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321

抑制剂 & 化合物

89

天然产物

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Cat. No. Product Name Target Signaling Pathways
T6945 Vps34-PIK-III

PIK-III,VPS34-IN2

PI3K; Autophagy Autophagy; PI3K/Akt/mTOR signaling
Vps34-PIK-III (VPS34-IN2) 是 VPS34 酶活性的选择性抑制剂,IC50值为18 nM。它可抑制自噬并导致自噬底物稳定。
T7577 Angiotensin III, human, mouse

血管紧张素III,Angiotensin III, human, mouse(3TFA)

RAAS Endocrinology/Hormones
Angiotensin III, human, mouse (Angiotensin III, human, mouse(3TFA)) 是一种七肽,是血管紧张素 2 型受体 (AT2R) 激动剂,能够作用于 AT2R (IC50:0.648 nM)及 AT1R (IC50:21.1nM)。
T5612 Sudan III

Solvent Red 23,Tetrazobenzene-β-naphthol,111440 Red,Sudan Red III,苏丹红Ⅲ

Others Others
Sudan III (Solvent Red 23) 是一种疏水性双偶氮染料。
T60108 PDGFR Tyrosine Kinase Inhibitor III

PDGF Receptor Tyrosine Kinase Inhibitor III

PDGFR Angiogenesis; Tyrosine Kinase/Adaptors
PDGFR Tyrosine Kinase Inhibitor III (PDGF Receptor Tyrosine Kinase Inhibitor III) (PDGF Receptor Tyrosine Kinase Inhibitor III)是一种多激酶抑制剂,可抑制 PDGFR、EGFR、FGFR、PKA 和 PKC 等。PDGFR Tyrosine Kinase Inhibitor III 可用于肌萎缩侧索硬化症的研究。
T35885 KRM-III

Others Others
KRM-III 是一种具有口服活性的 T 细胞抗原受体 (TCR) 抑制剂,具有抗炎活性,可有效抑制 TCR 和肉豆蔻酸乙酸酯/佛波霉素/离子霉素诱导的 NFAT 核因子活化和 T 细胞增殖,IC50 约为 5 μM。
T26091 Riparin III

Riparin III is an alcamide isolated from Aniba riparia that has exhibited effects of antidepressant and anxiolytic activities in acute stress behavioral models.
T77628 Bisindolylmaleimide III

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
Bisindolylmaleimide III is a potent and selective inhibitor of protein kinase C (PKC).Bisindolylmaleimide III selectively interacts with PKCα or ribosomal S6 protein kinase 1 upon activation of these kinases.
T14914 Cdk1/2 Inhibitor III

CDK Cell Cycle/Checkpoint
Cdk1/2 Inhibitor III 是一种具有选择性的 Cdk1/2抑制剂,对 CDK1/cyclin B 的 IC50值为2.1μM。
T7944 VPS34 inhibitor 1 (Compound 19, PIK-III analogue)

PIK-III analogue

PI3K PI3K/Akt/mTOR signaling
VPS34 inhibitor 1 (Compound 19, PIK-III analogue) (PIK-III analogue) 是一种有效的选择性 VPS34抑制剂( IC50 : 15 nM)。
T22353 Lanthanum(III) chloride heptahydrate

Calcium Channel Membrane transporter/Ion channel; Metabolism
Lanthanum(III) chloride heptahydrate 是一种无机化合物,用于生化研究,阻断二价阳离子通道,尤其是钙通道的活性。
T38164 MnTBAP chloride

Mn(III)TBAP

MnTBAP chloride (Mn(III)TBAP) 是一种具有细胞渗透性的超氧化物歧化酶 (SOD) 模拟物和过氧亚硝酸盐清除剂,能使SOD-大肠杆菌的加倍时间减少了2倍。 MnTBAP chloride 通过上调 BMPR-II 和抑制 NFκB 信号传导展现抗炎作用。MnTBAP chloride 是一种锰卟啉配合物,具有抗氧化性能,具有用于研究慢性肾脏疾病 (CKDs) 纤维化反应的潜力。
T6759 AP-III-a4

ENOblock

Glucokinase Metabolism
AP-III-a4 (ENOblock) 是第一个非底物类似物,可直接与烯醇酶结合,IC50=0.576 uM,可阻碍体内癌细胞转移。
T2470 MDL-28170

Calpain Inhibitor III

Cysteine Protease; Proteasome Proteases/Proteasome; Ubiquitination
MDL-28170 (Calpain Inhibitor III) 是一种选择性的、有效的、具有膜渗透性的半胱氨酸蛋白酶 (calpain)抑制剂,可在全身给药后迅速穿过血脑屏障。它还能阻断γ-secretase。
T3956 Sodium ionophore III

ETH2120

Sodium Channel Membrane transporter/Ion channel
Sodium ionophore III (ETH2120) 是一种Na+载体,适用于测定血液、血浆、血清中的钠活性。
T5524 Aurora kinase inhibitor-3

Aurora Kinase Inhibitor III

Aurora Kinase Cell Cycle/Checkpoint; Chromatin/Epigenetic
Aurora kinase inhibitor-3 (Aurora Kinase Inhibitor III) 是一种有效的,选择性 Aurora A 激酶抑制剂,IC50为 42 nM。
T38459 Chromium(III) acetate

Chromium triacetate,Chromic acetate,Chromium acetate

Others Others
Chromium(III) acetate (Chromium acetate) 是一种小分子离子交联剂,是用于合成其他化合物的原料。
T12058 MK2-IN-3 hydrate

MK-2 Inhibitor III

ERK; MAPK; MNK MAPK
MK2-IN-3 hydrate (MK-2 Inhibitor III) 是一种口服有活性的、ATP 竞争性的MAPKAP-K2 (MK-2)选择性抑制剂(IC50:0.85 nM)。
TP1700L LGnRH-III, lamprey acetate(147859-97-0 free base)

GNRH Receptor GPCR/G Protein
LGnRH-III, lamprey acetate(147859-97-0 free base) 是 GnRH 家族进化上保守的成员,可刺激促性腺激素的分泌,同时刺激促黄体激素和促卵泡激素的分泌。
T2157 M344

MS 344,Histone Deacetylase Inhibitor III

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
M344 (Histone Deacetylase Inhibitor III) 是一种组蛋白去乙酰化酶抑制剂,IC50为 100 nM。
T2683 IWP L6

Porcn Inhibitor III,IWP-L6,Porcn Inhibitor III

Porcupine Stem Cells
IWP L6 (Porcn Inhibitor III) 是一种高活性的 Porcn 抑制剂(EC50:0.5 nM)。
T6363 4μ8C

IRE1 Inhibitor III

IRE1 Cell Cycle/Checkpoint
4μ8C (IRE1 Inhibitor III) 是一种有效且特异性的 IRE1α 抑制剂。
T65550 Gefitinib analog III

4-((3-Chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl acetate

Others Others
Gefitinib analog III (4-((3-Chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl acetate) 具有潜在的抗炎和抗肿瘤活性,可用于研究其在生物体内的相互作用和活性。
T36941 Sporidesmolide III

Sporidesmolide III is a cyclodepsipeptide originally isolated from P. chartarum.
T38334 Corynecin III

Corynecin III is a chloramphenicol-like antibiotic originally isolated from Corynebacterium. It inhibits the growth of Gram-positive and Gram-negative bacteria, including S. faecalis, S. aureus, B. subtilis, E. coli, P. aeruginosa, P. vulgaris, S. sonnei, S. typhosa, and K. pneumoniae (MICs = 2.6-83 μg/ml).
T4637 R-7050

TNF-α Antagonist III

TNF Apoptosis
R-7050 (TNF-α Antagonist III) 是一种肿瘤坏死因子受体拮抗剂,对 TNFα具有更高选择性。
T35378 Iron (III) hexacyanoferrate (II)

Prussian Blue,Berlin blue,Iron (III) hexacyanoferrate (II)

Others Others
Iron (III) hexacyanoferrate (II) (Prussian Blue, Berlin blue) 用作吸附剂,用于有效去除水溶液中的重金属(Cu (II)、Co (II)、Ni (II) 和 Pb (II))。
T35420 (S)-p38 MAPK Inhibitor III

(S)-p38 MAPK Inhibitor III

(S)-p38 MAPK inhibitor III is a methylsulfanylimidazole that inhibits p38 MAP kinase (IC50 = 0.90 μM in vitro). It is cell-permeable, potently blocking the release of TNF-α and IL-1β from human peripheral blood mononuclear cells (IC50s = 0.37 and 0.044 μM, respectively).
T39589 Human PD-L1 inhibitor III

Human PD-L1 inhibitor III

Human PD-L1 inhibitor III is a human PD-L1 inhibitor.
T21915 TBCA

Casein Kinase II Inhibitor III, TBCA

Casein Kinase Metabolism; Stem Cells
TBCA (Casein Kinase II Inhibitor III, TBCA) 是高选择性的酪蛋白激酶II CK2 抑制剂,IC50 为 110 nM,Ki 为 77 nM。TBCA 对 CK1、DYRK1A 和 其它 27 个激酶表现出选择性。
T14322 ARP-100

MMP-2 Inhibitor III

MMP Proteases/Proteasome
ARP-100 (MMP-2 Inhibitor III) 是选择性基质金属蛋白酶MMP-2抑制剂 (IC50=12 nM)。它对 MMP-1 (>50 μM),MMP-3 (4.5 μM),MMP-7 (>50 μM) 和MMP-9 (0.2 μM) 的抑制活性较小。它与 MMP-2 的 S1'口袋相互作用,并在体外对基质胶的侵袭模型中显示抗侵袭特性。
T83663 Mn(III) Protoporphyrin IX Chloride

Manganese(III) Protoporphyrin IX Chloride

Mn(III) protoporphyrin IX chloride是一种金属卟啉,当浓度为10 µM时,能在鸡胚肝细胞中诱导δ-氨基酮戊二酸合成酶和血红素加氧酶(HO)基因的mRNA表达,这些酶分别催化血红素生物合成和降解的限速步骤。Mn(III) protoporphyrin IX chloride含纳米仿生物已被用于体外纤维蛋白凝块的磁共振成像(MRI)研究。此外,它还被用于Mn(III) protoporphyrin IX-6(7)-甘氨酰-甘氨酰-L-组氨酸甲酯(MnGGH)的合成,MnGGH是一种具有微过氧化物酶活性的金属卟啉衍生物。
T35966 Mn(III)TMPyP

Mn(III)TMPyP is a manganese-porphyrin which acts as a superoxide dismutase (SOD) mimetic and peroxynitrite decomposition catalyst. SOD mimetics described to date are unstable and are capable of catalyzing undesired side-reactions in addition to the dismutation of the superoxide radical (O2-). Mn(III)TMPyP is an SOD mimetic with increased stability to pH and hydrogen peroxide. The rate constant for superoxide dismutation and peroxynitrite decomposition are 3.9 x 107 M-1s-1 and ~2 x 106 M-1s-1, re...
T9034 MK2-IN-3

MK2 Inhibitor III

MAPK MAPK
MK2-IN-3 (MK2 Inhibitor III) 是选择性的 MAPKAP-K2 (MK-2)抑制剂(IC50:8.5 nM),能够抑制 U937 细胞及体内 TNFα 的生成。
T9209 PF-05221304

STAT5 Inhibitor III,NSC 170984,R 6238,,Clesacostat

Acetyl-CoA Carboxylase Metabolism
PF-05221304 (NSC-170984) 是一种具有口服活性的肝脏靶向乙酰辅酶A 羧化酶 (ACC) 抑制剂,ACC 是脂肪酸合成的限速酶。
T1900 LDN-212854

LDN212854,BMP Inhibitor III

ALK; TGF-beta/Smad Angiogenesis; Stem Cells; Tyrosine Kinase/Adaptors
LDN-212854 (BMP Inhibitor III) 是一种新型BMP 抑制剂,抑制 ALK2 的IC50=1.3 nM,比对ALK1,ALK3,ALK4和ALK5的抑制性高2,66,1641和7135倍。
T3195 CVT-313

CVT 313,Cdk2 Inhibitor III,CVT313,NG26

CDK Cell Cycle/Checkpoint
CVT-313 (NG26) 是一种有效的、选择性的、可逆的和 ATP 竞争性抑制剂,可抑制 CDC5L 磷酸化,对 CDK2的 IC50为 0.5 μM。
T40331 Ftase inhibitor III

Ftase Inhibitor III, derived from a phenotypic screen, functions as an anion-dependent inhibitor of Farnesyltransferase.
T39700 Ga(III) protoporphyrin IX

Ga(III)protoporphyrin-IX, a model for interporphyrin interactions in malaria pigment, possesses potent antibacterial effects against gram-negative, gram-positive, and acid-fast bacteria. It exhibits high solubility in methanol (MeOH) and serves as a malarial pigment analogue for drug development, as well as a potential antibacterial agent.
T10322 Angiotensin III

Others Others
Angiotensin III is an agonist of angiotensin 1 (AT1) and AT2 receptor.
T39300 BNM-III-170

BNM-III-170 is able to inhibit HIV-1 viral entry into target cells.
T6326 BMS-345541

BMS-345541 free base,IKK Inhibitor III,BMS345541

IκB/IKK NF-κB
BMS-345541 (IKK Inhibitor III) 是选择性的 IKK 催化亚基 IKK-1 和 IKK-2 抑制剂,抑制 IKK-2 (IC50=0.3 nM) 和 IKK-1 (IC50=4 nM)。它与 IKK 的变构位点结合。
TP1969 ProTx III

Potent Nav1.7 blocker (IC50 = 2.5 nM). Also inhibits Nav1.1, Nav1.2, Nav1.3 and Nav1.6 in the nanomolar range. Exhibits no effects on Cav channels or nAChR at 5 μM. Demonstrates analgesic activity in vivo; antagonizes effects of scorpion-venom toxin OD1 a
TP2263 Jingzhaotoxin III

Others Others
NaV1.5 channels blocker
T69502 HSP47 inhibitor III

HSP47 inhibitor III suppressed collagen type I expression in human and mouse cells and suppressed the viability and migration of lung fibroblasts.
T10322L Angiotensin III TFA (12687-51-3 free base)

Angiotensin III TFA

Others Others
Angiotensin III TFA is an agonist of angiotensin 1 (AT1) and AT2 receptor.
T9563 Type III-Intermediate7

Type III-Intermediate7 是一种有用的有机化合物,可用于生命科学领域的相关研究,其产品编号为 T9563。
T31994 Grayanotoxin III

Deacylasebotoxin I,Deacetylandromedotoxin,Andromedol

Grayanotoxins are a group of closely related neurotoxins named after Leucothoe grayana, a plant native to Japan originally. Extract from leaves Leucothoe grayana (Ericaceae).
T26206 Spiramycin III

Foromacidin C,Spiramycin 3,Foromacidine C

Spiramycin III is an antibiotic within the erythromycin/carbomycin group of compounds.
TP1700 LGnRH-III, lamprey

GnRH III, an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion of both luteinizing and follicle-stimulating hormones.
T19372 Indium(III) isopropoxide

Others Others
Indium(III) Isopropoxide is an organo-metallic compound commonly used as a metal precursor and a hydrogen transfer catalyst in chemical reactions. It facilitates the conversion of benzylic alcohols to aldehydes or ketones through Oppenauer oxidation.

化合物

Vps34-PIK-III
Cat.No: T6945
Synonym: PIK-III,VPS34-IN2
Target: PI3K, Autophagy
Angiotensin III, human, mouse
Cat.No: T7577
Synonym: 血管紧张素III,Angiotensin III, human, mouse(3TFA)
Target: RAAS
Sudan III
Cat.No: T5612
Synonym: Solvent Red 23,Tetrazobenzene-β-naphthol,111440 Red,Sudan Red III,苏丹红Ⅲ
Target: Others
PDGFR Tyrosine Kinase Inhibitor III
Cat.No: T60108
Synonym: PDGF Receptor Tyrosine Kinase Inhibitor III
Target: PDGFR
KRM-III
Cat.No: T35885
Synonym:
Target: Others
Riparin III
Cat.No: T26091
Synonym:
Target:
Bisindolylmaleimide III
Cat.No: T77628
Synonym:
Target: PKC
Cdk1/2 Inhibitor III
Cat.No: T14914
Synonym:
Target: CDK
VPS34 inhibitor 1 (Compound 19, PIK-III analogue)
Cat.No: T7944
Synonym: PIK-III analogue
Target: PI3K
Lanthanum(III) chloride heptahydrate
Cat.No: T22353
Synonym:
Target: Calcium Channel
MnTBAP chloride
Cat.No: T38164
Synonym: Mn(III)TBAP
Target:
AP-III-a4
Cat.No: T6759
Synonym: ENOblock
Target: Glucokinase
MDL-28170
Cat.No: T2470
Synonym: Calpain Inhibitor III
Target: Cysteine Protease, Proteasome
Sodium ionophore III
Cat.No: T3956
Synonym: ETH2120
Target: Sodium Channel
Aurora kinase inhibitor-3
Cat.No: T5524
Synonym: Aurora Kinase Inhibitor III
Target: Aurora Kinase
Chromium(III) acetate
Cat.No: T38459
Synonym: Chromium triacetate,Chromic acetate,Chromium acetate
Target: Others
MK2-IN-3 hydrate
Cat.No: T12058
Synonym: MK-2 Inhibitor III
Target: ERK, MAPK, MNK
LGnRH-III, lamprey acetate(147859-97-0 free base)
Cat.No: TP1700L
Synonym:
Target: GNRH Receptor
M344
Cat.No: T2157
Synonym: MS 344,Histone Deacetylase Inhibitor III
Target: HDAC
IWP L6
Cat.No: T2683
Synonym: Porcn Inhibitor III,IWP-L6,Porcn Inhibitor III
Target: Porcupine
4μ8C
Cat.No: T6363
Synonym: IRE1 Inhibitor III
Target: IRE1
Gefitinib analog III
Cat.No: T65550
Synonym: 4-((3-Chloro-4-fluorophenyl)amino)-7-methoxyquinazolin-6-yl acetate
Target: Others
Sporidesmolide III
Cat.No: T36941
Synonym:
Target:
Corynecin III
Cat.No: T38334
Synonym:
Target:
R-7050
Cat.No: T4637
Synonym: TNF-α Antagonist III
Target: TNF
Iron (III) hexacyanoferrate (II)
Cat.No: T35378
Synonym: Prussian Blue,Berlin blue,Iron (III) hexacyanoferrate (II)
Target: Others
(S)-p38 MAPK Inhibitor III
Cat.No: T35420
Synonym: (S)-p38 MAPK Inhibitor III
Target:
Human PD-L1 inhibitor III
Cat.No: T39589
Synonym: Human PD-L1 inhibitor III
Target:
TBCA
Cat.No: T21915
Synonym: Casein Kinase II Inhibitor III, TBCA
Target: Casein Kinase
ARP-100
Cat.No: T14322
Synonym: MMP-2 Inhibitor III
Target: MMP
Mn(III) Protoporphyrin IX Chloride
Cat.No: T83663
Synonym: Manganese(III) Protoporphyrin IX Chloride
Target:
Mn(III)TMPyP
Cat.No: T35966
Synonym:
Target:
MK2-IN-3
Cat.No: T9034
Synonym: MK2 Inhibitor III
Target: MAPK
PF-05221304
Cat.No: T9209
Synonym: STAT5 Inhibitor III,NSC 170984,R 6238,,Clesacostat
Target: Acetyl-CoA Carboxylase
LDN-212854
Cat.No: T1900
Synonym: LDN212854,BMP Inhibitor III
Target: ALK, TGF-beta/Smad
CVT-313
Cat.No: T3195
Synonym: CVT 313,Cdk2 Inhibitor III,CVT313,NG26
Target: CDK
Ftase inhibitor III
Cat.No: T40331
Synonym:
Target:
Ga(III) protoporphyrin IX
Cat.No: T39700
Synonym:
Target:
Angiotensin III
Cat.No: T10322
Synonym:
Target: Others
BNM-III-170
Cat.No: T39300
Synonym:
Target:
BMS-345541
Cat.No: T6326
Synonym: BMS-345541 free base,IKK Inhibitor III,BMS345541
Target: IκB/IKK
ProTx III
Cat.No: TP1969
Synonym:
Target:
Jingzhaotoxin III
Cat.No: TP2263
Synonym:
Target: Others
HSP47 inhibitor III
Cat.No: T69502
Synonym:
Target:
Angiotensin III TFA (12687-51-3 free base)
Cat.No: T10322L
Synonym: Angiotensin III TFA
Target: Others
Type III-Intermediate7
Cat.No: T9563
Synonym:
Target:
Grayanotoxin III
Cat.No: T31994
Synonym: Deacylasebotoxin I,Deacetylandromedotoxin,Andromedol
Target:
Spiramycin III
Cat.No: T26206
Synonym: Foromacidin C,Spiramycin 3,Foromacidine C
Target:
LGnRH-III, lamprey
Cat.No: TP1700
Synonym:
Target:
Indium(III) isopropoxide
Cat.No: T19372
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TN1720 Gymnoside III

手参苷III

Others Others
Gymnoside III 是一种 2-异丁基苹果酸葡糖氧基氧基苄酯,分离自 Gymnadenia conopsea 的块茎。
T2S1193 Mogroside III-A1

罗汉果苷 III-A1

Others Others
Mogroside III-A1 是一种来自罗汉果 Swingle 的三萜糖苷。 Mogroside III-A1 一种无糖甜味剂。
T3902 Atractylenolide III

白术内酯 III,ICodonolactone,8β-Hydroxyasterolide

Apoptosis Apoptosis
Atractylenolide III (ICodonolactone) 是白术根茎主要成分,通过诱导细胞色素 c 的释放、上调 Bax 的表达和易位凋亡诱导因子,是治疗人肺癌的潜力。
T2197 10-Deacetylbaccatin III

10-脱乙酰巴卡丁 III,10-脱乙酰基巴卡丁III

Others Others
10-Deacetylbaccatin-III 是一种紫杉醇类似物制剂的中间体,具有抗癌活性。
TN7052 Crocin III

西红花苷 III,Crocetin-mono-(β-D-gentiobiosyl)-ester

Others Others
Crocin III (Crocetin-mono-(β-D-gentiobiosyl)-ester) 是一种来自于藏红花 (Crocus sutivusL)的藏红花素。Crocins 可用作香料和着色剂。Crocins 具有抗炎作用,能够抑制肿瘤细胞的细胞生长。
T5S0527 Rhodojaponin III

闹羊花素 Ⅲ,闹羊花毒素III

Others Others
Rhodojaponin III 是二萜类化合物,提取于Rhododendron molle 叶子,具有抗炎作用。
T5132 9-dihydro-13-acetylbaccatin III

13-乙酰基-9-羟基巴卡丁 III,13-Acetyl-9-dihydrobaccatin III,9-DHAB III

Apoptosis Apoptosis
9-dihydro-13-acetylbaccatin III (9-DHAB III) 是一种制备紫杉醇类似物的中间体。
T2788 Baccatin III

巴卡亭 Ⅲ,浆果赤霉素III,Baccatin Ⅲ

Others Others
Baccatin III (Baccatin Ⅲ) 是一种分离自太平洋紫杉树和其近缘种中的天然产物,能够减少 MDSCs 积累并抑制其功能,延缓肿瘤发展进程。
T5S0733 Picroside III

Others Others
Picroside III(胡黄连苷 III)是一种环烯醚萜苷,分离自传统中药胡黄连中。
TCS1188 Mogroside III

Others Others
Mogroside III 是一种三萜糖苷和非糖甜味剂。 Mogroside III 被人体肠道细菌转化,释放出次生Mogroside IIA1 和苷元莫格罗。
T3696 polygalaxanthone III

Others; P450 Metabolism; Others
Polygalaxanthone III 提取自远志polygala tenuifolia wild,可抑制CYP450酶。它能够抑制由 CYP2E1 催化的氯唑沙宗 6-羟基化(IC50:50.56μM)。
TN2302 Viscidulin III

Ganhuangenin

Glucosidase Metabolism
Viscidulin III (Ganhuangenin) 存在于黄芩中,可作为α-葡萄糖苷酶抑制剂。
T20819 Ammonium iron(III) citrate

柠檬酸铁铵,柠檬酸铁 (III) 铵,Ferric ammonium citrate

Others; Ferroptosis Apoptosis; Others
Ammonium iron(III) citrate (Ferric ammonium citrate) 是一种非运铁蛋白结合的铁的生理形式,会引起的细胞内铁超负荷从而导致细胞铁死亡,能增强蛋白质产生。
T5S0833 Astragaloside III

Antioxidant oxidation-reduction
Astragaloside III 是一种分离自黄芪中的一种天然产物。
T4S1849 Tubeimoside III

Others Others
Tubeimoside III 是一种具有抗炎和抗肿瘤活性的三萜皂苷,在体内具急性毒性。
TN1264 3'-O-Methylbatatasin III

Antifungal Microbiology/Virology
3'-O-Methylbatatasin III 是一种来自兰科植物白芨的天然化合物,具有抗生素活性和解痉活性。3'-O-Methylbatatasin III 具有抗真菌活性。
TN1433 Batatasin III

FAK; Others; Akt Angiogenesis; Cytoskeletal Signaling; Others; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors
Batatasin III 通过抑制上皮间质转化和 FAK-AKT 信号来抑制癌症迁移和侵袭,并具有抗癌活性。 Batatasin III 对整株生长有长期抑制作用,显示出抑制萌发活性。
TN1936 Mogroside III-E

罗汉果皂苷ⅢE

IL Receptor; TNF; TLR Apoptosis; Immunology/Inflammation
Mogroside IIIe 是一种葫芦烷型化合物,从罗汉果中分离得到,可抑制 NO 的释放,具有抗肺纤维化作用。
TN1383 Timosaponin B III

Anemarsaponin BIII,知母皂苷B3,知母皂苷BIII

Others; Platelet aggregation Others
Timosaponin B III (Anemarsaponin BIII) 是一种具有生物活性的甾体皂苷,从知母中分离出来。Timosaponin B III 具有抗炎、抗血小板聚集和抗抑郁作用。
TN2303 Viscumneoside III

槲寄生新甙III,槲寄生新苷III

Tyrosinase Proteases/Proteasome
Viscumneoside III 是一种二氢黄酮 O-糖苷,抑制酪氨酸酶 (tyrosinase),IC50 为 0.5 mM。Viscumneoside III 具有抗心绞痛作用。
TN1183 11-​Oxomogroside III

11-Oxomogroside III,11-O-罗汉果苷III

Others Others
11-Oxomogroside III is a natural product from Siraitia grosvenorii Swingle.
T3395 Timosaponin AIII

Filiferin B,知母皂苷 A-III,AneMarsaponin A3,Timosaponin A3

AChE; mTOR Neuroscience; PI3K/Akt/mTOR signaling
Timosaponin AIII (Timosaponin A3) 是一种乙酰胆碱酯酶活性抑制剂,其IC50=35.4 μM。
T82970 Aristolactam A III

Aristololactam A III

Aristolactam A III (Aristololactam A III) 为一生物碱,具潜在细胞毒性,并可从鱼腥草中分离。
T81764 Monofucosyllacto-N-hexaose III

MFLNH III

Monofucosyllacto-N-hexaose III(MFLNH III)是一种具有特定生物学功能的中性人乳寡糖(HMO)。
TN1935 Mogroside III A2

Mogroside III-A2,罗汉果苷IIIA2,罗汉果苷 III A2

Others Others
Mogroside III-A2 exhibits inhibitory effects with IC50 values of 346-400 mol ratio/32 pmol TPA. and shows weak inhibitory effects on activation of (+/-)-(E)-methyl-2-[(E)-hydroxyimino]-5-nitro-6-methoxy-3-hexemide (NOR 1), a nitric oxide (NO) donor.
T36227 Beauveriolide III

Beauveriolide III is a cyclodepsipeptide that has been found inBeauveriaand an inhibitor of lipid droplet formation.1It inhibits lipid droplet formation when used at concentrations of 3 and 10 μM, as well as inhibits cholesterol synthesis (IC50= 0.41 μM), in primary mouse peritoneal macrophages.1,2Beauveriolide III also inhibits acyl-coenzyme A:cholesterol acyltransferase (ACAT) activity in mouse macrophage membranes (IC50= 5.5 μM).2Beauveriolide III (25 and 50 mg/kg) reduces the size of aortic ...
T11288 Filipin III

Antifungal Microbiology/Virology
Filipin III 是 从菌株KPE18H 中提取得到,具有显著的抗真菌活性。
T5S1252 Prosapogenin A

重楼皂苷E,Progenin III

Apoptosis; Others Apoptosis; Others
Prosapogenin A (Progenin III) 是藜芦中的一种天然产物,通过抑制 STAT3 信号通路和糖酵解,可诱导人癌细胞凋亡,有抗癌作用。
TN1382 Anemarrhenasaponin III

Others Others
Anemarrhenasaponin III is a natural product
T13897 Soyasaponin III

Others Others
Soyasaponin III is one of the main potentially bioactive saponins found in soy (Glycine max) and related products,and can induce apoptosis in Hep-G2 cells.
T2217 Cephalomannine

Baccatin III,三尖杉宁碱

Microtubule Associated Cytoskeletal Signaling
Cephalomannine (Baccatin III) 是一种从云南红豆杉中提取的紫杉醇衍生物,具有抗肿瘤活性,可用于癌症研究。
T3394 Timosaponin BII

知母皂苷BII,Prototimosaponin A III

Beta Amyloid; Others; BACE Neuroscience; Others
Timosaponin BII (Prototimosaponin A III) 是一种甾体皂苷,发现于知母根茎中,具有神经保护、抗炎和抗氧化作用。
TL0007 Bisdemethoxycurcumin

双去甲氧基姜黄素,Curcumin III,Didemethoxycurcumin

Epigenetic Reader Domain; Wnt/beta-catenin Chromatin/Epigenetic; Cytoskeletal Signaling; Stem Cells
Bisdemethoxycurcumin (Curcumin III) 是一种具有抗炎及抗氧化作用的姜黄素。
TN5600 Paniculoside III

Paniculoside III is a natural product from the metabolites of the algicolous fungus Stevia paniculata.
TN3485 Bakkenolide III

Others Others
Bakkenolide III may have cytotoxicity.
T24242 Kaikasaponin III

Kaikasaponin III is isolated from Abrus Cantoniensis. It also has an antihepatotoxic activity.
TN3842 Diarylcomosol III

Others Others
Diarylcomosol III shows inhibitory effects on melanogenesis in B16 melanoma cells, it is a promising therapeutic agent for the treatment of skin disorders.
TN5837 Creoside III

Creoside III 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5837,CAS号为 1038602-12-8。
T19247 Coproporphyrin III

Zincphyrin

Others Others
Coproporphyrin III is a derivative of porphyrin.
T6473 Dioscin

山药,CCRIS 4123,Collettiside III,Saponin

Apoptosis; Autophagy Apoptosis; Autophagy
Dioscin (Collettiside III) 是一种来源植物的天然甾体皂苷,针对多种癌细胞有较好的抗癌活性。
T30156 Asebotoxin III

Asebotoxin III is a diterpenoid obtained from the leaves of Asebi, Pieris japonica.
TN4757 Peucedanocoumarin III

Others Others
Peucedanocoumarin Ⅲ can induce rice resistance to blast disease.
TN2662 19-Hydroxybaccatin III

Others Others
19-Hydroxybaccatin III, 10-deacetylcephalomannine, and 10-deacetyltaxol are new antitumor taxanes from Taxus wallichiana.
TN5239 Viscidulin III tetraacetate

Others Others
Viscidulin III tetraacetate 是一种天然产物,可用于生命科学领域的相关研究。其产品编号为 TN5239,CAS号为 96684-81-0。
TN6544 24-Hydroxymomordicine III

24-Hydroxymomordicine III 可用于生命科学领域的相关研究,其产品编号为 TN6544。
TN2615 13-O-Cinnamoylbaccatin III

Others Others
13-O-Cinnamoylbaccatin III is a natural product from Taxus yunnanensis.
T1882 Meisoindigo

N-Methylisoindigotin,Methylisoindigotin,Natura-α,甲异靛,Dian III,异甲靛

Apoptosis Apoptosis
Meisoindigo (Natura-α) 是 Indirubin 的衍生物,可以造成急性髓细胞性白血病细胞周期在 G0/G1 期停滞,并诱导凋亡,具有高抗肿瘤活性。
TN3251 7-Xylosyl-10-deacetylbaccatin III

Others Others
7-Xylosyl-10-deacetylbaccatin III is a natural product from Taxus brevifolia.
T2822 Ginsenoside Rb1

Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III

ATPase; Mitophagy; IRAK; NF-κB; Autophagy; HSV Autophagy; Immunology/Inflammation; Membrane transporter/Ion channel; Microbiology/Virology; NF-κB
Ginsenoside Rb1 (Gypenoside Ⅲ) 是中药人参的成分,可能具有抑制或阻止肿瘤生长的特性。
T6S1688 (1E,6E)-Bis(demethoxy)curcumin

(1E,6E)-1,7-双(4-羟基苯基)庚-1,6-二烯-3,5-二酮,Curcumin III,双去甲氧基姜黄素,Didemethoxycurcumin,BDMC

Apoptosis; Others; Autophagy Apoptosis; Autophagy; Others
(1E,6E)-Bis(demethoxy)curcumin (Curcumin III) 是姜黄素的天然去甲氧基衍生物,具有抗炎和抗癌活性。
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天然产物

Gymnoside III
Cat.No: TN1720
Synonym: 手参苷III
Target: Others
Mogroside III-A1
Cat.No: T2S1193
Synonym: 罗汉果苷 III-A1
Target: Others
Atractylenolide III
Cat.No: T3902
Synonym: 白术内酯 III,ICodonolactone,8β-Hydroxyasterolide
Target: Apoptosis
10-Deacetylbaccatin III
Cat.No: T2197
Synonym: 10-脱乙酰巴卡丁 III,10-脱乙酰基巴卡丁III
Target: Others
Crocin III
Cat.No: TN7052
Synonym: 西红花苷 III,Crocetin-mono-(β-D-gentiobiosyl)-ester
Target: Others
Rhodojaponin III
Cat.No: T5S0527
Synonym: 闹羊花素 Ⅲ,闹羊花毒素III
Target: Others
9-dihydro-13-acetylbaccatin III
Cat.No: T5132
Synonym: 13-乙酰基-9-羟基巴卡丁 III,13-Acetyl-9-dihydrobaccatin III,9-DHAB III
Target: Apoptosis
Baccatin III
Cat.No: T2788
Synonym: 巴卡亭 Ⅲ,浆果赤霉素III,Baccatin Ⅲ
Target: Others
Picroside III
Cat.No: T5S0733
Synonym:
Target: Others
Mogroside III
Cat.No: TCS1188
Synonym:
Target: Others
polygalaxanthone III
Cat.No: T3696
Synonym:
Target: Others, P450
Viscidulin III
Cat.No: TN2302
Synonym: Ganhuangenin
Target: Glucosidase
Ammonium iron(III) citrate
Cat.No: T20819
Synonym: 柠檬酸铁铵,柠檬酸铁 (III) 铵,Ferric ammonium citrate
Target: Others, Ferroptosis
Astragaloside III
Cat.No: T5S0833
Synonym:
Target: Antioxidant
Tubeimoside III
Cat.No: T4S1849
Synonym:
Target: Others
3'-O-Methylbatatasin III
Cat.No: TN1264
Synonym:
Target: Antifungal
Batatasin III
Cat.No: TN1433
Synonym:
Target: FAK, Others, Akt
Mogroside III-E
Cat.No: TN1936
Synonym: 罗汉果皂苷ⅢE
Target: IL Receptor, TNF, TLR
Timosaponin B III
Cat.No: TN1383
Synonym: Anemarsaponin BIII,知母皂苷B3,知母皂苷BIII
Target: Others, Platelet aggregation
Viscumneoside III
Cat.No: TN2303
Synonym: 槲寄生新甙III,槲寄生新苷III
Target: Tyrosinase
11-​Oxomogroside III
Cat.No: TN1183
Synonym: 11-Oxomogroside III,11-O-罗汉果苷III
Target: Others
Timosaponin AIII
Cat.No: T3395
Synonym: Filiferin B,知母皂苷 A-III,AneMarsaponin A3,Timosaponin A3
Target: AChE, mTOR
Aristolactam A III
Cat.No: T82970
Synonym: Aristololactam A III
Target:
Monofucosyllacto-N-hexaose III
Cat.No: T81764
Synonym: MFLNH III
Target:
Mogroside III A2
Cat.No: TN1935
Synonym: Mogroside III-A2,罗汉果苷IIIA2,罗汉果苷 III A2
Target: Others
Beauveriolide III
Cat.No: T36227
Synonym:
Target:
Filipin III
Cat.No: T11288
Synonym:
Target: Antifungal
Prosapogenin A
Cat.No: T5S1252
Synonym: 重楼皂苷E,Progenin III
Target: Apoptosis, Others
Anemarrhenasaponin III
Cat.No: TN1382
Synonym:
Target: Others
Soyasaponin III
Cat.No: T13897
Synonym:
Target: Others
Cephalomannine
Cat.No: T2217
Synonym: Baccatin III,三尖杉宁碱
Target: Microtubule Associated
Timosaponin BII
Cat.No: T3394
Synonym: 知母皂苷BII,Prototimosaponin A III
Target: Beta Amyloid, Others, BACE
Bisdemethoxycurcumin
Cat.No: TL0007
Synonym: 双去甲氧基姜黄素,Curcumin III,Didemethoxycurcumin
Target: Epigenetic Reader Domain, Wnt/beta-catenin
Paniculoside III
Cat.No: TN5600
Synonym:
Target:
Bakkenolide III
Cat.No: TN3485
Synonym:
Target: Others
Kaikasaponin III
Cat.No: T24242
Synonym:
Target:
Diarylcomosol III
Cat.No: TN3842
Synonym:
Target: Others
Creoside III
Cat.No: TN5837
Synonym:
Target:
Coproporphyrin III
Cat.No: T19247
Synonym: Zincphyrin
Target: Others
Dioscin
Cat.No: T6473
Synonym: 山药,CCRIS 4123,Collettiside III,Saponin
Target: Apoptosis, Autophagy
Asebotoxin III
Cat.No: T30156
Synonym:
Target:
Peucedanocoumarin III
Cat.No: TN4757
Synonym:
Target: Others
19-Hydroxybaccatin III
Cat.No: TN2662
Synonym:
Target: Others
Viscidulin III tetraacetate
Cat.No: TN5239
Synonym:
Target: Others
24-Hydroxymomordicine III
Cat.No: TN6544
Synonym:
Target:
13-O-Cinnamoylbaccatin III
Cat.No: TN2615
Synonym:
Target: Others
Meisoindigo
Cat.No: T1882
Synonym: N-Methylisoindigotin,Methylisoindigotin,Natura-α,甲异靛,Dian III,异甲靛
Target: Apoptosis
7-Xylosyl-10-deacetylbaccatin III
Cat.No: TN3251
Synonym:
Target: Others
Ginsenoside Rb1
Cat.No: T2822
Synonym: Gypenoside Ⅲ,人参皂苷Rb1,人参皂苷 Rb1,Gypenoside III
Target: ATPase, Mitophagy, IRAK, NF-κB, Autophagy, HSV
(1E,6E)-Bis(demethoxy)curcumin
Cat.No: T6S1688
Synonym: (1E,6E)-1,7-双(4-羟基苯基)庚-1,6-二烯-3,5-二酮,Curcumin III,双去甲氧基姜黄素,Didemethoxycurcumin,BDMC
Target: Apoptosis, Others, Autophagy
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