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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T10404 ATP synthase inhibitor 1

ATPase Membrane transporter/Ion channel
ATP synthase inhibitor 1 是 F1/FO-ATP 合酶复合物 c 亚基的有效抑制剂,抑制线粒体通透性转换孔的开放。
T60032 BRM/BRG1 ATP Inhibitor-2

Epigenetic Reader Domain Chromatin/Epigenetic
BRM/BRG1 ATP Inhibitor-2 是 BRG1/BRM ATPase 的抑制剂,可用于治疗 BAF 相关疾病的研究。
T22592 ATPγS tetralithium salt

ATP-gamma-S tetralithium salt

PERK Apoptosis
ATPγS tetralithium salt 是真核生物翻译起始因子 eIF4A 的核苷酸水解和RNA解链活性的底物,与 p97 突变体和朊病毒相关。
T13541 α,β-Methylene ATP trisodium

Others Others
α,β-Methylene ATP trisodium is a ligand of P2X3 and P2X7 receptor.
T10616 BRM/BRG1 ATP Inhibitor-1

Epigenetic Reader Domain Chromatin/Epigenetic
BRM/BRG1 ATP Inhibitor-1 是变构双 Brahma 同源物 (BRM)/SWI/SNF 相关的基质相关肌动蛋白依赖性调节剂,染色质亚家族 A 成员 2 和 BRG1/SMARCA4 ATP 酶活性抑制剂,IC50值低于 0.005 μM。
T39891 8-Bromo-ATP

8-Bromoadenosine 5'-triphosphate,8-Bromo-ATP,8-Br-ATP

8-Bromo-ATP (8-Bromoadenosine 5'-triphosphate) is a purinergic P2X receptor agonist and an ATP analogue. It exhibits cytotoxicity towards multiple myeloma cells, with an IC50 of 23.1 μM.
T40616 8-Azido-ATP

8-Azidoadenosine 5'-triphosphate,8-N3-ATP,8-Azido-ATP

8-Azido-ATP is a nucleotide analog that demonstrates photo-reactivity properties. It offers utility in the precise labeling and identification of proteins, particularly those involved in DNA-dependent RNA polymerase activity.
T40455 8-NH2-ATP

8-Aminoadenosine-5'-O-triphosphate,8-NH2-ATP

8-NH2-ATP is an inactive derivative of adenosine triphosphate (ATP), synthesized from 8-NH2-Ado. It has been documented that 8-NH2-Ado exhibits potent properties, as evidenced by its ability to induce apoptosis-associated cleavage of poly(ADP-ribose) polymerase.
T40696 2'-NH2-ATP

2'-NH2-ATP,2'-Amino-2'-deoxyadenosine-5'-triphosphate

2'-NH2-ATP (2'-Amino-2'-deoxyadenosine-5'-triphosphate) is an adenosine derivative compound that acts as a weak competitive inhibitor of ATP with a K i value of 2.3 mM. It finds utility in nucleic acid labeling.
T22496 2-Methylthio-ATP tetrasodium

2-Methylthioadenosine triphosphate tetrasodium salt,2-methylthio-atp-tetrasodium

Others Others
P2 purinoceptor agonist
T17454 ATP-polyamine-biotin

Others Others
ATP-polyamine-biotin is a cell-permeable, efficient kinase cosubstrate with conversions and kinetics similar to those of other known ATP analogues. APB shows a cytotoxicity EC50 value of 19 ± 1 mM. ATP-polyamine-biotin is shown to promote biotin labeling
T38444 α,β-Methylene-ATP dilithium

α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors. It is a potent agonist specifically targeting P2X1 and P2X3 receptors while exerting negligible activity on P2X2, P2X4, P2X5, P2X6, and P2X7 receptors.
T18917 ATP-Red 1

Others Others
ATP-Red 1 is a multisite-binding switchable fluorescent probe. It can rapidly and selectively respond to intracellular concentrations of ATP in living cells.
T69111 2',3'-Dialdehyde ATP

2',3'-Dialdehyde ATP is a derivative of, and the oxidized form of, ATP. It has been found to be a specific, irreversible inhibitor of component A3 of the methylreductase system which plays a role in processing amino acids.
T40522 3'-Deoxy-3'-amino-ATP

3'-Deoxy-3'-amino-ATP, an ATP analogue, is a highly effective and competitive inhibitor of ATP, exhibiting a K i value of 2.3 μM. Its application includes the synthesis of 3′-Amino-3′-deoxy transfer RNA by integrating it into the 3' terminus of tRNA-C-C.
T22738 DMNPE-caged ATP diammonium salt

Others Others
DMNPE-caged ATP
TP2297 TNP-ATP triethylammonium salt

Others Others
P2X receptor antagonist
T75326 ATP ditromethamine

ATP ditromethamine(Adenosine 5'-triphosphate ditromethamine)作为体内能量储存和代谢的核心物质,不仅为代谢过程提供必需能量,而且在细胞中担任辅酶角色。此外,它在免疫和炎症反应中,扮演着关键的内源性信号分子角色。
T75325 ATP dimagnesium

ATP dimagnesium(Adenosine 5'-triphosphate dimagnesium)是生物体内关键的能量储存及代谢物质,不仅为代谢活动供能,而且还在细胞内扮演着辅酶的角色。此外,ATP dimagnesium 在免疫和炎症过程中,作为重要的内源性信号分子发挥作用。
T74033 6-Me-ATP

6-Me-ATP(N6-Methyl-ATP)为ATP的N6修饰衍生物。该化合物与GSK3β结合亲和力显著,能有效作为GSK3β催化底物肽磷酸化的磷酸基团供体。
T83802 TNP-ATP sodium

TNP-ATPATP的衍生物,同时是嘌呤P2Y1、P2X3和P2X2/3受体的拮抗剂(IC50s分别为6、0.9和7 nM,在表达人类受体的HEK293细胞中)。该化合物相对于嘌呤P2X2、P2X4和P2X7受体显示出选择性(IC50s分别为2、15.2和>30 µM,在表达人类受体的HEK293细胞中)。TNP-ATP能降低表达P2X3和P2X2/3受体的1321N1细胞中乙酸诱导的钙流量(IC50s分别为100和62 nM)。它还可以减轻小鼠模型中由乙酸诱发的痛性绞曲(ED50 = 6.35 µmol/kg)。在403 nm激发下,其发射最大峰值为547 nm,当结合于胰岛素降解酶(IDE)时,其相对荧光强度增加四倍,并且发射峰移至538 nm。
T82944 ATP Synthesis-IN-2

ATP Synthesis-IN-2 (Compound 5) 是一种有效的ATP合成活性抑制剂,对Pseudomonas aeruginosa (PA) 表现出抗菌活性,其IC50值为0.7 μg/mL。
T79586 3′-Acetate-ATP

3’-Acetate-ATPATP的乙酰化衍生物,表现为ATP类似物,其在中性pH值的水溶液中于259 nm波长处展现出最大的紫外线吸收。该化合物能够抑制核酸聚合酶活性,从而阻断核酸的延伸。
T78639 Oxidized ATP trisodium salt

oATP trisodium salt

P2X Receptor Membrane transporter/Ion channel; Neuroscience
Oxidized ATP (oATP) trisodium salt 是一种P2 受体广泛抑制剂,其不可逆地阻断P2X7R活化并抑制CRP引发的NLRP3炎性体激活,常用于动脉粥样硬化研究。
T82945 ATP Synthesis-IN-1

ATP Synthesis-IN-1(Compound 4)为喹啉衍生物,有效抑制PA ATP合成,IC50为11.1μg/mL。本化合物亦展示抗菌特性,适用于研究耐药PA感染。
T72590 α,β-Methylene-ATP

α,β-Methylene ATP,一种ATP的膦酸酯类似物,充当P2X3和P2X7受体的配体。该化合物对P2X1和P2X3表现出高选择性激动剂活性,而在P2X2, 4, 7受体上无活性。
T83786 8-Chloroadenosine-5'-triphosphate sodium

8-chloro ATP

8-Chloroadenosine-5’-triphosphate(8-chloro ATP)是抗癌剂8-chloro cAMP的活性代谢物,也是核苷酸腺苷5’-三磷酸(ATP)的衍生物。它通过8-chloro cAMP、8-chloroadenosine以及一磷酸和二磷酸中间体形成。应用8-chloro cAMP或8-chloroadenosine后,8-chloro ATP可累积长达12小时,与细胞生长抑制、内源性ATP水平下降以及患者源多发性骨髓瘤细胞中RNA合成减少(但DNA合成不受影响)相关。在1.5至8 mM浓度范围内,它抑制topoisomerase II-α依赖的超螺旋pUC19 DNA放松,同时在1 mM时减少了K562人髓性白血病细胞中topoisomerase II-α催化的ATP水解50%。
T83807 Rp-Adenosine-5'-O-(1-thiotriphosphate) sodium

Rp-ATP-α-S

Rp-Adenosine-5'-O-(1-thiotriphosphate)(Rp-ATP-α-S)是一种含硫核苷酸衍生物ATP-α-S的异构体,同时也是嘌呤P2Y1受体的激动剂。在表达人类P2Y1受体的HEK293细胞中,Rp-ATP-α-S能增加钙的动员(EC50 = 75 nM)。该化合物与洗涤的人类孤立血小板结合(Ki = 156 nM),抑制由ADP引发的人类富血小板血浆(PRP)的聚集(pA2 = 4.74),并且能够抑制前列腺素E1(PGE1)在人类孤立PRP中引发的cAMP产生(pA2 = 5.26)。同时,Rp-ATP-α-S还能引起用氨基甲酰胆碱预先缩紧的豚鼠结肠条带的松弛(EC50 = 56 nM)。此外,Rp-ATP-α-S已经被用于合成被细菌核糖开关识别的环状二核苷酸。
T61649 ATP synthase inhibitor 2

ATP synthase inhibitor2 是一个铜绿假单胞菌 (PA)ATP synthase 抑制剂 (IC50=10 μg/mL),在 128 μg/mL 时可完全抑制铜绿假单胞菌 (PA) 的 ATP 合成活性。
T74034 6-Me-ATP trisodium

6-Me-ATP trisodium (N6-Methyl-ATP) 是N6-修饰的ATP衍生物,展现对GSK3良好的结合亲和力,可作为GSK3β磷酸化底物肽的磷酸基团供体。
T83808 Sp-Adenosine-5'-O-(1-thiotriphosphate) sodium

Sp-ATP-α-S

Sp-Adenosine-5'-O-(1-thiotriphosphate) (Sp-ATP-α-S) 是一种含硫核苷酸衍生物 ATP-α-S 的异构体,也是嘌呤P2Y1受体的激动剂。在表达P2Y1受体的HEK293细胞中增加钙离子的流动(对人类受体的EC50 = 9.4 nM)。Sp-ATP-α-S 抑制了ADP诱导的孤立人类血小板聚集(Ki = 4 μM)。它还能引起经卡巴胆碱预收缩的豚鼠十二指肠松弛(EC50 = 426 nM)。
T83811 2'(3')-O-Anthraniloyladenosine-5'-O-triphosphate sodium

2'(3')-ANT-ATP

2'(3')-O-Anthraniloyladenosine-5'-O-triphosphate(2'-ANT-ATP)与3'-ANT-ATP是荧光ATP衍生物,可自发地进行异构化。在水中,2'(3')-ANT-ATP的激发波长为330 nm时,发射最大波长为428 nm。它对哺乳动物腺苷酸环化酶(AC1)、AC2及AC5显示出抑制作用,抑制常数(Kis)分别为130、640和120 nM。此外,它还能抑制百日咳杆菌腺苷酸环化酶毒素CyaA(在锰和镁存在下,Kis分别为1.3和20 µM)、炭疽杆菌腺苷酸环化酶毒素水肿因子(在锰和镁存在下,Kis分别为0.44和5.15 µM)以及大肠杆菌重组酶A(RecA;Ki = 6.3 µM)。
T72257 BRM/BRG1 ATP Inhibitor-3

BRM/BRG1 ATP Inhibitor-3为一种针对BRG1/BRM的抑制剂,具有分别针对BRM和BRG1的IC50值为10.4 nM及19.3 nM,适用于癌症与BAF复合物相关疾病的研究。
T15373 Gboxin

ATPase; Mitochondrial Metabolism Membrane transporter/Ion channel; Metabolism
Gboxin 是一种氧化磷酸化抑制剂,可靶向抑制胶质母细胞瘤生长,还抑制 F0F1 ATP 合成,具有抗肿瘤活性。
T79004 ATP synthase inhibitor 2 TFA

ATP synthase inhibitor2 (Compound 22) TFA 为针对铜绿假单胞菌 (PA) ATP synthase 的抑制剂,具IC50值为10 μg/mL,在浓度达到128 μg/mL 时能够全面阻断铜绿假单胞菌 (PA) ATP的合成活性。
T60877 Mtb ATP synthase-IN-1

Mtb ATP synthase-IN-1 (compound 6ab) 可用于研究抗结核分枝杆菌。Mtb ATP synthase-IN-1 具有低细胞毒性 (Vero IC50> 64 μg/mL)和可接受的口服生物利用度,具有良好的代谢稳定性。Mtb ATP synthase-IN-1 是结核分枝杆菌 (Mtb) ATP 合成酶的有效抑制剂(MIC 值为 0.452 ~ 0.499 μg/mL)。
T72258 BRM/BRG1 ATP Inhibitor-4

BRM/BRG1 ATP Inhibitor-4 是一种BRG1/BRM 抑制剂。BRM/BRG1 ATP Inhibitor-4 可用于癌症和 BAF 复合物相关疾病的研究。
T40862 Fludarabine triphosphate

三磷酸氟达拉滨,F-ara-ATP

Fludarabine triphosphate (F-ara-ATP), the cytotoxic metabolite of Fludarabine phosphate , inhibits ribonucleotide reductase and DNA polymerase and ultimately leads to cellular apoptosis.
T38511 AWL-II-38.3

Ephrin Receptor Tyrosine Kinase/Adaptors
AWL-II-38.3 is a highly effective inhibitor of EphA3, a receptor for ephrin-A. It demonstrates potent kinase inhibitory activity against EphA3 and does not show significant cellular activity against Src-family kinases or b-raf [1] [2].
T40456 8-Bromoadenosine 5'-triphosphate tetrasodium

8-Br-ATP tetrasodium,8-Bromoadenosine 5'-triphosphate tetrasodium

8-Bromoadenosine 5'-triphosphate tetrasodium (8-Br-ATP tetrasodium) is a tetrasodium ATP analogue, serving as a vital element for energy storage and metabolic processes in living organisms. ATP, a central component in vivo, plays a critical role in these functions.
T83818 Isoguanosine-5'-O-triphosphate sodium

2-Hydroxyadenosine 5’-triphosphate,2-hydroxy ATP,isoGTP

Isoguanosine-5'-O-triphosphate是guanosine 5'-triphosphate(GTP)的一个异构体且是crotonoside的磷酸化形式。与GTP不同,Isoguanosine-5'-O-triphosphate不促进微管组装。在逆转录酶实验中,Isoguanosine-5'-O-triphosphate(2 mM)能抑制转录并诱导T到C的突变。它已被用于确定phosphofructokinase和mutT homolog 1(MTH1)的底物特异性。
T83830 2'-Deoxy-2'-fluoroadenosine-5'-O-triphosphate sodium

2′-fluoro-2′-deoxy ATP,AfTP,2'-fluoro dATP

2'-Deoxy-2'-fluoroadenosine-5'-O-triphosphate是ATP的一种氟代衍生物,ATP是细胞代谢必需的能量底物。它抑制E. coli RNA聚合酶(Ki = 200 µM)。
T9626 Cycloleucine

NMDAR Neuroscience
Cycloleucine 是 NMDA 受体相关甘氨酸受体的拮抗剂,Ki 为 600 μM。Cycloleucine 也是 S-腺苷甲硫氨酸介导的甲基化的竞争性抑制剂,具有抗焦虑和细胞抑制作用。
T15385 Glibornuride

Potassium Channel Membrane transporter/Ion channel
Glibornuride 是对 ATP 敏感的 K+通道 (KATP 通道) 阻滞剂,pKi 为 5.75。Glibornuride 显示抗糖尿病活性。
T16861 SB 204990

ATP Citrate Lyase Metabolism
SB 204990是一种有效的、特异性 ATP 柠檬酸裂解酶抑制剂。
T7424 NDI-091143

ATP Citrate Lyase Metabolism
NDI-091143 是高亲和力人 ATP 柠檬酸裂解酶抑制剂,其IC50为 2.1 nM (ADP-Glo 分析),Ki 为 7.0 nM,Kd 为 2.2 nM。它能够稳定柠檬酸盐域中的大构象变化,间接抑制柠檬酸的结合和识别,进而抑制ACLY 催化变构反应。
T8535 GAK inhibitor 49

Serine/threonin kinase Cell Cycle/Checkpoint; Metabolism
GAK inhibitor 49 是 ATP 竞争性的细胞周期蛋白 G 相关激酶选择性抑制剂,Ki=0.54 nM,细胞 IC50=56 nM。它也具有与 RIPK2 结合的能力。
T7545 6-Aminonicotinamide

Others Others
6-Aminonicotinamide 是一种竞争性 NADP+依赖性酶,是一种烟酰胺抗代谢药,葡萄糖 6-磷酸脱氢酶抑制剂 (Ki=0.46 μM)。 它干扰糖酵解,导致 ATP 耗竭,并与 DNA 交联化学疗法药物,如Cisplatin,协同杀死癌细胞。
T2337 BMS-303141

BMS 303141

ATP Citrate Lyase Metabolism
BMS-303141是高效性和可渗透细胞的 ACL 抑制剂(IC50:0.13 μM)。
T22518 5-BDBD

P2X Receptor Membrane transporter/Ion channel; Neuroscience
5-BDBD 是选择性P2X4受体拮抗剂,抑制 rP2X4R 介导的电流,IC50为0.75μM。它可完全阻断硝酸甘油诱导的基础性和急性痛觉过敏。

化合物

ATP synthase inhibitor 1
Cat.No: T10404
Synonym:
Target: ATPase
BRM/BRG1 ATP Inhibitor-2
Cat.No: T60032
Synonym:
Target: Epigenetic Reader Domain
ATPγS tetralithium salt
Cat.No: T22592
Synonym: ATP-gamma-S tetralithium salt
Target: PERK
α,β-Methylene ATP trisodium
Cat.No: T13541
Synonym:
Target: Others
BRM/BRG1 ATP Inhibitor-1
Cat.No: T10616
Synonym:
Target: Epigenetic Reader Domain
8-Bromo-ATP
Cat.No: T39891
Synonym: 8-Bromoadenosine 5'-triphosphate,8-Bromo-ATP,8-Br-ATP
Target:
8-Azido-ATP
Cat.No: T40616
Synonym: 8-Azidoadenosine 5'-triphosphate,8-N3-ATP,8-Azido-ATP
Target:
8-NH2-ATP
Cat.No: T40455
Synonym: 8-Aminoadenosine-5'-O-triphosphate,8-NH2-ATP
Target:
2'-NH2-ATP
Cat.No: T40696
Synonym: 2'-NH2-ATP,2'-Amino-2'-deoxyadenosine-5'-triphosphate
Target:
2-Methylthio-ATP tetrasodium
Cat.No: T22496
Synonym: 2-Methylthioadenosine triphosphate tetrasodium salt,2-methylthio-atp-tetrasodium
Target: Others
ATP-polyamine-biotin
Cat.No: T17454
Synonym:
Target: Others
α,β-Methylene-ATP dilithium
Cat.No: T38444
Synonym:
Target:
ATP-Red 1
Cat.No: T18917
Synonym:
Target: Others
2',3'-Dialdehyde ATP
Cat.No: T69111
Synonym:
Target:
3'-Deoxy-3'-amino-ATP
Cat.No: T40522
Synonym:
Target:
DMNPE-caged ATP diammonium salt
Cat.No: T22738
Synonym:
Target: Others
TNP-ATP triethylammonium salt
Cat.No: TP2297
Synonym:
Target: Others
ATP ditromethamine
Cat.No: T75326
Synonym:
Target:
ATP dimagnesium
Cat.No: T75325
Synonym:
Target:
6-Me-ATP
Cat.No: T74033
Synonym:
Target:
TNP-ATP sodium
Cat.No: T83802
Synonym:
Target:
ATP Synthesis-IN-2
Cat.No: T82944
Synonym:
Target:
3′-Acetate-ATP
Cat.No: T79586
Synonym:
Target:
Oxidized ATP trisodium salt
Cat.No: T78639
Synonym: oATP trisodium salt
Target: P2X Receptor
ATP Synthesis-IN-1
Cat.No: T82945
Synonym:
Target:
α,β-Methylene-ATP
Cat.No: T72590
Synonym:
Target:
8-Chloroadenosine-5'-triphosphate sodium
Cat.No: T83786
Synonym: 8-chloro ATP
Target:
Rp-Adenosine-5'-O-(1-thiotriphosphate) sodium
Cat.No: T83807
Synonym: Rp-ATP-α-S
Target:
ATP synthase inhibitor 2
Cat.No: T61649
Synonym:
Target:
6-Me-ATP trisodium
Cat.No: T74034
Synonym:
Target:
Sp-Adenosine-5'-O-(1-thiotriphosphate) sodium
Cat.No: T83808
Synonym: Sp-ATP-α-S
Target:
2'(3')-O-Anthraniloyladenosine-5'-O-triphosphate sodium
Cat.No: T83811
Synonym: 2'(3')-ANT-ATP
Target:
BRM/BRG1 ATP Inhibitor-3
Cat.No: T72257
Synonym:
Target:
Gboxin
Cat.No: T15373
Synonym:
Target: ATPase, Mitochondrial Metabolism
ATP synthase inhibitor 2 TFA
Cat.No: T79004
Synonym:
Target:
Mtb ATP synthase-IN-1
Cat.No: T60877
Synonym:
Target:
BRM/BRG1 ATP Inhibitor-4
Cat.No: T72258
Synonym:
Target:
Fludarabine triphosphate
Cat.No: T40862
Synonym: 三磷酸氟达拉滨,F-ara-ATP
Target:
AWL-II-38.3
Cat.No: T38511
Synonym:
Target: Ephrin Receptor
8-Bromoadenosine 5'-triphosphate tetrasodium
Cat.No: T40456
Synonym: 8-Br-ATP tetrasodium,8-Bromoadenosine 5'-triphosphate tetrasodium
Target:
Isoguanosine-5'-O-triphosphate sodium
Cat.No: T83818
Synonym: 2-Hydroxyadenosine 5’-triphosphate,2-hydroxy ATP,isoGTP
Target:
2'-Deoxy-2'-fluoroadenosine-5'-O-triphosphate sodium
Cat.No: T83830
Synonym: 2′-fluoro-2′-deoxy ATP,AfTP,2'-fluoro dATP
Target:
Cycloleucine
Cat.No: T9626
Synonym:
Target: NMDAR
Glibornuride
Cat.No: T15385
Synonym:
Target: Potassium Channel
SB 204990
Cat.No: T16861
Synonym:
Target: ATP Citrate Lyase
NDI-091143
Cat.No: T7424
Synonym:
Target: ATP Citrate Lyase
GAK inhibitor 49
Cat.No: T8535
Synonym:
Target: Serine/threonin kinase
6-Aminonicotinamide
Cat.No: T7545
Synonym:
Target: Others
BMS-303141
Cat.No: T2337
Synonym: BMS 303141
Target: ATP Citrate Lyase
5-BDBD
Cat.No: T22518
Synonym:
Target: P2X Receptor
Cat. No. Product Name Target Signaling Pathways
T20089 ATP

Atipi,ATP disodium salt hydrate,Triphosphoric acid adenosine ester,Ara-ATP,Triphosphaden,Adenosine triphosphate;Ara-ATP,Adenosine triphosphate

Endogenous Metabolite Metabolism
ATP (Adenosine triphosphate) 可为细胞提供能量,参与整体能量平衡,维持细胞内稳态。ATP 可以通过与特异性嘌呤能受体的相互作用充当细胞外信号分子,以介导神经传递、炎症、细胞凋亡和骨重塑等多种过程。
T1352 ATP disodium salt

Adenosine 5'-triphosphate disodium salt,三磷酸腺苷二钠,ATP,ATP disodium,腺苷-5'-三磷酸二钠盐,Adetide,Adenosine-Triphosphate,Disodium adenosine triphosphate

P2X Receptor; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism; Neuroscience
ATP disodium salt (Adenosine-Triphosphate) 是体内能量储存的重要物质,为代谢提供能量,同时在细胞中作为辅酶发挥作用。Adenosine 5'-triphosphate disodium salt 也是免疫和炎症中重要的内源性信号分子。
T2812 ATP disodium salt hydrate

ATP disodium,ATP disodium salt,Adenosine disodium triphosphate,三磷酸腺苷二钠盐

Others; Endogenous Metabolite Metabolism; Others
ATP disodium salt hydrate (Adenosine disodium triphosphate) 是体内能量储存和代谢的重要物质,为代谢提供能量,同时在细胞中作为辅酶发挥作用。同时,它是也是免疫和炎症中重要的内源性信号分子。
T64980 ATP disodium trihydrate

Adenosine-5'-triphosphate disodium trihydrate

Endogenous Metabolite Metabolism
ATP disodium trihydrate (Adenosine-5'-triphosphate disodium trihydrate) 是体内能量储存和代谢的重要物质,是免疫和炎症中重要的内源性信号分子,可为机体代谢提供能量,同时在细胞中作为辅酶发挥作用。
T40526 ATP dipotassium

腺苷三磷酸二钾盐,Adenosine5'-triphosphatedipotassium

ATP dipotassium (Adenosine 5'-triphosphate dipotassium) is a vital compound involved in energy storage and metabolism within living organisms. It plays a crucial role in supplying metabolic energy for driving pumps and acts as a coenzyme in cellular processes. Additionally, ATP dipotassium functions as a significant endogenous signaling molecule contributing to immunity and inflammation.
T11590 (-)-Hydroxycitric acid

Garcinia acid,(-)-羟基柠檬酸

ATP Citrate Lyase Metabolism
(-)-Hydroxycitric acid (Garcinia acid) 是Garcinia cambogia 果皮中的主要酸。它是 ATP 柠檬酸裂解酶的竞争性抑制剂,能够抑制脂肪酸的合成,减少脂肪生成,控制食物摄入,从而减轻体重。
T6323 Oligomycin A

MCH 32,寡霉素A

ATPase; Antibiotic; Antifungal Membrane transporter/Ion channel; Microbiology/Virology
Oligomycin A (MCH 32) 是从链霉菌属中得到的一种线粒体F0F1-ATPase 抑制剂,抑制氧化磷酸化和线粒体偶联膜上发生的所有 ATP 依赖性过程。
T11589 Hydroxycitric acid tripotassium hydrate

柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate

ATP Citrate Lyase; HIF/HIF Prolyl-Hydroxylase; HIF Angiogenesis; Chromatin/Epigenetic; Metabolism
Hydroxycitric acid tripotassium hydrate (Potassium citrate monohydrate) 是一种藤黄果的主要活性成分,也是一种柠檬酸的衍生物。它可竞争性抑制柠檬酸裂解酶 (ATP citrate lyase) ,并具有减肥作用。它有效抑制结石形成,并抑制HIF,具有抗氧化,抗炎和抗肿瘤活性。
T3S0156 Atractyloside potassium salt

Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐

Others Others
Atractyloside potassium salt (Atractyloside Dipotassium Salt) 是一种从苍术果实中分离出得到的二萜苷类化合物,具有毒性。它能抑制大鼠心脏线粒体膜的氯离子通道。它是高效、特异性的线粒体 ADP/ATP 转运 (ADP/ATP transport) 抑制剂。
T12045 (-)-Hydroxycitric acid lactone

藤黄内酯,Garcinia lactone

ATP Citrate Lyase Metabolism
(-)-Hydroxycitric acid lactone (Garcinia lactone) 是一种有效的 ATP-柠檬酸裂解酶抑制剂,能够催化柠檬酸盐线粒体外裂解为草酰乙酸和乙酰辅酶 A,限制了脂肪酸合成所需乙酰辅酶 A 单位的可用性。它是一种减肥药,是一种广受欢迎的减肥食品补充剂。
T5544 2-Furoic acid

Furan-2-carboxylic acid,糠酸

Anti-infection; ATP Citrate Lyase; Endogenous Metabolite; Acyltransferase Metabolism; Microbiology/Virology
2-Furoic acid (Furan-2-carboxylic acid) 2-Furoic acid 能够降低血清中胆固醇和甘油三酯的水平,具有抗血脂作用。
T0256 Citric acid trilithium salt tetrahydrate

Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate

Dehydrogenase; GSK-3; HIF/HIF Prolyl-Hydroxylase; Antibacterial; GluR Chromatin/Epigenetic; Metabolism; Microbiology/Virology; Neuroscience; PI3K/Akt/mTOR signaling; Stem Cells
Citric acid trilithium salt tetrahydrate (Lithium citrate tribasic tetrahydrate) 是一种用于治疗精神疾病的药物。它也是一种医药和建筑材料, 可用于氨基酸定量分析时的梯度洗脱。
T3981 Acacetin

4'-Methoxyapigenin,金合欢素,5,7-Dihydroxy-4'-methoxyflavone,Linarigenin

Apoptosis; IAP; COX; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; Neuroscience
Acacetin (5,7-Dihydroxy-4'-methoxyflavone) 是一种来自狗舌草的口服有效类黄酮。它停在 PI3Kγ 的 ATP 结合口袋中,可导致癌细胞周期停滞,并诱导细胞凋亡和自噬。它有抗癌和抗炎活性,有潜力研究疼痛相关疾病。
TN2019 Orobol

3'-Hydroxygenistein,3’,4’,5,7-tetrahydroxy-isoflavon,3',4',5,7-四羟基异黄酮

BCL; Caspase; PI3K Apoptosis; PI3K/Akt/mTOR signaling; Proteases/Proteasome
Orobol (3’,4’,5,7-tetrahydroxy-isoflavon) 是酪氨酸特异性蛋白激酶和磷脂酰肌醇转换的抑制剂。Orobol 抑制 PI3K,对 PI3K α/β/γ/K/δ 的 IC50 为 3.46-5.27 μM。 Orobol 具有抗皮肤老化和抗肥胖的作用。
T40426 Cytidine 5'-diphosphate trisodium salt

CDP,胞苷5'-二磷酸三钠盐水合物,胞苷-5-二磷酸三钠盐,胞苷-5'-二磷酸三钠盐

Others Others
Cytidine 5'-diphosphate trisodium salt (CDP) 可通过尿苷单磷酸激酶 (UMPK) 催化将磷酸基从 ATP 转移到胞苷一磷酸 (CMP) 生成用于合成 DNA 和 RNA 的胞苷三磷酸。
T7475 S-Adenosyl-L-methionine

AdoMet,Ademetionine,SAMe,S-Adenosyl methionine,S-腺苷-L-蛋氨酸

Others; Endogenous Metabolite Metabolism; Others
S-Adenosyl-L-methionine (Ademetionine) 是一种具有有效的抗抑郁和减轻疼痛作用的膳食补充剂,是通过蛋氨酸腺苷转移酶的作用由蛋氨酸和 ATP 内源性生产的,是一种重要的口服具有活力的甲基供体,能够用于肝病和骨关节炎的研究。
T8170 Carboxyatractyloside

羧基苍术苷,Gummiferin,Carboxyatractyloside tripotassium salt

Others Others
Carboxyatractyloside (Carboxyatractyloside tripotassium salt) tripotassium salt 是一种 ADP/ATP 载体蛋白 (ADP/ATP carrier) 抑制剂,抑制线粒体 ADP/ATP 的转运。它是一种具有毒性的天然产物,
T0465 Ellagic acid

鞣花酸,Gallogen,Elagostasine

Hedgehog/Smoothened; Casein Kinase; Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; PKA; Syk; PKC; Carbonic Anhydrase Angiogenesis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; Metabolism; NF-κB; Stem Cells; Tyrosine Kinase/Adaptors
Ellagic acid (Gallogen) 是从 Eucalyptus maculata Hook 和 E. Hemipholia F. Muell 的 kino 中分离出来的稠合四环天然产物,是一种有效的,ATP 竞争性的CK2抑制剂,IC50和Ki 值分别为 40 nM 和 20 nM。
T3S0870 Paederosidic acid methyl ester

鸡屎藤苷酸甲酯,紫草酸甲酯

ATPase; Potassium Channel; NO Synthase Immunology/Inflammation; Membrane transporter/Ion channel
Paederosidic acid methyl ester 是 ATP 敏感的 K+channel 通道激活剂,分离自 P. scandens。它通过激活脑中和脊髓水平中 ATP 敏感型 K+通道提高了痛觉阈值,表现出显著的中枢缓解疼痛活性。
T4888 Phosphocreatine disodium hydrate

磷酸肌酸二钠盐,Phosphocreatine disodium salt hydrate

Others; Endogenous Metabolite Metabolism; Others
Phosphocreatine disodium hydrate 是内源性代谢产物的一种。
T21494 Oligomycin

HIF Angiogenesis; Chromatin/Epigenetic
Oligomycin 是一种抗真菌抗生素,是 H+-ATP 合成酶的抑制剂。Oligomycin 能够阻断氧化磷酸化和电子传递链。Oligomycin 对缺氧性肿瘤细胞 HIF-1alpha 表达具有抑制作用。
T3419 Chelerythrine chloride

白屈菜红碱,盐酸白屈菜红碱

Apoptosis; BCL; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling
Chelerythrine chloride 是一种可渗透细胞的蛋白激酶 C 抑制剂,对磷酸盐受体具有竞争性,而对 ATP 是非竞争性的。它诱导细胞凋亡和自噬。
T22300 Creatine monohydrate

Methylguanidoacetic acid monohydrate,一水肌酸

Others; Endogenous Metabolite Metabolism; Others
Creatine monohydrate (Methylguanidoacetic acid monohydrate) 是磷酸原能量系统的关键参与者,尤其是在肌肉和大脑中。 Creatine monohydrate 是高强度、短期活动中 ATP 的主要来源。
T20003 Acridone

Antibacterial; ABC Membrane transporter/Ion channel; Microbiology/Virology
Acridone 具有抗菌、抗疟、抗病毒和抗肿瘤活性。它可诱导细胞凋亡,抑制 ABCG2 蛋白,并调节激素水平。
Fr14207 (-)-Isopulegol

Others Others
(-)-Isopulegol 具有抗氧化和神经活性特性。它还具有由异胡薄荷醇诱导的胃保护作用,似乎至少部分由内源性前列腺素介导,K+ATP 通道开放和与 GSH 相关的抗氧化特性增加。
T6680 Staurosporine

Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素

Apoptosis; PKA; Antibacterial; Antibiotic; Src; PKC; Antifungal Angiogenesis; Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Tyrosine Kinase/Adaptors
Staurosporine (AM-2282) 是一种蛋白激酶抑制剂,对 PKC、PKA、c-Fgr、Phosphorylase kinase 和 TAOK2 均有抑制活性 (IC50=6/15/2/3/3000 nM),具有 ATP 竞争性和非选择性。Staurosporine 也可以诱导凋亡。
T25192 Butyrolactone I

Olomoucin,丁酸内酯I

CDK Cell Cycle/Checkpoint
Butyrolactone I (Olomoucin) 是 CDK 和 cdc2 激酶家族的 ATP 竞争性抑制剂。 Butyrolactone I 在非小细胞肺、小细胞肺和前列腺癌细胞系中显示出抗肿瘤作用。
T3313 D-Luciferin

Firefly luciferin,D-萤光素,D-荧光素,D-(-)-Luciferin

Others Others
D-Luciferin (D-(-)-Luciferin) 是一种萤光素酶的底物,能够催化生物发光昆虫产生典型的黄绿光。
T3929 Kaurenoic acid

Kauren-19-Oic Acid,异贝壳杉烯酸,kaurenoate,kaur-16-en-18-oic acid

Others Others
Kaurenoic acid (kaurenoate) 是一种二萜,来源于 Sphagneticola trilobata 中,可以抑制细胞因子的产生和激活 NO–cyclic GMP–PKG–ATP- 敏感型钾通道信号通路,并抑制炎症疼痛。
T4739 Sodium creatine phosphate dibasic tetrahydrate

磷酸肌酸二钠盐,Creatine phosphate disodium salt tetrahydrate

Others; Endogenous Metabolite Metabolism; Others
Sodium creatine phosphate dibasic tetrahydrate (Creatine phosphate disodium salt tetrahydrate) 主要存在于脊椎动物的骨骼肌中,是测定肌酸激酶的底物,能够用于骨骼肌收缩过程中 ATP 的再生。
T0064 Adenine

Vitamin B4,腺嘌呤,6-Aminopurine

DNA/RNA Synthesis; Endogenous Metabolite; AChR Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Neuroscience
Adenine (6-Aminopurine) 是一种嘌呤衍生物,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T17143 Toyocamycin

丰加霉素,Vengicide

Apoptosis; Others; IRE1; Antibiotic; Antifungal Apoptosis; Cell Cycle/Checkpoint; Microbiology/Virology; Others
Toyocamycin (Vengicide) 是放线菌类产生的腺苷类似物,为 X 盒结合蛋白 1 (XBP1) 抑制剂,抑制 IRE1α 诱导的 ATP 依赖性 XBP1 mRNA 的断裂,IC50值为 80 nM。它还诱导凋亡。
TL0009 coniferin

Coniferoside,松柏苷,Abietin

Others; Antifungal Microbiology/Virology; Others
Coniferin (Abietin) 是一种松柏醇中的葡萄糖苷。它抑制真菌生长和黑化反应,具有 ATP 依赖性转运活性并具有抗氧化作用。
T5079 Adenosine 5'-diphosphate sodium salt

腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt

Others; Endogenous Metabolite Metabolism; Others
Adenosine 5'-diphosphate sodium salt (ADP sodium salt) 是一种核苷二磷酸,是一种 ATP 酶对 ATP 去磷酸化的产物。它通过在 P2T-嘌呤受体上的作用诱导人血小板聚集并抑制刺激的腺苷酸环化酶。
TN4883 Quinine sulfate dihydrate

奎宁树

Others Others
Quinine sulfate dihydrate 在钾通道阻滞剂中起主要作用。它也被用作抗疟疾、抗胆碱能、抗高血压和降糖药。它抑制线粒体atp 调节的钾通道。它也被用来研究生物结晶血红素,血红素,在疟疾寄生虫的代谢和研究血红素(FP)复合物的毒性。
T5067 Flavin adenine dinucleotide disodium salt

Flavin Adenine Dinucleotide Disodium,黄素腺嘌呤二核苷酸二钠,FAD sodium salt,FAD-Na2

Others; Endogenous Metabolite Metabolism; Others
Flavin adenine dinucleotide disodium salt (FAD sodium salt) 是一种辅酶,作用是促进细胞氧化还原反应中黄素酶的电子转移。
T1723 Adenosine 5'-diphosphate

腺苷5'-二磷酸,Adenosine diphosphate,adenosine pyrophosphate,ADP

Endogenous Metabolite Metabolism
Adenosine 5'-diphosphate (ADP) 是一种嘌呤核糖核苷5'-二磷酸,是 ATPATP 酶作用下去磷酸化的产物。Adenosine 5'-diphosphate (adenosine pyrophosphate) 可诱导人血小板聚集并通过作用于P2T-嘌呤受体抑制受刺激的腺苷酸环化酶。
T4786 D-Ribose(mixture of isomers)

D-Ribose,D-(-)-Ribose,D-(-)-核糖

Others; Endogenous Metabolite Metabolism; Others
D-Ribose(mixture of isomers) (D-(-)-Ribose) 是 ATP 的糖部分,可作为能量增强剂,被广泛用作慢性疲劳综合症和心肌能量代谢的代谢疗法补充剂。它在蛋白质糖化中具有特性,能够 RAGE 依赖的方式诱导 NF-Κb 炎症。
T10857 Coenzyme A

Endogenous Metabolite Metabolism
Coenzyme A 是所有活细胞中必需的辅助因子,由泛酸,三磷酸腺苷和半胱氨酸合成的。Coenzyme A 与过氧化物酶 5 共价结合导致其过氧化物酶活性完全抑制,通过 DTT 还原能够逆转。Coenzyme A 及其硫酯衍生物是主要分解代谢,合成代谢途径和基因表达调控的关键参与者。
T4897 Inosine-5'-triphosphate trisodium salt

ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt

Others; Endogenous Metabolite Metabolism; Others
Inosine-5'-triphosphate trisodium salt (ITP) 是三磷酸核苷,能够作为 ATPases 和 GTPases 的底物。
T3228 Fosfructose

D-fructose-1,6-diphosphate,Betulanonaprenol,4937-84-2,Diphosphofructose,二磷酸果糖,Fructose 1,6-diphosphate,D-fructofuranose 1,6-bisphosphate,Esafosfan

Others; Endogenous Metabolite Metabolism; Others
D-fructose-1,6-diphosphate 是一种细胞保护性的天然糖磷酸盐,Fosfructose 通过刺激无氧糖酵解起作用,其在缺血条件下产生三磷酸腺苷,有潜力用于心血管缺血,镰状细胞性贫血和哮喘的研究。
T3375 Verbascoside

毛蕊花苷,麦角甾苷,Kusaginin,Acteoside,TJC160

Apoptosis; PARP; Antibacterial; PKC; p53; HSV Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; Microbiology/Virology
Verbascoside (Kusaginin) 是从Lantana camara 中得到的糖苷类物质,是具有ATP 竞争性的PKC 抑制剂,IC50值为 25 µM,它还有抗炎,抗肿瘤,抗神经性疼痛等作用。
T6354 (+)-Usnic acid

D-Usnic Acid,松萝酸,(+)-Usniacin,(+)-地衣酸

Antiviral; Antibacterial; mTOR Immunology/Inflammation; Microbiology/Virology; PI3K/Akt/mTOR signaling
(+)-Usnic acid (D-Usnic Acid) 是地衣中的二苯并呋喃衍生物,可结合 mTOR 的 ATP 结合口袋,抑制 mTORC1/2的活性。它诱导自噬,有抗菌和抗肿瘤活性。
T4737 2'-Deoxyadenosine-5'-monophosphate

D-AMP,2′-脱氧腺苷-5′-单磷酸,2'-Deoxyadenosine 5'-monophosphate,2'-脱氧腺苷-5'-单磷酸

Others; Endogenous Metabolite Metabolism; Others
2'-Deoxyadenosine-5'-monophosphate (D-AMP) 是一种存在于 DNA 中的脱氧核糖核苷酸,是一种核酸 AMP 衍生物。它能够用于研究 DNA 合成和 DNA 损伤过程中基于腺苷的相互作用。
T4826 L-Histidine monohydrochloride monohydrat

Others; Endogenous Metabolite Metabolism; Others
L-Histidine monohydrochloride monohydrat 是一种 α-氨基酸。 L-异构体是 22 种蛋白质氨基酸之一,即蛋白质的组成部分。
T8061 Citronellal

(±)-Citronellal,香茅醛

Others Others
Citronellal ((±)-Citronellal) 是多种芳香植物精油的单萜烯,具有促进睡眠、安定和抗伤害的作用。它可以降低机械伤害感受,且部分通过 NO-cGMP-ATP 敏感型 K⁺渠道通道介导的。
T6225 Adenine hydrochloride

Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Adenine hydrochloride (6-Aminopurine hydrochloride) 是一种嘌呤,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T4861 trans-Aconitic acid

ATPase; Endogenous Metabolite Membrane transporter/Ion channel; Metabolism
trans-Aconitic acid 是反式丙酮酸2-甲基转移酶的底物,存在于正常人尿液中,大量存在于 Reye 综合征和有机酸尿症。
T6369 Adenine hemisulfate

硫酸腺嘌呤,Diadenine sulphate,Adenine sulfate,Adeninsulfat,1H-嘌呤-6-胺硫酸盐

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Adenine hemisulfate (Diadenine sulphate) 是一种嘌呤,是一种核碱基。它在细胞呼吸、以富含能量的 ATP 和 NAD 和 FAD 的形式和蛋白质合成作用,作为 DNA 和 RNA 的化学成分。
T8270 Deserpidine

地舍平,Harmonyl

RAAS Endocrinology/Hormones
Deserpidine (Harmonyl) 是从 Rauwolfia canescens 的根中分离的生物碱。Deserpidine 与 Reserpine 相关。Deserpidine 是竞争性血管紧张素转化酶抑制剂,可以被用作抗高血压药以及镇定剂。Deserpidine 还减少了肾上腺皮质血管紧张素 II 诱导的醛固酮分泌。
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天然产物

ATP
Cat.No: T20089
Synonym: Atipi,ATP disodium salt hydrate,Triphosphoric acid adenosine ester,Ara-ATP,Triphosphaden,Adenosine triphosphate;Ara-ATP,Adenosine triphosphate
Target: Endogenous Metabolite
ATP disodium salt
Cat.No: T1352
Synonym: Adenosine 5'-triphosphate disodium salt,三磷酸腺苷二钠,ATP,ATP disodium,腺苷-5'-三磷酸二钠盐,Adetide,Adenosine-Triphosphate,Disodium adenosine triphosphate
Target: P2X Receptor, Endogenous Metabolite
ATP disodium salt hydrate
Cat.No: T2812
Synonym: ATP disodium,ATP disodium salt,Adenosine disodium triphosphate,三磷酸腺苷二钠盐
Target: Others, Endogenous Metabolite
ATP disodium trihydrate
Cat.No: T64980
Synonym: Adenosine-5'-triphosphate disodium trihydrate
Target: Endogenous Metabolite
ATP dipotassium
Cat.No: T40526
Synonym: 腺苷三磷酸二钾盐,Adenosine5'-triphosphatedipotassium
Target:
(-)-Hydroxycitric acid
Cat.No: T11590
Synonym: Garcinia acid,(-)-羟基柠檬酸
Target: ATP Citrate Lyase
Oligomycin A
Cat.No: T6323
Synonym: MCH 32,寡霉素A
Target: ATPase, Antibiotic, Antifungal
Hydroxycitric acid tripotassium hydrate
Cat.No: T11589
Synonym: 柠檬酸钾一水合物,三水合钾柠檬酸,Potassium citrate monohydrate
Target: ATP Citrate Lyase, HIF/HIF Prolyl-Hydroxylase, HIF
Atractyloside potassium salt
Cat.No: T3S0156
Synonym: Atractyloside Dipotassium Salt,苍术苷钾盐,苍术苷二钾盐
Target: Others
(-)-Hydroxycitric acid lactone
Cat.No: T12045
Synonym: 藤黄内酯,Garcinia lactone
Target: ATP Citrate Lyase
2-Furoic acid
Cat.No: T5544
Synonym: Furan-2-carboxylic acid,糠酸
Target: Anti-infection, ATP Citrate Lyase, Endogenous Metabolite, Acyltransferase
Citric acid trilithium salt tetrahydrate
Cat.No: T0256
Synonym: Lithium citrate tribasic tetrahydrate,柠檬酸三锂盐四水合物,Trilithium citrate tetrahydrate
Target: Dehydrogenase, GSK-3, HIF/HIF Prolyl-Hydroxylase, Antibacterial, GluR
Acacetin
Cat.No: T3981
Synonym: 4'-Methoxyapigenin,金合欢素,5,7-Dihydroxy-4'-methoxyflavone,Linarigenin
Target: Apoptosis, IAP, COX, Autophagy
Orobol
Cat.No: TN2019
Synonym: 3'-Hydroxygenistein,3’,4’,5,7-tetrahydroxy-isoflavon,3',4',5,7-四羟基异黄酮
Target: BCL, Caspase, PI3K
Cytidine 5'-diphosphate trisodium salt
Cat.No: T40426
Synonym: CDP,胞苷5'-二磷酸三钠盐水合物,胞苷-5-二磷酸三钠盐,胞苷-5'-二磷酸三钠盐
Target: Others
S-Adenosyl-L-methionine
Cat.No: T7475
Synonym: AdoMet,Ademetionine,SAMe,S-Adenosyl methionine,S-腺苷-L-蛋氨酸
Target: Others, Endogenous Metabolite
Carboxyatractyloside
Cat.No: T8170
Synonym: 羧基苍术苷,Gummiferin,Carboxyatractyloside tripotassium salt
Target: Others
Ellagic acid
Cat.No: T0465
Synonym: 鞣花酸,Gallogen,Elagostasine
Target: Hedgehog/Smoothened, Casein Kinase, Reactive Oxygen Species, Topoisomerase, Endogenous Metabolite, PKA, Syk, PKC, Carbonic Anhydrase
Paederosidic acid methyl ester
Cat.No: T3S0870
Synonym: 鸡屎藤苷酸甲酯,紫草酸甲酯
Target: ATPase, Potassium Channel, NO Synthase
Phosphocreatine disodium hydrate
Cat.No: T4888
Synonym: 磷酸肌酸二钠盐,Phosphocreatine disodium salt hydrate
Target: Others, Endogenous Metabolite
Oligomycin
Cat.No: T21494
Synonym:
Target: HIF
Chelerythrine chloride
Cat.No: T3419
Synonym: 白屈菜红碱,盐酸白屈菜红碱
Target: Apoptosis, BCL, PKC, Autophagy
Creatine monohydrate
Cat.No: T22300
Synonym: Methylguanidoacetic acid monohydrate,一水肌酸
Target: Others, Endogenous Metabolite
Acridone
Cat.No: T20003
Synonym:
Target: Antibacterial, ABC
(-)-Isopulegol
Cat.No: Fr14207
Synonym:
Target: Others
Staurosporine
Cat.No: T6680
Synonym: Antibiotic AM-2282,星形孢菌素,AM-2282,CGP 41251,星孢菌素
Target: Apoptosis, PKA, Antibacterial, Antibiotic, Src, PKC, Antifungal
Butyrolactone I
Cat.No: T25192
Synonym: Olomoucin,丁酸内酯I
Target: CDK
D-Luciferin
Cat.No: T3313
Synonym: Firefly luciferin,D-萤光素,D-荧光素,D-(-)-Luciferin
Target: Others
Kaurenoic acid
Cat.No: T3929
Synonym: Kauren-19-Oic Acid,异贝壳杉烯酸,kaurenoate,kaur-16-en-18-oic acid
Target: Others
Sodium creatine phosphate dibasic tetrahydrate
Cat.No: T4739
Synonym: 磷酸肌酸二钠盐,Creatine phosphate disodium salt tetrahydrate
Target: Others, Endogenous Metabolite
Adenine
Cat.No: T0064
Synonym: Vitamin B4,腺嘌呤,6-Aminopurine
Target: DNA/RNA Synthesis, Endogenous Metabolite, AChR
Toyocamycin
Cat.No: T17143
Synonym: 丰加霉素,Vengicide
Target: Apoptosis, Others, IRE1, Antibiotic, Antifungal
coniferin
Cat.No: TL0009
Synonym: Coniferoside,松柏苷,Abietin
Target: Others, Antifungal
Adenosine 5'-diphosphate sodium salt
Cat.No: T5079
Synonym: 腺苷-5‘-二磷酸钠盐,Adenosine-5'-diphosphate trisodium salt,ADP sodium salt
Target: Others, Endogenous Metabolite
Quinine sulfate dihydrate
Cat.No: TN4883
Synonym: 奎宁树
Target: Others
Flavin adenine dinucleotide disodium salt
Cat.No: T5067
Synonym: Flavin Adenine Dinucleotide Disodium,黄素腺嘌呤二核苷酸二钠,FAD sodium salt,FAD-Na2
Target: Others, Endogenous Metabolite
Adenosine 5'-diphosphate
Cat.No: T1723
Synonym: 腺苷5'-二磷酸,Adenosine diphosphate,adenosine pyrophosphate,ADP
Target: Endogenous Metabolite
D-Ribose(mixture of isomers)
Cat.No: T4786
Synonym: D-Ribose,D-(-)-Ribose,D-(-)-核糖
Target: Others, Endogenous Metabolite
Coenzyme A
Cat.No: T10857
Synonym:
Target: Endogenous Metabolite
Inosine-5'-triphosphate trisodium salt
Cat.No: T4897
Synonym: ITP,肌苷-5'-三磷酸三钠盐,三磷酸肌苷三钠盐,Inosine 5'-triphosphate trisodium salt
Target: Others, Endogenous Metabolite
Fosfructose
Cat.No: T3228
Synonym: D-fructose-1,6-diphosphate,Betulanonaprenol,4937-84-2,Diphosphofructose,二磷酸果糖,Fructose 1,6-diphosphate,D-fructofuranose 1,6-bisphosphate,Esafosfan
Target: Others, Endogenous Metabolite
Verbascoside
Cat.No: T3375
Synonym: 毛蕊花苷,麦角甾苷,Kusaginin,Acteoside,TJC160
Target: Apoptosis, PARP, Antibacterial, PKC, p53, HSV
(+)-Usnic acid
Cat.No: T6354
Synonym: D-Usnic Acid,松萝酸,(+)-Usniacin,(+)-地衣酸
Target: Antiviral, Antibacterial, mTOR
2'-Deoxyadenosine-5'-monophosphate
Cat.No: T4737
Synonym: D-AMP,2′-脱氧腺苷-5′-单磷酸,2'-Deoxyadenosine 5'-monophosphate,2'-脱氧腺苷-5'-单磷酸
Target: Others, Endogenous Metabolite
L-Histidine monohydrochloride monohydrat
Cat.No: T4826
Synonym:
Target: Others, Endogenous Metabolite
Citronellal
Cat.No: T8061
Synonym: (±)-Citronellal,香茅醛
Target: Others
Adenine hydrochloride
Cat.No: T6225
Synonym: Adenine HCl,腺嘌呤盐酸盐,6-Aminopurine hydrochloride
Target: DNA/RNA Synthesis, Endogenous Metabolite
trans-Aconitic acid
Cat.No: T4861
Synonym:
Target: ATPase, Endogenous Metabolite
Adenine hemisulfate
Cat.No: T6369
Synonym: 硫酸腺嘌呤,Diadenine sulphate,Adenine sulfate,Adeninsulfat,1H-嘌呤-6-胺硫酸盐
Target: DNA/RNA Synthesis, Endogenous Metabolite
Deserpidine
Cat.No: T8270
Synonym: 地舍平,Harmonyl
Target: RAAS
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