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459

抑制剂 & 化合物

68

天然产物

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Cat. No. Product Name Target Signaling Pathways
T34744 Sulfo-NHS-LC-Biotin

long chain Sulfo NHS Biotin

Sulfo-NHS-LC-Biotin, or Sulfosuccinimidyl 6-(biotinamido) Hexanoate, is a long-chain water-soluble biotinylating agent that targets cell surface proteins and is reactive to primary amine groups.
T5051 Isopropamide Iodide

AChR Neuroscience
Isopropamide iodide 是长效季铵盐抗胆碱能药物。它用于研究消化性溃疡和其他胃肠道疾病,尤其是胃酸过多和运动过度。
T8133 SulfadiMethoxine sodium

Anti-infection; Antibacterial; Antibiotic Microbiology/Virology
SulfadiMethoxine sodium 是一种磺胺类抗生素,可研究由多种感染引起的疾病。
T4985 Neticonazole Hydrochloride

Antifungal Microbiology/Virology
Neticonazole hydrochloride 是一种咪唑衍生物,具有抗感染和抗癌作用。它也是一种长效抗真菌剂。
T9778 KCNQ1 activator-1 

Potassium Channel Membrane transporter/Ion channel
KCNQ1 activator-1 是有效的 KCNQ1通道激活剂。它在研究长 QT 综合征中有研究的价值。
T1078 Sulfadimethoxine

Sulphadimethoxine,磺胺二甲氧嗪

Antibacterial; Antibiotic Microbiology/Virology
Sulfadimethoxine (Sulphadimethoxine) 是一种磺胺类抗生素,用于多种感染引起的疾病的研究。
T12103 MR-L2

PDE Metabolism
MR-L2 是可逆的、非竞争性的长型异构体磷酸二酯酶 -4激活剂,可以激活代表性的 PDE4 长型异构体 (PDE4A4、PDE4B1、PDE4C3、PDE4D5)。它可抑制 PGE2- 诱导的 MDCK 细胞囊肿形成,其EC50=1.2 µM。
T0388 Cilnidipine

FRC-8653,西尼地平

Calcium Channel Membrane transporter/Ion channel; Metabolism
Cilnidipine (FRC-8653) 是二氢吡啶类Ca2+通道阻断剂,可作用于 L 和 N 型 Ca2+通道,具有抗高血压活性。
T7808 Alacepril

Cetapril,阿拉普利,DU-1219

RAAS Endocrinology/Hormones
Alacepril (DU-1219) 是一种具有口服活性血管紧张素转换酶 (ACE) 抑制剂,具有长效抗高血压作用。
T8778 TTK21

Epigenetic Reader Domain Chromatin/Epigenetic
TTK21 是 CBP/p300 组蛋白乙酰转移酶活性的激活剂,与葡萄糖基碳纳米球结合时,可通过血脑屏障,对成人大脑神经发生和长期记忆功能有益。
T12732 Rezafungin

棘白菌素,SP-3025,CD101,Biafungin

Others; Antifungal Microbiology/Virology; Others
Rezafungin (SP-3025) 是一种长效的广谱棘皮菌素,对念珠菌、曲霉和肺孢子菌具有强效抗真菌活性。
T7943 Fluphenazine decanoate

Dopamine Receptor GPCR/G Protein; Neuroscience
Fluphenazine decanoate 是一种高度连续的多巴胺 D2受体阻滞剂,是一种长效吩噻嗪抗精神病药,用于精神分裂症的研究。
T3716 Rolapitant

罗拉吡坦,SCH619734,罗拉匹坦

Neurokinin receptor GPCR/G Protein; Neuroscience
Rolapitant (SCH619734) 是一种高效选择性具有口服活性的神经激肽 1 受体抑制剂,Ki 值为0.66 nM。
T6541 Ibutilide Fumarate

Corvert Fumarate,U70226E,富马酸伊布利特

Calcium Channel; Sodium Channel Membrane transporter/Ion channel; Metabolism
Ibutilide Fumarate (U70226E) 是一种 III 类抗心律失常药物,可作用于急性心梗阻塞。
T41323 Dihomo-γ-Linolenic acid methyl ester

Others Others
Dihomo-γ-Linolenic acid methyl ester 是 Dihomo-γ-Linolenic acid 的甲酯形式,Dihomo-γ-Linolenic acid 具有抗炎和抗增殖作用。
T9578 ELOVL1-IN-1

1-(2-Fluorophenyl)-N-(1-(2-fluoropyridin-4-YL)-1H-pyrazol-3-YL)cyclopropane-1-carboxamide

Others Others
ELOVL1-IN-1 (1-(2-Fluorophenyl)-N-(1-(2-fluoropyridin-4-YL)-1H-pyrazol-3-YL)cyclopropane-1-carboxamide) 是ELOVL1抑制剂,能够降低超长链脂肪酸的水平,可用于肾上腺脑白质营养不良的研究。
T5159 Olodaterol hydrochloride

BI-1744 HCl,盐酸奥达特罗,BI 1744 hydrochloride

Adrenergic Receptor GPCR/G Protein; Neuroscience
Olodaterol hydrochloride (BI-1744 HCl) 是一种长效的、选择性 β2-adrenoceptor(β2-AR) 激动剂 (EC50=0.1 nM;pKi= 9.14 for human β2-adrenoceptor),可用于慢性阻塞性肺疾病 (COPD) 和肺纤维化的研究。
T20720 Norethisterone enanthate

NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,炔诺酮庚酸酯,NSC-9564

Estrogen/progestogen Receptor Endocrinology/Hormones
Norethisterone enanthate (NSC-9564) 是一种口服有效的长效的孕激素。
T2390 Cevimeline hydrochloride hemihydrate

AChR Neuroscience
Cevimeline hydrochloride hemihydrate 是乙酰胆碱的奎尼丁衍生物,也是选择性的和口服活性的毒蕈碱型M1和M3受体激动剂。它可穿过血脑屏障,刺激唾液腺分泌,用作口干症的催涎剂。
T5358 Longdaysin

ERK; Casein Kinase; CDK Cell Cycle/Checkpoint; MAPK; Metabolism; Stem Cells
Longdaysin 是一种 CK1α 和 CK1δ 的抑制剂,IC50为5.6和8.8 µM。它还抑制ERK2,IC50值为52 µM。它是Wnt/β-catenin 信号通路的抑制剂,通过阻断CK1δ/ε依赖性 Wnt 信号通路发挥抗肿瘤作用。
T22774L eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species](TFA)

Others Others
eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species](TFA) 是延伸因子 1 亚基。真核翻译延伸因子 1 alpha 1 (EEF1A1) 编码延伸因子 alpha 亚基的同种型- 1 复合物,负责将氨酰 tRNA 酶促递送至核糖体。这种亚型(α 1)在脑、胎盘、肺、肝、肾和胰腺中表达,另一种亚型(α 2)在脑、心脏和骨骼肌中表达。这种亚型在 66% 的 Felty 综合征患者中被鉴定为自身抗原。已发现该基因在许多染色体上具有多个拷贝,其中一些(如果不是全部)代表不同的假基因。
T125797 Longilactone, delta-4(18)-Isomer, 2alpha-alcoho

Longilactone, delta-4(18)-Isomer, 2alpha-alcoho 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T125797,CAS号为 149155-28-2。
T32862 Longicin

Longicin is a cytotoxic agent isolated from Asimina longifolia.
T32863 Longicoricin

Longicoricin is a monotetrahydrofuran Annonaceous acetogenin from Asimina longifolia.
T60682 Elongation factor P-IN-2

Elongation factor P-IN-2可影响大肠杆菌的增殖率。Elongation factor P-IN-2 是 β-赖氨酸衍生化合物,是延伸因子 P (EFP)的有效抑制剂。
T124889 Isocalolongic acid

Isocalolongic acid 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124889,CAS号为 40737-92-6。
T72727 Huanglongmycin N

Huanglongmycin N为DNA拓扑异构酶I (DNA topoisomerase I) 抑制剂,表现出EC50值为14 μM。
T24429 Malonganenone A

Malonganenone-A,Malonganenone-E,Malonganenone E

Malonganenone A is a selective plasmodial Hsp70s modulator. It also has antimalarial activity.
T130680 Longicaulenone

Longicaulenone 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T130680。
T126352 (-)-Isolongifolol

(-)-Isolongifolol 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126352,CAS号为 1139-17-9。
T124874 Virolongin B

Virolongin B 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T124874,CAS号为 41535-94-8。
T130156 8,10-Dihydroxy-3-longipinen-5-one, diangeloyl

8,10-Dihydroxy-3-longipinen-5-one, diangeloyl 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T130156。
T60491 Elongation factor P-IN-1

Elongation factor P-IN-1 是 β-赖氨酸衍生化合物,是延伸因子 P (EFP) 的有效抑制剂,可影响大肠杆菌的增殖率。
T126080 Longilactone

Longilactone 是一种有用的有机化合物,可用于生命科学领域的相关研究。其产品编号为 T126080,CAS号为 129587-09-3。
T32859 Longanlactone

Longanlactone is a natural neurotrophic agent.
T22774 eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species]

Others Others
eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) encodes an isoform of the alpha subunit of the elongation factor-1 complex, which is responsible for the enzymatic delivery of aminoacyl tRNAs to the ribosome. This isoform (alpha 1) is expressed
T31716 Etidocaine Hydrochloride

W-19053,Duranest,W19053,W 19053

Sodium Channel Membrane transporter/Ion channel
Etidocaine Hydrochloride (W19053) 是一种长效麻醉剂和电压门控钠通道阻滞剂。
T12315 OR-1896

PDE Metabolism
OR-1896 is an active long-lived Levosimendan metabolite, is a highly selective inhibitor of phosphodiesterase (PDE) III isoformand a powerful vasodilator.
T0364L Dibucaine hydrochloride

Cinchocaine HCl,Dibucaine HCl,盐酸地布卡因,Cinchocaine hydrochloride

Sodium Channel; AChR Membrane transporter/Ion channel; Neuroscience
Dibucaine hydrochloride (Cinchocaine hydrochloride) 是钠通道抑制剂和有效的 SChE 抑制剂。
T0749 Succinylsulfathiazole

琥珀酰磺胺噻唑,Succinylsulphathiazole

Antibacterial; Antibiotic; Autophagy Autophagy; Microbiology/Virology
Succinylsulfathiazole (Succinylsulphathiazole) 是一种超长效磺胺类药物。
T6876 Liraglutide

利拉鲁肽,Liraglutidum,利拉糖肽,Victoza,Liraglutida,NN2211

Glucagon Receptor GPCR/G Protein
Liraglutide (Liraglutida) 是胰高血糖素样肽-1 受体激动剂,用于 2 型糖尿病的研究。
T28360 PF-00489791

PF-4634817,PF 4634817,PF00489791,PF 00489791,PF4634817

PDE Metabolism
PF-00489791 (PF4634817) 是一种长效 PDE5 抑制剂,具有降血压活性,可用于研究糖尿病肾病。
T11235 Estradiol 3-sulfamate

雌二醇 3-氨基磺酸,ES-J 995,E2MATE,BLE 00084

Others Others
.Estradiol 3-sulfamate inhibits estrone sulfatase with an IC50 of 251 nM and a Ki of 133 nM. Estradiol 3-sulfamate is a potent, long-acting, and orally active steroid sulfatase inhibitor.
T4499 Mequitazine

Metaplexan,Virginan,Primalan,LM-209,美喹他嗪

Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Mequitazine (Virginan) 是一种有效的、非镇静剂和长效组胺 H1 拮抗剂。
T1239 Indacaterol maleate

马来酸茚达特罗,QAB149

Adrenergic Receptor GPCR/G Protein; Neuroscience
Indacaterol maleate (QAB149) 是一种超长效的 β-肾上腺素受体激动剂。
T2431 ID-8

ID8

DYRK Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors
ID-8 是 DYRK 抑制剂,长时间培养能够维持胚胎干细胞的自我更新。
T33386 Milveterol HCl

Milveterol,GSK-159797,GSK 159797,GSK159797

Adrenergic Receptor GPCR/G Protein; Neuroscience
Milveterol HCl 是一种长效β(2)-肾上腺素能受体激动剂,可用于治疗慢性阻塞性肺病(COPD)。
T1629 Rifapentine

MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin

DNA/RNA Synthesis; Antibacterial; Antibiotic Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Rifapentine (Rifapentinum) 是可用于肺结核的抗生素。
T20435L Leuphasyl TFA

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Leuphasyl TFA 是一种酰胺肽,一种 δ-阿片受体激动剂,是一种抗降解的长效 Leu-脑啡肽类似物,用于研究 δ 阿片受体的信号通路。 它 是一种有效的长效 Leu-脑啡肽类似物,可抵抗酶促降解。
T0127 Glimepiride

Glimperide,HOE-490,格列美脲

Potassium Channel Membrane transporter/Ion channel
Glimepiride (HOE-490) 是一种中长效的磺酰脲类抗糖尿病化合物,其 ED50=182 μg/k。

化合物

Sulfo-NHS-LC-Biotin
Cat.No: T34744
Synonym: long chain Sulfo NHS Biotin
Target:
Isopropamide Iodide
Cat.No: T5051
Synonym:
Target: AChR
SulfadiMethoxine sodium
Cat.No: T8133
Synonym:
Target: Anti-infection, Antibacterial, Antibiotic
Neticonazole Hydrochloride
Cat.No: T4985
Synonym:
Target: Antifungal
KCNQ1 activator-1 
Cat.No: T9778
Synonym:
Target: Potassium Channel
Sulfadimethoxine
Cat.No: T1078
Synonym: Sulphadimethoxine,磺胺二甲氧嗪
Target: Antibacterial, Antibiotic
MR-L2
Cat.No: T12103
Synonym:
Target: PDE
Cilnidipine
Cat.No: T0388
Synonym: FRC-8653,西尼地平
Target: Calcium Channel
Alacepril
Cat.No: T7808
Synonym: Cetapril,阿拉普利,DU-1219
Target: RAAS
TTK21
Cat.No: T8778
Synonym:
Target: Epigenetic Reader Domain
Rezafungin
Cat.No: T12732
Synonym: 棘白菌素,SP-3025,CD101,Biafungin
Target: Others, Antifungal
Fluphenazine decanoate
Cat.No: T7943
Synonym:
Target: Dopamine Receptor
Rolapitant
Cat.No: T3716
Synonym: 罗拉吡坦,SCH619734,罗拉匹坦
Target: Neurokinin receptor
Ibutilide Fumarate
Cat.No: T6541
Synonym: Corvert Fumarate,U70226E,富马酸伊布利特
Target: Calcium Channel, Sodium Channel
Dihomo-γ-Linolenic acid methyl ester
Cat.No: T41323
Synonym:
Target: Others
ELOVL1-IN-1
Cat.No: T9578
Synonym: 1-(2-Fluorophenyl)-N-(1-(2-fluoropyridin-4-YL)-1H-pyrazol-3-YL)cyclopropane-1-carboxamide
Target: Others
Olodaterol hydrochloride
Cat.No: T5159
Synonym: BI-1744 HCl,盐酸奥达特罗,BI 1744 hydrochloride
Target: Adrenergic Receptor
Norethisterone enanthate
Cat.No: T20720
Synonym: NSC 9564,Norethindrone enanthate,LG-202,LG202,NSC9564,LG 202,炔诺酮庚酸酯,NSC-9564
Target: Estrogen/progestogen Receptor
Cevimeline hydrochloride hemihydrate
Cat.No: T2390
Synonym:
Target: AChR
Longdaysin
Cat.No: T5358
Synonym:
Target: ERK, Casein Kinase, CDK
eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species](TFA)
Cat.No: T22774L
Synonym:
Target: Others
Longilactone, delta-4(18)-Isomer, 2alpha-alcoho
Cat.No: T125797
Synonym:
Target:
Longicin
Cat.No: T32862
Synonym:
Target:
Longicoricin
Cat.No: T32863
Synonym:
Target:
Elongation factor P-IN-2
Cat.No: T60682
Synonym:
Target:
Isocalolongic acid
Cat.No: T124889
Synonym:
Target:
Huanglongmycin N
Cat.No: T72727
Synonym:
Target:
Malonganenone A
Cat.No: T24429
Synonym: Malonganenone-A,Malonganenone-E,Malonganenone E
Target:
Longicaulenone
Cat.No: T130680
Synonym:
Target:
(-)-Isolongifolol
Cat.No: T126352
Synonym:
Target:
Virolongin B
Cat.No: T124874
Synonym:
Target:
8,10-Dihydroxy-3-longipinen-5-one, diangeloyl
Cat.No: T130156
Synonym:
Target:
Elongation factor P-IN-1
Cat.No: T60491
Synonym:
Target:
Longilactone
Cat.No: T126080
Synonym:
Target:
Longanlactone
Cat.No: T32859
Synonym:
Target:
eukaryotic translation elongation factor 1 alpha 1 (EEF1A1) (387-394) [Multiple species]
Cat.No: T22774
Synonym:
Target: Others
Etidocaine Hydrochloride
Cat.No: T31716
Synonym: W-19053,Duranest,W19053,W 19053
Target: Sodium Channel
OR-1896
Cat.No: T12315
Synonym:
Target: PDE
Dibucaine hydrochloride
Cat.No: T0364L
Synonym: Cinchocaine HCl,Dibucaine HCl,盐酸地布卡因,Cinchocaine hydrochloride
Target: Sodium Channel, AChR
Succinylsulfathiazole
Cat.No: T0749
Synonym: 琥珀酰磺胺噻唑,Succinylsulphathiazole
Target: Antibacterial, Antibiotic, Autophagy
Liraglutide
Cat.No: T6876
Synonym: 利拉鲁肽,Liraglutidum,利拉糖肽,Victoza,Liraglutida,NN2211
Target: Glucagon Receptor
PF-00489791
Cat.No: T28360
Synonym: PF-4634817,PF 4634817,PF00489791,PF 00489791,PF4634817
Target: PDE
Estradiol 3-sulfamate
Cat.No: T11235
Synonym: 雌二醇 3-氨基磺酸,ES-J 995,E2MATE,BLE 00084
Target: Others
Mequitazine
Cat.No: T4499
Synonym: Metaplexan,Virginan,Primalan,LM-209,美喹他嗪
Target: Histamine Receptor
Indacaterol maleate
Cat.No: T1239
Synonym: 马来酸茚达特罗,QAB149
Target: Adrenergic Receptor
ID-8
Cat.No: T2431
Synonym: ID8
Target: DYRK
Milveterol HCl
Cat.No: T33386
Synonym: Milveterol,GSK-159797,GSK 159797,GSK159797
Target: Adrenergic Receptor
Rifapentine
Cat.No: T1629
Synonym: MDL473,Rifapentina,Rifapentinum,DL 473,利福喷丁,Priftin,Cyclopentylrifampicin
Target: DNA/RNA Synthesis, Antibacterial, Antibiotic
Leuphasyl TFA
Cat.No: T20435L
Synonym:
Target: Opioid Receptor
Glimepiride
Cat.No: T0127
Synonym: Glimperide,HOE-490,格列美脲
Target: Potassium Channel
Cat. No. Product Name Target Signaling Pathways
T12287 Octadecanedioic acid

Endogenous Metabolite Metabolism
Octadecanedioic acid 是内源性代谢物的一种,是一种长链二羧酸,曾在雷氏综合征的血清游离脂肪酸中被发现。
T5567 Tetradecanedioic acid

十四烷二酸,Tetradecanedicarboxylate

Others; Endogenous Metabolite Metabolism; Others
Tetradecanedioic acid (Tetradecanedicarboxylate) 是一种长链脂肪酸,属于内源性代谢物的一种。它能够作为有机阴离子转运多肽介导的药物-药物相互作用的候选生物标志物。
T5368 Eicosapentaenoic Acid

Histone Demethylase; Others; Endogenous Metabolite Chromatin/Epigenetic; Metabolism; Others
Eicosapentaenoic Acid 是一种 ω-3 脂肪酸。
T6947 Piperlongumine

PPLGM,荜茇酰胺,Piplartine

Apoptosis; ERK; Ferroptosis; Reactive Oxygen Species; ROS; Antibacterial; Autophagy Apoptosis; Autophagy; Immunology/Inflammation; MAPK; Metabolism; Microbiology/Virology; NF-κB
Piperlongumine (Piplartine) 是一种来自 Piper longum L. 的天然生物碱,具有抗炎、抗菌、抗血管生成、抗氧化、抗肿瘤和抗糖尿病等活性。它选择性地杀死癌细胞并增强活性氧的水平。它具有抗心肌纤维化的作用,通过抑制 ERK1/2 信号通路抑制肌成纤维细胞的转化。
TN6110 4,5-Dihydropiperlonguminine

二氢荜茇明宁碱,Dihydropiperlonguminine

Parasite Microbiology/Virology
4,5-Dihydropiperlonguminine (Dihydropiperlonguminine) 是一种从 Piper tuberculatum Jacq 的种子中分离出来的小分子化合物,具有杀虫和潜在的镇痛活性。
TN7157 (+/-)-Longamide

Pyrrolo[1,2-a]pyrazin-1(2H)-one, 6,7-dibromo-3,4-dihydro-4-hydroxy-,6,7-dibromo-4-hydroxy-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-1-one,6,7-dibromo-4-hydroxy-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-one

Others Others
(+/-)-Longamide (6,7-dibromo-4-hydroxy-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-one) 是一种海洋来源的天然产物,存在于Agelas flabelliformis。
T11685 Isolongifolene

异长叶烯,(-)-Isolongifolene

Apoptosis; Others Apoptosis; Others
Isolongifolene ((-)-Isolongifolene) 是一种从调料九里香中分离的三环倍半萜烯,具有抗氧化,抗炎,抗癌和神经保护的特性。它通过调节 PI3K/AKT/GSK-3β 信号通路来减轻鱼藤酮诱导的氧化应激,线粒体功能障碍和细胞凋亡。
TN2085 Piperlonguminine

Anti-infection; Antibacterial; Antifungal Microbiology/Virology
Piperlonguminine 是一种从 Piper 中分离出的生物碱酰胺。它具有多种生物活性,如神经保护、抗炎、抗肿瘤、抗血小板、抗黑素生成、抗真菌和抗菌活性。
T8110 (+)-Longifolene

Endogenous Metabolite Metabolism
(+)-Longifolen 是倍半萜类化合物。它也是家兔体内的代谢物,兔子体内转化为伯醇、仲醇或叔醇,其中以伯醇为主。
TN4591 Murralongin

Others Others
Murralongin exhibits cytotoxicity against cholangiocarcinoma cell line, KKU-100.
TN1223 23-Hydroxylongispinogenin

(3BETA,4ALPHA,16BETA)-齐墩果-12-烯-3,16,23,28-四醇,23-羟基龙吉苷元

Others Others
23-Hydroxylongispinogenin is a natural product
T32864 Longispinogenin

Longispinogenin is a triterpenetriol fatty acid ester isolated from Trichocereus chilensis.
TN4447 Longifloroside A

Others Others
Longifloroside A is a natural product from Ligustrum lucidum.
T75700 Longistyline A

Longistyline A (Longistylin A) 是一种天然二苯乙烯,可从木豆中提取。Longistyline A 对耐甲氧西林金黄色葡萄球菌具有抑菌效应,MIC 值为 1.56 μg/mL。Longistyline A 具有神经保护作用,可用于感染和神经系统疾病的研究。
TN4450 Longistylumphylline A

Others Others
Longistylumphylline A是一种天然产物,属于交让木科虎皮楠属,其产品编号为 TN4450,CAS号为 857672-34-5。Longistylumphylline A可用作对照参考。
TN4446 Longiferone B

NOS; COX Immunology/Inflammation; Neuroscience
Longiferone B shows anti-inflammatory activity against NO release with IC50 values of 21.0 uM, it also suppresses the iNOS and COX-2 mRNA expression.
T32861 Longicautadine

NSC377102,NSC 377102,NSC-377102

Longicautadine is an alkaloid isolated from stembark of Strychnos chrysophylla.
TN4449 Longistylin C

Antifection Microbiology/Virology
Longistylin A and longistylin C show some cytotoxic effects, with IC(50) values of 0.7-14.7 microM against the range of cancer cell lines. Longistylin A and longistylin C, and betulinic acid show a moderately high in vitro activity against the chloroquine
TN3767 Daphnilongeranin C

Others Others
Daphnilongeranin C是一种天然产物,属于交让木科虎皮楠属,其产品编号为 TN3767,CAS号为 750649-07-1。Daphnilongeranin C可用作对照参考。
TN3768 Daphnilongeridine

Others Others
Daphnilongeridine shows cytotoxicity against several tumor cell lines.
T32860 Longiborneol

Longiborneol is a sesquiterpene alcohol.
TN4982 Secolongifolenediol

Others Others
Secolongifolenediol 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN4982,CAS号为 53587-37-4。
TN3766 Daphnilongeranin A

Others Others
Daphnilongeranin A is a natural product from Cimicifuga foetida L.
TN4313 Isomurralonginol acetate

Others Others
Isomurralonginol acetate是一种天然产物,属于芸香科九里香属,其产品编号为 TN4313,CAS号为 139115-59-6。Isomurralonginol acetate可用作对照参考。
TN4448 Longipedlactone J

Others Others
Longipedlactone J是一种天然产物,属于五味子科南五味子属,其产品编号为 TN4448,CAS号为 1011762-93-8。Longipedlactone J可用作对照参考。
TN2001 Oblongine

Others Others
Oblongine chloride may have potential haemodynamic effects, it can cause a dose-dependent reduction of systolic and diastolic blood pressure, and that these effects are not mediated by α²-adrenergic receptor stimulation.
T17048 Tetradecanoylcarnitine

L-Myristoylcarnitine,Myristoyl-L-(-)-carnitine

Endogenous Metabolite Metabolism
Tetradecanoylcarnitine (L-Myristoylcarnitine) 是一种酰基肉碱,参与长链脂肪酸的β-氧化,是极长链酰辅酶A脱氢酶缺乏症的一种潜在标记物。
T8111 Triacontanoic Acid

蜂花酸,Melissic acid A

Others Others
Triacontanoic Acid (Melissic acid A) 是一种超长链脂肪酸。
T40637 Gondoic acid

cis-11-Eicosenoicacid,顺-11-二十碳烯酸

Others Others
Gondoic acid (cis-11-Eicosenoicacid) (cis-11-Eicosenoic acid) is a monounsaturated long-chain fatty acid that can be found in various plant oils and nuts [1].
T8271 10Z-Nonadecenoic acid

Endogenous Metabolite Metabolism
10Z-Nonadecenoic acid 是一种长链脂肪酸,具有抗肿瘤特性。
T8285 Methyl tricosanoate

Others Others
Methyl tricosanoate 是一种长链脂肪酸化合物,存在于各种抗微生物剂和抗菌剂中。
T8192 Pentacosanoic acid

Others; Endogenous Metabolite Metabolism; Others
Pentacosanoic acid 是戊酸的共轭酸,是 25 碳长链饱和脂肪酸。
T8070 Nonadecanoic acid

Others Others
Nonadecanoic acid 是19 C 长的饱和脂肪酸,是白蚁防御时分泌的主要物质。
T5942 Docosanoic acid

Behenic Acid,山嵛酸

DNA/RNA Synthesis; Endogenous Metabolite Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Metabolism
Docosanoic acid (Behenic Acid) 是一种较难吸收的饱和脂肪酸,能提高人类胆固醇水平。
T7095 Hexacosanoic acid

二十六酸,Cerotic acid

Endogenous Metabolite Metabolism
Hexacosanoic acid 是长链脂肪酸,与多种疾病有关(如肾上腺脑白质营养不良,肾上腺髓鞘病和动脉粥样硬化)。
T4903 Heptadecanoic acid

Others; Endogenous Metabolite Metabolism; Others
Heptadecanoic acid 是奇链饱和脂肪酸,与一些疾病(如冠心病、糖尿病前期和 2 型糖尿病以及多发性硬化症)有关。
T0086 Galanthamine hydrobromide

Galantamine hydrobromide,Galanthamine HBr,氢溴酸加兰他敏

AChR; AChE Neuroscience
Galanthamine hydrobromide (Galantamine hydrobromide) 是一种长效的中枢活性 AChE 抑制剂,IC50为 410 nM。它是神经元烟碱型 ACh 受体的变构增强剂,IC50值为 0.35 µM,可用于阿尔茨海默症的研究。
T4944 Nervonic acid

cis-15-Tetracosenoic acid,神经酸,Selacholeic acid

Endogenous Metabolite Metabolism
Nervonic acid (Selacholeic acid) 是在髓磷脂生物合成中很重要的单不饱和脂肪酸。
T6S2115 Ginkgolide J

BN 52024,7-beta-Hydroxyginkgolide A,银杏内酯 J,银杏内酯J

PDE Metabolism
Ginkgolide J (BN 52024) 是一种银杏叶中非黄酮部分的主要成分(IC50:12-54 µM),具有神经保护和抗神经元凋亡功能。
T14011 2-Arachidonoylglycerol

Cannabinoid Receptor; Endogenous Metabolite GPCR/G Protein; Metabolism
2-Arachidonoylglycerol 属于人内源性代谢物,是中枢神经系统中的一种内源性大麻素配体。
T8011 1,2-dioleoyl-sn-glycero-3-phosphocholine

二油酰磷脂酰胆碱,DOPC

Others Others
1,2-dioleoyl-sn-glycero-3-phosphocholine (DOPC) 是磷脂的一种,在胶束,脂质体和其他类型的人工膜的生成中通常单独使用或与其他组分一起使用。
TN2285 DL-Tryptophan

(±)-Tryptophan,Tryptophan,DL-色氨酸

Serotonin Transporter; Endogenous Metabolite Metabolism; Neuroscience
DL-Tryptophan ((±)-Tryptophan) 是内源性代谢产物的一种。
T9299 D-Leucine

D-亮氨酸,(R)-Leucine

Endogenous Metabolite Metabolism
D-Leucine ((R)-Leucine) 具有抗癫痫特性,活性比L-leucine,能够有效终止癫痫发作。在体外,它能够抑制长期点位,但基底突触传递无影响。
T1261 Medroxyprogesterone Acetate

Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)

Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; Androgen Receptor; Endogenous Metabolite Endocrinology/Hormones; Metabolism; Others
Medroxyprogesterone Acetate (Farlutin) 是广泛使用的合成类固醇,与雄激素,孕酮及糖皮质激素受体均有作用。
T4867 Erucic acid

Prifac 2990,芥酸,13(Z)-Docosenoic Acid,cis-13-docosenoic acid

PI3K; Endogenous Metabolite Metabolism; PI3K/Akt/mTOR signaling
Erucic acid (13(Z)-Docosenoic Acid) 是单不饱和脂肪酸,分离自萝卜的种子。Erucic acid 可以容易地穿过血脑屏障,使大脑中长链脂肪酸的积累正常化。Erucic acid 能够改善认知障碍并有效预防痴呆。
T3S2007 MRE-269

3-氧代-12-烯-28-乌苏酸,MRE 269,ACT-333679,MRE269

Prostaglandin Receptor GPCR/G Protein; Immunology/Inflammation
MRE-269 (ACT-333679) 是一种口服的长效前列环素受体激动剂前药,是 Selexipag 的活性代谢物,用于治疗肺动脉高压。
TN1433 Batatasin III

FAK; Others; Akt Angiogenesis; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Batatasin III 通过抑制上皮间质转化和 FAK-AKT 信号来抑制癌症迁移和侵袭,并具有抗癌活性。 Batatasin III 对整株生长有长期抑制作用,显示出抑制萌发活性。
T9143 D-Isoleucine

(2R,3R)-2-Amino-3-methylpentanoic acid,D-异亮氨酸,(R)-Isoleucine

Others Others
D-Isoleucine ((2R,3R)-2-Amino-3-methylpentanoic acid) 是一种异亮氨酸立体异构体,是 Asc-1 反转运蛋白的选择性激活剂。它能够释放内源性 D-丝氨酸,提高海马 CA1-CA3 的长期增效作用。
T3674 Hydroxysafflor yellow A

藏红花,羟基红花黄色素A,HSYA,Safflomin A

TGF-beta/Smad Stem Cells
Hydroxysafflor yellow A (Safflomin A) 是一种黄酮类天然产物,从中药红花中分离得到,具有抗癌作用。
T0012 Cinchonine

LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁

Apoptosis; P-gp; Parasite Apoptosis; Membrane transporter/Ion channel; Microbiology/Virology; Neuroscience
Cinchonine (LA40221) 是金鸡纳树皮中的一种天然产物。它可激活内质网应激诱导的人肝癌细胞凋亡。它是一种酰胺类局部麻醉剂。
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天然产物

Octadecanedioic acid
Cat.No: T12287
Synonym:
Target: Endogenous Metabolite
Tetradecanedioic acid
Cat.No: T5567
Synonym: 十四烷二酸,Tetradecanedicarboxylate
Target: Others, Endogenous Metabolite
Eicosapentaenoic Acid
Cat.No: T5368
Synonym:
Target: Histone Demethylase, Others, Endogenous Metabolite
Piperlongumine
Cat.No: T6947
Synonym: PPLGM,荜茇酰胺,Piplartine
Target: Apoptosis, ERK, Ferroptosis, Reactive Oxygen Species, ROS, Antibacterial, Autophagy
4,5-Dihydropiperlonguminine
Cat.No: TN6110
Synonym: 二氢荜茇明宁碱,Dihydropiperlonguminine
Target: Parasite
(+/-)-Longamide
Cat.No: TN7157
Synonym: Pyrrolo[1,2-a]pyrazin-1(2H)-one, 6,7-dibromo-3,4-dihydro-4-hydroxy-,6,7-dibromo-4-hydroxy-3,4-dihydro-2H-pyrrolo[1,2-a]pyrazin-1-one,6,7-dibromo-4-hydroxy-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-one
Target: Others
Isolongifolene
Cat.No: T11685
Synonym: 异长叶烯,(-)-Isolongifolene
Target: Apoptosis, Others
Piperlonguminine
Cat.No: TN2085
Synonym:
Target: Anti-infection, Antibacterial, Antifungal
(+)-Longifolene
Cat.No: T8110
Synonym:
Target: Endogenous Metabolite
Murralongin
Cat.No: TN4591
Synonym:
Target: Others
23-Hydroxylongispinogenin
Cat.No: TN1223
Synonym: (3BETA,4ALPHA,16BETA)-齐墩果-12-烯-3,16,23,28-四醇,23-羟基龙吉苷元
Target: Others
Longispinogenin
Cat.No: T32864
Synonym:
Target:
Longifloroside A
Cat.No: TN4447
Synonym:
Target: Others
Longistyline A
Cat.No: T75700
Synonym:
Target:
Longistylumphylline A
Cat.No: TN4450
Synonym:
Target: Others
Longiferone B
Cat.No: TN4446
Synonym:
Target: NOS, COX
Longicautadine
Cat.No: T32861
Synonym: NSC377102,NSC 377102,NSC-377102
Target:
Longistylin C
Cat.No: TN4449
Synonym:
Target: Antifection
Daphnilongeranin C
Cat.No: TN3767
Synonym:
Target: Others
Daphnilongeridine
Cat.No: TN3768
Synonym:
Target: Others
Longiborneol
Cat.No: T32860
Synonym:
Target:
Secolongifolenediol
Cat.No: TN4982
Synonym:
Target: Others
Daphnilongeranin A
Cat.No: TN3766
Synonym:
Target: Others
Isomurralonginol acetate
Cat.No: TN4313
Synonym:
Target: Others
Longipedlactone J
Cat.No: TN4448
Synonym:
Target: Others
Oblongine
Cat.No: TN2001
Synonym:
Target: Others
Tetradecanoylcarnitine
Cat.No: T17048
Synonym: L-Myristoylcarnitine,Myristoyl-L-(-)-carnitine
Target: Endogenous Metabolite
Triacontanoic Acid
Cat.No: T8111
Synonym: 蜂花酸,Melissic acid A
Target: Others
Gondoic acid
Cat.No: T40637
Synonym: cis-11-Eicosenoicacid,顺-11-二十碳烯酸
Target: Others
10Z-Nonadecenoic acid
Cat.No: T8271
Synonym:
Target: Endogenous Metabolite
Methyl tricosanoate
Cat.No: T8285
Synonym:
Target: Others
Pentacosanoic acid
Cat.No: T8192
Synonym:
Target: Others, Endogenous Metabolite
Nonadecanoic acid
Cat.No: T8070
Synonym:
Target: Others
Docosanoic acid
Cat.No: T5942
Synonym: Behenic Acid,山嵛酸
Target: DNA/RNA Synthesis, Endogenous Metabolite
Hexacosanoic acid
Cat.No: T7095
Synonym: 二十六酸,Cerotic acid
Target: Endogenous Metabolite
Heptadecanoic acid
Cat.No: T4903
Synonym:
Target: Others, Endogenous Metabolite
Galanthamine hydrobromide
Cat.No: T0086
Synonym: Galantamine hydrobromide,Galanthamine HBr,氢溴酸加兰他敏
Target: AChR, AChE
Nervonic acid
Cat.No: T4944
Synonym: cis-15-Tetracosenoic acid,神经酸,Selacholeic acid
Target: Endogenous Metabolite
Ginkgolide J
Cat.No: T6S2115
Synonym: BN 52024,7-beta-Hydroxyginkgolide A,银杏内酯 J,银杏内酯J
Target: PDE
2-Arachidonoylglycerol
Cat.No: T14011
Synonym:
Target: Cannabinoid Receptor, Endogenous Metabolite
1,2-dioleoyl-sn-glycero-3-phosphocholine
Cat.No: T8011
Synonym: 二油酰磷脂酰胆碱,DOPC
Target: Others
DL-Tryptophan
Cat.No: TN2285
Synonym: (±)-Tryptophan,Tryptophan,DL-色氨酸
Target: Serotonin Transporter, Endogenous Metabolite
D-Leucine
Cat.No: T9299
Synonym: D-亮氨酸,(R)-Leucine
Target: Endogenous Metabolite
Medroxyprogesterone Acetate
Cat.No: T1261
Synonym: Medroxyprogesterone 17-acetate,Provera,Metigestrona,NSC-26386,醋酸甲羟孕酮,Farlutin,安宫黄体酮,Medroxyprogesterone (acetate)
Target: Glucocorticoid Receptor, Estrogen/progestogen Receptor, Progesterone Receptor, Androgen Receptor, Endogenous Metabolite
Erucic acid
Cat.No: T4867
Synonym: Prifac 2990,芥酸,13(Z)-Docosenoic Acid,cis-13-docosenoic acid
Target: PI3K, Endogenous Metabolite
MRE-269
Cat.No: T3S2007
Synonym: 3-氧代-12-烯-28-乌苏酸,MRE 269,ACT-333679,MRE269
Target: Prostaglandin Receptor
Batatasin III
Cat.No: TN1433
Synonym:
Target: FAK, Others, Akt
D-Isoleucine
Cat.No: T9143
Synonym: (2R,3R)-2-Amino-3-methylpentanoic acid,D-异亮氨酸,(R)-Isoleucine
Target: Others
Hydroxysafflor yellow A
Cat.No: T3674
Synonym: 藏红花,羟基红花黄色素A,HSYA,Safflomin A
Target: TGF-beta/Smad
Cinchonine
Cat.No: T0012
Synonym: LA40221,(8R,9S)-Cinchonine,奎宁树,辛可宁
Target: Apoptosis, P-gp, Parasite
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