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30

抑制剂 & 化合物

32

天然产物

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Cat. No. Product Name Target Signaling Pathways
T11020 DHODH-IN-11

Dehydrogenase; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
DHODH-IN-11 是一种来氟米特衍生物和弱二氢乳清酸脱氢酶 (DHODH) 抑制剂,pKa 为 5.03
T21606L Anti-Inflammatory Peptide 1 Acetate

Anti-Inflammatory Peptide 1 Acetate(118850-70-8 Free base)

Phospholipase Metabolism
Anti-Inflammatory Peptide 1 Acetate 在体内具有有效的抗炎活性,是磷脂酶 A2 (PLA2) 的强抑制剂,其存在和活性增加会导致某些身体部位的炎症和疼痛。
T41302 Itaconate-alkyne

ITalk

Others Others
Itaconate-alkyne (ITalk) 是一种生物正交探针,用于对炎症性巨噬细胞中的衣康酸进行定量和位点特异性化学蛋白质组学分析,并能够对其直接靶标进行生化评估和蛋白质组学分析。
T22358 Etalocib

LY293111,VML295

Apoptosis; Leukotriene Receptor; LTR Apoptosis; GPCR/G Protein; Immunology/Inflammation
Etalocib (LY293111) 是一种具有口服活性的白三烯(LTB4)受体的拮抗剂,抑制 [3H]LTB4结合的 Ki 值为 25 nM。它还可诱导凋亡。它抑制 LTB4诱导的钙动员,lC50值为 20 nM。
T1163 Betamethasone valerate

Betnovate,倍他米松戊酸酯,Betaderm,Betamethasone 17-valerate,Luxiq

Glucocorticoid Receptor Endocrinology/Hormones
Betamethasone valerate (Luxiq) 的 17 戊酸酯,是一种具有抗炎活性的局部皮质类固醇。它能够抑制放射标记的糖皮质激素地塞米松与人表皮(IC50:5 nM)及小鼠皮肤(IC50:6 nM)的结合。它可用于研究复发性口疮。
T0383 Fenspiride hydrochloride

Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利

Adrenergic Receptor; PDE; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Metabolism; Neuroscience
Fenspiride hydrochloride (Decaspiride) 是一种口服活性的非甾体抗炎剂,是 H1-组胺受体的拮抗剂,可用于呼吸系统疾病的研究。
T12856 SC-26196

ALPHA,ALPHA-二苯基-4-[(3-吡啶亚甲基)氨基]-1-吡嗪戊腈

Others Others
SC-26196 是一种 Delta6 去饱和酶 (D6D, FADS2) 抑制剂 (在大鼠肝微粒体中,IC50=0.2 µM),具有口服活性,具有抗炎作用。
T10091 Anti-inflammatory agent 1

Others Others
Anti-inflammatory agent 1 is an anti-inflammatory compound.
T64332 Glimepiride sulfonamide

Immunology/Inflammation related Immunology/Inflammation
Glimepiride sulfonamide 是一种抗炎活性化合物。
T0270 Hydrocortisone 17-butyrate

丁酸氢化可的松,Cortisol 17-butyrate,Hydrocortisone butyrate

Glucocorticoid Receptor; Annexin A; Adrenergic Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) 是一种肾上腺皮质激素类药物。
T40380 17α-Hydroxyprogesterone acetate

Others Others
17α-Hydroxyprogesterone acetate 具有孕激素活性和抗炎活性。
T19694 Hydronidone

F351,F-351,F 351

Others Others
Hydronidone (F-351) 是一种 pyridine 衍生物。Hydronidone 对肝纤维化具有潜在的治疗作用。
T1586 Tenoxicam

Ro-12-0068,替诺昔康,Tenoxicamum,Mobiflex,Tilcotil

COX Immunology/Inflammation; Neuroscience
Tenoxicam (Tilcotil) 是一种抗炎化合物,具有退热止痛作用。
T27167 Diclofenac Acyl Glucuronide

Diclofenac Acyl Glucuronide is a major biliary metabolite of Diclofenac (GLXC-07892), a nonsteroidal antiinflammatory drug and COX inhibitor.
T15774 Losmiprofen

Others Others
Losmiprofen is a nonsteroidal compound of antiinflammatory.
T11271 Fenclozine

Others Others
Fenclozine is a non-steroidal antiinflammatory drug.
T7710L Mofebutazone sodium

BRN0213056,BRN 0213056,BRN-0213056

Mofebutazone sodium is, a nonsteroidal antiinflammatory drug (NSAID), is used to treat joint and muscular pain.
T15126 Diflumidone

二氟米酮,R807

Others Others
Diflumidone, a non-steroidal, is an antiinflammatory drug.
T12063 MK-447

Others Others
MK-447 is a nonsteroidal antiinflammatory agent.
T11196 Enazadrem

Lipoxygenase Metabolism
Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.
T26912 Broperamole

Broperamole, an antiinflammatory, has been found to help with gastrointestinal microbleeding.
T12535 Prednisolone Tebutate

Others Others
Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.
T27573 Ibuproxam

Ibuproxamum,G-277

Ibuproxam, a nonsteroidal antiinflammatory drug (NSAID), is used for the treatment of musculoskeletal pain, arthritis, and soft-tissue disorders.
T40461 Ibuprofen alcohol

Ibuprofen alcohol, a nonsteroidal antiinflammatory drug (NSAID), exhibits very little activity for acid-sensing ion channels (ASICs).
T68926 Indomethacin salicylate

Indomethacin salicylate is an antiinflammatory drug. It has shown remarkable inhibitory effects on carrageenin edema, ultraviolet erythema and adjuvant arthritis.
T27658 JNJ-10191584

VUF-6002,JNJ10191584

JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation.
T15021 CV-159

Others Others
CV-159 is a unique dihydropyridine Ca2+ antagonist with antiinflammatory activities. It has an anti-calmodulin (CaM) action.
T60816 Protizinic acid

Protizinic acid 抑制磷脂酶 A2 (PLA2),IC50值为 210 μM。Protizinic acid 是具有抗炎和解热活性的,口服非甾体抗炎剂。
T11998 Meloxicam-d3

Meloxicam D4

Others Others
Meloxicam D4 is deuterium labeled Meloxicam. Meloxicam is a non-steroidal antiinflammatory agent, inhibits COX activity,(Target:COX-1; IC50: 36.6 μM ;(Target:COX-2; IC50: 0.49 μM).
T69491 (E/Z)-Ensifentrine

(E/Z)-Ensifentrine is a potent and selective PDE3/4 inhibitor. (E/Z)-Ensifentrine acts as a long-acting inhibitor of the phosphodiesterase enzymes PDE-3 and PDE-4, producing both bronchodilator and antiinflammatory effects. It is being developed by Verona Pharma as a potential treatment for asthma and hay fever, and is currently in clinical trials.

化合物

DHODH-IN-11
Cat.No: T11020
Synonym:
Target: Dehydrogenase, DNA/RNA Synthesis
Anti-Inflammatory Peptide 1 Acetate
Cat.No: T21606L
Synonym: Anti-Inflammatory Peptide 1 Acetate(118850-70-8 Free base)
Target: Phospholipase
Itaconate-alkyne
Cat.No: T41302
Synonym: ITalk
Target: Others
Etalocib
Cat.No: T22358
Synonym: LY293111,VML295
Target: Apoptosis, Leukotriene Receptor, LTR
Betamethasone valerate
Cat.No: T1163
Synonym: Betnovate,倍他米松戊酸酯,Betaderm,Betamethasone 17-valerate,Luxiq
Target: Glucocorticoid Receptor
Fenspiride hydrochloride
Cat.No: T0383
Synonym: Fenspiride HCl,Pneumorel,Fluiden,Decaspiride,盐酸芬司必利
Target: Adrenergic Receptor, PDE, Histamine Receptor
SC-26196
Cat.No: T12856
Synonym: ALPHA,ALPHA-二苯基-4-[(3-吡啶亚甲基)氨基]-1-吡嗪戊腈
Target: Others
Anti-inflammatory agent 1
Cat.No: T10091
Synonym:
Target: Others
Glimepiride sulfonamide
Cat.No: T64332
Synonym:
Target: Immunology/Inflammation related
Hydrocortisone 17-butyrate
Cat.No: T0270
Synonym: 丁酸氢化可的松,Cortisol 17-butyrate,Hydrocortisone butyrate
Target: Glucocorticoid Receptor, Annexin A, Adrenergic Receptor
17α-Hydroxyprogesterone acetate
Cat.No: T40380
Synonym:
Target: Others
Hydronidone
Cat.No: T19694
Synonym: F351,F-351,F 351
Target: Others
Tenoxicam
Cat.No: T1586
Synonym: Ro-12-0068,替诺昔康,Tenoxicamum,Mobiflex,Tilcotil
Target: COX
Diclofenac Acyl Glucuronide
Cat.No: T27167
Synonym:
Target:
Losmiprofen
Cat.No: T15774
Synonym:
Target: Others
Fenclozine
Cat.No: T11271
Synonym:
Target: Others
Mofebutazone sodium
Cat.No: T7710L
Synonym: BRN0213056,BRN 0213056,BRN-0213056
Target:
Diflumidone
Cat.No: T15126
Synonym: 二氟米酮,R807
Target: Others
MK-447
Cat.No: T12063
Synonym:
Target: Others
Enazadrem
Cat.No: T11196
Synonym:
Target: Lipoxygenase
Broperamole
Cat.No: T26912
Synonym:
Target:
Prednisolone Tebutate
Cat.No: T12535
Synonym:
Target: Others
Ibuproxam
Cat.No: T27573
Synonym: Ibuproxamum,G-277
Target:
Ibuprofen alcohol
Cat.No: T40461
Synonym:
Target:
Indomethacin salicylate
Cat.No: T68926
Synonym:
Target:
JNJ-10191584
Cat.No: T27658
Synonym: VUF-6002,JNJ10191584
Target:
CV-159
Cat.No: T15021
Synonym:
Target: Others
Protizinic acid
Cat.No: T60816
Synonym:
Target:
Meloxicam-d3
Cat.No: T11998
Synonym: Meloxicam D4
Target: Others
(E/Z)-Ensifentrine
Cat.No: T69491
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
TN1006 Tirucallol

NOS; NO Synthase; Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
Tirucallol 是一种四环三萜,分离自Euphorbia lacteal 乳胶。它能够抑制小鼠模型中的耳部水肿,并阻碍脂多糖刺激的巨噬细胞中亚硝酸盐的产生,具有局部消炎作用。
TN1712 Gossypin

NF-κB; S6 Kinase MAPK; NF-κB; PI3K/Akt/mTOR signaling
Gossypin 是一种从Hibiscus vitifolius 中分离得到的黄酮,能够抑制NF-κB 和 NF-κB 的调节基因表达。在小鼠原代骨髓细胞和 RAW264.7 细胞中,它也可抑制 RANKL 诱导的破骨细胞形成。它具有抗氧化、抗炎、抗癌、抗衰老、抗糖尿病和保护肝脏的活性。
T6S2384 Poliumoside

Reductase Endocrinology/Hormones; Metabolism
Poliumoside 是从 Brandisia hancei 的茎和叶中分离出来的咖啡酰化的苯丙烷糖苷。Poliumoside 能够抑制晚期糖基化终产物的形成和大鼠晶状体醛糖还原酶,IC50分别为 19.69 和 8.47 μM。Poliumoside 具有抗炎和抗氧化特性。
TL0007 Bisdemethoxycurcumin

双去甲氧基姜黄素,Curcumin III,Didemethoxycurcumin

Epigenetic Reader Domain; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; Stem Cells
Bisdemethoxycurcumin (Curcumin III) 是一种具有抗炎及抗氧化作用的姜黄素。
T3S0153 Xanthatin

苍耳亭,叶黄制菌素

Apoptosis; VEGFR; Lipoxygenase; Wnt/beta-catenin; Antibacterial Angiogenesis; Apoptosis; Cytoskeletal Signaling; Metabolism; Microbiology/Virology; Stem Cells; Tyrosine Kinase/Adaptors
Xanthatin 是一种从Xanthium strumarium 叶子中提取的天然产物,可诱导细胞凋亡。它抑制布鲁氏菌的IC50值为 2.63 μg/ mL,对寄生虫特异性锥虫硫磷还原酶具有不可逆的弱抑制作用。它通过抑制PGE2的合成和 5-脂氧合酶的活性而显示出抗炎活性。
T8293 γ-Tocopherol

D-gamma-生育酚,γ-生育酚,(+)-γ-Tocopherol

COX Immunology/Inflammation; Neuroscience
γ-Tocopherol ((+)-γ-Tocopherol) 是有效的环氧合酶抑制剂,是存在于玉米油和大豆中的维生素 E,具有抗炎特性和抗癌活性。
T6S1369 Vitexin

牡荆素,Apigenin-8-C-glucoside

Antioxidant oxidation-reduction
Vitexin 是一种存在于多种药用植物(如榕树、螺旋藻)中的 c-糖基化的黄酮。 它具有广泛的药理作用,包括抗氧化,抗癌,抗炎,抗痛觉过敏和神经保护作用。
T3836 Eudesmin

MAPK; S6 Kinase MAPK; PI3K/Akt/mTOR signaling
Eudesmin 通过抑制S6K1信号通路来干扰成脂分化,具有抗肿瘤、抗炎和抗菌活性。
TN1563 Dehydropachymic acid

Autophagy; Immunology/Inflammation related Autophagy; Immunology/Inflammation
Dehydropachymic acid 是从茯苓中分离出的一种三萜类天然产物,有抗炎活性。
TN1047 Ingenol mebutate

Ingenol 3-Angelate,巨大戟醇甲基丁烯酸酯,PEP005

gp120/CD4; HIV Protease; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Ingenol mebutate (Ingenol 3-Angelate) 是 PKC 的有效激动剂,包括 PKC-α、PKC-β、PKC-γ、PKC-δ 和 PKC-ε,Kis 为 0.3、0.105、0.162、0.376 和 0.171 nM。 Ingenol mebutate 具有抗炎和抗肿瘤活性。
T5783 Rosamultin

野蔷薇苷,罗莎白素

Antioxidant; HIV Protease Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Rosamultin 是从Potentilla anserina L 分离的 19 α-羟基型三萜。它抑制 HIV-1 蛋白酶,具有抗氧化、抗炎和镇痛作用。
T3021 Bulleyaconitine A

草乌甲素,Bulleyaconi cine A

Sodium Channel Membrane transporter/Ion channel
Bulleyaconitine A (Bulleyaconi cine A) 是一种分离自乌头属植物的抗炎活性化合物,也可用于缓解疼痛的研究。
TN1490 Chrysoeriol

ERK; p38 MAPK; Akt Cytoskeletal Signaling; MAPK; PI3K/Akt/mTOR signaling
Chrysoeriol 是一种天然黄酮,可从热带植物Coronopus didymus 中提取获得,具有强大的抗氧化功能,能够抑制脂质的过氧化。
T2838 Naringenin

柚皮素,Naringetol,S-Dihydrogenistein,Pelargidanon,Salipurol,NSC 11855,NSC 34875

P450; Influenza Virus; Reactive Oxygen Species; Endogenous Metabolite; PPAR DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Naringenin (NSC-11855) 是葡萄柚中主要的黄烷酮,可作为抗氧化剂、自由基清除剂、抗炎剂、碳水化合物代谢促进剂、免疫系统调节剂。
TCS0862 p-Anisic acid

大茴香酸,对甲氧基苯甲酸,4-Methoxybenzoic acid,Draconic Acid,4-Anisic Acid

Endogenous Metabolite; Antibacterial Metabolism; Microbiology/Virology
4-Methoxybenzoic acid 是anisic acid 的一个异构体,具有抗菌和防腐活性。它可用作化妆品和皮肤科产品的原料,以及食品中的芳香成分。
T0492 Dimethyl fumarate

富马酸二甲酯,DMF

Reactive Oxygen Species; HIV Protease; Nrf2; Endogenous Metabolite; Autophagy Autophagy; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Dimethyl fumarate (DMF) 是具有口服活性且可透过血脑屏障的Nrf2激活剂,可诱导抗氧化剂基因表达上调。它是一种富马酸盐衍生物,可作抗炎和免疫调节剂,可研究多发性硬化症。
T6S0627 Mesaconitine

新乌碱,新乌头碱;中乌头碱

TNF Apoptosis
Mesaconitine 是乌头属植物的一种主要活性成分,通过循环 AMP 和刺激中枢 β-肾上腺素能系统具有镇痛活性,还有抗炎活性。
TN4660 Niranthin

Anti-infection; HBV; PAFR; Topoisomerase DNA Damage/DNA Repair; GPCR/G Protein; Microbiology/Virology
Niranthin 是一种木脂素,具有广泛的药理活性。它是L. donovaniIB 拓扑异构酶的非竞争性抑制剂,可用于研究耐药利什曼病的治疗。
TN1249 3-Epiursolic acid

Cysteine Protease; Immunology/Inflammation related Immunology/Inflammation; Proteases/Proteasome
3-Epiursolic Acid 是一种三萜类物质,分离自桃金娘科植物,是组织蛋白酶 L 的竞争性抑制剂(IC50=6.5 μM,Ki=19.5 μM),对 cathepsin B 无明显作用。
TN1413 Atranorin

荔枝素,巴美灵,荔枝素

Endogenous Metabolite; NO Synthase; Ras GPCR/G Protein; Immunology/Inflammation; MAPK; Metabolism
Atranorin 是地衣的次生代谢产物,具有显着的抗伤害、抗炎和氧化还原活性,对 H(2)O(2) 诱导的氧化应激下的细胞具有细胞保护作用。
T2897 (Rac)-Shikonin

(±)-Shikonin,Alkanet extract,Anchusin,紫草素,Anchusa acid

Others Others
(Rac)-Shikonin (Anchusin) 具有抗肿瘤作用。它能够诱导坏死死亡来绕过癌症耐药性。
TN2080 Pinoresinol

松脂酚,松脂素,(+)-Pinoresinol

Apoptosis; NF-κB; CDK; p53 Apoptosis; Cell Cycle/Checkpoint; NF-κB
Pinoresinol ((+)-Pinoresinol) 是一种植物来源的木质素,具有抗炎、保肝和杀真菌活性。它导致 CDK 抑制剂 p21(WAF1/Cip1) 在 mRNA 和蛋白质水平上调,抑制 NF-kappaB 和激活蛋白 1 。
T4958 (-)-Alkannin

Alkannin,左旋紫草素,紫草素,Shikonin

Apoptosis; PI3K Apoptosis; PI3K/Akt/mTOR signaling
(-)-Alkannin (Shikonin) 是从紫朱草中发现的一种天然产物,具有抗癌活性,可抑制细胞周期,诱导细胞凋亡,用作食品着色剂,在 Rho 激酶途径中可改善肝脏炎症。
T4S0145 Corylifol A

Corylinin,补骨脂异黄酮A

hCE; STAT; UGT JAK/STAT signaling; Metabolism; Stem Cells
Corylifol A (Corylinin) 是补骨脂中的一种天然产物,可抑制IL-6 诱导的STAT3激活和磷酸化,IC50值为0.81 μM。
T4S1472 Cucurbitacin S

Cucurbitacins from Wilbrandia ebracteata have analgesic effects. Cucurbitacin S has anticancer and antiinflammatory activities.
TN2002 Obovatol

BCL; Caspase; JAK Angiogenesis; Apoptosis; Chromatin/Epigenetic; JAK/STAT signaling; Proteases/Proteasome; Stem Cells
Obovatol has antioxidant, neuroprotective, antiinflammatory, antithrombotic and antitumour effects, it is a potent NF-κB inhibitors for Alzheimer's disease treatment.
TN3436 ar-Curcumene

Others Others
ar-Curcumene has antiinflammatory activity, it could be used as antiinflammatory drugs in respiratory infections. ar-Curcumene is effective as oviposition deterrents against Anopheles stephensi, Aedes aegypti, and Culex quinquefasciatus, it can be conside
TN7116 6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone

Others Others
6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone 是一种来自 Piper obliquum 的烯基酚,具有抗炎和抗菌活性。
TN3620 Celaphanol A

NF-κB NF-κB
Celaphanol A shows moderate inhibition in both NF-κB activation and nitric oxide production, suggests that it is a possible inhibitor of the NF-kappaB pathway and has antiinflammatory activity.
TN1080 Kaji-ichigoside F1

蔷薇苷

Kaji-ichigoside F1 shows antiinflammatory/antinociceptive action in acetic acid-induced writhing and hot plate testing and in a carrageenan-induced paw edema model in mice and rats. Kaji-ichigoside F1 exhibits in vivo hepatoprotective effects, it inhibite
TN3444 Aristolactam BII

HIV Protease Microbiology/Virology; Proteases/Proteasome
Aristolactam BII exhibits antimicrobial and antiinflammatory activity, it shows significant activity towards DPPH radical scavenging and potent inhibitory effects against tyrosinase mushroom. Aristolactam BII also exerts its significant neuroprotective ef
TN4648 Nepetoidin B

IL Receptor; p38 MAPK; TNF; NOS; NF-κB; COX; Antibacterial; JNK; Antifection; Antifungal Apoptosis; Immunology/Inflammation; MAPK; Microbiology/Virology; Neuroscience; NF-κB
Nepetoidin B 具有抗真菌、抗细菌和抗炎作用,它可以抑制 LPS 刺激的 NO 生成,可能是通过调节 RAW 264.7 细胞中由 MKP-5/NF-κB 通路介导的 iNOS 。

天然产物

Tirucallol
Cat.No: TN1006
Synonym:
Target: NOS, NO Synthase, Prostaglandin Receptor
Gossypin
Cat.No: TN1712
Synonym:
Target: NF-κB, S6 Kinase
Poliumoside
Cat.No: T6S2384
Synonym:
Target: Reductase
Bisdemethoxycurcumin
Cat.No: TL0007
Synonym: 双去甲氧基姜黄素,Curcumin III,Didemethoxycurcumin
Target: Epigenetic Reader Domain, Wnt/beta-catenin
Xanthatin
Cat.No: T3S0153
Synonym: 苍耳亭,叶黄制菌素
Target: Apoptosis, VEGFR, Lipoxygenase, Wnt/beta-catenin, Antibacterial
γ-Tocopherol
Cat.No: T8293
Synonym: D-gamma-生育酚,γ-生育酚,(+)-γ-Tocopherol
Target: COX
Vitexin
Cat.No: T6S1369
Synonym: 牡荆素,Apigenin-8-C-glucoside
Target: Antioxidant
Eudesmin
Cat.No: T3836
Synonym:
Target: MAPK, S6 Kinase
Dehydropachymic acid
Cat.No: TN1563
Synonym:
Target: Autophagy, Immunology/Inflammation related
Ingenol mebutate
Cat.No: TN1047
Synonym: Ingenol 3-Angelate,巨大戟醇甲基丁烯酸酯,PEP005
Target: gp120/CD4, HIV Protease, PKC
Rosamultin
Cat.No: T5783
Synonym: 野蔷薇苷,罗莎白素
Target: Antioxidant, HIV Protease
Bulleyaconitine A
Cat.No: T3021
Synonym: 草乌甲素,Bulleyaconi cine A
Target: Sodium Channel
Chrysoeriol
Cat.No: TN1490
Synonym:
Target: ERK, p38 MAPK, Akt
Naringenin
Cat.No: T2838
Synonym: 柚皮素,Naringetol,S-Dihydrogenistein,Pelargidanon,Salipurol,NSC 11855,NSC 34875
Target: P450, Influenza Virus, Reactive Oxygen Species, Endogenous Metabolite, PPAR
p-Anisic acid
Cat.No: TCS0862
Synonym: 大茴香酸,对甲氧基苯甲酸,4-Methoxybenzoic acid,Draconic Acid,4-Anisic Acid
Target: Endogenous Metabolite, Antibacterial
Dimethyl fumarate
Cat.No: T0492
Synonym: 富马酸二甲酯,DMF
Target: Reactive Oxygen Species, HIV Protease, Nrf2, Endogenous Metabolite, Autophagy
Mesaconitine
Cat.No: T6S0627
Synonym: 新乌碱,新乌头碱;中乌头碱
Target: TNF
Niranthin
Cat.No: TN4660
Synonym:
Target: Anti-infection, HBV, PAFR, Topoisomerase
3-Epiursolic acid
Cat.No: TN1249
Synonym:
Target: Cysteine Protease, Immunology/Inflammation related
Atranorin
Cat.No: TN1413
Synonym: 荔枝素,巴美灵,荔枝素
Target: Endogenous Metabolite, NO Synthase, Ras
(Rac)-Shikonin
Cat.No: T2897
Synonym: (±)-Shikonin,Alkanet extract,Anchusin,紫草素,Anchusa acid
Target: Others
Pinoresinol
Cat.No: TN2080
Synonym: 松脂酚,松脂素,(+)-Pinoresinol
Target: Apoptosis, NF-κB, CDK, p53
(-)-Alkannin
Cat.No: T4958
Synonym: Alkannin,左旋紫草素,紫草素,Shikonin
Target: Apoptosis, PI3K
Corylifol A
Cat.No: T4S0145
Synonym: Corylinin,补骨脂异黄酮A
Target: hCE, STAT, UGT
Cucurbitacin S
Cat.No: T4S1472
Synonym:
Target:
Obovatol
Cat.No: TN2002
Synonym:
Target: BCL, Caspase, JAK
ar-Curcumene
Cat.No: TN3436
Synonym:
Target: Others
6'-Hydroxy-3,4,2',3',4'-pentamethoxychalcone
Cat.No: TN7116
Synonym:
Target: Others
Celaphanol A
Cat.No: TN3620
Synonym:
Target: NF-κB
Kaji-ichigoside F1
Cat.No: TN1080
Synonym: 蔷薇苷
Target:
Aristolactam BII
Cat.No: TN3444
Synonym:
Target: HIV Protease
Nepetoidin B
Cat.No: TN4648
Synonym:
Target: IL Receptor, p38 MAPK, TNF, NOS, NF-κB, COX, Antibacterial, JNK, Antifection, Antifungal
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