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263

抑制剂 & 化合物

59

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Cat. No. Product Name Target Signaling Pathways
T22605 Bifemelane hydrochloride

MAO; Monoamine Oxidase Metabolism; Neuroscience
Bifemelane hydrochloride 是一种选择性的,有效的,和竞争性的单胺氧化酶A (MAO-A)抑制剂,Ki=4.20 μM,它也非竞争性地抑制MAO-B,Ki=46.0 μM。它具有显著的抗抑郁作用,可用于研究与脑血管疾病有关的认知和情绪障碍。
T0084 Moclobemide

吗氯贝胺,Ro111163

MAO; Monoamine Oxidase Metabolism; Neuroscience
Moclobemide (Ro111163) 是可逆的、可透过血脑屏障的单胺氧化酶 (MAO-A) 抑制剂,能够抑制 hMAO-A (IC50=6.061 μM)。它上调慢性应激小鼠海马祖细胞的增殖。
T7048 1,4-Naphthoquinone

α-Naphthoquinone,Naphthalene-1,4-Dione,P-Naphthoquinone,1,4-萘醌,para-naphthoquinone

Others; MAO; Topoisomerase DNA Damage/DNA Repair; Metabolism; Neuroscience; Others
1,4-Naphthoquinone (P-Naphthoquinone) 被用作单胺氧化酶和 DNA 拓扑异构酶活性的潜在抑制剂,还用于抑制乙酰转移酶活性。
T6073 OG-L002

Histone Demethylase; Monoamine Oxidase; HSV Chromatin/Epigenetic; Microbiology/Virology; Neuroscience
OG-L002 是一种高度选择性的 LSD1有效抑制剂,IC50为 0.02 μM。它抑制HSV IE 基因的表达,还是单胺氧化酶抑制剂,对 MAO-A 和 MAO-B 的IC50分别为 1.38 μM 和 0.72 μM。
T0006 Methylene Blue trihydrate

碱性亚甲蓝三水合物,Methylthionine chloride,Basic blue 9,亚甲蓝三水合物,Methylene Blue

Guanylate cyclase; Microtubule Associated; NO Synthase; Parasite; Monoamine Oxidase Cytoskeletal Signaling; GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience
Methylene Blue trihydrate (Basic blue 9) 是鸟苷酸环化酶,单胺氧化酶 A 和 NO 合酶抑制剂。它是血管加压药,在医疗中通常用作染料。它具有抗伤害感受,抗疟疾,抗抑郁和抗焦虑作用,可用于高铁血红蛋白血症,神经退行性疾病和异环磷酰胺引起的脑病的研究。
T78984 Xanthine oxidase-IN-10

XO8 analog

ROS Immunology/Inflammation
Xanthine oxidase-IN-10 (XO8 analog) 是一种黄嘌呤氧化酶 (XO) 抑制剂,可用于研究痛风。
T0692 Allopurinol

Zyloric,别嘌醇,Zyloprim,Lopurin,别嘌呤醇

ROS; Xanthine Oxidase Immunology/Inflammation; Metabolism
Allopurinol (Zyloric) 是一种黄嘌呤氧化酶(XO)抑制剂,IC50=7.82±0.12 μM。
T67850 FCE 28073

MAO Metabolism; Neuroscience
FCE 28073是一种 Monoamine oxidase B 抑制剂,IC50=0.45 μM。
T10509 Xanthine oxidase-IN-1

4-(3-Cyano-5,6-difluoroindol-1-yl)-2-hydroxybenzoic acid

Xanthine Oxidase Metabolism
Xanthine oxidase-IN-1是一种有效的黄嘌呤氧化酶抑制剂(IC50值:6.5 nM),是一种利用核酸和核苷酸介质降解产生的生物活性核苷酸在嘌呤分解代谢中起核心作用的化合物,
T20719 Oxadiargyl

RP 020630,RP-020630,RP020630,丙炔恶草酮,Topstar

Others Others
Oxadiargyl (RP020630) 是原卟啉原氧化酶抑制剂,在我国被用作除草剂。
T0773 Febuxostat

非布索坦,TMX 67,非布司他,TEI 6720

ROS; Xanthine Oxidase Immunology/Inflammation; Metabolism
Febuxostat (TEI 6720) 是一种选择性黄嘌呤氧化酶(XO)抑制剂,Ki=0.6 nM。
T6376 Allopurinol Sodium

1H-吡唑并[3,4-D]嘧啶-4-醇单钠盐,Allopurinol sodium salt,Sodium allopurinol

ROS Immunology/Inflammation
Allopurinol Sodium 是黄嘌呤氧化酶抑制剂,其IC50= 0.2~50 μM。它能够抗利什曼原虫,也可用于研究痛风以及高尿酸血症。
T67789 Bazinaprine

MAO Metabolism; Neuroscience
Bazinaprine 是一种选择性的、可逆的单胺氧化酶抑制剂(MAOI),是治疗抑郁症的候选化合物。Bazinaprine 对A 型单胺氧化酶显示出较强的抑制作用,对b 型单胺氧化酶只显示出较弱的抑制作用。Bazinaprine 在体内可逆,但在体外不可逆。
T38863 Luvadaxistat

TAK-831,Luvadaxistat

TAK-831 is a potent and highly selective inhibitor of D-amino acid oxidase (DAAO), offering great potential for utilization in schizophrenia research.
T20622 Fomesafen

氟磺胺草醚,PP021,PP-021,PP 021

Others Others
Fomesafen (PP-021) 是原卟啉原 IX 氧化酶的选择性抑制剂。Fomesafen (PP-021) 用作除草剂,具有低毒性和高选择性的优点。
T10079 MAO-IN-1

MAO Metabolism; Neuroscience
MAO-IN-1是一种高效的单胺氧化酶B (MAO B)抑制剂(IC50:20 nM),可用于研究神经系统相关疾病。
T38655 Trifludimoxazin

Others Others
Trifludimoxazin 可用作除草剂,是一种原卟啉原氧化酶的抑制剂。
T8567 amflutizole

Xanthine Oxidase Metabolism
amflutizole 用于治疗痛风,是一种黄嘌呤氧化酶抑制剂。
T5206 DAAO inhibitor-1

Others Others
DAAO inhibitor-1是 D-氨基酸氧化酶抑制剂(IC50:0.12 μM)。
T0821 Iproniazid Phosphate

磷酸异丙烟肼,Isoproniazid phosphate

MAO; Monoamine Oxidase Metabolism; Neuroscience
Iproniazid Phosphate 是一种非选择性的,不可逆的单胺氧化酶抑制剂,具有抗抑郁作用。
T5053 Eprobemide

LIS 630,依普贝胺

MAO; Monoamine Oxidase Metabolism; Neuroscience
Eprobemide (LIS 630) 是一种非竞争性的、可逆的单胺氧化酶 A 抑制剂。
T0300 Pargyline

Pargylamine,Paragyline,优降宁

MAO; Monoamine Oxidase Metabolism; Neuroscience
Pargyline (Pargylamine) 是不可逆的单胺氧化酶抑制剂,对MAO-A 和MAO-B 的Ki 分别为 13 μM 和 0.5 μM,具有降压和抗癌作用。
T5323 Toloxatone

托洛沙酮,MD 69276

MAO; Monoamine Oxidase Metabolism; Neuroscience
Toloxatone (MD 69276) 是可逆的单胺氧化酶 A (MAOA) 抑制剂,是一种抗抑郁剂。
T39280 Nitrofen

Others Others
Nitrofen 是选择性接触除草剂,也是视原卟啉原氧化酶和网膜脱氢酶抑制剂。
T6099 Setanaxib

GKT137831

NADPH-oxidase; Ferroptosis; NADPH Apoptosis; Immunology/Inflammation; Metabolism
Setanaxib (GKT137831) 是一种有效的特异性双重 NADPH 氧化酶 (NOX1/4) 抑制剂,Ki 分别为140和110nM。
T1117 Clorgyline hydrochloride

盐酸氯吉林,Clorgiline hydrochloride,N-[3-(2,4-二氯苯氧基)丙基]-N-甲基-2-丙炔胺盐酸盐

MAO; Monoamine Oxidase Metabolism; Neuroscience
Clorgyline hydrochloride (Clorgiline hydrochloride) 是一种选择性、不可逆的单胺氧化酶A 抑制剂,结构上与Pargyline 相关。
T15023 CX-157

KP 157

MAO Metabolism; Neuroscience
CX-157 (KP 157) 是一种新型单胺氧化酶-A(MAO-A)抑制剂,可用于研究抑郁症类的神经系统疾病和癌症。
T77564 Coumarin102

Exciton 480

Coumarin102 (Exciton 480)是一种荧光染料。Coumarin102对Monoamine oxidase B、MAO-B和MAO-A具有较弱的抑制活性,可用来研究神经系统疾病。
T16803 RS 8359

MAO Metabolism; Neuroscience
RS 8359 是单胺氧化酶 A (MAO-A) 的可逆抑制剂,对 A:B 酶类型的特异性比约为 2200。 RS 8359 具有抗抑郁活性。
T0358 Aminoguanidine hydrochloride

Imino semicarbazide,Pimagedine hydrochloride,CP-12009-18 tartrate,Hydrazinecarboximidamide,肼甲酰亚胺酰胺一氯化氢(氨基胍盐酸盐),氨基胍盐酸盐,Guanyl hydrazine,Pimagedine

NOS; NO Synthase Immunology/Inflammation
Aminoguanidine hydrochloride (Hydrazinecarboximidamide) 是二胺氧化酶抑制剂,也是一氧化氮合酶抑制剂,可用于糖尿病肾病的研究。
T24444 Medifoxamine

LG 152,Medifoxamina,LG-152,LG152

Dopamine Receptor; Monoamine Oxidase GPCR/G Protein; Neuroscience
Medifoxamine (LG 152) 是一种选择性非单胺氧化酶抑制剂,通过对5 HT 再摄取的抑制展现其抗抑郁活性。Medifoxamine 优先抑制多巴胺再摄取 (dopamine reuptake)。
T24680 PSB-1491

MAO Metabolism; Neuroscience
PSB-1491 是一种选择性和竞争性的单胺氧化酶 B 抑制剂,IC50 为 0.386 nM,是 MAO-A 的 25000 倍以上。
T4559 Isocarboxazid

Monoamine Oxidase Neuroscience
Isocarboxazid 是不可逆的、非选择性的单胺氧化酶 monoamine oxidase 抑制剂,其在大鼠大脑中测得的 IC50值为4.8 μM。
T22965 MDL 72527

N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride

Others Others
MDL 72527 (N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride) 是一种多胺氧化酶 (POA) 抑制剂
T22304 Desciclovir

BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV

Antifection Microbiology/Virology
Desciclovir (DCV) 是抗疱疹药物阿昔洛韦的前药,口服有活性,在体内被黄嘌呤氧化酶转化成为阿昔洛韦。
T12441 Phenelzine sulfate

硫酸苯乙肼,苯肼,硫酸盐

Monoamine Oxidase Neuroscience
Phenelzine sulfate 是一种非选择性的、不可逆的单胺氧化酶抑制剂 (MAOI),可用作抗抑郁药和抗焦虑药。
T8124 Sodium benzoate

Benzoic acid sodium salt,苯甲酸钠

Others Others
Sodium benzoate (Benzoic acid sodium salt) 是一种 D-氨基酸氧化酶抑制剂。它是一种食品防腐剂。
T24679 PSB-1434

PSB 1434,PSB1434

MAO Metabolism; Neuroscience
PSB-1434 是一种选择性和竞争性的单胺氧化酶 B 抑制剂,IC50 为 1.59 nM,相对于 MAO-A 的选择性>6000 倍。
T1025 Tranylcypromine (2-PCPA) hydrochloride

反苯环丙胺盐酸盐,Tranylcypromine (2-PCPA) HCl,SKF-385 HCl

Histone Demethylase; MAO Chromatin/Epigenetic; Metabolism; Neuroscience
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl) 是一种单胺氧化酶抑制剂,对治疗重度抑郁症、心境恶劣障碍和非典型抑郁症有效。
T60625 Tigulixostat

Tigulixostat 是吲哚基杂芳羧酸的新型衍生物。Tigulixostat 是一种非嘌呤选择性的黄嘌呤氧化酶抑制剂,可降低尿酸的生成。
T0948 Adrenalone hydrochloride

Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮

Adrenergic Receptor GPCR/G Protein; Neuroscience
Adrenalone hydrochloride (Adrenalone HCl) 是一种多巴胺β氧化酶 (dopamine β oxidase) 抑制剂,结构与去甲肾上腺素转运蛋白 (NET) 配体相似,IC50=36.9 μM。它是一种肾上腺素能 (adrenergic) 激动剂,用作局部血管收缩剂和止血剂。
T1578 Pargyline hydrochloride

优降宁盐酸盐,Pargylamine hydrochloride

MAO; Monoamine Oxidase Metabolism; Neuroscience
Pargyline hydrochloride (Pargylamine hydrochloride) 是不可逆的单胺氧化酶抑制剂,可作用于 MAO-A (Ki=13 μM) 和 MAO-B (Ki=0.5 μM) ,具有降压和抗癌作用。
TP1886L1 NoxA1ds acetate(1435893-78-9 free base)

NADPH-oxidase Immunology/Inflammation
NoxA1ds acetate(1435893-78-9 free base) 是一种有效的选择性 NADPH 氧化酶 1 (NOX1) 抑制剂 (IC50 : 20 nM)。对 NOX1 的选择性优于对 NOX2、NOX4、NOX5 和黄嘌呤氧化酶的选择性。它抑制 HT-29 人结肠癌细胞中 NOX1 衍生的 O2 产生。在体外缺氧条件下减弱 VEGF 诱导的人肺动脉内皮细胞迁移。
T83625 iNOS-IN-14

3-bromo-1H-indazole-7-carbonitrile

NOS Immunology/Inflammation
iNOS-IN-14 (3-bromo-1H-indazole-7-carbonitrile) 是一种有效的一氧化氮合酶(NOS)抑制剂,抑制nNOS的NADPH氧化酶活性。
T77615 ND-011992

ND011992

Mitochondrial Metabolism; Antibacterial Metabolism; Microbiology/Virology
ND-011992 是一种靶向醌还原酶 (quinone reductases) 和醌氧化酶 (quinol oxidases)的喹唑啉类抑制剂,具有可逆性和选择性。ND-011992 对大肠杆菌 BL21*Δcyo 呼吸复合体I (respiratory complex I) 、 bo3 氧化酶(bo3 oxidase)、 bd-I 氧化酶 (bd-I oxidases) 和 bd-II 氧化酶 (bd-II oxidases)具有抑制作用,IC50 分别为 0.12、2.47、0.63 和 1.3 μM。ND-011992 可以用于研究肺结核。
T29097 VAS 3947

VA-S3947,VA S3947,VAS3947

Apoptosis; NADPH-oxidase Apoptosis; Immunology/Inflammation
VAS 3947 是一种特异的 NADPH 氧化酶 (NOX) 抑制剂。VAS 3947具有强大的抗血小板作用, 通过 UPR 激活,主要由于蛋白质聚集和错误折叠,独立于抗 NOX 活性诱导细胞凋亡。
T0235 Modaline sulfate

MAO; Monoamine Oxidase Metabolism; Neuroscience
Modaline sulfate 是一种 MAO 抑制剂,用于研究抑郁症。
T7942 Tranylcypromine hemisulfate

Tranylcypromine Sulfate,Tranylcypromine (hemisulfate),反苯环丙胺半硫酸盐

Histone Demethylase; MAO; Monoamine Oxidase Chromatin/Epigenetic; Metabolism; Neuroscience
Tranylcypromine hemisulfate (Tranylcypromine Sulfate) 是单胺氧化酶(MAO) 和赖氨酸特异性去甲基化酶 1 (LSD1) 的抑制剂,可用于研究抑郁症和子宫内膜异位症。
T2397 Topiroxostat

托匹司他,FYX-051

P450; ROS; Xanthine Oxidase Immunology/Inflammation; Metabolism
Topiroxostat (FYX-051) 是一种有效的口服黄嘌呤氧化还原酶 (XOR) 抑制剂,IC50=5.3 nM,Ki=5.7 nM。它还表现出弱的CYP3A4抑制活性 (18.6%)。它有用于高尿酸血症的研究潜力。
T19533 Pyraclonil

Others Others
Pyraclonil 作为一种除草剂,有效地控制了敏感型(S)和多重抗药性(MHR)E. indica群体。Pyraclonil 作为丙啶类光 敏色素原氧化酶(PPO)抑制剂发挥作用。

化合物

Bifemelane hydrochloride
Cat.No: T22605
Synonym:
Target: MAO, Monoamine Oxidase
Moclobemide
Cat.No: T0084
Synonym: 吗氯贝胺,Ro111163
Target: MAO, Monoamine Oxidase
1,4-Naphthoquinone
Cat.No: T7048
Synonym: α-Naphthoquinone,Naphthalene-1,4-Dione,P-Naphthoquinone,1,4-萘醌,para-naphthoquinone
Target: Others, MAO, Topoisomerase
OG-L002
Cat.No: T6073
Synonym:
Target: Histone Demethylase, Monoamine Oxidase, HSV
Methylene Blue trihydrate
Cat.No: T0006
Synonym: 碱性亚甲蓝三水合物,Methylthionine chloride,Basic blue 9,亚甲蓝三水合物,Methylene Blue
Target: Guanylate cyclase, Microtubule Associated, NO Synthase, Parasite, Monoamine Oxidase
Xanthine oxidase-IN-10
Cat.No: T78984
Synonym: XO8 analog
Target: ROS
Allopurinol
Cat.No: T0692
Synonym: Zyloric,别嘌醇,Zyloprim,Lopurin,别嘌呤醇
Target: ROS, Xanthine Oxidase
FCE 28073
Cat.No: T67850
Synonym:
Target: MAO
Xanthine oxidase-IN-1
Cat.No: T10509
Synonym: 4-(3-Cyano-5,6-difluoroindol-1-yl)-2-hydroxybenzoic acid
Target: Xanthine Oxidase
Oxadiargyl
Cat.No: T20719
Synonym: RP 020630,RP-020630,RP020630,丙炔恶草酮,Topstar
Target: Others
Febuxostat
Cat.No: T0773
Synonym: 非布索坦,TMX 67,非布司他,TEI 6720
Target: ROS, Xanthine Oxidase
Allopurinol Sodium
Cat.No: T6376
Synonym: 1H-吡唑并[3,4-D]嘧啶-4-醇单钠盐,Allopurinol sodium salt,Sodium allopurinol
Target: ROS
Bazinaprine
Cat.No: T67789
Synonym:
Target: MAO
Luvadaxistat
Cat.No: T38863
Synonym: TAK-831,Luvadaxistat
Target:
Fomesafen
Cat.No: T20622
Synonym: 氟磺胺草醚,PP021,PP-021,PP 021
Target: Others
MAO-IN-1
Cat.No: T10079
Synonym:
Target: MAO
Trifludimoxazin
Cat.No: T38655
Synonym:
Target: Others
amflutizole
Cat.No: T8567
Synonym:
Target: Xanthine Oxidase
DAAO inhibitor-1
Cat.No: T5206
Synonym:
Target: Others
Iproniazid Phosphate
Cat.No: T0821
Synonym: 磷酸异丙烟肼,Isoproniazid phosphate
Target: MAO, Monoamine Oxidase
Eprobemide
Cat.No: T5053
Synonym: LIS 630,依普贝胺
Target: MAO, Monoamine Oxidase
Pargyline
Cat.No: T0300
Synonym: Pargylamine,Paragyline,优降宁
Target: MAO, Monoamine Oxidase
Toloxatone
Cat.No: T5323
Synonym: 托洛沙酮,MD 69276
Target: MAO, Monoamine Oxidase
Nitrofen
Cat.No: T39280
Synonym:
Target: Others
Setanaxib
Cat.No: T6099
Synonym: GKT137831
Target: NADPH-oxidase, Ferroptosis, NADPH
Clorgyline hydrochloride
Cat.No: T1117
Synonym: 盐酸氯吉林,Clorgiline hydrochloride,N-[3-(2,4-二氯苯氧基)丙基]-N-甲基-2-丙炔胺盐酸盐
Target: MAO, Monoamine Oxidase
CX-157
Cat.No: T15023
Synonym: KP 157
Target: MAO
Coumarin102
Cat.No: T77564
Synonym: Exciton 480
Target:
RS 8359
Cat.No: T16803
Synonym:
Target: MAO
Aminoguanidine hydrochloride
Cat.No: T0358
Synonym: Imino semicarbazide,Pimagedine hydrochloride,CP-12009-18 tartrate,Hydrazinecarboximidamide,肼甲酰亚胺酰胺一氯化氢(氨基胍盐酸盐),氨基胍盐酸盐,Guanyl hydrazine,Pimagedine
Target: NOS, NO Synthase
Medifoxamine
Cat.No: T24444
Synonym: LG 152,Medifoxamina,LG-152,LG152
Target: Dopamine Receptor, Monoamine Oxidase
PSB-1491
Cat.No: T24680
Synonym:
Target: MAO
Isocarboxazid
Cat.No: T4559
Synonym:
Target: Monoamine Oxidase
MDL 72527
Cat.No: T22965
Synonym: N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride
Target: Others
Desciclovir
Cat.No: T22304
Synonym: BW A515U,地昔洛韦,6-Deoxyacyclovir,DCV
Target: Antifection
Phenelzine sulfate
Cat.No: T12441
Synonym: 硫酸苯乙肼,苯肼,硫酸盐
Target: Monoamine Oxidase
Sodium benzoate
Cat.No: T8124
Synonym: Benzoic acid sodium salt,苯甲酸钠
Target: Others
PSB-1434
Cat.No: T24679
Synonym: PSB 1434,PSB1434
Target: MAO
Tranylcypromine (2-PCPA) hydrochloride
Cat.No: T1025
Synonym: 反苯环丙胺盐酸盐,Tranylcypromine (2-PCPA) HCl,SKF-385 HCl
Target: Histone Demethylase, MAO
Tigulixostat
Cat.No: T60625
Synonym:
Target:
Adrenalone hydrochloride
Cat.No: T0948
Synonym: Adrenalone HCl,肾上腺酮盐酸盐,盐酸肾上腺酮
Target: Adrenergic Receptor
Pargyline hydrochloride
Cat.No: T1578
Synonym: 优降宁盐酸盐,Pargylamine hydrochloride
Target: MAO, Monoamine Oxidase
NoxA1ds acetate(1435893-78-9 free base)
Cat.No: TP1886L1
Synonym:
Target: NADPH-oxidase
iNOS-IN-14
Cat.No: T83625
Synonym: 3-bromo-1H-indazole-7-carbonitrile
Target: NOS
ND-011992
Cat.No: T77615
Synonym: ND011992
Target: Mitochondrial Metabolism, Antibacterial
VAS 3947
Cat.No: T29097
Synonym: VA-S3947,VA S3947,VAS3947
Target: Apoptosis, NADPH-oxidase
Modaline sulfate
Cat.No: T0235
Synonym:
Target: MAO, Monoamine Oxidase
Tranylcypromine hemisulfate
Cat.No: T7942
Synonym: Tranylcypromine Sulfate,Tranylcypromine (hemisulfate),反苯环丙胺半硫酸盐
Target: Histone Demethylase, MAO, Monoamine Oxidase
Topiroxostat
Cat.No: T2397
Synonym: 托匹司他,FYX-051
Target: P450, ROS, Xanthine Oxidase
Pyraclonil
Cat.No: T19533
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN2004 Obtusin

1,7-二羟基-2,3,8-三甲氧基-6-甲基蒽-9,10-二酮,决明素

MAO; Monoamine Oxidase Metabolism; Neuroscience
Obtusin 是来自决明子种子,是一种高度选择性和竞争性的人单胺氧化酶-A 抑制剂,IC50=11.12 μM,Ki=6.15 μM。它在神经退行性疾病,尤其是焦虑和抑郁中起预防作用。
T3885 ROSIRIDIN

6'-O-Deacetylrosiridoside C,络塞定,(-)-Rosiridin

Others; Monoamine Oxidase Neuroscience; Others
Rosiridin (6'-O-Deacetylrosiridoside C) 能够抑制 MAO A 和 MAO B,有潜在的抑郁症和老年性痴呆作用。它在 10 μM 时对 MAO B 的抑制率为 83.8% (pIC50=5.38)。
TN7211 Tetrahydroharmine

Leptaflorine

MAO Metabolism; Neuroscience
Tetrahydroharmine (Leptaflorine) 是一种天然产物,存在于植物Banisteriopsis caapi cultivar Da Vine 的茎和枝中。四氢骆驼蓬碱是一种Monoamine oxidase A 抑制剂。
Fr12415 Ethyl 4-hydroxyphenylacetate

Others Others
Ethyl 4-hydroxyphenylacetate 是单胺氧化酶 A 的选择性抑制剂。
T13475 β-Aminopropionitrile

3-氨基丙腈,3-Aminopropionitrile,BAPN

Others; Endogenous Metabolite Metabolism; Others
β-Aminopropionitrile (3-Aminopropionitrile) 是赖氨酰氧化酶的特异性抑制剂。
T1694 Oxypurinol

Oxipurinol,羟基嘌呤

ROS; Xanthine Oxidase; Endogenous Metabolite Immunology/Inflammation; Metabolism
Oxypurinol 是一种黄嘌呤氧化酶 (xanthine oxidase) 抑制剂,是 Allopurinol 的主要特性代谢产物。它能够用于调节血尿酸水平,有潜力用于痛风的研究。
T6391 Apocynin

香草乙酮,Acetovanillone,Acetoguaiacone,NSC 2146,罗布麻宁

Apoptosis; NADPH; Autophagy Apoptosis; Autophagy; Metabolism
Apocynin (NSC 2146) 是一种选择性NADPH-氧化酶抑制剂,IC50为10 μM。
T2858 Baicalein

5,6,7-Trihydroxyflavone,黄芩素,黄芩黄素

Ferroptosis; Influenza Virus; ROS; Xanthine Oxidase Apoptosis; Immunology/Inflammation; Metabolism; Microbiology/Virology
Baicalein (5,6,7-Trihydroxyflavone) 是一种黄嘌呤氧化酶抑制剂,其IC50值为 3.12 μM。
TN1705 Glycyrrhisoflavone

MAO; Tyrosinase; NO Synthase; Immunology/Inflammation related Immunology/Inflammation; Metabolism; Neuroscience; Proteases/Proteasome
Glycyrrhisoflavone 是一种具有抗炎作用的酪氨酸酶抑制剂。 Glycyrrhisoflavone 抑制 α-葡萄糖苷酶和单胺氧化酶。
TQ0188 Miquelianin

槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide

stilbene oxidase; Endogenous Metabolite Metabolism
Miquelianin (Quercetin 3-glucuronide) 是槲皮素的代谢产物,属于类黄酮化合物。
T4716 Pyrrole-2-carboxylic acid

吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline

Endogenous Metabolite Metabolism
Pyrrole-2-carboxylic acid (Minaline) 是一种天然生物碱类,从海洋细菌Pelomonas puraquaesp. Nov 中分离得到。
T3750 4-Hydroxyacetophenone

对羟基苯乙酮,4-Acetylphenol,Piceol,p-Acetylphenol,4'-Hydroxyacetophenone

HBV; Xanthine Oxidase Metabolism; Microbiology/Virology
4-Hydroxyacetophenone (4-Acetylphenol) 是蒿属植物和木香属植物中的一种黄嘌呤氧化酶抑制剂,具有保肝促胆、抗乙型肝炎病毒和抗炎作用。
T3740 Isovanillin

3-羟基-4-甲氧基苯甲醛,3-Hydroxy-p-anisaldehyde,3-Hydroxy-4-methoxybenzaldehyde,5-Formylguaiacol

Others Others
Isovanillin (5-Formylguaiacol) 是一种醛氧化酶抑制剂,具有解痉挛和止泻活性。
T21164 Sulfentrazone

甲磺草胺,FP-846

Others Others
Sulfentrazone (FP-846) 是苯基三唑啉酮除草剂,能够抑制原卟啉原氧化酶,导致脂质细胞膜破裂,可用于控制某些阔叶和禾本科杂草。
T12564 Prudomestin

3,5,7-Trihydroxy-4',8-dimethoxyflavone,3,5,7-三羟基-8,4'-二甲氧基黄酮

Xanthine Oxidase Metabolism
Prudomestin (3,5,7-Trihydroxy-4',8-dimethoxyflavone) 是一种分离自 Prunus domestica 心材中,具有很强的黄嘌呤氧化酶(XO)抑制活性(IC50≈6 µM)。
T16685 Purpurogallin

红倍酚,红陪酚

Xanthine Oxidase Metabolism
Purpurogallin 是一种从栎属植物中提取的天然酚,具有显著的黄嘌呤氧化酶抑制作用,其IC50=0.2 µM,具有抗氧化和抗炎作用。
T3158 Harmane

Loturine,Harman,Aribine,哈尔满碱

Adrenergic Receptor; Monoamine Oxidase; Imidazoline Receptor GPCR/G Protein; Neuroscience
Harmane (Loturine) 是一种在咖啡和烟草烟雾中发现的 β-咔啉生物碱,是有效的神经毒素,可引起严重的动作震颤和精神病学表现。它还是选择性的单胺氧化酶抑制剂,具有致突变作用,对 MAO A/B 的 IC50值分别为 0.5 和 5 μM。
T4455 DL-3-Phenyllactic acid

DL-3-苯乳酸,3-Phenyllactic acid,2-Hydroxy-3-phenylpropanoic acid

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
DL-3-Phenyllactic acid (3-Phenyllactic acid) 是广谱抗菌化合物,对细菌和真菌具有活性。
T0617 Nicotinamide N-oxide

Nicotinamide-N-oxide,Nicotinamide 1-oxide,N-氧代烟酰胺,烟酰胺-N-氧化物,1-oxynicotinamide

c-Myc; Endogenous Metabolite; CXCR; Drug Metabolite Autophagy; Cell Cycle/Checkpoint; GPCR/G Protein; Immunology/Inflammation; Metabolism
Nicotinamide N-oxide (Nicotinamide 1-oxide) 是生物体内烟酰胺分解代谢物,是高效选择性CXCR2受体拮抗剂。
T16527 Phytic acid dodecasodium salt hydrate

植酸十二钠盐,myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate,Inositol hexaphosphate dodecasodium salt hydrate

Others; Xanthine Oxidase; Endogenous Metabolite Metabolism; Others
Phytic acid dodecasodium salt hydrate (myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate) 是种子和谷物的磷储存化合物。 Phytic acid dodecasodium salt hydrate 抑制酶促超氧化物源黄嘌呤氧化酶,IC50 为 6 mM,并具有抗氧化、神经保护和抗炎作用。
T10938 D-Kynurenine

D-尿嘧啶,(R)-2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid,ZINC901103

GPR; AhR; Endogenous Metabolite Endocrinology/Hormones; GPCR/G Protein; Immunology/Inflammation; Metabolism
D-Kynurenine (ZINC901103) 是 D-色氨酸的代谢物和 GPR109B 的激动剂。 D-Kynurenine 激活 AhR 并促进上皮细胞向间充质的转化。 D-Kynurenine 在 D-氨基酸氧化酶的荧光分析中用作底物。
TN1120 Osthenol

MAO; Monoamine Oxidase Metabolism; Neuroscience
Osthenol 是一种前酰化香豆素,从独活干根中分离得到。它对重组 hMAO-A 具有潜在的选择性抑制作用,IC50=0.74 µM,对 hMAO-A 和 hMAO-B 表现出较高的选择性指数。它是一种可逆的,选择性的竞争性人单胺氧化酶-A(hMAO-A)抑制剂 (Ki=0.26 µM)。
T3095 Tyramine

4-hydroxyphenethylamine,酪胺,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine

MAO; Endogenous Metabolite Metabolism; Neuroscience
Tyramine (Uteramine) 是天然存在于体内或某些食物中的氨基酸。Tyramine 有助于调节血压。
T3933 Jatrorrhizine

Yatrorizine,neprotin,药根碱

MAO; 5-HT Receptor; Antibacterial; AChE GPCR/G Protein; Metabolism; Microbiology/Virology; Neuroscience
Jatrorrhizine (neprotin) 是一种从黄连中分离得到的生物碱,具有抗菌、抗氧化、抗疟原虫和神经保护活性。它通过抑制 uptake-2 transporter 的活性减少血清素和去甲肾上腺素的摄取。它是一种有口服活性的乙酰胆碱酯酶制剂。
TN1470 Cassiaside B2

决明子苷B2

Phosphatase; MAO; 5-HT Receptor GPCR/G Protein; Metabolism; Neuroscience
Cassiaside B2 是蛋白酪氨酸磷酸酶1B (PTP1B) 和人单胺氧化酶A (hMAO-A) 的抑制剂。Cassiaside B2是 5-HT2C 受体的激动剂, 具有抗过敏活性。Cassiaside B2 是萘吡喃酮参比提取物(NRE)的有效成分之一。
TMA0958 Forsythoside F

连翘酯苷F,Arenarioside,三糖苯丙素苷

Xanthine Oxidase Metabolism
Forsythoside F (Arenarioside) 是一种黄嘌呤氧化酶 (xanthine oxidase) 抑制剂,具有抗高尿酸活性。
T5S0281 Tubuloside A

NOS Immunology/Inflammation
Tubuloside A 是一种苯乙醇苷,具有抗氧化活性和保肝活性。
T10933 D-Cysteine

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
D-Cysteine 是一种大肠杆菌生长的有力抑制剂,是半胱氨酸的 D 型异构体。它由 D-氨基酸氧化酶介导产生 H2S,是一种对抗小脑共济失调的神经保护剂。 D-半胱氨酸可以抑制由变形链球菌和链球菌血红蛋白形成的两种生物膜的生长和致龋性。
T5S2343 Acetylshikonin

乙酰紫草素,Acetyl shikonin

Others; P450; AChE Metabolism; Neuroscience; Others
Acetylshikonin 来源于紫草根,具有抗癌、抗炎作用。它是一种 AChE 抑制剂,具有很强的抗凋亡活性。它是一种非选择性的细胞色素 P450抑制剂,对所有 P450 亚型抑制的 IC50值范围为 1.4-4.0 μM。
T4746 Purine

7H-Imidazo(4,5-d)pyrimidine,嘌呤

Others; Endogenous Metabolite Metabolism; Others
Purine (7H-Imidazo(4,5-d)pyrimidine) 是内源性代谢产物的一种。
T19117 3-Deoxyglucosone

3-Deoxy-D-glucosone,2-keto-3-Deoxyglucose

GPX; Glucagon Receptor GPCR/G Protein; oxidation-reduction
3-Deoxyglucosone(3-Deoxy-D-glucosone) 是美拉德反应和多元醇反应的中间体途径合成。3-Deoxyglucosone 与蛋白质氨基快速反应形成晚期糖基化末端蛋白 (AGEs)。3-Deoxyglucosone 可使谷胱甘肽过氧化物酶失活,可与低葡萄糖协同作用以增强 GLP-1 分泌,可以作为糖尿病生物学检测的标志物。
T1362 Hypoxanthine

次黄嘌呤,6-羟基嘌呤,6-Hydroxypurine,Purin-6-ol,Sarcine,Sarkin

Others; Endogenous Metabolite Metabolism; Others
Hypoxanthine (Purin-6-ol),也被称为 purine-6-ol 或 Hyp,是一种天然存在的嘌呤衍生物,是腺苷代谢和核苷酸补救途径形成核酸的反应中间体。在正常情况下,Hypoxanthine 很容易转化为尿酸。Hypoxanthine 首先被氧化为黄嘌呤,黄嘌呤再被黄嘌呤氧化酶氧化为尿酸。
T4848 Mandelic acid

acidomandelico,DL-Mandelic acid,扁桃酸

Others; Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology; Others
DL-Mandelic acid (acidomandelico) 是一种 α-羟基羧酸,有抗菌活性,广泛用作医药和精细化学品的中间体,已用于研究尿路感染和阴道滴虫病,还具有较高的精子固定活性和较低的阴道刺激性。
T1311 4-aminobenzoic acid

PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸

Endogenous Metabolite Metabolism
4-aminobenzoic acid (para-Aminobenzoic acid) 是一种具有紫外线吸收和抗纤维化特性的有机酸。当暴露在光线下时,4-aminobenzoic acid 吸收紫外线并通过光化学反应释放多余的能量,这可能会对DNA造成损害。4-aminobenzoic acid 还可以增加组织水平的摄氧量,并可能增强单胺氧化酶(MAO)活性以促进血清素的降解,过量可能导致纤维化变化。
T4827 Trimethylammonium chloride

三甲胺盐酸盐,Trimethylamine hydrochloride

Others; Endogenous Metabolite Metabolism; Others
Trimethylammonium chloride (Trimethylamine hydrochloride) 是动植物分解的产物。它是造成鱼腥味的主要物质,通常与脏鱼、细菌性阴道感染和口臭有关。它也与服用大剂量胆碱有关。三甲胺尿是一种遗传性疾病,身体无法从食物中代谢三甲胺。食用富含胆碱的食物后,患者的汗液、尿液和呼吸中会出现特有的鱼腥味。三甲胺尿症是一种常染色体隐性遗传病,涉及三甲胺氧化酶缺乏症。三甲氨基尿症在罗德岛红鸡中也有发现,这种鸡产的蛋有腥味。尿液中的 Trimethylammonium chloride 是食用豆类的生物标志物。
TN2180 Sappanchalcone

苏木查耳酮

IL Receptor; BCL; TNF Apoptosis; Immunology/Inflammation
Sappanchalcone shows xanthine oxidase inhibitory activity, is a xanthine oxidase inhibitor.
TN5670 Protosappanin A dimethyl acetal

Protosappanin A dimethyl acetal shows significant xanthine oxidase inhibitory activity in a concentration-dependent manner.
TN4080 Fraxamoside

Xanthine Oxidase Metabolism
Fraxamoside is a xanthine oxidase inhibitor (XOI) comparable in potency in vitro to the standard antigout drug allopurinol. It shows significant free radical scavenging effect against DPPH(EC50=62.6 uM).
T38777 Ilexoside O

Ilexoside O, a triterpene saponin derived from Ilex pubescens roots, demonstrates modest inhibition of xanthine oxidase (XOD) activity with an IC50 value of 53.05 μM.
T36950 Rubrofusarin triglucoside

Rubrofusarin triglucoside is a glycoside compound isolated from Cassia obtusifolia Linn seeds. Rubrofusarin triglucoside inhibits human monoamine oxidase A (hMAO-A) with an IC50 of 85.5 μM[1]. [1]. Pradeep Paudel, et al. Rubrofusarin as a Dual Protein Tyrosine Phosphate 1B and Human Monoamine Oxidase-A Inhibitor: An in Vitro and in Silico Study. ACS Omega. 2019 Jul 3;4(7):11621-11630.
TN3208 7,3',4'-Trihydroxy-3-benzyl-2H-chromene

ROS Immunology/Inflammation
7,3',4'-Trihydroxy-3-benzyl-2H-chromene is a potential xanthine oxidase inhibitor.
T40244 Methyl citrate

Methyl citrate, obtained from Opuntia ficus-indica var. saboten Makino fruits, serves as a potent Monoamine oxidase B (MAO-B) inhibitor with an IC50 value of 0.23 mM.
TN2790 2'-O-Methylperlatolic acid

MAO Metabolism; Neuroscience
2'-O-Methylperlatolic acid and confluentic acid are monoamine oxidase B inhibitors in a Brazilian plant, Himatanthus sucuuba.
TN4137 Glicoricone

MAO Metabolism; Neuroscience
Glicoricone acts as a partial estrogen antagonist. Glicoricone inhibited the monoamine oxidase with the IC50 values of 6.0 x 10(-5)-1.4 x 10(-4) M.
T32208 Isogentisin

BRN 0258402,BRN-0258402,BRN0258402

MAO Metabolism; Neuroscience
Isogentisin (BRN 0258402) 是一种从龙胆科植物中分离出来的化合物,是一种用于预防吸烟引起的内皮损伤的新型化合物。Isogentisin 对单胺氧化酶具有抑制作用。
TN3116 5-Hydroxy-1-methoxyxanthone

MAO; Antifection Metabolism; Microbiology/Virology; Neuroscience
5-Hydroxy-1-methoxyxanthone, 1,5-dihydroxyxanthone and 6-deoxyjacareubin are all antifungal against Cladosporium cucumerinum, while they show differing degrees of inhibition of monoamine oxidase A and B.
T40576 (S)-Salsolidine

(S)-Salsolidine, a chemical compound, functions as a weak inhibitor of monoamine oxidase (MAO), exhibiting an inhibition constant (K i ) of 63 μM. R enantiomer demonstrating a greater efficacy than (S)-Salsolidine, boasting a K i value of 26 μM compared to the S form.
TN3726 Cudraflavone B

IκB/IKK; MAO; ROS; Akt; COX; PI3K; Nrf2; Autophagy Autophagy; Cytoskeletal Signaling; Immunology/Inflammation; Metabolism; Neuroscience; NF-κB; PI3K/Akt/mTOR signaling
Cudraflavone B has anti-proliferative activity, mouse brain monoamine oxidase (MAO) inhibitory effects, apoptotic actions in human gastric carcinoma cells and mouse melanoma cells, and hepatoprotective activity. It may be a lead for the development of a potential candidate for human oral squamous cell carcinoma cells.
TN2039 Panaxydol

cAMP; p38 MAPK; JNK GPCR/G Protein; MAPK
Panaxydol has anti-cancer activity, can inhibit the growth and apoptosis of cancer cells, the signaling mechanisms involve a [Ca(2+)](i) increase, JNK and p38 MAPK activation, cAMP, MAP kinase and ROS generation through NADPH oxidase and mitochondria.
TN4433 Licoarylcoumarin

cAMP; HIV Protease; Antifection GPCR/G Protein; Microbiology/Virology; Proteases/Proteasome
Licoarylcoumarin is a strong inhibitor of adenosine 3',5'-cyclic monophosphate (cAMP) phosphodiesterase. Licoarylcoumarin has antibacterial effects on the VRE strains; it has anti-HIV activity, and it has inhibitory effects on xanthine oxidase.
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天然产物

Obtusin
Cat.No: TN2004
Synonym: 1,7-二羟基-2,3,8-三甲氧基-6-甲基蒽-9,10-二酮,决明素
Target: MAO, Monoamine Oxidase
ROSIRIDIN
Cat.No: T3885
Synonym: 6'-O-Deacetylrosiridoside C,络塞定,(-)-Rosiridin
Target: Others, Monoamine Oxidase
Tetrahydroharmine
Cat.No: TN7211
Synonym: Leptaflorine
Target: MAO
Ethyl 4-hydroxyphenylacetate
Cat.No: Fr12415
Synonym:
Target: Others
β-Aminopropionitrile
Cat.No: T13475
Synonym: 3-氨基丙腈,3-Aminopropionitrile,BAPN
Target: Others, Endogenous Metabolite
Oxypurinol
Cat.No: T1694
Synonym: Oxipurinol,羟基嘌呤
Target: ROS, Xanthine Oxidase, Endogenous Metabolite
Apocynin
Cat.No: T6391
Synonym: 香草乙酮,Acetovanillone,Acetoguaiacone,NSC 2146,罗布麻宁
Target: Apoptosis, NADPH, Autophagy
Baicalein
Cat.No: T2858
Synonym: 5,6,7-Trihydroxyflavone,黄芩素,黄芩黄素
Target: Ferroptosis, Influenza Virus, ROS, Xanthine Oxidase
Glycyrrhisoflavone
Cat.No: TN1705
Synonym:
Target: MAO, Tyrosinase, NO Synthase, Immunology/Inflammation related
Miquelianin
Cat.No: TQ0188
Synonym: 槲皮素-3-O-葡萄糖醛酸苷,Quercetin 3-glucuronide,Quercetin 3-O-glucuronide
Target: stilbene oxidase, Endogenous Metabolite
Pyrrole-2-carboxylic acid
Cat.No: T4716
Synonym: 吡咯-2-羧酸,2-Pyrrolecarboxylic acid,Minaline
Target: Endogenous Metabolite
4-Hydroxyacetophenone
Cat.No: T3750
Synonym: 对羟基苯乙酮,4-Acetylphenol,Piceol,p-Acetylphenol,4'-Hydroxyacetophenone
Target: HBV, Xanthine Oxidase
Isovanillin
Cat.No: T3740
Synonym: 3-羟基-4-甲氧基苯甲醛,3-Hydroxy-p-anisaldehyde,3-Hydroxy-4-methoxybenzaldehyde,5-Formylguaiacol
Target: Others
Sulfentrazone
Cat.No: T21164
Synonym: 甲磺草胺,FP-846
Target: Others
Prudomestin
Cat.No: T12564
Synonym: 3,5,7-Trihydroxy-4',8-dimethoxyflavone,3,5,7-三羟基-8,4'-二甲氧基黄酮
Target: Xanthine Oxidase
Purpurogallin
Cat.No: T16685
Synonym: 红倍酚,红陪酚
Target: Xanthine Oxidase
Harmane
Cat.No: T3158
Synonym: Loturine,Harman,Aribine,哈尔满碱
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
DL-3-Phenyllactic acid
Cat.No: T4455
Synonym: DL-3-苯乳酸,3-Phenyllactic acid,2-Hydroxy-3-phenylpropanoic acid
Target: Others, Endogenous Metabolite, Antibacterial
Nicotinamide N-oxide
Cat.No: T0617
Synonym: Nicotinamide-N-oxide,Nicotinamide 1-oxide,N-氧代烟酰胺,烟酰胺-N-氧化物,1-oxynicotinamide
Target: c-Myc, Endogenous Metabolite, CXCR, Drug Metabolite
Phytic acid dodecasodium salt hydrate
Cat.No: T16527
Synonym: 植酸十二钠盐,myo-Inositol, hexakis(dihydrogen phosphate) dodecasodium salt hydrate,Inositol hexaphosphate dodecasodium salt hydrate
Target: Others, Xanthine Oxidase, Endogenous Metabolite
D-Kynurenine
Cat.No: T10938
Synonym: D-尿嘧啶,(R)-2-Amino-4-(2-aminophenyl)-4-oxobutanoic acid,ZINC901103
Target: GPR, AhR, Endogenous Metabolite
Osthenol
Cat.No: TN1120
Synonym:
Target: MAO, Monoamine Oxidase
Tyramine
Cat.No: T3095
Synonym: 4-hydroxyphenethylamine,酪胺,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine
Target: MAO, Endogenous Metabolite
Jatrorrhizine
Cat.No: T3933
Synonym: Yatrorizine,neprotin,药根碱
Target: MAO, 5-HT Receptor, Antibacterial, AChE
Cassiaside B2
Cat.No: TN1470
Synonym: 决明子苷B2
Target: Phosphatase, MAO, 5-HT Receptor
Forsythoside F
Cat.No: TMA0958
Synonym: 连翘酯苷F,Arenarioside,三糖苯丙素苷
Target: Xanthine Oxidase
Tubuloside A
Cat.No: T5S0281
Synonym:
Target: NOS
D-Cysteine
Cat.No: T10933
Synonym:
Target: Endogenous Metabolite, Antibacterial
Acetylshikonin
Cat.No: T5S2343
Synonym: 乙酰紫草素,Acetyl shikonin
Target: Others, P450, AChE
Purine
Cat.No: T4746
Synonym: 7H-Imidazo(4,5-d)pyrimidine,嘌呤
Target: Others, Endogenous Metabolite
3-Deoxyglucosone
Cat.No: T19117
Synonym: 3-Deoxy-D-glucosone,2-keto-3-Deoxyglucose
Target: GPX, Glucagon Receptor
Hypoxanthine
Cat.No: T1362
Synonym: 次黄嘌呤,6-羟基嘌呤,6-Hydroxypurine,Purin-6-ol,Sarcine,Sarkin
Target: Others, Endogenous Metabolite
Mandelic acid
Cat.No: T4848
Synonym: acidomandelico,DL-Mandelic acid,扁桃酸
Target: Others, Endogenous Metabolite, Antibacterial
4-aminobenzoic acid
Cat.No: T1311
Synonym: PABA,Vitamin H1,Vitamin Bx,para-Aminobenzoic acid,对氨基苯甲酸
Target: Endogenous Metabolite
Trimethylammonium chloride
Cat.No: T4827
Synonym: 三甲胺盐酸盐,Trimethylamine hydrochloride
Target: Others, Endogenous Metabolite
Sappanchalcone
Cat.No: TN2180
Synonym: 苏木查耳酮
Target: IL Receptor, BCL, TNF
Protosappanin A dimethyl acetal
Cat.No: TN5670
Synonym:
Target:
Fraxamoside
Cat.No: TN4080
Synonym:
Target: Xanthine Oxidase
Ilexoside O
Cat.No: T38777
Synonym:
Target:
Rubrofusarin triglucoside
Cat.No: T36950
Synonym:
Target:
7,3',4'-Trihydroxy-3-benzyl-2H-chromene
Cat.No: TN3208
Synonym:
Target: ROS
Methyl citrate
Cat.No: T40244
Synonym:
Target:
2'-O-Methylperlatolic acid
Cat.No: TN2790
Synonym:
Target: MAO
Glicoricone
Cat.No: TN4137
Synonym:
Target: MAO
Isogentisin
Cat.No: T32208
Synonym: BRN 0258402,BRN-0258402,BRN0258402
Target: MAO
5-Hydroxy-1-methoxyxanthone
Cat.No: TN3116
Synonym:
Target: MAO, Antifection
(S)-Salsolidine
Cat.No: T40576
Synonym:
Target:
Cudraflavone B
Cat.No: TN3726
Synonym:
Target: IκB/IKK, MAO, ROS, Akt, COX, PI3K, Nrf2, Autophagy
Panaxydol
Cat.No: TN2039
Synonym:
Target: cAMP, p38 MAPK, JNK
Licoarylcoumarin
Cat.No: TN4433
Synonym:
Target: cAMP, HIV Protease, Antifection
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