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95

抑制剂 & 化合物

14

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T18892	5(6)-Aminofluorescein 5(6)-氨基荧光素,Fluoresceinamine mixed isomers,5(6)-AFM	Others	Others
	5(6)-Aminofluorescein (5(6)-AFM) 是一种合成 5(6)-FITC 的前体。其中5(6)-FITC 是胺活性衍生物的荧光染料。
T37607	Rhodamine B isothiocyanate (mixed isomers)
	Rhodamine B isothiocyanate (RITC) is a cell-permeant fluorogenic dye most often used as a conjugate to antibodies and proteins for fluorescence detection in microscopy. It displays excitation/emission maxima of 570/595 nm, respectively, and can be used in conjunction with immunohistochemistry for multi-labeling studies. It has also been used as an anterograde and retrograde tracer in neurons and in nanoparticles to detect apoptosis.
T18893	5(6)-Carboxyfluorescein 5(6)-羧基荧光素,5-(and-6)-Carboxyfluorescein mixed isomers,5(6)-FAM	Others	Others
	5(6)-Carboxyfluorescein (5-(and-6)-Carboxyfluorescein mixed isomers) 是一种胺反应性 pH 敏感的绿色荧光标记物，能够标记蛋白质、多肽和氨基酸，可用于体内实验检测肿瘤位置。
TD0066	5(6)-TAMRA [5-(and-6)-Carboxytetramethylrhodamine] *Mixed isomers*
	5(6)-TAMRA contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid. This bright, orange-fluorescent dye produces conjugates with absorption/emission maxima of ~555/580 nm.
TD0067	5(6)-ROX [5-(and 6)-Carboxy-X-rhodamine] *Mixed isomers*
	ROX dyes have a strong red fluorescence.Their excitation and emission wavelengths are longer than those of traditional rhodamine dyes.They are used as labels for peptides, proteins, and other biological ligands.5-ROX, 6-ROx, and their mixture of 5(6) -RoX
TD0100	5(6)-TRITC [Tetramethylrhodamine-5-(and-6)-isothiocyanate] *Mixed isomers*
	5(6)-TRITC [Tetramethylrhodamine-5-(and-6) -Isothiocyanate] *Mixed isomers* is used to label antibodies with strong fluorescent dyes
TD0060	5(6)-CR110 [5-(and 6)-Carboxyrhodamine 110] *Mixed isomers* 5(6)-羧基罗丹明110（混合物）
	5(6)-CR110 [5-(and 6)-Carboxyrhodamine 110] *Mixed isomers* is a Fluorescein for peptide and oligonucleotide labeling. Compared to fluorescein labeling reagents such as FITC and FAM, CR110 reagents give more photostable and pH-independent bioconjugates that have the absorption maximum around the preferred 488 nm excitation wavelength. They are photostable alternative reagents superior to FITC and FAM.
TD0063	5(6)-CR110, SE [5-(and 6)-Carboxyrhodamine 110, succinimidyl ester] *Mixed isomers* 5(6)-羧基罗丹明110琥珀酰亚胺酯（混合物）
	5(6)-CR110, SE [5-(and 6)-Carboxyrhodamine 110, succinimidyl ester] *Mixed isomers* is a Fluorescein for peptide and oligonucleotide labeling. Compared to fluorescein labeling reagents such as FITC and FAM, CR110 reagents give more photostable and pH-independent bioconjugates that have the absorption maximum around the preferred 488 nm excitation wavelength. They are photostable alternative reagents superior to FITC and FAM.
T6057	URMC-099	ROCK; MLK; VEGFR; SGK; DNA Alkylation; Trk receptor; c-Met/HGFR; LRRK2; MEK; IGF-1R; Syk; Bcr-Abl; CDK; Src; Aurora Kinase; Autophagy	Angiogenesis; Autophagy; Cell Cycle/Checkpoint; Chromatin/Epigenetic; Cytoskeletal Signaling; DNA Damage/DNA Repair; MAPK; Metabolism; Stem Cells; Tyrosine Kinase/Adaptors
	URMC-099 是一种具有优异的血脑屏障穿透性的，可口服的混合谱系激酶 3 抑制剂，IC50为14 nM。
T11520	GW806742X	MLK; VEGFR	Angiogenesis; MAPK; Tyrosine Kinase/Adaptors
	GW806742X 是ATP 模拟物，是MLKL 抑制剂，可结合 MLKL 假激酶结构域，Kd 值为 9.3μM。它对VEGFR2的IC50为 2 nM，延缓 MLKL 膜移位并抑制坏死。
T6904	Necrosulfonamide (E)-Necrosulfonamide	MLK	MAPK
	Necrosulfonamide ((E)-Necrosulfonamide) 是一种坏死性凋亡抑制剂，通过选择性靶向(MLKL)，可阻止 MLKL-RIP1-RIP3 坏死小体复合体与其下游效应子相互作用。MLKL 是诱导坏死过程中 RIP3 的重要底物。
T9399	Menin-MLL inhibitor 20	Epigenetic Reader Domain; Histone Methyltransferase	Chromatin/Epigenetic
	Menin-MLL inhibitor 20 是一种不可逆的menin-MLL 相互作用抑制剂，具有抗肿瘤活性。
T8961	GW280264X Carbamic acid	MMP	Proteases/Proteasome
	GW280264X (Carbamic acid) 是一种 ADAM10/TACE (ADAM17)金属蛋白酶抑制剂。它有效阻断 TACE (ADAM17)和 ADAM10的 IC50分别为 8.0 nM 和 11.5 nM。其中ADAM10/17 能够调节胶质母细胞瘤起始细胞的免疫原性。
T14496	BAMB-4 ITPKA-IN-C14	Others	Others
	BAMB-4 (ITPKA-IN-C14) 是一种新型的膜渗透型ITPKA 抑制剂，在ADP-Glo 实验中的IC50值为37uM。
T18895	5(6)-FAM SE 5(6)-羧基荧光素琥珀酰亚胺酯,5(6)-Carboxyfluorescein N-hydroxysuccinimide ester	Others	Others
	5(6)-FAM SE (5(6)-Carboxyfluorescein N-hydroxysuccinimide ester) 是绿色荧光染料，普遍用于标记蛋白质。
TD0068	5(6)-ROX N-succinimidyl ester 5(6)-ROX, SE [5-(and-6)-Carboxy-X-rhodamine, succinimidyl ester] *Mixed isomers*,5(6)-羧基-X-罗丹明琥珀酰亚胺酯（混合物）
	5(6)-ROX, SE is an amine-reactive fluorescent probe that is widely used for oligonucleotide labeling and automated DNA sequencing applications.
T24488	MLS000545091 MLS-000545091,MLS 000545091
	MLS000545091 is a potent and selective human epithelial 15-lipoxygenase-2 mixed-type inhibitor.
T31640	Enrasentan SB-217242,SB 217242,SB217242	Endothelin Receptor	GPCR/G Protein
	Enrasentan（sb-217242）是一种 ET（A）和 ET（B）受体的混合拮抗剂，可降低血压、防止心肌肥大和保护心肌功能。
T3587	NOD-IN-1 Compound 4	NOD-like Receptor (NLR); NOD	Immunology/Inflammation; NF-κB
	NOD-IN-1 (Compound 4) 是核苷酸结合寡聚化结构域样受体 NOD1(IC50:5.74 μM)和 NOD2 (IC50:6.45 μM)的抑制剂。
T20080	Exifone NSC 680919,NSC680919,NSC-680919,依昔苯酮	HDAC	Chromatin/Epigenetic; DNA Damage/DNA Repair
	Exifone (NSC-680919) 是一种混合的、非必需的 HDAC1 激活剂，能够与游离酶和底物结合酶结合，从而提高 HDAC1 催化的去乙酰化的相对最大速率。
T68023L	Tolnapersine TFA Tolnapersine TFA(70312-00-4 Free base)	Dopamine Receptor; Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Tolnapersine TFA 是混合多巴胺激动剂和α肾上腺素受体拮抗剂。
T3082	SGC0946	Histone Methyltransferase	Chromatin/Epigenetic
	SGC0946是一种组蛋白甲基转移酶DOT1L 高选择性抑制剂，IC50值为0.3nM，可选择性地杀死混合谱系白血病细胞。
T6774	AZD-8835 AZD8835	PI3K	PI3K/Akt/mTOR signaling
	AZD-8835 是选择性的 PI3Kα (IC50:6.2 nM) 和 PI3Kδ (IC50:5.7 nM) 抑制剂。
T23631	Adatanserin WY-50324,WY 50324,WAY SEB 324,WY50324	5-HT Receptor	GPCR/G Protein; Neuroscience
	Adatanserin (WY 50324) 是一种混合型 5-HT1A 受体部分激动剂，也是一种 5-HT2A 和 5-HT2C 受体拮抗剂，具有潜在的神经保护活性，可用于研究焦虑和抑郁症。
T17227	Vernakalant Hydrochloride RSD1235 hydrochloride	Potassium Channel; Sodium Channel	Membrane transporter/Ion channel
	Vernakalant Hydrochloride (RSD1235 hydrochloride) 是一种混合电压和频率依赖性的 Na+ 和 K+ 通道阻断剂。Vernakalant 抑制 Kv1.5 channelwt，Kv1.5 channelI508F，Kv1.5 channelT479A，IC50 分别为 13.35±0.93 μM。
T15792	Luminol 鲁米诺,Diogenes reagent	Others	Others
	Luminol (Diogenes reagent) 是化学发光物质，pKa 值为 6.74 和 15.1。它的最适荧光波长为 425 nm。它在刑事侦查、生物工程、化学示踪等领域中可用作法医检测血迹的诊断工具。
T23397	ST 91	Others; Adrenergic Receptor	GPCR/G Protein; Neuroscience; Others
	ST-91 是一种 α2-肾上腺素能受体激动剂，具有混合的 α-肾上腺素能受体类型/亚型选择特征。
T67743	4-Pyridinecarboxaldehyde, 2-(2-pyridinyl)hydrazone, [C(E)]-	Others	Others
	4-Pyridinecarboxaldehyde, 2-(2-pyridinyl)hydrazone, [C(E)]-是混合配体配位聚合物[Zn4(bdc)4(ppmh)2(H2O)]n 的配体。
T27832	Lifibrol U 83860,K-12148,K-12.148,U-83860,K12148	Lipid	Metabolism
	Lifibrol (U-83860) 是一种胆固醇合成抑制剂。Lifibrol 具有抗胆固醇和降血脂的作用，可促进高胆固醇血症和混合型高脂血症患者体内低密度脂蛋白载脂蛋白 B-100 的转化。
T5023	Propiverine hydrochloride	Others; Calcium Channel; AChR	Membrane transporter/Ion channel; Metabolism; Neuroscience; Others
	Propiverine hydrochloride 是一种痉挛剂，具有钙拮抗和抗胆碱能特性，用于研究膀胱过度活动和尿失禁。
T18898	5(6)-TAMRA SE 5(6)-Carboxytetramethylrhodamine N-succinimidyl ester,5(6)-羧基四甲基罗丹明琥珀酰亚胺酯	Others	Others
	5(6)-TAMRA SE (5(6)-Carboxytetramethylrhodamine N-succinimidyl ester) 是荧光染料，能够结合寡聚核苷酸，并用于DNA 测序。
T34573	SCH-900271 SCH 900271	AChR	Neuroscience
	SCH-900271是一种有效的尼古丁酸受体，用于治疗血脂异常,常用来研究混合性高脂血症和原发性高胆固醇血症。
T38507	Renzapride BRL 24924	5-HT Receptor	GPCR/G Protein; Neuroscience
	Renzapride (BRL 24924) 是一种混合 5-羟色胺 4 型（5-HT4）激动剂和 5-HT3 受体拮抗剂。Renzapride 可用于研究以便秘为主的肠易激综合征（C-IBS）。
T27119L	(Rac)-Daglutril SLV 306 acetic acid,2-((3S)-3-(1-(2-(ethoxycarbonyl)-4-phenylbutyl)cyclopentane-1-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)acetic acid	Others	Others
	(Rac)-Daglutril (SLV 306 acetic acid) 是 Daglutril 的消旋体。Daglutril 是一种口服活性的混合中性内肽酶/内皮素转化酶抑制剂，正在开发用于治疗原发性高血压和充血性心力衰竭。
T3465	Vesnarinone 维司力农,OPC-8212,Arkin,Piteranometozine	HIV Protease; PDE	Metabolism; Microbiology/Virology; Proteases/Proteasome
	Vesnarinone (Arkin) 是一种喹啉酮衍生物，可抑制磷酸二酯酶III 活性，增加钙通量和减小钾通量。
T8691	PD 168368 PD168368	Bombesin Receptor	GPCR/G Protein
	PD 168368 是一种新型有效且具有竞争性和选择性的非肽类神经调节蛋白 B 受体 (NMB-R) 拮抗剂，对胃泌素释放肽受体 (GRPR)具有抑制作用。PD 168368 是一种高效的 FPR1/FPR2/FPR3 的混合激动剂。
T11925	M‑89	Epigenetic Reader Domain; Histone Methyltransferase	Chromatin/Epigenetic
	M-89 可抑制 Menin-MLL 蛋白之间的相互作用，有研究混合谱系白血病的潜力。它是一种强特异性 menin 抑制剂，结合到 menin 的Kd 值为 1.4 nM。
T20570	Labetalol Apo-Labetalol,Albetol,Trandate,Dilevalol,拉贝洛尔,Normodyne	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Labetalol (Apo-Labetalol) 是一种抗高血压药物，可用于心血管疾病的研究，如妊娠期高血压。它是一种口服具有活性的选择性 α1- 和非选择性 β-肾上腺素能受体 (adrenergic receptor) 竞争性拮抗剂。
T8768	MM-102 TFA HMTase Inhibitor IX TFA	Histone Methyltransferase	Chromatin/Epigenetic
	MM-102 TFA (HMTase Inhibitor IX TFA) 是一种有效的 WDR5/MLL 相互作用抑制剂，在 WDR5 结合检测中，IC50为 2.4 nM，Ki 小于 1 nM。
T1951	Asenapine Maleate Org 5222 maleate,Org 5222,马来酸阿塞那平,阿塞那平马来酸盐	5-HT Receptor	GPCR/G Protein; Neuroscience
	Asenapine Maleate (Org 5222 maleate) 是5-HT 和D2的拮抗剂，Ki 值分别为 0.03-4.0 nM, 1.3 nM。它也是抗精神病药物，用于治疗与双相 1 型障碍相关的精神分裂症和躁狂或混合发作。
T0976	Propoxur 残杀威,Aprocarb,Propoxure,Baygon	AChR; Antifungal	Microbiology/Virology; Neuroscience
	Propoxur (Propoxure) 是一种氨基甲酸酯类杀虫剂，用于控制蟑螂、苍蝇、蚊子以及草坪和草坪昆虫。
T4616	Metoclopramide 甲氧氯普胺,胃复安,5-Chloro-2-methoxyprocainamide	Dopamine Receptor; 5-HT Receptor	GPCR/G Protein; Neuroscience
	Metoclopramide (5-Chloro-2-methoxyprocainamide) 是5-HT3和多巴胺D2受体拮抗剂，IC50值分别为 308 和 483 nM，可用于恶心呕吐、胃食管反流和胃轻瘫的研究。
T67956L	Litoxetine HCl litoxetine HCL(86811-09-8 Free base)	5-HT Receptor	GPCR/G Protein; Neuroscience
	Litoxetine HCl 是一种选择性5-羟色胺（5-HT）再摄取抑制剂（SSRI）和混合5-羟色胺拮抗剂，可用于治疗尿失禁。Litoxetine HCl 在没有抗毒蕈碱特性的浓度下（10 nM-1 microM）引起大鼠离体食道肌肉粘膜的浓度依赖性松弛，使卡巴胆碱张力降低达37%,更高浓度的Litoxetine HCl（3微摩-300微摩）与明显的松弛有关，直至取消卡巴胆碱张力。以前在离体豚鼠肠道中证明的利托西汀的抗心律失常活性，在浓度大于1 microM 时在大鼠离体食道肌肉粘膜中发挥了作用。 Litoxetine HCl 的5-HT 释放作用可以解释利托西汀对未处理的大鼠组织中的5-HT 诱导的松弛的效力，这种效力被pCPA 处理所逆转。
T28452	Profadol hydrochloride Centrac,A-2205,CI 572,Profadol HCl,CI-572
	Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.
T27358	FQ
	FQ is a novel reversible inhibitor of mixed-type tyrosinase.
T28568	Ro 23-0364 Ro-23-0364
	Ro 23-0364 an imidazobenzodiazepine with mixed benzodiazepine agonist/antagonist properties.
T12002	Menin-MLL inhibitor 4	Others	Others
	Menin-MLL inhibitor 4 has antitumor activity.Menin-MLL inhibitor 4 is an inhibitor of Menin- MLL (mixed-lineage leukemia protein) interaction .
T12091L	MM-589 TFA	JAK	Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells
	MM-589 TFA is a potent WD repeat domain 5 (WDR5)inhibitor and mixed lineage leukemia (MLL) protein-protein interaction.
T24471	MIV-6
	MIV-6 is an inhibitor of the menin-mixed lineage leukemia interaction.
T69370	Cyclazocine
	Cyclazocine is an analgesic with mixed narcotic agonist-antagonist properties.

化合物

5(6)-Aminofluorescein

Cat.No: T18892

Synonym: 5(6)-氨基荧光素,Fluoresceinamine mixed isomers,5(6)-AFM

Target: Others

Rhodamine B isothiocyanate (mixed isomers)

Cat.No: T37607

5(6)-Carboxyfluorescein

Cat.No: T18893

Synonym: 5(6)-羧基荧光素,5-(and-6)-Carboxyfluorescein mixed isomers,5(6)-FAM

Target: Others

5(6)-TAMRA [5-(and-6)-Carboxytetramethylrhodamine] *Mixed isomers*

Cat.No: TD0066

5(6)-ROX [5-(and 6)-Carboxy-X-rhodamine] *Mixed isomers*

Cat.No: TD0067

5(6)-TRITC [Tetramethylrhodamine-5-(and-6)-isothiocyanate] *Mixed isomers*

Cat.No: TD0100

5(6)-CR110 [5-(and 6)-Carboxyrhodamine 110] *Mixed isomers*

Cat.No: TD0060

Synonym: 5(6)-羧基罗丹明110（混合物）

5(6)-CR110, SE [5-(and 6)-Carboxyrhodamine 110, succinimidyl ester] *Mixed isomers*

Cat.No: TD0063

Synonym: 5(6)-羧基罗丹明110琥珀酰亚胺酯（混合物）

Cat.No: T6057

Target: ROCK, MLK, VEGFR, SGK, DNA Alkylation, Trk receptor, c-Met/HGFR, LRRK2, MEK, IGF-1R, Syk, Bcr-Abl, CDK, Src, Aurora Kinase, Autophagy

Cat.No: T11520

Target: MLK, VEGFR

Necrosulfonamide

Cat.No: T6904

Synonym: (E)-Necrosulfonamide

Target: MLK

Menin-MLL inhibitor 20

Cat.No: T9399

Target: Epigenetic Reader Domain, Histone Methyltransferase

Cat.No: T8961

Synonym: Carbamic acid

Target: MMP

Cat.No: T14496

Synonym: ITPKA-IN-C14

Target: Others

Cat.No: T18895

Synonym: 5(6)-羧基荧光素琥珀酰亚胺酯,5(6)-Carboxyfluorescein N-hydroxysuccinimide ester

Target: Others

5(6)-ROX N-succinimidyl ester

Cat.No: TD0068

Synonym: 5(6)-ROX, SE [5-(and-6)-Carboxy-X-rhodamine, succinimidyl ester] *Mixed isomers*,5(6)-羧基-X-罗丹明琥珀酰亚胺酯（混合物）

Cat.No: T24488

Synonym: MLS-000545091,MLS 000545091

Cat.No: T31640

Synonym: SB-217242,SB 217242,SB217242

Target: Endothelin Receptor

Cat.No: T3587

Synonym: Compound 4

Target: NOD-like Receptor (NLR), NOD

Cat.No: T20080

Synonym: NSC 680919,NSC680919,NSC-680919,依昔苯酮

Target: HDAC

Tolnapersine TFA

Cat.No: T68023L

Synonym: Tolnapersine TFA(70312-00-4 Free base)

Target: Dopamine Receptor, Adrenergic Receptor

Cat.No: T3082

Target: Histone Methyltransferase

Cat.No: T6774

Synonym: AZD8835

Target: PI3K

Cat.No: T23631

Synonym: WY-50324,WY 50324,WAY SEB 324,WY50324

Target: 5-HT Receptor

Vernakalant Hydrochloride

Cat.No: T17227

Synonym: RSD1235 hydrochloride

Target: Potassium Channel, Sodium Channel

Cat.No: T15792

Synonym: 鲁米诺,Diogenes reagent

Target: Others

Cat.No: T23397

Target: Others, Adrenergic Receptor

4-Pyridinecarboxaldehyde, 2-(2-pyridinyl)hydrazone, [C(E)]-

Cat.No: T67743

Target: Others

Cat.No: T27832

Synonym: U 83860,K-12148,K-12.148,U-83860,K12148

Target: Lipid

Propiverine hydrochloride

Cat.No: T5023

Target: Others, Calcium Channel, AChR

Cat.No: T18898

Synonym: 5(6)-Carboxytetramethylrhodamine N-succinimidyl ester,5(6)-羧基四甲基罗丹明琥珀酰亚胺酯

Target: Others

Cat.No: T34573

Synonym: SCH 900271

Target: AChR

Cat.No: T38507

Synonym: BRL 24924

Target: 5-HT Receptor

(Rac)-Daglutril

Cat.No: T27119L

Synonym: SLV 306 acetic acid,2-((3S)-3-(1-(2-(ethoxycarbonyl)-4-phenylbutyl)cyclopentane-1-carboxamido)-2-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepin-1-yl)acetic acid

Target: Others

Cat.No: T3465

Synonym: 维司力农,OPC-8212,Arkin,Piteranometozine

Target: HIV Protease, PDE

Cat.No: T8691

Synonym: PD168368

Target: Bombesin Receptor

Cat.No: T11925

Target: Epigenetic Reader Domain, Histone Methyltransferase

Cat.No: T20570

Synonym: Apo-Labetalol,Albetol,Trandate,Dilevalol,拉贝洛尔,Normodyne

Target: Adrenergic Receptor

Cat.No: T8768

Synonym: HMTase Inhibitor IX TFA

Target: Histone Methyltransferase

Asenapine Maleate

Cat.No: T1951

Synonym: Org 5222 maleate,Org 5222,马来酸阿塞那平,阿塞那平马来酸盐

Target: 5-HT Receptor

Cat.No: T0976

Synonym: 残杀威,Aprocarb,Propoxure,Baygon

Target: AChR, Antifungal

Cat.No: T4616

Synonym: 甲氧氯普胺,胃复安,5-Chloro-2-methoxyprocainamide

Target: Dopamine Receptor, 5-HT Receptor

Cat.No: T67956L

Synonym: litoxetine HCL(86811-09-8 Free base)

Target: 5-HT Receptor

Profadol hydrochloride

Cat.No: T28452

Synonym: Centrac,A-2205,CI 572,Profadol HCl,CI-572

Cat.No: T27358

Cat.No: T28568

Synonym: Ro-23-0364

Menin-MLL inhibitor 4

Cat.No: T12002

Target: Others

Cat.No: T12091L

Target: JAK

Cat.No: T24471

Cat.No: T69370

Cat. No.	Product Name	Target	Signaling Pathways
T6752	S-Adenosyl-L-methionine disulfate tosylate S-腺苷蛋氨酸对甲苯磺酸硫酸盐,Ademetionine disulfate tosylate	DNA/RNA Synthesis	Cell Cycle/Checkpoint; DNA Damage/DNA Repair
	S-Adenosyl-L-methionine disulfate tosylate (Ademetionine disulfate tosylate) 是一种主要生物甲基供体，在所有哺乳动物细胞中合成，但在肝脏中含量较高。
TN1016	Kukoamine A	NF-κB; Lipoxygenase; DNA/RNA Synthesis; Parasite	Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB
	Kukoamine A 是一种天然的精胺衍生物，具有抗癌、抗高血压、细胞保护、抗氧化和抗炎活性。它是锥虫硫磷还原酶抑制剂，Ki 值为 1.8 μM。
T3S2259	Methyl eugenol 4-allylveratrole,eugenyl methyl ether,O-methyleugenol,Eugenol Methyl ether,丁香酚甲醚,丁子香酚甲醚	GABA Receptor	Membrane transporter/Ion channel; Neuroscience
	Methyl eugenol (4-allylveratrole) 是一种苯丙类化合物，存在于植物叶子、果实、根茎中，当植物相应的部位因食草动物进食而受损时，就会释放。它可用于消灭雄性东方果蝇。
TMA2563	Pedalitin	Tyrosinase	Proteases/Proteasome
	Pedalitin is a mixed-type inhibitor of tyrosinase. In the assay of α-glucosidase inhibition, rosmarinic acid is a competitive inhibitor, whereas both methyl rosmarinate and Pedalitin are mixed-type inhibitors.
T20309	Anise alcohol AI301170,AI3-01170,AI3 01170
	Anise drinks is a family of alcoholic drinks with unique characteristics. Crystallization and color-changing when mixed with other liquids.
TN3899	Drupacine	Others	Others
	Drupacine and a crude alkaloid extract suppress nematode hatch, activity of mixed life stages, and population numbers on plant roots.
T62625	11-O-Methylpseurotin A
	11-O-Methylpseurotin A为一种(PKS/NRPS)混合聚酮合成酶-非核糖体肽合成酶化合物，其特性为选择性抑制Hof1缺失菌株。
T81735	Mycestericin C
	Mycestericin C, 分离自 Mycelia sterilia ATCC 20349 的培养液, 能在小鼠同种异体混合淋巴细胞反应中抑制淋巴细胞的增殖。
T5276	4,4'-Disulfanediylbis(2-aminobutanoic acid) DL-Homocystine,DL-高胱氨酸	Others; Endogenous Metabolite	Metabolism; Others
	4,4'-Disulfanediylbis(2-aminobutanoic acid) (DL-Homocystine) 是内源性代谢产物的一种。
TN2913	3-Acetoxy-11-ursen-28,13-olide	Phosphatase	Metabolism
	3β-Acetoxy-urs-11-en-28,13-olide exhibits significant protein tyrosine phosphatase 1B (PTP1B) inhibitory activity, it is a mixed-type PTP1B inhibitor. It exhibits weak-moderate antiproliferative activity against the A2780 human ovarian cancer cell line.
T75511	BChE-IN-10
	BChE-IN-10 (compound 6)，一种从白芨 (Bletilla striata) 分离提取的丁酰胆碱酯酶 (BChE) 混合型抑制剂，具有 6.4 μM 的IC50，适用于阿尔兹海默症 (AD) 研究。
TN2280	Trametenolic acid	Tyrosinase	Proteases/Proteasome
	Trametenolic acid is a cytotoxic agent.It exhibits a mode of mixed inhibition with a K I of 0.9μM, K IS of 0.5μM, and an IC50 of 7.25μM.Trametenolic acid and Betulin as a new candidate of potent tyrosinase inhibitors, can decrease tyrosinase activity and melanin content.
TN2217	Sophoflavescenol 槐苦参醇,槐黄醇	Others; Beta-Secretase; BACE; PDE; AChR; AChE	Metabolism; Neuroscience; Others
	Sophoflavescenol 是异戊烯基黄酮类化合物，能够抑制PDE5的活性，IC50=0.013 μM。它也抑制 RLAR，HRAR，BACE1，AChE 和 BChE，IC50值分别为 0.30 µM，0.17 µM，10.98 µM，8.37 µM 和 8.21 µM。
T75514	Blestrin D
	Blestrin D，作为一种丁酰胆碱酯酶(BChE)的有效混合型抑制剂，具有8.1 μM的IC50值，可从白芨(Bletilla striata)中分离提取，适用于阿尔兹海默症(AD)研究。

天然产物

S-Adenosyl-L-methionine disulfate tosylate

Cat.No: T6752

Synonym: S-腺苷蛋氨酸对甲苯磺酸硫酸盐,Ademetionine disulfate tosylate

Target: DNA/RNA Synthesis

Cat.No: TN1016

Target: NF-κB, Lipoxygenase, DNA/RNA Synthesis, Parasite

Cat.No: T3S2259

Synonym: 4-allylveratrole,eugenyl methyl ether,O-methyleugenol,Eugenol Methyl ether,丁香酚甲醚,丁子香酚甲醚

Target: GABA Receptor

Cat.No: TMA2563

Target: Tyrosinase

Cat.No: T20309

Synonym: AI301170,AI3-01170,AI3 01170

Cat.No: TN3899

Target: Others

11-O-Methylpseurotin A

Cat.No: T62625

Cat.No: T81735

4,4'-Disulfanediylbis(2-aminobutanoic acid)

Cat.No: T5276

Synonym: DL-Homocystine,DL-高胱氨酸

Target: Others, Endogenous Metabolite

3-Acetoxy-11-ursen-28,13-olide

Cat.No: TN2913

Target: Phosphatase

Cat.No: T75511

Trametenolic acid

Cat.No: TN2280

Target: Tyrosinase

Sophoflavescenol

Cat.No: TN2217

Synonym: 槐苦参醇,槐黄醇

Target: Others, Beta-Secretase, BACE, PDE, AChR, AChE

Cat.No: T75514

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