于合成 MCH-R1 拮抗剂 piperidin-4-yl-urea 衍生物。
T26235 Sulfaperin

磺胺培林,Methylsulfadiazin,Archisulfa,Chemiopen,Demosulfan,Anastaf,Isosulfamerazine

Antibacterial Microbiology/Virology
Sulfaperin (Chemiopen) 是一种磺胺类抗菌剂。
T50083 12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide

Others Others
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide 可用作分子结构单元,用于多种化合物的合成。
T7843 4-phenoxypiperidine

Others Others
4-phenoxypiperidine 具有肌肉松弛和抗惊厥活性。
TP1220L Carperitide acetate

醋酸卡培立肽,Carperitide acetate (89213-87-6 Free base),Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate

Endothelin Receptor GPCR/G Protein
Carperitide acetate (Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate) 是一种由 28 个氨基酸组成的激素,由心脏产生并分泌,以响应心脏损伤和机械拉伸。Carperitide acetate 抑制内皮素-1 (endothelin-1) 分泌。
T62461 Benzyl-piperazine-CO-benzothiazole-4-methylpiperidine

Others Others
Benzyl-piperazine-CO-benzothiazole-4-methylpiperidine 可用于改变真核生物寿命。

化合物

Perifosine
Cat.No: T2492
Synonym: NSC 639966,D21266,KRX-0401,哌立福新
Target: Apoptosis, Akt, Autophagy
Perindoprilat
Cat.No: T1484
Synonym: Perindoprilate,培哚普利
Target: RAAS, MRP, AChR
Roluperidone
Cat.No: T15034
Synonym: CYR-101,MIN-101,MT-210
Target: Sigma receptor, 5-HT Receptor
Perindopril erbumine
Cat.No: T1484L
Synonym: 培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt
Target: Apoptosis, RAAS, MRP
BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride
Cat.No: T40111L
Synonym:
Target: PD-1/PD-L1
Droperidol
Cat.No: T0990
Synonym: 氟派利多,NSC 169874,Dehydrobenzperidol,氟哌啶
Target: Dopamine Receptor
Velneperit
Cat.No: T17222
Synonym: 韦利贝特,S2367
Target: Neuropeptide Y Receptor
Ethyl 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate
Cat.No: T66256
Synonym:
Target: Factor Xa
Tresperimus TFA
Cat.No: T34921L1
Synonym: Tresperimus TFA(160677-67-8 Free base)
Target: Others
4-(4-chlorophenyl)piperidin-4-ol
Cat.No: Fr13199
Synonym:
Target:
Domperidone
Cat.No: T0082
Synonym: R33812,多潘立酮
Target: Dopamine Receptor
3-​Phenyl-​N-​[1-​(phenylmethyl)​-​4-​piperidinyl]​-tricyclo[3.3.1.13,​7]​decane-​1-​carboxamide
Cat.No: T8501
Synonym:
Target: Influenza Virus
4-Bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione
Cat.No: T40018
Synonym:
Target: Others
Piperidolate
Cat.No: T7405
Synonym: 二苯哌酯,哌立度酯
Target: AChR
Haloperidol
Cat.No: T0025
Synonym: Aloperidin,氟哌啶醇,Serenace,Haldol
Target: Dopamine Receptor, 5-HT Receptor
Anisole-piperazine-methanone-benzothiazole-p-methylpiperidine
Cat.No: T77598
Synonym: (4-(4-methoxyphenyl)piperazin-1-yl)(2-(4-methylpiperidin-1-yl)benzo[d]thiazol-6-yl)methanone
Target: Others
Piperidolate hydrochloride
Cat.No: T7555
Synonym:
Target: AChR
Pericyazine
Cat.No: T16472
Synonym: Propericiazine,氰噻嗪,RP 8909
Target: Dopamine Receptor
1-Benzyl-4-hydroxypiperidine
Cat.No: Fr12729
Synonym: 1-Benzylpiperidin-4-ol
Target:
Abaperidone
Cat.No: T14083
Synonym:
Target: Dopamine Receptor, 5-HT Receptor
Anisperimus HCl
Cat.No: T30077L
Synonym: LF 150195 HCl,Anisperimus HCl(170368-04-4 Free base)
Target: Others
3-amino-1-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one dihydrochloride
Cat.No: T50072
Synonym:
Target: Others
5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione
Cat.No: T9361
Synonym: 5-bromo-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione
Target: Others
2-(2,6-dioxopiperidin-3-yl)-4-((7-hydroxyheptyl)oxy)isoindoline-1,3-dione
Cat.No: T9385
Synonym:
Target: Others
3-Morpholino-1-(4-(2-oxopiperidin-1-yl)phenyl)-5,6-dihydropyridin-2(1H)-one
Cat.No: T77687
Synonym:
Target: Others
4-benzyloxycarbonylamino-piperidine-1,4-dicarboxylic acid mono-tert-butyl ester
Cat.No: T64319
Synonym:
Target: Others
Thioquinapiperifil dihydrochloride
Cat.No: T9773
Synonym: KF-31327
Target: PDE
N-piperidine Ibrutinib hydrochloride
Cat.No: T12152
Synonym:
Target: BTK
Tolperisone hydrochloride
Cat.No: T0511
Synonym: 盐酸托哌酮,Muscalm,Midocalm,托哌酮盐酸盐,Tolperisone HCl
Target: Sodium Channel
Benproperine phosphate
Cat.No: T5007
Synonym: 磷酸苯丙哌林,Blascorid,Pirexyl phosphate
Target: Others, Microtubule Associated
Haloperidol decanoate
Cat.No: T25487
Synonym: KD 16,KD-136,KD 136,Neoperidole,Haldol
Target: Others
Benperidol
Cat.No: T26360
Synonym: R4584,R-4584,Anquil,McN-JR-4584,R 4584
Target:
Inaperisone
Cat.No: T68087
Synonym:
Target: Others
Ocaperidone
Cat.No: T3497
Synonym: 奥卡哌酮,Ocaperidona,R79598
Target: Dopamine Receptor, 5-HT Receptor
2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]amino}acetic acid
Cat.No: T50060
Synonym:
Target: Others
2-(2,6-dioxopiperidin-3-yl)-4-((9-hydroxynonyl)oxy)isoindoline-1,3-dione
Cat.No: T9386
Synonym:
Target: Others
Ibrutinib deacryloylpiperidine
Cat.No: T8636
Synonym: IBT4A,5-(4-phenoxyphenyl)-7H-pyrrolo[2,3-d]pyriMidin-4-ylaMine,伊布替尼中间体N-2
Target: BTK
2-Phenyl-2-(1-piperidinyl)propane
Cat.No: T7788
Synonym:
Target: Others
Lusaperidone
Cat.No: T11894
Synonym: R107474
Target: Adrenergic Receptor
Risperidone
Cat.No: T0351
Synonym: Risperidal,R 64 766,利培酮
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, P-gp
Iloperidone
Cat.No: T1539
Synonym: 伊潘立酮,HP 873
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Bromperidol
Cat.No: T14830
Synonym: 溴哌利多,R-11333
Target: 5-HT Receptor
Silperisone HCl
Cat.No: T28778
Synonym: RGH5002,SILA336,RGH-5002,Silperisone hydrochloride,SILA-336
Target:
Anisperimus
Cat.No: T30077
Synonym: LF 150195,LF-150195,LF 15-0195,LF-15-0195,LF15-0195
Target: Caspase
3-Piperidinyl(1-pyrrolidinyl)methanone hydrochloride
Cat.No: T9968
Synonym:
Target: Others
Sulfaperin
Cat.No: T26235
Synonym: 磺胺培林,Methylsulfadiazin,Archisulfa,Chemiopen,Demosulfan,Anastaf,Isosulfamerazine
Target: Antibacterial
12-oxo-N-[1-(propan-2-yl)piperidin-4-yl]-6H,7H,8H,9H,10H,12H-azepino[2,1-b]quinazoline-3-carboxamide
Cat.No: T50083
Synonym:
Target: Others
4-phenoxypiperidine
Cat.No: T7843
Synonym:
Target: Others
Carperitide acetate
Cat.No: TP1220L
Synonym: 醋酸卡培立肽,Carperitide acetate (89213-87-6 Free base),Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
Target: Endothelin Receptor
Benzyl-piperazine-CO-benzothiazole-4-methylpiperidine
Cat.No: T62461
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T2S1992 Perillartine

Perilla sugar,Peryllartine,紫苏葶,DL-Perillartine

Others; Endogenous Metabolite Metabolism; Others
Perillartine (DL-Perillartine) 是甜味剂,能够激活味觉受体 1 型成员 2 。
TN2054 Periplocymarin

Calcium Channel Membrane transporter/Ion channel; Metabolism
Periplocymarin 是一种强心苷,从 Periploca sepium 和 Periploca graeca 中分离得到,具有抗癌潜力。
TN2213 Imperialine 3-β-D-glucoside

Sipeimine-3-beta-D-glucoside,西贝母碱苷

Others Others
Imperialine 3-β-D-glucoside (Sipeimine-3-beta-D-glucoside) 是 Imperialine 的糖苷。它对多重耐药肿瘤细胞表现出抗肿瘤特性。
T5S1982 Periplocin

Periplocoside,杠柳毒苷

Apoptosis; Others Apoptosis; Others
Periplocin (Periplocoside) 是从黑龙骨中分离出的一种强心类固醇。它可促进肿瘤细胞凋亡并抑制肿瘤生长。它通过激活 Na/K-ATPase 介导的 Src/ERK 和 PI3K/Akt 途径,具有促进伤口愈合的潜力。
T4S1983 Periplogenin

5-beta-Hydroxydigitoxigenin,Desoxostrophanthidin,杠柳苷元

Others Others
Periplogenin (Desoxostrophanthidin) 是一种天然呋喃香豆素,存在于白芷根中,可以诱导脂肪细胞分化,具有高抗银屑病作用。
T6377 Aloperine

Apoptosis; Virus Protease; HIV Protease; Antibiotic; Autophagy Apoptosis; Autophagy; Microbiology/Virology; Proteases/Proteasome
Aloperine 是一种在苦参类植物中的生物碱,其具有抗癌,抗炎、抗肿瘤和抗病毒特性,可用于研究过敏性接触性皮炎湿疹和其他皮肤炎症。
T1035 Hesperidin

橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷

Apoptosis; Reactive Oxygen Species; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Metabolism; NF-κB
Hesperidin (Cirantin) 是一种广泛存在于柑橘类水果中黄烷酮糖苷,具有减少炎症介质并发挥重要的抗氧化作用,还有抗肿瘤和抗过敏活性。
T6S0923 Hypericin

Hypericine,金丝桃素,Cyclosan

Apoptosis; Antiviral; Influenza Virus; Tyrosine Kinases; Antibacterial; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Tyrosine Kinase/Adaptors
Hypericin (Cyclosan) 是贯叶连翘的提取物,有抗菌、抗病毒、抗肿瘤和抗抑郁作用。
T3S2381 Perillene

3-Isohexenylfuran,紫苏烯,Perillen

Others; Antibacterial Microbiology/Virology; Others
Perillene (3-Isohexenylfuran) 是促进肠蠕动的药物中的活性成分,它对金黄色葡萄球菌和大肠杆菌具有很强的抗药性。
TN2108 Protohypericin

Others Others
Protohypericin 是一种从贯叶连翘中提取的天然石脑粉。放射性碘化 Protohypericin 能用于肿瘤坏死靶向放射研究。
T0076 Paliperidone

9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Paliperidone (9-hydroxyrisperidone) 是 Risperidone 的主要活性代谢产物,是多巴胺 D2 拮抗剂和5-HT2A 拮抗剂。它用作非典型抗精神病药,用于精神分裂症的急性及维持治疗。它对α1和α2肾上腺素能受体和 H1组胺能受体也有拮抗作用。
T29756 1-piperoylpiperidine

AI3 01439,胡椒碱,AI3-01439,AI 3-01439,piperine

Others Others
1-piperoylpiperidine (AI3-01439) 是一种生化物质。
T0228 Methyl-Hesperidin

甲基橙皮甙

Akt; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling
Methyl hesperidin 是一种血管扩张剂。
T13495 3-Amino-2-piperidinone

Cyclo-ornithine

Endogenous Metabolite Metabolism
3-Amino-2-piperidinone 是来自生物体的代谢物,可用作环状鸟氨酸类似物。
T3314 Perillyl alcohol

Isocarveol,Perilla alcohol,紫苏醇

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
Perillyl alcohol (Isocarveol) 是一种单萜,可在不影响正常细胞的情况下诱导肿瘤细胞凋亡。
T2767 Neohesperidin Dihydrochalcone

NHDC,新橙皮苷二氢查尔酮,新橙皮苷二氢查耳酮,Neohesperidin DC,NCI-c60764

Reactive Oxygen Species Immunology/Inflammation; Metabolism; NF-κB
Neohesperidin Dihydrochalcone (Neohesperidin DC) 是一种合成的糖苷查耳酮,可用作低热量人造甜味剂,添加到各种食品和饮料中。
T6S0920 2"-O-Galloylhyperin

2”-O-没食子酰基金丝桃苷,2''-O-Galloylhyperin,Q-100605,FT-0689359

Others Others
2"-O-Galloylhyperin (FT-0689359) 是一种分离自Pyrola incarnateFisch. 中的活性化合物,具有抗氧化和抗炎作用,对氧化应激诱导的肝损伤具有肝保护作用。
T3002 Piperine

胡椒碱,1-Piperoylpiperidine,Bioperine

P450; Endogenous Metabolite; P-gp; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism; Neuroscience
Piperine (Bioperine) 是从胡椒中分离的一种生物碱,可以抑制P-糖蛋白和 CYP3A4 的活性,在HeLa 细胞中的IC50值为61.94±0.054 μg/mL。它已用于研究治疗多发性骨髓瘤和吞咽障碍的试验。
T8282 (S)-(−)-Perillyl alcohol

Perillyl alcohol,(-)-Perillyl Alcohol,L-紫苏醇

Apoptosis; Endogenous Metabolite Apoptosis; Metabolism
(S)-(−)-Perillyl alcohol (Perillyl alcohol) 是一种在薰衣草中发现的单萜,可抑制 Ras 的法尼基化,上调 6-磷酸甘露糖受体并诱导细胞凋亡。 它还具有抗癌活性。
T5786 TETRAHYDROPIPERINE

四氢胡椒碱,Cosmoperine

P450; TRP/TRPV Channel Membrane transporter/Ion channel; Metabolism
Tetrahydropiperine (Cosmoperine) 是胡椒碱的环己基类似物,也是一种天然芳基戊酰胺,从Piper longum 分离得到。它对细胞色素 P450 (CYP) 同工型 CYP1A1/芳基烃羟化酶 (AHH;IC50=23 µM)具有抑制作用。
T8256 piperitone

胡椒酮,3甲基-6-(1-甲基乙基)-2-环己烯-1-酮

Others Others
Piperitone 是强大的驱虫剂和抗食欲剂。它对 Cymbopogon schoenanthus(C. schoenanthus) 成虫、新产卵和新生幼虫有很大的毒性。
TN1819 Kaempferol 3-neohesperidoside

Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷

GSK-3; MEK; PI3K MAPK; PI3K/Akt/mTOR signaling; Stem Cells
Kaempferol 3-neohesperidoside (Kaempferol 3-O-neohesperidoside) 是一种类黄酮,对大鼠比目鱼肌具有拟胰岛素作用。
T2737 Neohesperidin

Hesperetin 7-O-neohesperidoside,NSC 31048,新橙皮苷

Antioxidant oxidation-reduction
Neohesperidin (NSC-31048) 是一种类黄酮化合物,存在于葫芦科植物中,具有抗氧化和抗炎活性。
TN1164 1-(3,4-Dimethoxycinnamoyl)piperidine

Others Others
1-(3,4-Dimethoxycinnamoyl)piperidine is a natural product
T9112 (-)-Perillaldehyde

AhR; ROS; Nrf2 Immunology/Inflammation; Metabolism
L-Perillaldehyde 是紫苏草精油的主要成分,吸入后经由嗅觉神经功能表现出抗抑郁功能。
TN2055 Periplogenin 3-[O-β-glucopyranosyl-(1→4)-β-sarmentopyranoside]

4)-beta-sarmentopyranoside]'>Periplogenin 3-[O-beta-glucopyranosyl-(1->4)-beta-sarmentopyranoside],异杠柳毒苷

Others Others
Periplogenin 3-[O-beta-glucopyranosyl-(1->4)-beta-sarmentopyranoside] is a natural product from Periploca sepiumBge.
TN2109 Protopseudohypericin

Others Others
Protopseudohypericin is a natural product
TN5312 Periplocogenin

Periplocogenin 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5312,CAS号为 112899-63-5。
TN4751 Periglaucine B

HBV Microbiology/Virology
Periglaucine B can inhibit hepatitis B virus (HBV) surface antigen (HBsAg) secretion in Hep G2.2.15 cells.
TN1044 Quercetin 3-O-neohesperidoside

Others Others
Quercetin 3-O-neohesperidoside shows anti-atherosclerosis, and antiplatelet aggregation activities.
T40252 Peritassine A

Peritassine A, an alkaloid derived from Tripterygium wilfordii Hook. f., exhibits anti-HIV properties.
T40640 Glycoperine

Glycoperine is a alkaloid from haplophyllum perforatum.
TN2758 2-Ethyl-2,6,6-trimethylpiperidin-4-one

Others Others
2-Ethyl-2,6,6-trimethylpiperidin-4-one 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN2758,CAS号为 133568-79-3。
TN4148 Glyasperin C

Tyrosinase; Antifection Microbiology/Virology; Proteases/Proteasome
Glyasperin C acts as a partial estrogen antagonist, it shows tyrosinase inhibitory activity (IC (50) = 0.13 +/- 0.01 microg/mL), it could be a promising candidate in the design of skin-whitening agents. Glyasperin C shows potent anti-vancomycin-resistant
TN4750 Periglaucine A

HBV Microbiology/Virology
Periglaucine A inhibits hepatitis B virus (HBV) surface antigen (HBsAg) secretion in Hep G2.2.15 cells.
TN4372 Kaempferol-7-O-neohesperidoside

Others Others
Kaempferol-7-O-neohesperidoside 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4372,CAS号为 17353-03-6。
T83353 3'-Methoxy-3,5,4'-trihydroxyflavone-7-neohesperidoside

3'-Methoxy-3,5,4'-triHydroxyflavone-7-neheesperidoside,一种从Cleome droserifolia中分离的黄酮类化合物,显示出中等程度的保肝活性。
TN4825 Prenylpiperitol

Others Others
Prenylpiperitol是一种天然产物,属于芸香科石南芸木属,其产品编号为 TN4825,CAS号为 157659-20-6。Prenylpiperitol可用作对照参考。
TN2056 Perisesaccharide B

Others Others
Perisesaccharide B is a natural product
TN4149 Glyasperin F

Others Others
Glyasperin F has antinociceptive, and anti-inflammatory effects, it could inhibit NO production in RAW 264.7 macrophages to some extent. Glyasperin F displayed cytotoxic effects against the four tested cancer cell lines with IC50values below 85 μM.
TN3806 Dehydroglyasperin C

ERK; IκB/IKK; p38 MAPK; TNF; NF-κB; Akt; COX; PI3K; NADPH; DNA/RNA Synthesis; Nrf2; JNK; Autophagy Apoptosis; Autophagy; Cell Cycle/Checkpoint; Cytoskeletal Signaling; DNA Damage/DNA Repair; Immunology/Inflammation; MAPK; Metabolism; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling
Dehydroglyasperin C is a potent NAD(P)H:oxidoquinone reductase (NQO1) and phase 2 enzyme inducer. Dehydroglyasperin C possesses potent antioxidant, cancer chemopreventive, and neuroprotective activities, it has protective effects against chronic diseases
TN4147 Glyasperin A

Others Others
Glyasperin A has cytotoxic properties against P-388 cells, its IC50 values being 6.0 microM.
T4110 Perivine

Perivin,派利文碱

Others Others
Perivine (Perivin) 以视网膜母细胞瘤相关蛋白 (RbAp48) 为靶点,能够解决 RbAp48-FOG-1 复合物的不稳定性。Perivine 可用于研究阿尔茨海默病。
T7980 Hesperidin methylchalcone

NF-κB NF-κB
Hesperidin methylchalcone 抑制氧化应激,细胞因子产生和NF-κB 活化。它能够抑制炎症和疼痛,具有血管保护作用。
TN7049 6''-Acetylhyperin

6''-Acetylhyperin 在生命科学相关研究中具有广泛的应用。
TN3810 Dehydroperilloxin

COX Immunology/Inflammation; Neuroscience
Dehydroperilloxin possesses inhibitory activity against cyclooxygenase-1, with the IC(50) value of 30.4 microM.
TN2052 Periplocoside M

Others Others
Periplocoside M possesses observably antitumor activity against SMMC-7721( IC 50=12.9 ng/L),Hela( IC 50=8.63 ng/L) and MCF-7( IC 50=18.5 ng/L) cancer cell lines.
TN5315 Periplocoside F

Periploside F

Periplocoside F 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5315,CAS号为 119902-17-9。
TN2084 Piperitol

Others Others
Piperitol has in vitro antioxidant potential, it also exhibits a stronger CNS depressant effect than that of M. rotundifolia.
TN1356 Acetyl Perisesaccharide C

乙酰杠柳寡糖 C,乙酰杠柳寡糖C

Others Others
Acetyl Perisesaccharide C is a natural product
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天然产物

Perillartine
Cat.No: T2S1992
Synonym: Perilla sugar,Peryllartine,紫苏葶,DL-Perillartine
Target: Others, Endogenous Metabolite
Periplocymarin
Cat.No: TN2054
Synonym:
Target: Calcium Channel
Imperialine 3-β-D-glucoside
Cat.No: TN2213
Synonym: Sipeimine-3-beta-D-glucoside,西贝母碱苷
Target: Others
Periplocin
Cat.No: T5S1982
Synonym: Periplocoside,杠柳毒苷
Target: Apoptosis, Others
Periplogenin
Cat.No: T4S1983
Synonym: 5-beta-Hydroxydigitoxigenin,Desoxostrophanthidin,杠柳苷元
Target: Others
Aloperine
Cat.No: T6377
Synonym:
Target: Apoptosis, Virus Protease, HIV Protease, Antibiotic, Autophagy
Hesperidin
Cat.No: T1035
Synonym: 橙皮甙,Hesperetin 7-rutinoside,Cirantin,橙皮苷
Target: Apoptosis, Reactive Oxygen Species, Endogenous Metabolite, Autophagy
Hypericin
Cat.No: T6S0923
Synonym: Hypericine,金丝桃素,Cyclosan
Target: Apoptosis, Antiviral, Influenza Virus, Tyrosine Kinases, Antibacterial, PKC
Perillene
Cat.No: T3S2381
Synonym: 3-Isohexenylfuran,紫苏烯,Perillen
Target: Others, Antibacterial
Protohypericin
Cat.No: TN2108
Synonym:
Target: Others
Paliperidone
Cat.No: T0076
Synonym: 9-羟基利培酮,帕潘立酮,9-hydroxyrisperidone
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
1-piperoylpiperidine
Cat.No: T29756
Synonym: AI3 01439,胡椒碱,AI3-01439,AI 3-01439,piperine
Target: Others
Methyl-Hesperidin
Cat.No: T0228
Synonym: 甲基橙皮甙
Target: Akt, PKC
3-Amino-2-piperidinone
Cat.No: T13495
Synonym: Cyclo-ornithine
Target: Endogenous Metabolite
Perillyl alcohol
Cat.No: T3314
Synonym: Isocarveol,Perilla alcohol,紫苏醇
Target: Apoptosis, Endogenous Metabolite
Neohesperidin Dihydrochalcone
Cat.No: T2767
Synonym: NHDC,新橙皮苷二氢查尔酮,新橙皮苷二氢查耳酮,Neohesperidin DC,NCI-c60764
Target: Reactive Oxygen Species
2"-O-Galloylhyperin
Cat.No: T6S0920
Synonym: 2”-O-没食子酰基金丝桃苷,2''-O-Galloylhyperin,Q-100605,FT-0689359
Target: Others
Piperine
Cat.No: T3002
Synonym: 胡椒碱,1-Piperoylpiperidine,Bioperine
Target: P450, Endogenous Metabolite, P-gp, Autophagy
(S)-(−)-Perillyl alcohol
Cat.No: T8282
Synonym: Perillyl alcohol,(-)-Perillyl Alcohol,L-紫苏醇
Target: Apoptosis, Endogenous Metabolite
TETRAHYDROPIPERINE
Cat.No: T5786
Synonym: 四氢胡椒碱,Cosmoperine
Target: P450, TRP/TRPV Channel
piperitone
Cat.No: T8256
Synonym: 胡椒酮,3甲基-6-(1-甲基乙基)-2-环己烯-1-酮
Target: Others
Kaempferol 3-neohesperidoside
Cat.No: TN1819
Synonym: Kaempferol 3-O-neohesperidoside,堪非醇 3-新橙皮糖苷
Target: GSK-3, MEK, PI3K
Neohesperidin
Cat.No: T2737
Synonym: Hesperetin 7-O-neohesperidoside,NSC 31048,新橙皮苷
Target: Antioxidant
1-(3,4-Dimethoxycinnamoyl)piperidine
Cat.No: TN1164
Synonym:
Target: Others
(-)-Perillaldehyde
Cat.No: T9112
Synonym:
Target: AhR, ROS, Nrf2
Periplogenin 3-[O-β-glucopyranosyl-(1→4)-β-sarmentopyranoside]
Cat.No: TN2055
Synonym: 4)-beta-sarmentopyranoside]'>Periplogenin 3-[O-beta-glucopyranosyl-(1->4)-beta-sarmentopyranoside],异杠柳毒苷
Target: Others
Protopseudohypericin
Cat.No: TN2109
Synonym:
Target: Others
Periplocogenin
Cat.No: TN5312
Synonym:
Target:
Periglaucine B
Cat.No: TN4751
Synonym:
Target: HBV
Quercetin 3-O-neohesperidoside
Cat.No: TN1044
Synonym:
Target: Others
Peritassine A
Cat.No: T40252
Synonym:
Target:
Glycoperine
Cat.No: T40640
Synonym:
Target:
2-Ethyl-2,6,6-trimethylpiperidin-4-one
Cat.No: TN2758
Synonym:
Target: Others
Glyasperin C
Cat.No: TN4148
Synonym:
Target: Tyrosinase, Antifection
Periglaucine A
Cat.No: TN4750
Synonym:
Target: HBV
Kaempferol-7-O-neohesperidoside
Cat.No: TN4372
Synonym:
Target: Others
3'-Methoxy-3,5,4'-trihydroxyflavone-7-neohesperidoside
Cat.No: T83353
Synonym:
Target:
Prenylpiperitol
Cat.No: TN4825
Synonym:
Target: Others
Perisesaccharide B
Cat.No: TN2056
Synonym:
Target: Others
Glyasperin F
Cat.No: TN4149
Synonym:
Target: Others
Dehydroglyasperin C
Cat.No: TN3806
Synonym:
Target: ERK, IκB/IKK, p38 MAPK, TNF, NF-κB, Akt, COX, PI3K, NADPH, DNA/RNA Synthesis, Nrf2, JNK, Autophagy
Glyasperin A
Cat.No: TN4147
Synonym:
Target: Others
Perivine
Cat.No: T4110
Synonym: Perivin,派利文碱
Target: Others
Hesperidin methylchalcone
Cat.No: T7980
Synonym:
Target: NF-κB
6''-Acetylhyperin
Cat.No: TN7049
Synonym:
Target:
Dehydroperilloxin
Cat.No: TN3810
Synonym:
Target: COX
Periplocoside M
Cat.No: TN2052
Synonym:
Target: Others
Periplocoside F
Cat.No: TN5315
Synonym: Periploside F
Target:
Piperitol
Cat.No: TN2084
Synonym:
Target: Others
Acetyl Perisesaccharide C
Cat.No: TN1356
Synonym: 乙酰杠柳寡糖 C,乙酰杠柳寡糖C
Target: Others
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Cat. No. Product Name Species Expression System
TMPY-01613 Periostin/OSF-2 Protein, Mouse, Recombinant (His)

A630052E07Rik,OSF-2,Osf2,PLF,AI747096,peri,PN,p...

Mouse HEK293 Cells
Periostin/OSF-2 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 89 kDa and the accession number is Q62009-2.
TMPY-01020 Periostin/OSF-2 Protein, Human, Recombinant (His)

PN,OSF-2,OSF2,periostin,periostin, osteobl...

Human HEK293 Cells
Periostin/OSF-2 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 86.4 kDa and the accession number is Q15063-3.
TMPK-01032 Periostin/OSF-2 Protein, Mouse, Recombinant (aa 24-811, His)

POSTN,OSF2,Periostin,TRIF52,PNRP11-412K4.1,PN,Fasci...

Mouse HEK293 Cells
Periostin/OSF-2 Protein, Mouse, Recombinant (aa 24-811, His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 88.7 kDa and the accession number is Q62009-1.
TMPK-00973 Periostin/OSF-2 Protein, Human, Recombinant (aa 22-836, His)

Periostin,POSTN,Fasciclin I-like,TRIF52,OSF-2,PNRP1...

Human HEK293 Cells
Periostin/OSF-2 Protein, Human, Recombinant (aa 22-836, His) is expressed in HEK293 mammalian cells with C-His tag. The predicted molecular weight is 92.1 kDa and the accession number is Q15063.
TMPY-05190 Per a 1 Protein, Periplaneta americana, Recombinant (His)

Periplaneta americana E. coli
Per a 1 Protein, Periplaneta americana, Recombinant (His) is expressed in E. coli expression system with His tag. The predicted molecular weight is 27.2 kDa and the accession number is Q9TZR6.
TMPY-04853 TSHR Protein, Human, Recombinant (His)

TSHR,hTSHR-I,TSH Receptor,LGR3,CHNG1

Human Baculovirus Insect Cells
Thyroid-stimulating hormone (TSH) is secreted by the pituitary gland and promotes thyroid growth and function, with increased TSH levels typically associated with hypothyroidism. Immunohistochemical analysis revealed predominantly nuclei/peri-nuclei localization of TSHR in cancerous tissues but cell membrane localization in non-cancerous parts. Overexpression of TSHR was found in a great majority of HCC tissues and associated with unfavorable prognosis.

重组蛋白

Periostin/OSF-2 Protein, Mouse, Recombinant (His)
Cat.No: TMPY-01613
Species: Mouse
Expression System: HEK293 Cells
Periostin/OSF-2 Protein, Human, Recombinant (His)
Cat.No: TMPY-01020
Species: Human
Expression System: HEK293 Cells
Periostin/OSF-2 Protein, Mouse, Recombinant (aa 24-811, His)
Cat.No: TMPK-01032
Species: Mouse
Expression System: HEK293 Cells
Periostin/OSF-2 Protein, Human, Recombinant (aa 22-836, His)
Cat.No: TMPK-00973
Species: Human
Expression System: HEK293 Cells
Per a 1 Protein, Periplaneta americana, Recombinant (His)
Cat.No: TMPY-05190
Species: Periplaneta americana
Expression System: E. coli
TSHR Protein, Human, Recombinant (His)
Cat.No: TMPY-04853
Species: Human
Expression System: Baculovirus Insect Cells
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