store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year
1-Deoxymannojirimycin hydrochloride 是一种选择性的 α1,2-甘露糖苷酶抑制剂,IC50值为 20 μM。它还抑制 HIV-1 毒株,抗病毒活性较差。
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
1 mg | ¥ 490 | 4-5周 | ||
5 mg | ¥ 1,470 | 4-5周 | ||
10 mg | ¥ 2,200 | 4-5周 | ||
25 mg | ¥ 3,670 | 4-5周 |
产品描述 | 1-Deoxymannojirimycin hydrochloride is a selective α1,2-mannosidase inhibitor(IC50: 20 μM). 1-Deoxymannojirimycin hydrochloride also inhibits HIV‐1 strains and has poor antiviral activity. |
靶点活性 | α1/2 mannosidase I:20 μM |
体外活性 | Exposure of such mutant virus strains to 1-Deoxymannojirimycin results in an enhanced suppression of mutant virus-induced cytopathicity in CEM cell cultures[1].When combined with CBAs at concentrations that showed poor if any suppression of mutant virus replication as single drugs, a synergistic antiviral activity of 1-Deoxymannojirimycin was observed[1]. |
分子量 | 199.63 |
分子式 | C6H14ClNO4 |
CAS No. | 73465-43-7 |
store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 20 mg/ml(100.19 mM)
H2O: 20 mg/ml(100.19 mM)
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO / H2O | 1 mM | 5.0093 mL | 25.0463 mL | 50.0927 mL | 125.2317 mL |
5 mM | 1.0019 mL | 5.0093 mL | 10.0185 mL | 25.0463 mL | |
10 mM | 0.5009 mL | 2.5046 mL | 5.0093 mL | 12.5232 mL | |
20 mM | 0.2505 mL | 1.2523 mL | 2.5046 mL | 6.2616 mL | |
50 mM | 0.1002 mL | 0.5009 mL | 1.0019 mL | 2.5046 mL | |
100 mM | 0.0501 mL | 0.2505 mL | 0.5009 mL | 1.2523 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
1-Deoxymannojirimycin hydrochloride 73465-43-7 Microbiology/Virology Others Proteases/Proteasome Influenza Virus HIV Protease 1 Deoxymannojirimycin hydrochloride HIV-1 inhibit glycosylation antiviral reticulum HIV α1,2-mannosidase Human immunodeficiency virus N-linked 1-Deoxymannojirimycin Hydrochloride Inhibitor 1Deoxymannojirimycin hydrochloride 1-Deoxymannojirimycin Endoplasmic inhibitor