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7

抑制剂 & 化合物

178

天然产物

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Cat. No. Product Name Target Signaling Pathways
T0923 Busulfan

Myleran,Sulphabutin,白消安,Busulphan

Apoptosis; DNA Alkylator/Crosslinker; DNA Alkylation Apoptosis; DNA Damage/DNA Repair
Busulfan (Busulphan) 是二甲磺酸盐的合成衍生物,具有抗肿瘤和细胞毒特性。是一种烷化剂,对骨髓具有选择性免疫抑制作用。
T24962 10-Formylfolic acid

DHFR Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
10-Formylfolic acid 是一种新型有效的二氢叶酸还原酶 (dihydrofolate reductase) 抑制剂,可用于研究白血病。
T36898 Sandacanol

Sandranol,2-Ethyl-4-(2,2,3-trimethylcyclopent-3-en-yl)-but-2-en-1-ol

Apoptosis Apoptosis
Sandacanol(Sandranol) 是一种选择性嗅觉受体(OR10H1)激动剂。Sandacanol可诱导膀胱癌细胞的细胞周期停止和部分凋亡,可降低细胞迁移率和增殖率。
T19557 Sanshool

Others Others
Sanshool is a natural product isolated from Zanthoxylum bungeanum. Sanshool improves UVB-induced skin photodamage by targeting JAK2/STAT3-dependent autophagy.
T24776 Secologanate

Secologanic Acid

Secologanate is an inhibitor of plant growth.
T37680 3-hydroxy Palmitic Acid methyl ester

3-hydroxy Palmitic acid methyl ester (3-hydroxy PAME) is an esterized long-chain fatty acid involved in quorum sensing in R. solanacearum, a bacteria that causes lethal wilting in plants. 3-hydroxy-PAME (175 nM) increases levels of PhcA-regulated virulence factors, greater than 20-, 30-, and 25-fold for EPS I, EGL, and PME, respectively, in the AW1-83 strain of R. solanacearum.
T32269 Jasmone, (E)-

EINECS 228-410-7

Jasmone, (E)- is a type of perfuming agent.

化合物

Busulfan
Cat.No: T0923
Synonym: Myleran,Sulphabutin,白消安,Busulphan
Target: Apoptosis, DNA Alkylator/Crosslinker, DNA Alkylation
10-Formylfolic acid
Cat.No: T24962
Synonym:
Target: DHFR
Sandacanol
Cat.No: T36898
Synonym: Sandranol,2-Ethyl-4-(2,2,3-trimethylcyclopent-3-en-yl)-but-2-en-1-ol
Target: Apoptosis
Sanshool
Cat.No: T19557
Synonym:
Target: Others
Secologanate
Cat.No: T24776
Synonym: Secologanic Acid
Target:
3-hydroxy Palmitic Acid methyl ester
Cat.No: T37680
Synonym:
Target:
Jasmone, (E)-
Cat.No: T32269
Synonym: EINECS 228-410-7
Target:
Cat. No. Product Name Target Signaling Pathways
T2S1086 Nepitrin

假荆芥属苷,Nepetin-7-glucoside

Antioxidant oxidation-reduction
Nepitrin (Nepetin-7-glucoside) 分离自Scrophularia striata 中,具有强大的抗炎、抗关节炎作用。
TN2117 Pulsatilloside E

3-O-B-D-葡萄糖( 1→4)-[ A -L-鼠李糖(1→2)]- A-L-阿拉伯糖 23-羟基羽扇豆20(29)-烯-28–酸- 28-O-鼠李糖(1→4)葡萄糖(1→6)葡萄糖苷,Pulchinenoside E,白头翁皂苷E

Others Others
Pulsatilloside E (Pulchinenoside E) 是一种从毛茛科白头翁Pulsatilla chinensis (Ranunculaceae)的根中分离出来的天然产物。
TN1539 Cussosaponin C

Others Others
Cussosaponin C 是从 Pulsatilla koreana Nakai 中分离得到的天然产物。
T3818 Fraxinol

Others; P450 Metabolism; Others
Fraxinol 是一种分离自半边莲中的化合物。
T6S2391 L-Chicoric Acid

(-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸,是一种选择性可逆的 HIV-1 整合酶抑制剂,IC50约为 100 nM。它还可抑制 HIV-1 复制。
T3370 Hederacoside C

常春藤苷C,Kalopanaxsaponin B,Hederasaponin C

Others; Antibacterial Microbiology/Virology; Others
Hederacoside C (Hederasaponin C) 是常春藤的叶子组分中的主要成分,具有祛痰、抗菌、支气管扩张等作用,可研究呼吸系统疾病。
T3910 Pulchinenoside C

Anemoside B4,Chinensioside A,Pulchinenoside B4,白头翁皂苷 B4,Pulsatilla saponin B4

IL Receptor Immunology/Inflammation
Pulchinenoside C (Anemoside B4) 是一种从 P. chinensis 中分离出来的丰富的三萜皂苷,具有抗炎和抗氧化作用。
TN6760 1-Eicosanol

Others Others
1-Eicosanol 是从金丝桃分离得到的天然产物,具有抗氧化作用。
T0562 Protocatechuic acid

3, 4-Dihydroxybenzoic acid,3,4-二羟基苯甲酸,Protocatechuate,原儿茶酸,3,4-Dihydroxybenzoic acid

Others Others
Protocatechuic acid (3, 4-Dihydroxybenzoic acid) 是天然的多酚类物质,具有神经保护活性。
T6S0781 Phellodendrine

黄柏碱,Phallodendrin

Others; NF-κB; Akt Cytoskeletal Signaling; NF-κB; Others; PI3K/Akt/mTOR signaling
Phellodendrine (Phallodendrin) 是异喹啉生物碱,是黄柏皮层中的重要特征成分之一。它具有良好的抗氧化,抗炎作用。它通过调节AKT/NF-κB 途径抵抗 AAPH 诱导的氧化应激。
T3790 Hederacoside D

常春藤苷 D,常春藤苷D;常春藤皂苷D

TNF Apoptosis
Hederacoside D 是从常春藤中分离到的皂苷,具有很高的生物活性。
TN5634 Aureusidin

Auresudidin,金鱼草素,Auresidin

Antioxidant; Reactive Oxygen Species; Lipoxygenase Immunology/Inflammation; Metabolism; NF-κB; oxidation-reduction
Aureusidin (Auresidin) 具有抗氧化和脂氧合酶抑制活性,具有抗炎作用。
TN1377 α-Spinasterol

Α-波菜甾醇,alpha-Spinasterol,菠甾醇

COX; Antibacterial; TRP/TRPV Channel Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
α-Spinasterol 是一种从Spinacia oleracea 分离的瞬时受体电位香草酸 1 拮抗剂,具有抗菌、抗炎、抗抑郁、抗氧化和抗伤害作用。它抑制COX-1和COX-2活性,IC50值分别为 16.17 μM 和 7.76 μM。
TN1142 8-Oxocoptisine

8-Oxycoptisine,8-氧黄连碱

Others Others
8-Oxocoptisine (8-Oxycoptisine) 是天然原小檗碱生物碱,具有抗癌作用。
T5S0055 Chelidonine

Helidonine,Khelidonin,白屈菜碱,Stylophorin

Apoptosis; Others; Influenza Virus Apoptosis; Microbiology/Virology; Others
Chelidonine (Stylophorin) 是白屈菜中的一种异喹啉生物碱,有抗肿瘤和抗病毒作用。它可导致细胞周期 G2/M 停滞,诱导 caspase 依赖和非依赖性的细胞凋亡。
T0878 Diosmin

Venosmine,Diosmil,Barosmin,地奥司明,地奥司明(7-芸香糖甙)

Aryl Hydrocarbon Receptor; Norepinephrine Immunology/Inflammation; Neuroscience
Diosmin (Venosmine) 是在各种柑橘类水果中发现的类黄酮,也是芳烃受体激动剂,有增强血管壁的作用。
T3428 Helicid

Hilicidum,4-formylphenyl-O-β-d-allopyranoside,Helicide,豆腐果苷

Others Others
Helicid (Helicide) 是 Helicia nilgirica Bedd 的主要组成部分。它被用于精神神经症的相关研究,可用于促进安定、睡眠和缓解疼痛。
T2881 Crustecdysone

Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,β-蜕皮甾酮,Hydroxyecdysone,羟基蜕皮激素

Others; Caspase; Endogenous Metabolite; Autophagy Apoptosis; Autophagy; Metabolism; Others; Proteases/Proteasome
Crustecdysone (Hydroxyecdysone) 是来源于露水草的一种蜕皮激素,可调节昆虫的蜕皮或蜕皮过程。它是 Ecdysone 的活性代谢物,通过 20E 核受体复合物 EcR-USP 抑制半胱天冬酶活性并诱导自噬,在心血管系统中具有调节或保护作用。
T5S1959 (-)-Asarinin

Fagarol,Sesamin,细辛脂素,Pseudocubebin,Eleutheroside B4,Episesamin,Asarinin

Antibacterial Microbiology/Virology
(-)-Asarinin (Eleutheroside B4) 是一种主要从 Zanthoxylum armatum 根部提取到的木脂素。
TQ0160 Hydrastine

北美黄连碱,(-)-β-Hydrastine,(1R,9S)-β-Hydrastine

Others Others
Hydrastine ((-)-β-Hydrastine) 是一种天然生物碱,存在于Hydrastis canadensis 和Ranunculaceae 家族其他植物。
T0479 Cytisinicline

野靛碱,Baptitoxine,Cytisine,Baphitoxine,Sophorine,金雀花碱

AChR Neuroscience
Cytisinicline (Sophorine) 是从染料木中提取的一种生物碱,可用于帮助戒烟。它是 α4β2 烟碱乙酰胆碱能受体的部分激动剂,也是含 β4 受体和 α7 受体的偏完全性激动剂。
T8859 NITIDINE

Others Others
NITIDINE 是一种从花椒根中分离出来的具有生物活性的植物苯并菲啶生物碱。它具有抗癌、神经保护、抗疟疾、抗 HIV、镇痛、抗炎和抗真菌活性。
T0965 Histamine

Ergamine,组胺

5-HT Receptor; Endogenous Metabolite; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Histamine (Ergamine) 是通过组胺的酶促脱羧衍生的胺。它是一种强大的胃分泌兴奋剂、支气管平滑肌的收缩剂、血管扩张剂以及中枢作用的神经递质。
T3095 Tyramine

4-hydroxyphenethylamine,酪胺,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine

MAO; Endogenous Metabolite Metabolism; Neuroscience
Tyramine (Uteramine) 是天然存在于体内或某些食物中的氨基酸。Tyramine 有助于调节血压。
T0847 Chenodeoxycholic acid

CDCA,鹅去氧胆酸,Chenodiol

Potassium Channel; FXR; Endogenous Metabolite; Autophagy Autophagy; Membrane transporter/Ion channel; Metabolism
Chenodeoxycholic acid (CDCA) 是一种胆汁酸,通常与甘氨酸或牛磺酸结合。它作为清洁剂溶解脂肪以供肠道吸收,并被小肠重新吸收。它被用作利胆剂、利胆泻药,以及预防或溶解胆结石。
TC0027 beta-Sitosterol acetate

Others Others
beta-Sitosterol acetate 是几种被称为植物甾醇的植物性物质之一。
T3S2152 23-Hydroxybetulinic acid

Anemosapogenin,23-羟基白桦酸

Others Others
23-Hydroxybetulinic acid (Anemosapogenin) 是一种具有抗癌作用的生物化合物。
T5S0803 Columbamine

非洲防己碱,Columbamin,Dehydroisocorypalmine

Others Others
Columbamine (Columbamin) 是一种从植物中提取的季异喹啉生物碱。
TQ0036 Anemarrhenasaponin I

Others Others
Anemarrhenasaponin I 是一种对血小板聚集有显著的抑制作用的传统中药。
T4396 Officinalisinin I

Others Others
Officinalisinin I 是一种甾体皂苷,分离自 Anemarrhena asphodeloides。
T3394 Timosaponin BII

知母皂苷BII,Prototimosaponin A III

Beta Amyloid; Others; BACE Neuroscience; Others
Timosaponin BII (Prototimosaponin A III) 是一种甾体皂苷,发现于知母根茎中,具有神经保护、抗炎和抗氧化作用。
T0760 Cholesterol

Cholesterin,Cholesteryl alcohol,胆固醇

Estrogen Receptor/ERR; MRP; Endogenous Metabolite; ROR Endocrinology/Hormones; Immunology/Inflammation; Metabolism
Cholesterol (Cholesteryl alcohol) 属于天然产物,是哺乳动物中的主要固醇,是一种雌激素相关受体 α (ERRα) 的激动剂。Cholesterol 广泛存在于动物的细胞膜,也是合成几种重要荷尔蒙及胆酸的材料。
T8195 Lotusine

Others Others
Lotusine 是一种提取自Nelumbo nucifera Gaertn 的绿色种胚中的纯生物碱。它能够作用于心肌中动作电位及心脏浦肯野纤维缓慢内向电流。
T5S0802 Palmatine

巴马汀,Berbericinine,Burasaine

Indoleamine 2,3-Dioxygenase (IDO); AChR; AChE; Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic; Metabolism; Neuroscience
Palmatine (Burasaine) 是口服具有活力的、不可逆IDO-1抑制剂。它可以减轻结肠损伤,预防肠道菌群失调和调节色氨酸分解代谢,从而改善DSS (Dextran Sulphate Sodium Salt) 诱发的结肠炎。它有用于结肠炎的研究潜力。
T2910 Flavonol

3-羟基黄酮,3-Hydroxyflavone,3-HF,Flavon-3-ol,3-Hydroxy-2-phenylchromone

Others; Endogenous Metabolite Metabolism; Others
Flavonol (3-Hydroxyflavone) 是内源性代谢产物的一种。
T2870 Matrine

Vegard,苦参碱,Matridin-15-one,Matrinium,α-Matrine,(+)-Matrine

Mitophagy; Ferroptosis; Opioid Receptor; Autophagy Apoptosis; Autophagy; Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Matrine (Vegard) 是一种从槐属植物中分离出来的生物碱,可作为一种κ阿片受体激动剂,有抗肿瘤活性。
T4593 ISOPIMPINELLIN

5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen

Antiviral; DNA/RNA Synthesis; Parasite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Immunology/Inflammation; Microbiology/Virology
Isopimpinellin (4,9-Dimethoxypsoralen) 是从 Pimpinella saxifrage 根部分离得到的一种天然产物,具有抗病毒和抗利什曼病活性。
T2698 Asperosaponin VI

Akebia saponin D,Asperosaponin Ⅵ,川续断皂苷 VI

Apoptosis; Others; Caspase Apoptosis; Others; Proteases/Proteasome
Asperosaponin VI (Akebia saponin D) 是一种来自续断壁的皂苷组分。它通过增加 Bcl-2/Bax 比值,降低活性 caspase-3 表达,以及增强 p-Akt 和 p-CREB,从而抑制缺氧诱导的心肌细胞凋亡。它通过 BMP-2/p38 和 ERK1/2 信号途径诱导成骨细胞分化。
T3804 Neomangiferin

Mangiferin 7-glucoside,新芒果苷

Phosphatase Metabolism
Neomangiferin (Mangiferin 7-glucoside) 是一种天然的 C-glucosyl xanthone,分离自干燥的Anemarrhena asphodeloides 的根茎中。它能够减轻大鼠高脂饮食诱导的非酒精性脂肪性肝病 (NAFLD)。
T2S2295 Timosaponin A1

知母皂苷A1

Others Others
Timosaponin A1 是一种黄酮类甾体皂苷,分离自知母中。
T3395 Timosaponin AIII

Filiferin B,知母皂苷 A-III,AneMarsaponin A3,Timosaponin A3

AChE; mTOR Neuroscience; PI3K/Akt/mTOR signaling
Timosaponin AIII (Timosaponin A3) 是一种乙酰胆碱酯酶活性抑制剂,其IC50=35.4 μM。
T7030 anemarsaponin B

知母皂苷B,知母皂苷 B

p38 MAPK; NF-κB; MEK; COX; NO Synthase Immunology/Inflammation; MAPK; Neuroscience; NF-κB
Anemarsaponin B 是一种甾体皂苷,可降低iNOS 和COX-2的蛋白和 mRNA 水平,减少促炎细胞因子的表达和产生。它通过阻断 IκBα 的磷酸化来抑制NF-κB 的 p65 亚基的核转位,还抑制 MAP 激酶激酶 3/6 (MKK3/6) 和混合谱系激酶 3 的磷酸化。
TN6931 Anemarrhenasaponin Ia

知母皂苷IA,(2S,3R,4S,5S,6R)-2-{[(2R,3R,4S,5R,6R)-4,5-dihydroxy-2-{[(1R,3R,4R,7S,9S,12S,13S,16S,18R)-3-hydroxy-6-methoxy-7,9,13-trimethyl-6-(3-methylbutyl)-5-oxapentacyclo[10.8.0.02,?.0?,?.013,1?]icosan-16-yl]oxy}-6-(hydroxymethyl)oxan-3-yl]oxy}-6-(hydroxymethyl)oxan

Others Others
Anemarrhenasaponin Ia ((2S,3R,4S,5S,6R)-2-{[(2R,3R,4S,5R,6R)-4,5-dihydroxy-2-{[(1R,3R,4R,7S,9S,12S,13S,16S,18R)-3-hydroxy-6-methoxy-7,9,13-trimethyl-6-(3-methylbutyl)-5-oxapentacyclo[10.8.0.02,?.0?,?.013,1?]icosan-16-yl]oxy}-6-(hydroxymethyl)oxan-3-yl]oxy}-6-(hydroxymethyl)oxan) 具有抗炎活性。Anemarrhenasaponin Ia 具有抗炎作用,从知母根茎中分离得到。 Anemarrhenasaponin Ia 抑制 N-甲酰-甲硫氨酰-亮氨酰-苯丙氨酸 (fMLP) 诱导的超氧化物的进一步产生。
TN7064 Candicine

4-Hydroxy-N-Benzeneethanaminium,N, N, N-trimethyltyramine chloride,Candicin,N-Methylhordenine,Tyramine Impurity 1,4-羟基-N,N,N-三甲基-苯乙铵,2-(4-hydroxyphenyl)ethyl-trimethylazanium

Others Others
Candicine (N, N, N-trimethyltyramine chloride) 是来自 Stapelia gigantea 的天然产品。
T5237 Hexadecanedioic acid

1,14-Tetradecanedicarboxylic acid,1,16-Hexadecanedioic acid,Thapsic acid,十六碳二酸

Others; Endogenous Metabolite Metabolism; Others
Hexadecanedioic acid (1,16-Hexadecanedioic acid) 能够与 Sepharose 4B 以共价键结合,比染料树脂更具有特异性,用于去除血浆中的血清白蛋白。
T6S2123 Ginkgolic Acid

Romanicardic acid,Ginkgolic acid I,Ginkgolic acid (15:1),银杏酸C15:1,银杏酸,Ginkgolic acid C15:1

Others; E1/E2/E3 Enzyme Others; Ubiquitination
Ginkgolic Acid (Romanicardic acid) 是一种天然化合物, 在体外实验中抑制SUMOylation,IC50=3.0 μM。
TN1217 2'-O-Methylisoliquiritigenin

Dopamine Receptor; 5-HT Receptor; GABA Receptor GPCR/G Protein; Membrane transporter/Ion channel; Neuroscience
2'-O-Methylisoliquiritigenin 是从洋甘草中分离出来的一种天然产物,是由 NR 中特异性诱导的酶合成的。它上调 5-HT、NE、DA 和 GABA 途径,对 NE 通路有显著影响。
T0937 Riboflavin

Vitamin B2,维生素B2,E101

Endogenous Metabolite Metabolism
Riboflavin (E101),一种人内源性代谢物, 是极易吸收的微量营养素。
TN2703 2,3-Dihydroxy-4-methoxyacetophenone

2',3'-Dihydroxy-4'-methoxyacetophenone,2,3-二羟基-4-甲氧基苯乙酮水合物

Calcium Channel Membrane transporter/Ion channel; Metabolism
2,3-Dihydroxy-4-methoxyacetophenone (2',3'-Dihydroxy-4'-methoxyacetophenone) 是一种从圆锥花草取得的的神经保护化合物。它能够改善认知功能,对阿尔茨海默氏病具有潜在的研究价值。
T7468 (-​)​-​α-​Terpineol

alpha-松油醇,(-)-α-松油醇,α-Terpineol

Others Others
(-​)​-​α-​Terpineol 是白葡萄酒中重要的香气化合物,是一种单萜化合物。
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天然产物

Nepitrin
Cat.No: T2S1086
Synonym: 假荆芥属苷,Nepetin-7-glucoside
Target: Antioxidant
Pulsatilloside E
Cat.No: TN2117
Synonym: 3-O-B-D-葡萄糖( 1→4)-[ A -L-鼠李糖(1→2)]- A-L-阿拉伯糖 23-羟基羽扇豆20(29)-烯-28–酸- 28-O-鼠李糖(1→4)葡萄糖(1→6)葡萄糖苷,Pulchinenoside E,白头翁皂苷E
Target: Others
Cussosaponin C
Cat.No: TN1539
Synonym:
Target: Others
Fraxinol
Cat.No: T3818
Synonym:
Target: Others, P450
L-Chicoric Acid
Cat.No: T6S2391
Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸
Target: Others, HIV Protease
Hederacoside C
Cat.No: T3370
Synonym: 常春藤苷C,Kalopanaxsaponin B,Hederasaponin C
Target: Others, Antibacterial
Pulchinenoside C
Cat.No: T3910
Synonym: Anemoside B4,Chinensioside A,Pulchinenoside B4,白头翁皂苷 B4,Pulsatilla saponin B4
Target: IL Receptor
1-Eicosanol
Cat.No: TN6760
Synonym:
Target: Others
Protocatechuic acid
Cat.No: T0562
Synonym: 3, 4-Dihydroxybenzoic acid,3,4-二羟基苯甲酸,Protocatechuate,原儿茶酸,3,4-Dihydroxybenzoic acid
Target: Others
Phellodendrine
Cat.No: T6S0781
Synonym: 黄柏碱,Phallodendrin
Target: Others, NF-κB, Akt
Hederacoside D
Cat.No: T3790
Synonym: 常春藤苷 D,常春藤苷D;常春藤皂苷D
Target: TNF
Aureusidin
Cat.No: TN5634
Synonym: Auresudidin,金鱼草素,Auresidin
Target: Antioxidant, Reactive Oxygen Species, Lipoxygenase
α-Spinasterol
Cat.No: TN1377
Synonym: Α-波菜甾醇,alpha-Spinasterol,菠甾醇
Target: COX, Antibacterial, TRP/TRPV Channel
8-Oxocoptisine
Cat.No: TN1142
Synonym: 8-Oxycoptisine,8-氧黄连碱
Target: Others
Chelidonine
Cat.No: T5S0055
Synonym: Helidonine,Khelidonin,白屈菜碱,Stylophorin
Target: Apoptosis, Others, Influenza Virus
Diosmin
Cat.No: T0878
Synonym: Venosmine,Diosmil,Barosmin,地奥司明,地奥司明(7-芸香糖甙)
Target: Aryl Hydrocarbon Receptor, Norepinephrine
Helicid
Cat.No: T3428
Synonym: Hilicidum,4-formylphenyl-O-β-d-allopyranoside,Helicide,豆腐果苷
Target: Others
Crustecdysone
Cat.No: T2881
Synonym: Commisterone,B-ecdysone,Commisterone,20-Hydroxyecdysone,Ecdysterone,B-ecdysone,β-蜕皮甾酮,Hydroxyecdysone,羟基蜕皮激素
Target: Others, Caspase, Endogenous Metabolite, Autophagy
(-)-Asarinin
Cat.No: T5S1959
Synonym: Fagarol,Sesamin,细辛脂素,Pseudocubebin,Eleutheroside B4,Episesamin,Asarinin
Target: Antibacterial
Hydrastine
Cat.No: TQ0160
Synonym: 北美黄连碱,(-)-β-Hydrastine,(1R,9S)-β-Hydrastine
Target: Others
Cytisinicline
Cat.No: T0479
Synonym: 野靛碱,Baptitoxine,Cytisine,Baphitoxine,Sophorine,金雀花碱
Target: AChR
NITIDINE
Cat.No: T8859
Synonym:
Target: Others
Histamine
Cat.No: T0965
Synonym: Ergamine,组胺
Target: 5-HT Receptor, Endogenous Metabolite, Histamine Receptor
Tyramine
Cat.No: T3095
Synonym: 4-hydroxyphenethylamine,酪胺,para-tyramine,p-Tyramine,mydrial,Tocosine,Uteramine
Target: MAO, Endogenous Metabolite
Chenodeoxycholic acid
Cat.No: T0847
Synonym: CDCA,鹅去氧胆酸,Chenodiol
Target: Potassium Channel, FXR, Endogenous Metabolite, Autophagy
beta-Sitosterol acetate
Cat.No: TC0027
Synonym:
Target: Others
23-Hydroxybetulinic acid
Cat.No: T3S2152
Synonym: Anemosapogenin,23-羟基白桦酸
Target: Others
Columbamine
Cat.No: T5S0803
Synonym: 非洲防己碱,Columbamin,Dehydroisocorypalmine
Target: Others
Anemarrhenasaponin I
Cat.No: TQ0036
Synonym:
Target: Others
Officinalisinin I
Cat.No: T4396
Synonym:
Target: Others
Timosaponin BII
Cat.No: T3394
Synonym: 知母皂苷BII,Prototimosaponin A III
Target: Beta Amyloid, Others, BACE
Cholesterol
Cat.No: T0760
Synonym: Cholesterin,Cholesteryl alcohol,胆固醇
Target: Estrogen Receptor/ERR, MRP, Endogenous Metabolite, ROR
Lotusine
Cat.No: T8195
Synonym:
Target: Others
Palmatine
Cat.No: T5S0802
Synonym: 巴马汀,Berbericinine,Burasaine
Target: Indoleamine 2,3-Dioxygenase (IDO), AChR, AChE, Aurora Kinase
Flavonol
Cat.No: T2910
Synonym: 3-羟基黄酮,3-Hydroxyflavone,3-HF,Flavon-3-ol,3-Hydroxy-2-phenylchromone
Target: Others, Endogenous Metabolite
Matrine
Cat.No: T2870
Synonym: Vegard,苦参碱,Matridin-15-one,Matrinium,α-Matrine,(+)-Matrine
Target: Mitophagy, Ferroptosis, Opioid Receptor, Autophagy
ISOPIMPINELLIN
Cat.No: T4593
Synonym: 5,8-Dimethoxypsoralen,异茴芹内酯,4,9-Dimethoxypsoralen
Target: Antiviral, DNA/RNA Synthesis, Parasite
Asperosaponin VI
Cat.No: T2698
Synonym: Akebia saponin D,Asperosaponin Ⅵ,川续断皂苷 VI
Target: Apoptosis, Others, Caspase
Neomangiferin
Cat.No: T3804
Synonym: Mangiferin 7-glucoside,新芒果苷
Target: Phosphatase
Timosaponin A1
Cat.No: T2S2295
Synonym: 知母皂苷A1
Target: Others
Timosaponin AIII
Cat.No: T3395
Synonym: Filiferin B,知母皂苷 A-III,AneMarsaponin A3,Timosaponin A3
Target: AChE, mTOR
anemarsaponin B
Cat.No: T7030
Synonym: 知母皂苷B,知母皂苷 B
Target: p38 MAPK, NF-κB, MEK, COX, NO Synthase
Anemarrhenasaponin Ia
Cat.No: TN6931
Synonym: 知母皂苷IA,(2S,3R,4S,5S,6R)-2-{[(2R,3R,4S,5R,6R)-4,5-dihydroxy-2-{[(1R,3R,4R,7S,9S,12S,13S,16S,18R)-3-hydroxy-6-methoxy-7,9,13-trimethyl-6-(3-methylbutyl)-5-oxapentacyclo[10.8.0.02,?.0?,?.013,1?]icosan-16-yl]oxy}-6-(hydroxymethyl)oxan-3-yl]oxy}-6-(hydroxymethyl)oxan
Target: Others
Candicine
Cat.No: TN7064
Synonym: 4-Hydroxy-N-Benzeneethanaminium,N, N, N-trimethyltyramine chloride,Candicin,N-Methylhordenine,Tyramine Impurity 1,4-羟基-N,N,N-三甲基-苯乙铵,2-(4-hydroxyphenyl)ethyl-trimethylazanium
Target: Others
Hexadecanedioic acid
Cat.No: T5237
Synonym: 1,14-Tetradecanedicarboxylic acid,1,16-Hexadecanedioic acid,Thapsic acid,十六碳二酸
Target: Others, Endogenous Metabolite
Ginkgolic Acid
Cat.No: T6S2123
Synonym: Romanicardic acid,Ginkgolic acid I,Ginkgolic acid (15:1),银杏酸C15:1,银杏酸,Ginkgolic acid C15:1
Target: Others, E1/E2/E3 Enzyme
2'-O-Methylisoliquiritigenin
Cat.No: TN1217
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, GABA Receptor
Riboflavin
Cat.No: T0937
Synonym: Vitamin B2,维生素B2,E101
Target: Endogenous Metabolite
2,3-Dihydroxy-4-methoxyacetophenone
Cat.No: TN2703
Synonym: 2',3'-Dihydroxy-4'-methoxyacetophenone,2,3-二羟基-4-甲氧基苯乙酮水合物
Target: Calcium Channel
(-​)​-​α-​Terpineol
Cat.No: T7468
Synonym: alpha-松油醇,(-)-α-松油醇,α-Terpineol
Target: Others
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