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108

抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T10480 Bay 41-4109 (less active enantiomer)

HBV Microbiology/Virology
Bay 41-4109 less active enantiomer shows less activity than Bay 41-4109. BAY 41-4109 is a potent HBV inhibitor (IC50: 53 nM).
T6352 (-)-Dizocilpine maleate

C13737,(-)-MK 801 (Maleate),(-)-MK 801马来酸,(-)-MK 801 Maleate

NMDAR; iGluR Membrane transporter/Ion channel; Neuroscience
(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) 是一种选择性且非竞争性的 N-甲基-D-天冬氨酸 (NMDA) 受体拮抗剂,Ki 为 211.7 nM。它是一种 Dizocilpine 的活性较低的 (-)-对映体,具有抗抑郁作用。
T12814 (S)-Tenofovir

(S)-替诺福韦,(S)-PMPA,(S)-GS 1278,(S)-TDF

Others Others
(S)-Tenofovir ((S)-PMPA) 是Tenofovir 的活性较低的S-对映体,Tenofovir 是一种核苷酸逆转录酶抑制剂。
T12664 (Rac)-BRD0705

Others Others
(Rac)-BRD0705 是 BRD0705 的活性较低的外消旋体。 BRD0705 是一种有效的特异性 GSK3α 抑制剂。
T12831 SAR405 R enantiomer

Others Others
SAR405 R enantiomer 是一种 PIK3C3/Vps34 抑制剂,也是活性低于 SAR405 的对映体。
T68051L RS 15385-198

Adrenergic Receptor GPCR/G Protein; Neuroscience
RS 15385-198 是 Delequamine 的低活性异构体。Delequamine 是一种选择性 α2-肾上腺素受体拮抗剂。
T10376 ARS-1630

Ras GPCR/G Protein; MAPK
ARS-1630 是一种突变型 K-ras G12C 抑制剂。 它是 ARS-1620 的活性较低的对映异构体。
T7080 CCT245737

SRA737

Chk Cell Cycle/Checkpoint
CCT245737 (SRA737) 是一种具有口服活性的选择性 Chk1 抑制剂,IC50值为 1.3 nM。
T9554 SN-008

STING Immunology/Inflammation
SN-008 是 SN-011 的低活性类似物,可作为阴性对照。
T11129L Duvelisib (R enantiomer) hydrochloride

IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl

PI3K PI3K/Akt/mTOR signaling
Duvelisib (R enantiomer) hydrochloride (INK1197 R enantiomer HCl) 是 PI3K 抑制剂。Duvelisib (R enantiomer) hydrochloride 是 Duvelisib 的活性较低的对映体。
T22450 Tyrphostin B44, (+) enantiomer

酪氨酸磷酸化抑制剂AG 835

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Tyrphostin B44, (+) enantiomer 是一种表皮生长因子受体 (EGFR) 激酶抑制剂,IC50 为 0.86 μM,活性低于 (-) 对映体。
T6205 AT7519

Apoptosis; GSK-3; CDK Apoptosis; Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Stem Cells
AT7519 是一种CDK 抑制剂,对 CDK1,CDK2,CDK4-CDK6 以及 CDK9 的IC50值分别为 210,47,100,13,170 和 <10 nM。
T22818 GSK9027

GR agonist 23a,GSK 9027,GSK-9027

Glucocorticoid Receptor Endocrinology/Hormones
GSK9027 (GR agonist 23a) 是一种非甾体糖皮质激素受体 (GR) 激动剂。GSK9027 (GR agonist 23a) 在2×GRE报告基因上对比地塞米松的活性属于部分激动剂,活性较地塞米松活性较弱。
T9042 Teriflunomide impurity 3

4-Amino-N-(4-trifluoromethylphenyl)benzamide

COX Immunology/Inflammation; Neuroscience
Teriflunomide impurity 3 (4-Amino-N-(4-trifluoromethylphenyl)benzamide) 是一种选择性COX-1抑制剂,IC50为 30 µM。
T16759 Ritanserin

利坦丝林,R 55667

Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; Histamine Receptor GPCR/G Protein; Immunology/Inflammation; Neuroscience
Ritanserin (R 55667) 是一种长效、高效、相对选择性、可口服的5-HT2受体拮抗剂,IC50值为 0.9 nM。
T67905 GS-829845

JAK; Drug Metabolite Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Metabolism; Stem Cells
GS-829845 是一种 JAK1 抑制剂,是 Filgotinib 活性代谢物的主要成分,其效力比母体低约 10 倍且半衰期更长。
T12146 N-Desmethyl-Apalutamide

N-Desmethyl Apalutamide,N-去甲基阿帕鲁胺杂质

P450; Androgen Receptor Endocrinology/Hormones; Metabolism
N-Desmethyl-Apalutamide 是一种 Apalutamide 的活性代谢产物,主要由 CYP2C8 和 CYP3A4 介导形成。它是一种低活性的雄激素受体拮抗剂,其作用力是 Apalutamide 活性的三分之一。它是中等至强的CYP3A4和CYP2B6诱导剂,并具有优异的血浆蛋白结合浓度。
T6104 Cerdulatinib hydrochloride

Cerdulatinib,PRT2070,PRT062070 hydrochloride,PRT062070,PRT2070 hydrochloride

MLK; c-Fms; Tyrosine Kinases; Hippo pathway; JAK; Syk Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; MAPK; Stem Cells; Tyrosine Kinase/Adaptors
Cerdulatinib hydrochloride (PRT2070 hydrochloride) 是一种选择性可逆,具有口服活性、 ATP 竞争性的 SYK 和 JAK 的双重抑制剂,抑制 JAK1、2、3、SYK 和 Tyk2的 IC50值分别为12、6、8、32 和 0.5 nM。它可用于研究自身免疫性疾病和B 细胞恶性肿瘤。
T15545 ICA-27243

Potassium Channel Membrane transporter/Ion channel
ICA-27243 是选择性的,口服有效的 KCNQ2/Q3钾通道开放剂,EC50为 0.38 μM。对 KCNQ4 和 KCNQ3/Q5 的激活效果较差。它具有抗惊厥和抗癫痫作用。
T12695 RBN-2397

PARP Chromatin/Epigenetic; DNA Damage/DNA Repair
RBN-2397 是一种有效的、选择性的、具有口服活性的跨物种 NAD+ 竞争性 PARP7 抑制剂,IC50 小于 3 nM。它选择性结合 PARP7 ,Kd 为0.001 μM,可恢复干扰素 I 型信号转导,有用于晚期或转移性实体肿瘤的研究潜力。
T21938 AS-041164

PI3K PI3K/Akt/mTOR signaling
AS-041164 是选择性的,具有口服活性的PI3Kγ亚型抑制剂,IC50=70 nM。它对 PI3Kα (IC50:240 μM),PI3Kβ (IC50:1.45 μM) 和 PI3Kδ (IC50:1.70 μM) 的活性较低。它具有抗炎活性。
T4481 Tucidinostat

HBI-8000,Chidamide,西达本胺,CS 055

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
Tucidinostat (Chidamide) 是一种可口服的 HDAC I 类 HDAC1/2/3和第 IIb 类 HDAC10的抑制剂,IC50值分别为 95、160、67 和 78 nM。
T6458 CYC-116

噻氯匹定

VEGFR; FLT; CDK; S6 Kinase; Aurora Kinase Angiogenesis; Cell Cycle/Checkpoint; Chromatin/Epigenetic; MAPK; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
CYC116是一种有效的极光激酶 A 和 B 的抑制剂,Ki 值分别为8和9 nM。
T13140 Umbralisib R-enantiomer

TGR-1202 R-enantiomer,RP5264 R-enantiomer

PI3K PI3K/Akt/mTOR signaling
Umbralisib R-enantiomer (RP5264 R-enantiomer) 是 PI3K 的δ型抑制剂,是 TGR-1202 活性较低的对映体。Umbralisib R-enantiomer 对δ型 pi3激酶的 IC50,至少比抑制剂对其他 PI3K 亚型(A, β和γ)的 IC50低20倍。
T11991 Mefentrifluconazole

P450; Antifungal Metabolism; Microbiology/Virology
Mefentrifluconazole 是一种有效的、选择性的和具有口服活性的真菌 CYP51 (Kd= 0.5 nM) 抑制剂,但对人芳香酶的抑制活性较低,IC50值为0.92 μM。它是一种新型唑类衍生物,用作农用广谱抗真菌剂。
T0932 Cefixime

FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635

Antibacterial; Antibiotic Microbiology/Virology
Cefixime (FR-17027) 是一种头孢菌素类抗生素, 可研究一些细菌感染。
T20898 (R)-Propranolol hydrochloride

Dexpropranolol hydrochloride,(R)-(+)-Propranolol,盐酸普奈洛尔

Adrenergic Receptor GPCR/G Protein; Neuroscience
(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) 是一种抗肾上腺素受体拮抗剂,是一种普萘洛尔的活性较低的对映体。Dexpropranolol 是一种非选择性的β-adrenergic receptor 拮抗剂,对 β1AR 和 β2AR 具有高亲和力。
T35528L TD52 dihydrochloride

TD52 dihydrochloride(1798328-24-1 Free base),TD52 2HCl

Others Others
TD52 dihydrochloride (TD52 2HCl), a derivative of Erlotinib, is a potent and orally active inhibitor of protein phosphatase 2A (CIP2A). It exhibits strong anti-cancer properties by regulating the CIP2A/PP2A/p-Akt signaling pathway, resulting in the induction of apoptosis in triple-negative breast cancer (TNBC) cells. Mechanistically, TD52 dihydrochloride disrupts the binding of Elk1 to the CIP2A promoter, effectively reducing CIP2A levels. Notably, TD52 dihydrochloride demonstrates powerful anti...
T15199 Edicotinib

JNJ-527,JNJ-40346527

c-Fms; FLT; CSF-1R; c-Kit Angiogenesis; Tyrosine Kinase/Adaptors
Edicotinib (JNJ-527) 是能够透过血脑屏障的、口服具有活性的、选择性的CSF-1R 抑制剂 (IC50:3.2 nM)。它对 KIT (IC50:20 nM) 和 FLT3 (IC50:190 nM) 的抑制作用较小。它抑制小胶质细胞的扩张,减弱小胶质细胞的增殖和神经退行性变。它可用于研究阿尔茨海默病和类风湿性关节炎。
T6446 Clevudine

L-FMAU,克拉夫定,Levovir

HBV; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Microbiology/Virology
Clevudine (Levovir) 是一种非自然 L-构型的核苷类似物,是一种与聚合酶结合的非竞争性抑制剂,具有较强的抗 HBV 活性,半衰期长,毒性低的特点。
T60336 CCR4 antagonist 3-1

CCR Immunology/Inflammation; Microbiology/Virology
CCR4 antagonist 3-1 是一种具有较低活性的趋化因子受体 4 (CCR4) 拮抗剂,对 [125I]TARC (胸腺和活化调节趋化因子) 具有抑制作用,IC50 值为 1.7 μM。CCR4 antagonist 3-1 对放射标记的[125I]TARC和巨噬细胞来源的趋化因子(MDC) 与 CEM 细胞表面的CCR4 受体的结合有抑制作用, 并对 TARC 介导的 CEM 细胞的体外迁移有抑制作用,IC50 值为 6.4 μM。
T13438 (R,S)-Ivosidenib

(R,S)-AG-120

Opioid Receptor Endocrinology/Hormones; GPCR/G Protein; Neuroscience
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
T13450 (S)-GNE-140

Others Others
(S)-GNE-140 is the less active enantiomer of GNE-140.
T13426L (3S,4S)-Tofacitinib

(3S,4S)-托法替尼

Others Others
(3S,4S)-Tofacitinib, a less active enantiomer of tofacitinib, is a Janus kinases inhibitor.
T13451 (S)-Mapracorat

(S)-ZK-245186,(S)-BOL-303242X

Others Others
(S)-Mapracorat is a selective and less active agonist of glucocorticoid receptor.
T26371 (2S,3R)-LP99

(2S,3R)-LP99 is a less active enantiomer of LP99.
T11801 l-Atabrine dihydrochloride

Others Others
l-Atabrine dihydrochloride displays antiprion activity. l-Atabrine dihydrochloride is a less active enantiomer of quinacrine.
T26163 Rubradirin B

Rubradirin B has an antibacterial activity similar to rubradirin, but the antibiotic is less active.
T10564 (8R,9S)-Talazoparib

(8R,9S)-BMN-673,他拉唑帕利 (8R,9S)

Others Others
(8R,9S)-Talazoparib is Talazoparib enantiomer , less active than Talazoparib on the inhibition of PARP1 (IC50: 144 nM).
T19549 Ro18-5362

Others Others
Ro18-5362 is the less active prodrug of Ro 18-5364.
T12635 (R)-Plevitrexed

(R)-ZD 9331,(R)-BGC9331,(R)-普来曲塞

Others Others
(R)-Plevitrexed is a less active enantiomer of Plevitrexed. Plevitrexed is an orally active and potent inhibitor of thymidylate synthase (TS).
T11156 Nazartinib S-enantiomer

EGF816 (S-enantiomer)

Others Others
Nazartinib is an EGFR inhibitor. Nazartinib S-enantiomer is the less active S-enantiomer of Nazartinib.
T10856 Cobimetinib (R-enantiomer)

考比替尼 (R 型对映体),XL-518 R-enantiomer,Cobimetinib R-enantiomer,GDC-0973 R-enantiomer

Others Others
Cobimetinib R-enantiomer is the less active R-enantiomer of Cobimetinib which is a selective MEK inhibitor.
T12636 (R)-(+)-Anatabine

Others Others
(R)-(+)-Anatabine is an less active R-enantiomer of Anatabine. Anatabine is a potent agonist of α4β2 nAChR.
T6493L (R)-Citalopram oxalate

(R)-Citalopram oxalate is a less active enantiomer of Escitalopram Oxalate. Escitalopram Oxalate is a potent and selective serotonin reuptake inhibitor.
T13427 (3S,4R)-Tofacitinib

Others Others
(3S,4R)-Tofacitinib is an less active enantiomer of Tofacitinib. Tofacitinib is a JAK3 inhibitor(IC50 : 1 nM).
T13426 (3R,4S)-Tofacitinib

Others Others
(3R,4S)-Tofacitinib is an less active enantiomer of Tofacitinib. Tofacitinib is a JAK3 inhibitor(IC50 : 1 nM).
T11334 Fulvestrant (R enantiomer)

ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer

Others Others
Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T11335 Fulvestrant (S enantiomer)

ZM 182780 S enantiomer,ICI 182780 S enantiomer,Fulvestrant S enantiomer,ZD 9238 S enantiomer

Others Others
Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.
T12641 (R)-SCH 42495

Others Others
(R)-SCH 42495 is the less active enantiomer of SCH 42495. SCH 42495 is an orally active inhibitor of neutral metalloendopeptidase (NEP), with antihypertensive effect.

化合物

Bay 41-4109 (less active enantiomer)
Cat.No: T10480
Synonym:
Target: HBV
(-)-Dizocilpine maleate
Cat.No: T6352
Synonym: C13737,(-)-MK 801 (Maleate),(-)-MK 801马来酸,(-)-MK 801 Maleate
Target: NMDAR, iGluR
(S)-Tenofovir
Cat.No: T12814
Synonym: (S)-替诺福韦,(S)-PMPA,(S)-GS 1278,(S)-TDF
Target: Others
(Rac)-BRD0705
Cat.No: T12664
Synonym:
Target: Others
SAR405 R enantiomer
Cat.No: T12831
Synonym:
Target: Others
RS 15385-198
Cat.No: T68051L
Synonym:
Target: Adrenergic Receptor
ARS-1630
Cat.No: T10376
Synonym:
Target: Ras
CCT245737
Cat.No: T7080
Synonym: SRA737
Target: Chk
SN-008
Cat.No: T9554
Synonym:
Target: STING
Duvelisib (R enantiomer) hydrochloride
Cat.No: T11129L
Synonym: IPI-145 R enantiomer HCl,Duvelisib (R enantiomer) hydrochloride(1261590-48-0 Free base),INK1197 R enantiomer HCl
Target: PI3K
Tyrphostin B44, (+) enantiomer
Cat.No: T22450
Synonym: 酪氨酸磷酸化抑制剂AG 835
Target: EGFR
AT7519
Cat.No: T6205
Synonym:
Target: Apoptosis, GSK-3, CDK
GSK9027
Cat.No: T22818
Synonym: GR agonist 23a,GSK 9027,GSK-9027
Target: Glucocorticoid Receptor
Teriflunomide impurity 3
Cat.No: T9042
Synonym: 4-Amino-N-(4-trifluoromethylphenyl)benzamide
Target: COX
Ritanserin
Cat.No: T16759
Synonym: 利坦丝林,R 55667
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
GS-829845
Cat.No: T67905
Synonym:
Target: JAK, Drug Metabolite
N-Desmethyl-Apalutamide
Cat.No: T12146
Synonym: N-Desmethyl Apalutamide,N-去甲基阿帕鲁胺杂质
Target: P450, Androgen Receptor
Cerdulatinib hydrochloride
Cat.No: T6104
Synonym: Cerdulatinib,PRT2070,PRT062070 hydrochloride,PRT062070,PRT2070 hydrochloride
Target: MLK, c-Fms, Tyrosine Kinases, Hippo pathway, JAK, Syk
ICA-27243
Cat.No: T15545
Synonym:
Target: Potassium Channel
RBN-2397
Cat.No: T12695
Synonym:
Target: PARP
AS-041164
Cat.No: T21938
Synonym:
Target: PI3K
Tucidinostat
Cat.No: T4481
Synonym: HBI-8000,Chidamide,西达本胺,CS 055
Target: HDAC
CYC-116
Cat.No: T6458
Synonym: 噻氯匹定
Target: VEGFR, FLT, CDK, S6 Kinase, Aurora Kinase
Umbralisib R-enantiomer
Cat.No: T13140
Synonym: TGR-1202 R-enantiomer,RP5264 R-enantiomer
Target: PI3K
Mefentrifluconazole
Cat.No: T11991
Synonym:
Target: P450, Antifungal
Cefixime
Cat.No: T0932
Synonym: FK-027,头孢克肟,Cefspan,Cefiximum,Cephoral,FR-17027,CL-284635
Target: Antibacterial, Antibiotic
(R)-Propranolol hydrochloride
Cat.No: T20898
Synonym: Dexpropranolol hydrochloride,(R)-(+)-Propranolol,盐酸普奈洛尔
Target: Adrenergic Receptor
TD52 dihydrochloride
Cat.No: T35528L
Synonym: TD52 dihydrochloride(1798328-24-1 Free base),TD52 2HCl
Target: Others
Edicotinib
Cat.No: T15199
Synonym: JNJ-527,JNJ-40346527
Target: c-Fms, FLT, CSF-1R, c-Kit
Clevudine
Cat.No: T6446
Synonym: L-FMAU,克拉夫定,Levovir
Target: HBV, DNA/RNA Synthesis
CCR4 antagonist 3-1
Cat.No: T60336
Synonym:
Target: CCR
(R,S)-Ivosidenib
Cat.No: T13438
Synonym: (R,S)-AG-120
Target: Opioid Receptor
(S)-GNE-140
Cat.No: T13450
Synonym:
Target: Others
(3S,4S)-Tofacitinib
Cat.No: T13426L
Synonym: (3S,4S)-托法替尼
Target: Others
(S)-Mapracorat
Cat.No: T13451
Synonym: (S)-ZK-245186,(S)-BOL-303242X
Target: Others
(2S,3R)-LP99
Cat.No: T26371
Synonym:
Target:
l-Atabrine dihydrochloride
Cat.No: T11801
Synonym:
Target: Others
Rubradirin B
Cat.No: T26163
Synonym:
Target:
(8R,9S)-Talazoparib
Cat.No: T10564
Synonym: (8R,9S)-BMN-673,他拉唑帕利 (8R,9S)
Target: Others
Ro18-5362
Cat.No: T19549
Synonym:
Target: Others
(R)-Plevitrexed
Cat.No: T12635
Synonym: (R)-ZD 9331,(R)-BGC9331,(R)-普来曲塞
Target: Others
Nazartinib S-enantiomer
Cat.No: T11156
Synonym: EGF816 (S-enantiomer)
Target: Others
Cobimetinib (R-enantiomer)
Cat.No: T10856
Synonym: 考比替尼 (R 型对映体),XL-518 R-enantiomer,Cobimetinib R-enantiomer,GDC-0973 R-enantiomer
Target: Others
(R)-(+)-Anatabine
Cat.No: T12636
Synonym:
Target: Others
(R)-Citalopram oxalate
Cat.No: T6493L
Synonym:
Target:
(3S,4R)-Tofacitinib
Cat.No: T13427
Synonym:
Target: Others
(3R,4S)-Tofacitinib
Cat.No: T13426
Synonym:
Target: Others
Fulvestrant (R enantiomer)
Cat.No: T11334
Synonym: ICI 182780 R enantiomer,ZD 9238 R enantiomer,ZM 182780 R enantiomer,Fulvestrant R enantiomer
Target: Others
Fulvestrant (S enantiomer)
Cat.No: T11335
Synonym: ZM 182780 S enantiomer,ICI 182780 S enantiomer,Fulvestrant S enantiomer,ZD 9238 S enantiomer
Target: Others
(R)-SCH 42495
Cat.No: T12641
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T20191 (-)-Camphoric acid

(-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-

GluR Neuroscience
(-)-Camphoric acid (L-Camphoric acid) 是一种活性较低的樟脑酸对映异构体,樟脑酸可诱导 GluR 表达。
T13669 (E)-Cinnamamide

trans-Cinnamamide,肉桂酰胺

Others Others
(E)-Cinnamamide (trans-Cinnamamide) 是 Cinnamamide 的活性较低的异构体,Cinnamamide 是一种有效的非致命化学驱虫剂,适用于减少鸟类害虫的损害。
TN1448 (-)-Bornyl acetate

L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯

p38 MAPK; NF-κB; JNK; Antifungal MAPK; Microbiology/Virology; NF-κB
(-)-Bornyl acetate (L-(-)-Bornyl acetate) 是存在于牛膝草油中的一种具有抗真菌活性的 (+)-Bornyl acetate 低活性异构体。
T36585 Isodeoxycholic Acid

isoDCA

Chloride channel; Antibacterial Membrane transporter/Ion channel; Microbiology/Virology
Isodeoxycholic Acid 是一种胆汁酸,由肠道细菌通过脱氧胆酸的表聚作用形成。Isodeoxycholic acid 的临界胶束浓度高于二氯苯甲醚,这表明它的去污活性降低了,而且在抑制七种肠道共生细菌生长方面的活性低于二氯苯甲醚。Isodeoxycholic Acid(0.1%)能抑制几种艰难梭菌菌株在牛磺胆酸诱导下的孢子萌发,并能降低艰难梭菌培养上清对 Vero 细胞的细胞毒性。在高脂饮食诱发肥胖的大鼠模型中,血浆中的Isodeoxycholic acid 水平比正常饮食的大鼠低。
TN2931 3-Epikatonic acid

Antifection Microbiology/Virology
Epikatonic acid shows less active against T. (S.) cruzi trypanosome.
T38497 (-)-Taxifolin

(-)-二氢槲皮素,(-)-Dihydroquercetin

(-)-Taxifolin is the less active enantiomer of Taxifolin, demonstrating vital anti-tyrosinase activity and notable inhibition against collagenase (IC50 = 193.3 μM). It is valued as an essential natural compound showing antifibrotic potential, while also acting as a capable free radical scavenger and possessing antioxidant capacity.
TN4471 Lysicamine

IL Receptor; Antifection Immunology/Inflammation; Microbiology/Virology
Lysicamine shows significant antioxidant capacity in the ORAC(FL) assay and it is active against S. epidermidis and C. dubliniensis, with MIC values in the range 12.5-100 microg mL(-1). Lysicamine has antimicrobial and anti-inflammation activity, the mini

天然产物

(-)-Camphoric acid
Cat.No: T20191
Synonym: (-)-樟脑酸,L-Camphoric acid,Camphoric acid, (-)-
Target: GluR
(E)-Cinnamamide
Cat.No: T13669
Synonym: trans-Cinnamamide,肉桂酰胺
Target: Others
(-)-Bornyl acetate
Cat.No: TN1448
Synonym: L-(-)-Bornyl acetate,左旋乙酸冰片酯,Bornyl acetate,(-)-乙酸龙脑酯
Target: p38 MAPK, NF-κB, JNK, Antifungal
Isodeoxycholic Acid
Cat.No: T36585
Synonym: isoDCA
Target: Chloride channel, Antibacterial
3-Epikatonic acid
Cat.No: TN2931
Synonym:
Target: Antifection
(-)-Taxifolin
Cat.No: T38497
Synonym: (-)-二氢槲皮素,(-)-Dihydroquercetin
Target:
Lysicamine
Cat.No: TN4471
Synonym:
Target: IL Receptor, Antifection
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