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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T24141 HIV-1 Inhibitor 18A

HIV-1 Inhibitor-18A

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 Inhibitor 18A (HIV-1 Inhibitor-18A) 特异性抑制多种 HIV-1 分离株的进入。
T9039 HIV-1 Nef-IN-1

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 Nef-IN-1HIV-1 Nef 蛋白的抑制剂。 它有效地竞争 Nef-SH3Hck 相互作用,Kd 值为 6.7 μM。
TP1149 HIV-1 Rev (34-50)

HIV-1 Rev 34-50,HIV-1 rev Protein (34-50)

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 Rev (34-50) (HIV-1 rev Protein (34-50)) 是一种具有抗 HIV-1 活性的 17 个氨基酸多肽。 HIV-1 Rev (34-50) 源自 HIV-1 中 Rev 的 Rev 响应元件结合域。
T67833 HIV-1 inhibitor-54

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 inhibitor-54 是一种有效的 HIV-1 抑制剂,在 MT-4 细胞中对 WT HIV-1 (菌株 IIIB) x 显示出抗 HIV 活性(EC50 : 32 nM)。HIV-1 inhibitor-54 可用于研究病毒感染。
T9854 HIV-1 inhibitor-6 

3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) 是一种有效的HIV-1 pre-mRNA 选择性剪接抑制剂,可以阻断HIV 复制。
TP1809 TAT

HIV Protease Microbiology/Virology; Proteases/Proteasome
TAT 源自人免疫缺陷病毒的转录反式激活因子,是一种细胞穿透肽。它可以增加异源蛋白质的产量和溶解度。
T1883 Des(benzylpyridyl) Atazanavi

HIV Protease Microbiology/Virology; Proteases/Proteasome
Des(benzylpyridyl) Atazanavi 是 Atazanavir 的 N-脱烷基代谢物 (M1),一种 HIV 蛋白酶抑制剂。
T39729 HIV Protease Substrate 1

HIV Protease Substrate 1 is a fluorogenic compound that offers insights into the enzymatic activity of HIV protease, making it a valuable tool for studying this aspect.
T11564 HIV-1 inhibitor-3

Others Others
HIV-1 inhibitor-3 is an HIV infection inhibitor.
T11566 HIV-1 integrase inhibitor

Others Others
Hiv-1 integrase inhibitor is an effective anti-HIV drug.
T40719 (Cys47)-HIV-1 tat Protein (47-57)

(Cys47)-HIV-1 tat Protein (47-57)

(Cys47)-HIV-1 tat Protein (47-57) possesses membrane translocation functionality and can serve as a surface derivatization agent for magnetic pharmaceuticals, thereby enhancing their uptake into specific target cells.
TP1776 HIV-1 TAT 48-60

HIV-1 TAT (48-60) is a cell-penetrating peptide derived from the human immunodeficient virus (HIV)-1 Tat protein residue 48-60. This is one of the cell-penetrating peptides generated from the human immunodeficient virus -1 Tat protein residue 48-60.
T11565 HIV-1 integrase inhibitor 7

Others Others
HIV-1 integrase inhibitor 7 is a potent HIV-1 integrase inhibitor (IC50: 33.3 nM).
T11568 HIV-1 integrase inhibitor 4

Others Others
HIV-1 integrase inhibitor 4 is an HIV-1 integrase strand transfer (INST) inhibitor (IC50: 3.7 nM).
T11567 HIV-1 integrase inhibitor 3

Others Others
HIV-1 integrase inhibitor 3 is an HIV-1 integrase strand transfer (INST) inhibitor (IC50: 2.7 nM).
T60742 HIV-1 integrase inhibitor 8

HIV Protease Microbiology/Virology; Proteases/Proteasome
HIV-1 integrase inhibitor 8 是一种 HIV-1 整合酶抑制剂,整合是HIV 复制的必要步骤。
T9212 IMB-301

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
IMB-301是根据 hA3G 模型通过虚拟筛选的一种小分子抑制剂。
T15371 Gardiquimod

TLR; HIV Protease Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Gardiquimod 可抑制巨噬细胞和活化的外周血单个核细胞的HIV-1感染。 它是一种咪唑喹啉类似物,是一种 TLR7/8 激动剂。
T4182 lavendustin B

薰草菌素B

Tyrosinase; transporter; HIV Protease Metabolism; Microbiology/Virology; Proteases/Proteasome
Lavendustin B 是一种酪氨酸激酶抑制剂,是 HIV-1 整合酶 (IN) 与其同源细胞辅助因子、晶状体上皮衍生生长因子 (LEDGF/p75) 相互作用的抑制剂。
T12715 Reverse transcriptase-IN-1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Reverse transcriptase-IN-1 是一种二芳基苯并嘧啶类似物,是一种有效的 HIV-1 非核苷类逆转录酶抑制剂,IC50 为 13.7 nM。
T16276 NBD-556

HIV Protease Microbiology/Virology; Proteases/Proteasome
NBD-556是一种 CD4 模拟物,识别 HIV-1 包膜蛋白 gp120 并诱导 gp120 重组,类似于 CD4 结合,可阻断 gp120-CD4 的相互作用。
T11465 Lenacapavir

GS-6207

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
Lenacapavir (GS-6207) 是一种有效的靶向衣壳的 HIV 复制抑制剂。 Lenacapavir 在 MT-4 细胞中显示出抗 HIV 活性,EC50 为 100 pM。
T8233 BRD3308

Apoptosis; HIV Protease; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
BRD3308 是一种高选择性的HDAC3抑制剂,IC50为 54 nM。它可激活HIV-1转录并破坏HIV-1潜伏期。它抑制由炎性细胞因子或糖脂毒性应激诱导的胰腺 β 细胞凋亡,并增加功能性胰岛素释放。
T9063 Clathrin-IN-1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Clathrin-IN-1 是一种网格蛋白抑制剂,可通过与网格蛋白的末端域相关联来抑制网格蛋白介导的内吞作用,有潜力用于抗癌的研究。
T28578 Ro24-7429

Ro 24-7429,Ro-24-7429,Ro 247429

HIV Protease Microbiology/Virology; Proteases/Proteasome
Ro24-7429 是一种有效的口服活性 HIV-1 反式激活蛋白 Tat 拮抗剂和一种矮小相关转录因子 1 的抑制剂。Ro24-7429 具有抗 HIV、抗纤维化和抗炎作用。
T20062 Thiamine disulfide

二硫化硫胺,TDS,Daiomin,Algoneurina

HIV Protease; Endogenous Metabolite Metabolism; Microbiology/Virology; Proteases/Proteasome
Thiamine disulfide (Algoneurina) 是一种存在于食物中的维生素,可作为膳食补充剂和药物生产。 它还充当许多中枢代谢酶的辅助因子。
T6246 Cobicistat

Tybost,GS-9350,考西司他

P450; HIV Protease Metabolism; Microbiology/Virology; Proteases/Proteasome
Cobicistat (GS-9350) 是一种细胞色素酶P450 3A 的选择性抑制剂,IC50值为30-285 nM。它是一种药代动力学增强剂,可增强抗 HIV 药物的吸收。
T11538 Hck-IN-1

HIV Protease; Src; Hck Angiogenesis; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Hck-IN-1 是二苯基吡唑啉化合物,选择性的 Nef 依赖性 Hck 抑制剂。它是广泛的 HIV-1 Nef 直接拮抗剂,对于野生型 HIV-1 复制的IC50为 100-300 nM。它结合口袋残基 Asn126,具有抗逆转录病毒活性。
T9223 RO-0335

Reverse Transcriptase Microbiology/Virology
RO-0335 是新高效二苯醚非核苷逆转录酶抑制剂。它 (IC50= 1.1 nM) 可以抑制Wt HIV-1病毒,对 92% 的 NNRTI 耐药临床分离株具有保留活性 (IC50<100 nM)。
T6420 BMS-707035

N-[(4-氟苯基)甲基1,6-二氢-5-羟基-1-甲基-6-氧代-2-(四氢-1,1-二氧-2H-1,2-噻嗪-2-基)-4-嘧啶甲酰胺

HIV Protease Microbiology/Virology; Proteases/Proteasome
BMS707035是一种 HIV-1 整合酶抑制剂,IC50为15 nM。
T3199 PTACH

NCH-51,Cpd 51

HIV Protease; HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Proteases/Proteasome
PTACH (Cpd 51) 是一种有效的 HDAC 抑制剂,对 HDAC1,HDAC4和 HDAC6的 IC50分别为 48 nM,32 nM 和 41 nM。PTACH 对多种癌细胞具有强大的生长抑制作用 (EC50为 1.1-9.1 µM)。
T11281L FGI-106 tetrahydrochloride

Virus Protease; HCV Protease; Influenza Virus; HIV Protease Microbiology/Virology; Proteases/Proteasome
FGI-106 tetrahydrochloride 对多种病毒具有抑制活性,有抗埃博拉病毒,裂谷病毒和登革热病毒的 EC50分别为 100 nM,800 nM 和 400-900 nM,抑制非失血性发热病毒HCV 和HIV-1的EC50分别为 200 nM 和 150 nM 。
T27030 CK176

HIV-1 inhibitor-34,HIV-1 inhibitor 34,CK 176,CK-176,HIV-1 inhibitor34

CK176 is a capsid targeted inhibitor of HIV-1 replication. CK176 shows an 11-fold improvement over I-XW-053 in blocking HIV-1 replication in primary human peripheral blood mononuclear cells (PBMCs).
T6255 Bromosporine

Epigenetic Reader Domain; CDK Cell Cycle/Checkpoint; Chromatin/Epigenetic
Bromosporine 是广谱 BRD2/4/9 和 CECR2 溴结构域抑制剂,IC50为0.41、0.29、0.122和0.017 μM。
T0100L Atazanavir

Zrivada,Reyataz,Latazanavir,阿扎那韦,BMS-232632

P450; SARS-CoV; HIV Protease; P-gp Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Atazanavir (BMS-232632) 是一种高选择性的HIV-1蛋白酶抑制剂,可研究艾滋病毒感染。它也是SARS-CoV 3CLpro 的抑制剂,IC50为 3.49 μM。它是CYP3A4的底物和抑制剂,也是P-糖蛋白的抑制剂和诱导剂。
T7212 Delavirdine mesylate

U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate)

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Delavirdine mesylate (BHAP-U 90152(mesylate)) 是一种口服活性非核苷逆转录酶抑制剂。它抑制 HIV-1 病毒复制,可以用于艾滋病的相关研究。它选择性地抑制 HIV-1 逆转录酶,其选择性超过 DNA 聚合酶 α 和 DNA 聚合酶 δ 。
T11074 Dolutegravir intermediate-1

1-(2,2-dimethoxyethyl)-5-methoxy-6-methoxycarbonyl-4-oxopyridine-3-carboxylic acid,1-(2,2-dimethoxyethyl)-5-methoxy-6-(methoxycarbonyl)-4-oxo-1,4-dihydropyridine-3-carboxylic acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
Dolutegravir intermediate-1 (1-(2,2-dimethoxyethyl)-5-methoxy-6-(methoxycarbonyl)-4-oxo-1,4-dihydropyridine-3-carboxylic acid) 是 Dolutegravir 的一种新合成中间体。 它是一种整合酶抑制剂,有潜力研究人类免疫缺陷病毒 (HIV)-1 感染。
T15483 LEDGIN6

HIV-1 integrase inhibitor 2

Others Others
HIV-1 integrase inhibitor 2 is used for the treatment of human immunodeficiency virus (HIV) infection.
T7700 Lersivirine

3-氰基-5-[[3,5-二乙基-1-(2-羟基乙基)-1H-吡唑-4-基]氧基]苯腈,Lersivirine(UK 453061),UK-453061

HIV Protease; Reverse Transcriptase Microbiology/Virology; Proteases/Proteasome
Lersivirine (UK-453061) 是非核苷逆转录的抑制剂 (NNRTI),有效抑制 NNRTI 耐药病毒。它对野生型人类免疫缺陷病毒和临床相关 NNRTI 耐药菌株显示出强大的抗逆转录病毒活性。
T76502 HIV-1, HIV-2 Protease Substrate

HIV-1,HIV-2Protease Substrate 是HIV-1HIV-2蛋白酶的底物。HIV-1HIV-2蛋白酶底物结合残基有 4 个保守取代残基。
T27154 Dexelvucitabine

D-D-4FC,DPC-817,RVT,beta-D-D-4FC,DFC

Reverse Transcriptase Microbiology/Virology
Dexelvucitabine (RVT) 是一种胞苷类似物,一种口服有活性的核苷逆转录酶抑制剂。它是一种 2'-脱氧胞苷抗逆转录病毒剂。它是一种有效的抗 HIV-1病毒剂,这些病毒聚合酶中含有胸苷类似物和/或 M184V 突变。
T0100 Atazanavir sulfate

阿扎那韦硫酸盐,BMS-232632,BMS-232632 sulfate,硫酸阿扎那韦

P450; SARS-CoV; HIV Protease; P-gp Membrane transporter/Ion channel; Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Atazanavir sulfate (BMS-232632 sulfate) 是一种氮杂肽和 HIV 蛋白酶抑制剂,与其他抗 HIV 药物联合用于治疗 HIV 感染和艾滋病。它也是SARS-CoV 3CLpro 抑制剂,IC50为 3.49 μM。
T72565 HIV-1 inhibitor-52

HIV-1inhibitor-52 是高效广谱HIV-1活性抑制剂,具备对 WT HIV-1HIV-1 V370A、HIV-1 ΔV370、HIV-1 V362I/V370A、HIV-1 T332S/V362I/prR41G、HIV-1 A326T/V362I/V370A、和HIV-1 R361K/V362I/L363M 等变异株的强效抑制作用,其EC50值范围为 1.6 nM至6.4 nM。
T63813 HIV-1 inhibitor-39

HIV-1 inhibitor-39 是 HIV-1 的有效抑制剂 (EC50>112.88 μM)。 HIV-1 inhibitor-39 具有抗 RT (HIV-1 逆转录酶) 作用 (IC50: 15.75 μM)。HIV-1 inhibitor-39 对 MT-4 细胞表现出细胞毒性 (CC50: 112.9 μM)。
T62431 HIV-1 inhibitor-25

HIV-1 inhibitor-25 (compound R-12a) 是一种 HIV-1 逆转录 (HIV-1 RT) 的高效抑制剂 (IC50: 0.1061 nM)。HIV-1 inhibitor-25 对野生型 HIV-1 表现出较高的抗病毒效果,其 EC50 值为 13.6 nM,且细胞毒性较低 (对 MT-4 细胞的 CC50 值为 33.13 μM)。HIV-1 inhibitor-25 也能够抑制 HIV-1 突变株 (L100I, K103 N, Y181C, Y188L, E138K, F227L+V106A),EC50=0.1961 ~ 5.8136 μM。HIV-1 inhibitor-25 能够用于研究艾滋病。
T61797 HIV-1 inhibitor-15

HIV-1 inhibitor-15 (compound 9d) is a potent and broad-spectrum inhibitor targeting HIV-1. It exhibits inhibitory activity against HIV-1 WT, L100I, K103N, Y181C, and E138K with respective EC50 values of 1.7 nM, 4 nM, 2 nM, 6 nM, and 9 nM. In addition to its high efficacy, HIV-1 inhibitor-15 possesses favorable solubility, safety profiles, and oral bioavailability [1].
T61670 HIV-1 inhibitor-38

HIV-1 inhibitor-38 (Compound 91) is a powerful agent that inhibits the activity of HIV-1. It exhibits great potential as a novel latency reversing agent, making it a promising candidate for further development [1].
T61844 HIV-1 inhibitor-9

HIV-1 inhibitor-9 exhibits potent inhibition activity at low nanomolar concentrations against both the wild-type (WT) HIV-1 strain and multiple strains that have developed resistance to non-nucleoside reverse transcriptase inhibitors (NNRTIs).
T62452 HIV-1 inhibitor-40

HIV-1 inhibitor-40 (Compound 4ab) 是一种 HIV-1 非核苷型逆转录酶抑制剂 (NNRTI) (EC50: 1.9 nM),体内没有明显急性毒性。HIV-1 inhibitor-40 对 CYP 的敏感性较低,作用于 CYP2C9 (IC50: 5.16 μM) 和 CYP2C19 (IC50: 4.51 μM)。
T61311 HIV-1 inhibitor-30

HIV-1 inhibitor-30 (compound 10i) is a potent inhibitor of HIV-1, specifically targeting the RT DNA polymerase enzyme. It exhibits strong antiretroviral activity, with an EC 50 value of 40 nM and an IC 50 value of 80 nM. Furthermore, HIV-1 inhibitor-30 demonstrates significant effectiveness against seven NNRTI-resistant strains of HIV-1 (RT-K103N; RT-Y181C; RT-K103N, Y181C; RT-L100I, K103N; RT-Y188L; RT-K103N, G190A; RT-K103N, V108I), with IC 50 values ranging from 0.04 to 1.42 μM. This compound...

化合物

HIV-1 Inhibitor 18A
Cat.No: T24141
Synonym: HIV-1 Inhibitor-18A
Target: HIV Protease
HIV-1 Nef-IN-1
Cat.No: T9039
Synonym:
Target: HIV Protease
HIV-1 Rev (34-50)
Cat.No: TP1149
Synonym: HIV-1 Rev 34-50,HIV-1 rev Protein (34-50)
Target: HIV Protease
HIV-1 inhibitor-54
Cat.No: T67833
Synonym:
Target: HIV Protease
HIV-1 inhibitor-6 
Cat.No: T9854
Synonym: 3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-
Target: HIV Protease
TAT
Cat.No: TP1809
Synonym:
Target: HIV Protease
Des(benzylpyridyl) Atazanavi
Cat.No: T1883
Synonym:
Target: HIV Protease
HIV Protease Substrate 1
Cat.No: T39729
Synonym:
Target:
HIV-1 inhibitor-3
Cat.No: T11564
Synonym:
Target: Others
HIV-1 integrase inhibitor
Cat.No: T11566
Synonym:
Target: Others
(Cys47)-HIV-1 tat Protein (47-57)
Cat.No: T40719
Synonym: (Cys47)-HIV-1 tat Protein (47-57)
Target:
HIV-1 TAT 48-60
Cat.No: TP1776
Synonym:
Target:
HIV-1 integrase inhibitor 7
Cat.No: T11565
Synonym:
Target: Others
HIV-1 integrase inhibitor 4
Cat.No: T11568
Synonym:
Target: Others
HIV-1 integrase inhibitor 3
Cat.No: T11567
Synonym:
Target: Others
HIV-1 integrase inhibitor 8
Cat.No: T60742
Synonym:
Target: HIV Protease
IMB-301
Cat.No: T9212
Synonym:
Target: Others, HIV Protease
Gardiquimod
Cat.No: T15371
Synonym:
Target: TLR, HIV Protease
lavendustin B
Cat.No: T4182
Synonym: 薰草菌素B
Target: Tyrosinase, transporter, HIV Protease
Reverse transcriptase-IN-1
Cat.No: T12715
Synonym:
Target: HIV Protease
NBD-556
Cat.No: T16276
Synonym:
Target: HIV Protease
Lenacapavir
Cat.No: T11465
Synonym: GS-6207
Target: Others, HIV Protease
BRD3308
Cat.No: T8233
Synonym:
Target: Apoptosis, HIV Protease, HDAC
Clathrin-IN-1
Cat.No: T9063
Synonym:
Target: HIV Protease
Ro24-7429
Cat.No: T28578
Synonym: Ro 24-7429,Ro-24-7429,Ro 247429
Target: HIV Protease
Thiamine disulfide
Cat.No: T20062
Synonym: 二硫化硫胺,TDS,Daiomin,Algoneurina
Target: HIV Protease, Endogenous Metabolite
Cobicistat
Cat.No: T6246
Synonym: Tybost,GS-9350,考西司他
Target: P450, HIV Protease
Hck-IN-1
Cat.No: T11538
Synonym:
Target: HIV Protease, Src, Hck
RO-0335
Cat.No: T9223
Synonym:
Target: Reverse Transcriptase
BMS-707035
Cat.No: T6420
Synonym: N-[(4-氟苯基)甲基1,6-二氢-5-羟基-1-甲基-6-氧代-2-(四氢-1,1-二氧-2H-1,2-噻嗪-2-基)-4-嘧啶甲酰胺
Target: HIV Protease
PTACH
Cat.No: T3199
Synonym: NCH-51,Cpd 51
Target: HIV Protease, HDAC
FGI-106 tetrahydrochloride
Cat.No: T11281L
Synonym:
Target: Virus Protease, HCV Protease, Influenza Virus, HIV Protease
CK176
Cat.No: T27030
Synonym: HIV-1 inhibitor-34,HIV-1 inhibitor 34,CK 176,CK-176,HIV-1 inhibitor34
Target:
Bromosporine
Cat.No: T6255
Synonym:
Target: Epigenetic Reader Domain, CDK
Atazanavir
Cat.No: T0100L
Synonym: Zrivada,Reyataz,Latazanavir,阿扎那韦,BMS-232632
Target: P450, SARS-CoV, HIV Protease, P-gp
Delavirdine mesylate
Cat.No: T7212
Synonym: U 90152 (mesylate),BHAP-U 90152 (mesylate),Delavirdine (mesylate)
Target: HIV Protease, Reverse Transcriptase
Dolutegravir intermediate-1
Cat.No: T11074
Synonym: 1-(2,2-dimethoxyethyl)-5-methoxy-6-methoxycarbonyl-4-oxopyridine-3-carboxylic acid,1-(2,2-dimethoxyethyl)-5-methoxy-6-(methoxycarbonyl)-4-oxo-1,4-dihydropyridine-3-carboxylic acid
Target: HIV Protease
LEDGIN6
Cat.No: T15483
Synonym: HIV-1 integrase inhibitor 2
Target: Others
Lersivirine
Cat.No: T7700
Synonym: 3-氰基-5-[[3,5-二乙基-1-(2-羟基乙基)-1H-吡唑-4-基]氧基]苯腈,Lersivirine(UK 453061),UK-453061
Target: HIV Protease, Reverse Transcriptase
HIV-1, HIV-2 Protease Substrate
Cat.No: T76502
Synonym:
Target:
Dexelvucitabine
Cat.No: T27154
Synonym: D-D-4FC,DPC-817,RVT,beta-D-D-4FC,DFC
Target: Reverse Transcriptase
Atazanavir sulfate
Cat.No: T0100
Synonym: 阿扎那韦硫酸盐,BMS-232632,BMS-232632 sulfate,硫酸阿扎那韦
Target: P450, SARS-CoV, HIV Protease, P-gp
HIV-1 inhibitor-52
Cat.No: T72565
Synonym:
Target:
HIV-1 inhibitor-39
Cat.No: T63813
Synonym:
Target:
HIV-1 inhibitor-25
Cat.No: T62431
Synonym:
Target:
HIV-1 inhibitor-15
Cat.No: T61797
Synonym:
Target:
HIV-1 inhibitor-38
Cat.No: T61670
Synonym:
Target:
HIV-1 inhibitor-9
Cat.No: T61844
Synonym:
Target:
HIV-1 inhibitor-40
Cat.No: T62452
Synonym:
Target:
HIV-1 inhibitor-30
Cat.No: T61311
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T5783 Rosamultin

野蔷薇苷,罗莎白素

Antioxidant; HIV Protease Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Rosamultin 是从Potentilla anserina L 分离的 19 α-羟基型三萜。它抑制 HIV-1 蛋白酶,具有抗氧化、抗炎和镇痛作用。
TN1103 Diphyllin

山荷叶素,二叶草素

ATPase; Proton pump; Influenza Virus; HIV Protease Membrane transporter/Ion channel; Microbiology/Virology; Proteases/Proteasome
Diphyllin 是一种从Justicia procumbens 中分离的芳基萘木脂素,是HIV-1的有效抑制剂,IC50 为 0.38 μM。它是V-ATPase 抑制剂,IC50值为 17 nM,可抑制人破骨细胞中的溶酶体酸化。它抑制NO 产生,IC50值为 50 μM ,具有抗癌和抗炎活性。
T6S2391 L-Chicoric Acid

(-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸

Others; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
L-Chicoric Acid (trans-Caffeoyltartaric acid) 是一种二咖啡酰酒石酸,是一种选择性可逆的 HIV-1 整合酶抑制剂,IC50约为 100 nM。它还可抑制 HIV-1 复制。
T4962 Zingibroside R1

Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1

HIV Protease Microbiology/Virology; Proteases/Proteasome
Zingibroside R1 (Ginsenoside Z-R1) 是分离自Panax japonicasC. A. Meyer 根部的一种三萜皂苷,有HIV-1、抗肿瘤和抗血管生成活性。它对 EAT 细胞的 2-脱氧-D-葡萄糖的摄取具有抑制作用,IC50值为91.3 μM。
T22468 1-Deoxymannojirimycin hydrochloride

Others; Influenza Virus; HIV Protease Microbiology/Virology; Others; Proteases/Proteasome
1-Deoxymannojirimycin hydrochloride 是一种选择性的 α1,2-甘露糖苷酶抑制剂,IC50值为 20 μM。它还抑制 HIV-1 毒株,抗病毒活性较差。
T0200 α-Lipoic Acid

Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid,α-硫辛酸,硫辛酸

Apoptosis; NF-κB; HIV Protease; Mitochondrial Metabolism; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
α-Lipoic Acid (DL-α-Lipoic acid) 是线粒体酶复合物的重要辅助因子,是一种抗氧化剂,可抑制NF-κB 依赖性的HIV-1LTR 活化。它还可诱导内质网应激介导的肝癌细胞凋亡。
T4S1383 Escin IA

Aescin IA,Escin IA;Aescin IA,Escin IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Escin IA (Escin IA;Aescin IA);Aescin IA 是从马蹄中七叶树分离出的一种三萜皂苷,抑制HIV-1蛋白酶,IC50值为 35 μM。它具有抗 TNBC 转移活性,其作用机制涉及通过下调 LOXL2 表达抑制上皮-间质转化过程。
T4S1718 Punicalin

HBV; HIV Protease Microbiology/Virology; Proteases/Proteasome
Punicalin 是从Punica granatumL. 或Terminalia catappaL. 的叶子中分离的,一种可水解的单宁,具有抗炎活性。它是一种抗乙型肝炎病毒药物。
T3730 Methyl gallate

NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯

Reactive Oxygen Species; HIV Protease; Reverse Transcriptase; Antibacterial Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Methyl gallate (Gallincin) 是具有抗氧化,抗癌和抗炎活性的植物酚类。它也可抑制细菌活性。它还具有抗HIV-1HIV-1酶的抑制活性。
T2S0223 Isosinensetin

异橙黄酮,6-Demethoxynobiletin

Antioxidant; HIV Protease; Antibacterial; P-gp Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience; oxidation-reduction; Proteases/Proteasome
Isosinensetin (6-Demethoxynobiletin) 是从青皮中提取的一种甲氧基黄酮,具有抗氧化和抑制 HIV-1 蛋白酶的活性。
T4S1387 Isoescin IA

七叶皂苷C,异七叶皂苷 IA

HIV Protease Microbiology/Virology; Proteases/Proteasome
Isoescin IA 是一种从七叶树种子中分离出来的三萜皂苷。它具有抗HIV-1蛋白酶活性。
TN2283 Tripterifordin

HIV Protease Microbiology/Virology; Proteases/Proteasome
Tripterifordin 在 H9 淋巴细胞中显示出抗 HIV 复制活性,EC50值为 3100 nM。
TN5263 1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one

Xanthohumol,黄腐酚

Apoptosis; BCL; PARP; HCV Protease; IAP; Caspase; HIV Protease; NMDAR; p53 Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Microbiology/Virology; Neuroscience; Proteases/Proteasome
1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one (Xanthohumol) 是一种从蛇麻草中提纯的具有多种生物功能的天然产物。黄腐酚对 HIV-1 有效,可能是一种有趣的先导化合物。它可能代表一种用于 HIV-1 感染的新型化疗药物。
T3323 Ursonic Acid

CCRIS 7123,NSC4060,熊果酮酸,Prunol,3-Ketoursolic acid,Malol,TOS-BB-0966

Apoptosis; HIV Protease; Endogenous Metabolite Apoptosis; Metabolism; Microbiology/Virology; Proteases/Proteasome
Ursonic Acid (TOS-BB-0966) 是一种天然三萜酸,属于熊果烷三萜类,其结构基于五环熊果烷骨架。 它具有作为 HIV-1 蛋白酶抑制剂的潜力。
T5782 Bevirimat

YK FH312,MPC-4326,PA-457,贝韦立马

HIV Protease Microbiology/Virology; Proteases/Proteasome
Bevirimat (PA-457) 是一种 HIV-1 成熟抑制剂,可在病毒体成熟过程中阻断 Gag 衣壳 (CA) 前体 CA-SPI 裂解为成熟的 CA 蛋白。
TJS1779 Protosappanin A

原苏木素A,PTA

NADPH-oxidase; IL Receptor; IκB/IKK; TNF; NF-κB; TLR; ROS; COX; HIV Protease; JAK; NO Synthase; STAT Angiogenesis; Apoptosis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Microbiology/Virology; Neuroscience; NF-κB; Proteases/Proteasome; Stem Cells
Protosappanin A (PTA) 是从苏木中分离得到的免疫抑制成分和主要联苯化合物,通过下调 JAK2和 STAT3的磷酸化,抑制 JAK2/STAT3依赖的炎症通路。
T2S1158 4,5-Dicaffeoylquinic acid

3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C

Others; HBV; Endogenous Metabolite Metabolism; Microbiology/Virology; Others
4,5-Dicaffeoylquinic acid (Isochlorogenic acid C) 是一种天然产物,有抗病毒、抗肝毒性活性。
T4S1521 1,4-Dicaffeoylquinic acid

1,4-二咖啡酰奎宁酸,洋蓟素

HIV Protease Microbiology/Virology; Proteases/Proteasome
1,4-Dicaffeoylquinic acid 是一种苯丙素类物质,从苍耳子中获得,可以减少 LPS 诱导的 TNF-α 的生成,具有抗炎活性。
T4537 Cholic acid sodium

胆酸钠,[胆酸钠],SodiumCholate

HIV Protease; Endogenous Metabolite Metabolism; Microbiology/Virology; Proteases/Proteasome
Cholic acid sodium (SodiumCholate) 是肝脏中产生的主要胆汁酸,通常与牛磺酸或甘氨酸结合,有助于脂肪吸收和胆固醇排泄。
TL0006 Cichoric Acid

菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Cichoric Acid (Dicaffeoyltartaric acid) 是一种天然化合物,具有抗氧化作用。
T6841 Fumagillin

NSC9168,烟曲霉素,Amebacilin

Others; HIV Protease; Antibiotic; Parasite Microbiology/Virology; Others; Proteases/Proteasome
Fumagillin (Amebacilin) 由烟曲霉菌中提取的一种抗菌药,有抗阿米巴活性。它通过抑制 HIV-1 viral protein R 活性来抑制 HIV1感染。
T4S0295 Apigenin 7-glucoside

波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin

Reactive Oxygen Species; HIV Protease Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Apigenin 7-glucoside (Cosmosiin) 是一种 ROS 清除剂,具有抗增殖、抗氧化作用。
T8689 Chloroquine

CQ,氯喹

SARS-CoV; TLR; HIV Protease; Antibiotic; Parasite; Autophagy Autophagy; Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Chloroquine 是一种 Toll 样受体抑制剂,可以抑制自噬。Chloroquine 具有抗疟疾和抗炎活性,广泛用于治疗疟疾和类风湿性关节炎。Chloroquine 还具有抗 SARS-CoV-2 (COVID-19) 活性、抗 HIV-1 活性。
T2930 α-Lipoic Acid

Lipoic acid,Alphalipoic acid,硫辛酸

NF-κB; HIV Protease; Mitochondrial Metabolism; Endogenous Metabolite Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
α-Lipoic Acid (Alphalipoic acid) 抑制 NF-κB 依赖性 HIV-1 LTR 活化。 α-硫辛酸诱导内质网 (ER) 应激介导的肝癌细胞凋亡。α-硫辛酸是一种抗氧化剂,是线粒体酶复合物的重要辅助因子。
T3122 Fangchinoline

Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline

Apoptosis; FAK; HIV Protease; Autophagy Angiogenesis; Apoptosis; Autophagy; Cytoskeletal Signaling; Microbiology/Virology; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Fangchinoline (Tetrandrine B) 是从Stephaniatetrandra 中分离出来的,一种具有广泛生物学活性的天然产物。它是新型HIV-1抑制剂,通过损害 gp160 蛋白水解过程来抑制 HIV-1 复制。它靶向Focal adhesion kinase (FAK)并抑制肿瘤细胞中 FAK 介导的的信号传导途径。
TN1622 Ermanin

堪非醇3,4'-二-O-甲醚

NOS; Influenza Virus; COX; HIV Protease; Antibacterial; Antibiotic Immunology/Inflammation; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Ermanin 是一种从 Tanacetum microphyllum 中分离出来的类黄酮。Ermanin抑制血小板聚集,具有抗结核和抗病毒/细菌特性。Ermanin 可抑制 iNOS 和 COX-2 的表达,从而具有抗炎活性。Ermanin 可能具有抗 HIV-1 活性。Ermanin 在较低浓度下可有效地抑制 Dione juno 幼虫。
T5S2017 Ingenol

(-)-Ingenol,巨大戟二萜醇,巨大戟醇

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Ingenol ((-)-Ingenol) 是一种PKC 激活剂,Ki 值为 30 μM,具有抗肿瘤活性。 从 Ingenol 酯中配制新的衍生物可能是开发新的先导化合物以重新激活潜伏 HIV 的创新方法。Ingenol mebutate 是治疗光化性角化病的有效方法。
TN1059 Ganoderic acid B

IL Receptor; HIV Protease; JAK; STAT Angiogenesis; Chromatin/Epigenetic; Immunology/Inflammation; JAK/STAT signaling; Microbiology/Virology; Proteases/Proteasome; Stem Cells
Ganoderic acid B 是从灵芝中分离的一种三萜类天然产物。它是端粒酶抑制剂,抑制 Epstein-Barr 病毒抗原的活化。它是 HIV-1 蛋白酶抑制剂。
T4839 Ac-Ala-OH

N-Acetylalanine,N-Acetyl-L-alanine,N-乙酰-L-丙氨酸

Others; Endogenous Metabolite Metabolism; Others
Ac-Ala-OH (N-Acetyl-L-alanine) 是鸟嘌呤核苷酸结合蛋白G(I)/G(S)/G(O) γ -2亚基、髓鞘碱性蛋白、GTP-结合核蛋白 Ran、原肌球蛋白 α - 4链、HIV-1 Rev 结合蛋白2、Xaa-Pro 二肽酶、胸腺酶 β -10、肌动蛋白样蛋白3、丙氨酸转氨酶、丝氨酸/苏氨酸蛋白磷酸酶PP1 - β催化亚基、10 kda 热休克蛋白(线粒体)、钙调蛋白和 β -1-syntrophin 的底物。
TN1727 Helichrysetin

4,2',4'-三羟基-6'-甲氧基查耳酮,蜡菊亭

Apoptosis; HIV Protease Apoptosis; Microbiology/Virology; Proteases/Proteasome
Helichrysetin 是从豆蔻果实中分离出的一种天然产物,是一种 DNA 结合抑制剂,可抑制原位导管癌DCIS 的形成。它抑制细胞生长,可诱导 A549 细胞凋亡。
T5S1103 Isoliensinine

异莲心碱,Isoliensinin

Apoptosis; Antioxidant Apoptosis; oxidation-reduction
Isoliensinine (Isoliensinin) 是从水芙蓉种子胚中提取的一种双苄基异喹啉生物碱,能诱导三阴性乳腺癌细胞凋亡,具有抗氧化、抗炎、抗癌活性。
T0474 Erythromycin ethylsuccinate

EES,琥乙红霉素

ribosome; HIV Protease; Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology; Proteases/Proteasome
Erythromycin ethylsuccinate (EES) 是一种由红链霉菌产生的大环内酯类抗生素,有潜力用于多种细菌感染。它具有抗 HIV-1病毒活性。
T3321 Oleanonic acid

3-Oxooleanolic acid,3-Oxoolean-12-en-28-oic Acid,Oleanonic Acid,齐墩果酮酸,3-Ketooleanolic Acid

HIV Protease Microbiology/Virology; Proteases/Proteasome
Oleanonic acid (3-Ketooleanolic Acid) 是一种三萜,可以抑制 HIV-1 对细胞的感染。它具有保肝作用,并具有抗肿瘤和抗病毒特性。
T0966 Sennoside A

番泻苷A,NSC 112929,番泻苷 A

MAO; HIV Protease Metabolism; Microbiology/Virology; Neuroscience; Proteases/Proteasome
Sennoside A (NSC-112929) 是在番泻叶的叶子和豆荚中大量发现的蒽醌苷,抑制 HIV-1 复制。
T16791 Rottlerin

Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525

CaMK; Apoptosis; Others; HIV Protease; PKA; PKC; Autophagy Apoptosis; Autophagy; Chromatin/Epigenetic; Cytoskeletal Signaling; Microbiology/Virology; Neuroscience; Others; Proteases/Proteasome; Tyrosine Kinase/Adaptors
Rottlerin (NSC-56346) 是一种从Mallotus Philippinensis 中得到的天然产物, 是 PKC 的特异性抑制剂,抑制HIV-1整合和狂犬病病毒感染。它通过活化 caspase 3 诱导细胞凋亡.
T5429 Theaflavin 3,3'-digallate

茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG

Virus Protease; Antioxidant; HIV Protease; HSV Microbiology/Virology; oxidation-reduction; Proteases/Proteasome
Theaflavin 3,3'-digallate (8-Gingerol) 是一种寨卡病毒蛋白酶抑制剂,IC50为 2.3 μM。它直接与 ZIKVpro 结合并抑制 ZIKV 复制,可抑制 gp41 和 NS2B-3 蛋白酶的活性,并具有抗 HSV 和 HIV-1病毒活性。它是红茶中的主要多酚,有抗肿瘤作用。
T2S0731 Trilobatin

三叶苷,三叶甙,P-Phlorizin

Amylase Metabolism
Trilobatin (P-Phlorizin) 是源自Lithocarpus polystachyusRehd 的甜味剂,是一种HIV-1抑制剂,靶向 Gp41 包膜蛋白,具有神经保护作用。它还是SGLT1/2抑制剂,可选择性诱导人肝母细胞瘤细胞增殖。
T4S0797 Berberine

小檗碱,Berberin,Umbellatine,黄连素

Reactive Oxygen Species; Topoisomerase; Endogenous Metabolite; Antibacterial; Antibiotic; Autophagy Autophagy; DNA Damage/DNA Repair; Immunology/Inflammation; Metabolism; Microbiology/Virology; NF-κB
Berberine (Umbellatine) 是从中草药黄连中分离出来的一种生物碱抗生素。它诱导活性氧生成并抑制 DNA 拓扑异构酶,具有抗肿瘤特性。
T2830 Betulinic acid

白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid

Apoptosis; Mitophagy; NF-κB; HIV Protease; Topoisomerase; Endogenous Metabolite; Aminopeptidase; Autophagy Apoptosis; Autophagy; DNA Damage/DNA Repair; Metabolism; Microbiology/Virology; NF-κB; Proteases/Proteasome
Betulinic acid (ALS-357) 是从白桦树皮中分离出来的一种五环三萜类天然产物,是真核细胞拓扑异构酶 I 的抑制剂,IC50值为 5 μM,具有抗逆转录病毒、抗疟疾、抗癌和抗炎特性。
TN5675 Ganomycin I

Ganomycin I inhibits the activity of HIV-1 protease.
TN6541 Cleomiscosin B

Cleomiscosins A, B and C exhibit liver-protective properties. Cleomiscosin B shows the potent anti-HIV-1 activity in vitro and also has protective effects on MT4 cells infected by HIV-1(IIIB).
TN5012 Shizukaol C

HIV Protease; Antifection Microbiology/Virology; Proteases/Proteasome
1. Shizukaol C shows anti-HIV-1 replication activities in both wild-type HIV-1 and two NNRTIs-resistant strains. <br/> 2. Shizukaol C has significant cytotoxicities against C8166 cells. <br/>
TN4820 Pre-schisanartanin B

HIV Protease Microbiology/Virology; Proteases/Proteasome
Pre-schisanartanin B has cytotoxicity, it also has anti-HIV-1 activity.
TN4555 Methyl salvionolate A

HIV Protease Microbiology/Virology; Proteases/Proteasome
Methyl salvionolate A has anti-HIV-1 activity.
T73758 Glycolithocholic acid 3-sulfate

Glycolithocholic acid 3-sulfate (SLCG) 为一种胆汁酸衍生物及甘胆酸的代谢产物,具有抑制HIV-1复制的作用。该化合物在HIV感染和胆囊疾病的研究中有潜在应用价值。
T25445 Ganoderiol B

Ganoderiol B is a moderately active HIV-1 PR inhibitor (IC50: 0.17-0.23 mM).
T75553 Salvianan A

1,6,11-Trimethyl-1,2-dihydrofuro[2',3':1,2]phenanthro[4,3-d]oxazole (compound 1) 是一种有效的抗HIV-1剂。
TN4835 Przewalskin

HIV Protease Microbiology/Virology; Proteases/Proteasome
Przewalskin A and Przewalskin B showed modest anti-HIV-1 activity with EC50 = 41 and 30 microg/mL, respectively.
T2S0605 Liquidambaric lactone

HIV Protease Microbiology/Virology; Proteases/Proteasome
Liquidambaric lactone 是一种分离自Euonymus grandiflorusWall 中的化合物。
T80952 Tremuloidin

Tremuloidin (Compound 2)为源自Homalium cochinchinensis的水杨酸衍生物,其对HIV-1活性表现出较弱的抑制效果。
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天然产物

Rosamultin
Cat.No: T5783
Synonym: 野蔷薇苷,罗莎白素
Target: Antioxidant, HIV Protease
Diphyllin
Cat.No: TN1103
Synonym: 山荷叶素,二叶草素
Target: ATPase, Proton pump, Influenza Virus, HIV Protease
L-Chicoric Acid
Cat.No: T6S2391
Synonym: (-)-Chicoric acid,trans-Caffeoyltartaric acid,Chicoric acid,L-菊苣酸,dicaffeoyltartaric acid,菊苣酸
Target: Others, HIV Protease
Zingibroside R1
Cat.No: T4962
Synonym: Ginsenoside Z-R1,姜状三七皂苷R1,姜状三七苷R1
Target: HIV Protease
1-Deoxymannojirimycin hydrochloride
Cat.No: T22468
Synonym:
Target: Others, Influenza Virus, HIV Protease
α-Lipoic Acid
Cat.No: T0200
Synonym: Thioctic acid,DL-α-Lipoic acid,(±)-α-Lipoic acid,α-硫辛酸,硫辛酸
Target: Apoptosis, NF-κB, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite
Escin IA
Cat.No: T4S1383
Synonym: Aescin IA,Escin IA;Aescin IA,Escin IA
Target: HIV Protease
Punicalin
Cat.No: T4S1718
Synonym:
Target: HBV, HIV Protease
Methyl gallate
Cat.No: T3730
Synonym: NSC 363001,Gallicin,Gallic acid methyl ester,Gallincin,没食子酸甲酯
Target: Reactive Oxygen Species, HIV Protease, Reverse Transcriptase, Antibacterial
Isosinensetin
Cat.No: T2S0223
Synonym: 异橙黄酮,6-Demethoxynobiletin
Target: Antioxidant, HIV Protease, Antibacterial, P-gp
Isoescin IA
Cat.No: T4S1387
Synonym: 七叶皂苷C,异七叶皂苷 IA
Target: HIV Protease
Tripterifordin
Cat.No: TN2283
Synonym:
Target: HIV Protease
1-[2,4-Dihydroxy-6-methoxy-3-(3-methyl-2-buten-1-yl)phenyl]-3-(4-hydroxyphenyl)-2-propen-1-one
Cat.No: TN5263
Synonym: Xanthohumol,黄腐酚
Target: Apoptosis, BCL, PARP, HCV Protease, IAP, Caspase, HIV Protease, NMDAR, p53
Ursonic Acid
Cat.No: T3323
Synonym: CCRIS 7123,NSC4060,熊果酮酸,Prunol,3-Ketoursolic acid,Malol,TOS-BB-0966
Target: Apoptosis, HIV Protease, Endogenous Metabolite
Bevirimat
Cat.No: T5782
Synonym: YK FH312,MPC-4326,PA-457,贝韦立马
Target: HIV Protease
Protosappanin A
Cat.No: TJS1779
Synonym: 原苏木素A,PTA
Target: NADPH-oxidase, IL Receptor, IκB/IKK, TNF, NF-κB, TLR, ROS, COX, HIV Protease, JAK, NO Synthase, STAT
4,5-Dicaffeoylquinic acid
Cat.No: T2S1158
Synonym: 3,4-Dicaffeoylquinic acid,异绿原酸C(4,5),Isochlorogenic acid C
Target: Others, HBV, Endogenous Metabolite
1,4-Dicaffeoylquinic acid
Cat.No: T4S1521
Synonym: 1,4-二咖啡酰奎宁酸,洋蓟素
Target: HIV Protease
Cholic acid sodium
Cat.No: T4537
Synonym: 胆酸钠,[胆酸钠],SodiumCholate
Target: HIV Protease, Endogenous Metabolite
Cichoric Acid
Cat.No: TL0006
Synonym: 菊苣酸,Dicaffeoyltartaric acid,Chicoric Acid
Target: Reactive Oxygen Species, HIV Protease
Fumagillin
Cat.No: T6841
Synonym: NSC9168,烟曲霉素,Amebacilin
Target: Others, HIV Protease, Antibiotic, Parasite
Apigenin 7-glucoside
Cat.No: T4S0295
Synonym: 波斯菊,Cosmetin,Cosmosiin,Cosmosioside,Apigenin-7-O-β-D-glucopyranoside,芹甙元-7-葡萄糖苷,Thalictiin,Apigetrin
Target: Reactive Oxygen Species, HIV Protease
Chloroquine
Cat.No: T8689
Synonym: CQ,氯喹
Target: SARS-CoV, TLR, HIV Protease, Antibiotic, Parasite, Autophagy
α-Lipoic Acid
Cat.No: T2930
Synonym: Lipoic acid,Alphalipoic acid,硫辛酸
Target: NF-κB, HIV Protease, Mitochondrial Metabolism, Endogenous Metabolite
Fangchinoline
Cat.No: T3122
Synonym: Tetrandrine B,防己诺林碱,(+)-Limacine,Hanfangichin B,防己醇灵,(+)-Fangchinoline
Target: Apoptosis, FAK, HIV Protease, Autophagy
Ermanin
Cat.No: TN1622
Synonym: 堪非醇3,4'-二-O-甲醚
Target: NOS, Influenza Virus, COX, HIV Protease, Antibacterial, Antibiotic
Ingenol
Cat.No: T5S2017
Synonym: (-)-Ingenol,巨大戟二萜醇,巨大戟醇
Target: PKC
Ganoderic acid B
Cat.No: TN1059
Synonym:
Target: IL Receptor, HIV Protease, JAK, STAT
Ac-Ala-OH
Cat.No: T4839
Synonym: N-Acetylalanine,N-Acetyl-L-alanine,N-乙酰-L-丙氨酸
Target: Others, Endogenous Metabolite
Helichrysetin
Cat.No: TN1727
Synonym: 4,2',4'-三羟基-6'-甲氧基查耳酮,蜡菊亭
Target: Apoptosis, HIV Protease
Isoliensinine
Cat.No: T5S1103
Synonym: 异莲心碱,Isoliensinin
Target: Apoptosis, Antioxidant
Erythromycin ethylsuccinate
Cat.No: T0474
Synonym: EES,琥乙红霉素
Target: ribosome, HIV Protease, Antibacterial, Antibiotic, Autophagy
Oleanonic acid
Cat.No: T3321
Synonym: 3-Oxooleanolic acid,3-Oxoolean-12-en-28-oic Acid,Oleanonic Acid,齐墩果酮酸,3-Ketooleanolic Acid
Target: HIV Protease
Sennoside A
Cat.No: T0966
Synonym: 番泻苷A,NSC 112929,番泻苷 A
Target: MAO, HIV Protease
Rottlerin
Cat.No: T16791
Synonym: Mallotoxin,NSC 56346,粗糠柴苦素,NSC 94525
Target: CaMK, Apoptosis, Others, HIV Protease, PKA, PKC, Autophagy
Theaflavin 3,3'-digallate
Cat.No: T5429
Synonym: 茶黄素-3,3'-双没食子酸,8-Gingerol,TFDG
Target: Virus Protease, Antioxidant, HIV Protease, HSV
Trilobatin
Cat.No: T2S0731
Synonym: 三叶苷,三叶甙,P-Phlorizin
Target: Amylase
Berberine
Cat.No: T4S0797
Synonym: 小檗碱,Berberin,Umbellatine,黄连素
Target: Reactive Oxygen Species, Topoisomerase, Endogenous Metabolite, Antibacterial, Antibiotic, Autophagy
Betulinic acid
Cat.No: T2830
Synonym: 白桦脂酸,桦木酸,ALS-357,Lupatic acid,Betulic acid
Target: Apoptosis, Mitophagy, NF-κB, HIV Protease, Topoisomerase, Endogenous Metabolite, Aminopeptidase, Autophagy
Ganomycin I
Cat.No: TN5675
Synonym:
Target:
Cleomiscosin B
Cat.No: TN6541
Synonym:
Target:
Shizukaol C
Cat.No: TN5012
Synonym:
Target: HIV Protease, Antifection
Pre-schisanartanin B
Cat.No: TN4820
Synonym:
Target: HIV Protease
Methyl salvionolate A
Cat.No: TN4555
Synonym:
Target: HIV Protease
Glycolithocholic acid 3-sulfate
Cat.No: T73758
Synonym:
Target:
Ganoderiol B
Cat.No: T25445
Synonym:
Target:
Salvianan A
Cat.No: T75553
Synonym:
Target:
Przewalskin
Cat.No: TN4835
Synonym:
Target: HIV Protease
Liquidambaric lactone
Cat.No: T2S0605
Synonym:
Target: HIV Protease
Tremuloidin
Cat.No: T80952
Synonym:
Target:
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